Safety and Efficacy Study of YZJ-1139 Tablets in Insomnia Disorder

NCT ID: NCT06975514

Last Updated: 2025-07-15

Study Results

Results pending

The study team has not published outcome measurements, participant flow, or safety data for this trial yet. Check back later for updates.

Basic Information

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Recruitment Status

RECRUITING

Clinical Phase

PHASE3

Total Enrollment

60 participants

Study Classification

INTERVENTIONAL

Study Start Date

2025-03-25

Study Completion Date

2025-09-30

Brief Summary

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The main purpose of this study is to assess efficacy of YZJ-1139 for 28 days in adult subjects with insomnia disorder. Efficacy will be evaluated on objective and subjective sleep parameters.

Detailed Description

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Conditions

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Insomnia Disorder

Study Design

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Allocation Method

RANDOMIZED

Intervention Model

PARALLEL

Primary Study Purpose

TREATMENT

Blinding Strategy

DOUBLE

Participants Investigators

Study Groups

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YZJ-1139 group

Group Type EXPERIMENTAL

YZJ-1139

Intervention Type DRUG

YZJ-1139 20mg tablets, once daily in the evening

Zolpidem group

Group Type ACTIVE_COMPARATOR

Zolpidem

Intervention Type DRUG

Zolpidem 10mg tablets, once daily in the evening

Interventions

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YZJ-1139

YZJ-1139 20mg tablets, once daily in the evening

Intervention Type DRUG

Zolpidem

Zolpidem 10mg tablets, once daily in the evening

Intervention Type DRUG

Eligibility Criteria

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Inclusion Criteria

1. Males and females, aged ≥ 18 to \< 65 years.
2. Meet the clinical diagnostic criteria for insomnia disorder as defined in ICSD-3 criteria.
3. sTSO ≥ 30 min for at least 3 nights per week and/or sWASO ≥ 60 min for at least 3 nights per week within 4 weeks prior to screening.
4. Able to recognize 26 English letters and MMSE score indicats no cognitive impairment.
5. During the run-in period and on Day 1 of the treatment period, sTSO ≥ 30 min for at least 3 nights in the last 7 sleep diaries and/or sWASO ≥ 60 min for at least 3 nights out of 7 nights as confirmed by the sleep diary prior to PSG monitoring.
6. PSG results for 2 consecutive nights during the run-in period should meet the following conditions:

1. The mean LPS ≥ 30 min for 2 nights and ≥ 20 min for any one night; And/or the mean WASO ≥ 60 min for 2 nights, and ≥ 45 min either night.
2. The mean SE ≤ 85% for 2nights, with the SE ≤ 87.5% for both nights .
7. ISI score ≥ 15 at screening and on Day 1 of the treatment period .
8. Have a bedtime between 9 p.m. and 1 a.m., wake up between 5 a.m. and 10 a.m., and stay in bed for 6.5 to 9 hours for at least 5 nights in the last 7 sleep diaries as confirmed by the sleep diary prior to PSG monitoring during the run-in period and on Day 1 of the treatment period.
9. Reproductive-age male and female participants must agree to use effective contraceptive measures from the screening visit through at least 30 days after the last dose of double-blind study treatment, and must not be planning to become pregnant or donate sperm/eggs during this period.
10. Understand the study procedures and contents, voluntarily participate in the clinical study and sign the written Informed Consent Form, have good compliance during participation in the study, and are willing to attend the visits.

Exclusion Criteria

1. Hypersensitivity to YZJ-1139 tablets or zolpidem or to their excipients.
2. Have serious endocrine diseases, hematological diseases, cardiovascular and cerebrovascular diseases, gastrointestinal diseases, liver and kidney diseases, autoimmune diseases, impaired respiratory function or other related diseases, or have other medical history that may affect the safety of the subjects or interfere with the study assessments in the opinion of the investigator.
3. Have insomnia disorder due to other causes such as chronic pain, headache, eczema, neurodermatitis, allergic rhinitis, and serious dermatitis (difficulty sleeping due to physical reasons, difficulty falling asleep due to medical reasons).
4. Current or previous history of psychiatric or neurological disease such as epilepsy, schizophrenia, bipolar mental disorder, neurodevelopmental retardation, and cognitive disorder, or previous history of other mental illness that may affect the safety of the subjects or interfere with the study assessments in the opinion of the investigator.
5. Previous history of sleep-related respiratory disorders including obstructive sleep apnea (with or without continuous positive airway pressure \[CPAP\] therapy), periodic limb movement disorder, myasthenia gravis, restless legs syndrome, circadian rhythm sleep disturbances, narcolepsy or other sleep disorders: subjects with restless legs syndrome which is diagnosed by relevant diagnostic and treatment guidelines should be excluded. Those who have been cured of the above diseases can be enrolled.
6. Have previous complex sleep behaviors, such as sleep driving, sleep eating, and sleep phone calls.
7. Have nocturia increased caused by urinary tract infection, urinary tract injury or prostatic disorder.
8. Hyperthyroidism.
9. History of alcohol abuse (defined as regular daily alcohol consumption exceeding the following criteria: approximately 720 mL of beer, or 240 mL of wine, or 60 mL of liquor) within the past 6 months.
10. Regular daily consumption of excessive tea and coffee drinks (defined as consumption of \> 4 cups of caffeinated beverages or \> 400 mg of caffeine per day), or daily habituation to drinking caffeinated beverages beyond 18:00.
12. Have any lifestyle that interferes with the study process or may interfere with sleep: for example, there will be travels across 3 or more time zones (mainland China is considered as 1 time zone) within the next 2 weeks or during the study period, or there will be shift work (night and daytime shift).
13. History of drug abuse within the past 2 years, or positive urine drug screening for any indicator; history of drug taking or addiction, which is known through questioning.
14. Have received any hypnotics, antidepressants, antipsychotic drugs, anticholinergics, memory-enhancing drugs, antihistamines, centrally acting analgesics, centrally acting muscle relaxants, central nervous system stimulants, CYP3A inducers, CYP3A inhibitors, traditional Chinese medicines and traditional Chinese medicinal products with sleep-improving effects, or any other therapies for insomnia disorder within 1 week prior to the run-in period or within 5 half-lives of the investigational product, whichever is longer.
15. Plan to undergo surgery during the study.
16. Depression: Hamilton Depression Scale (HAMD) score ≥ 18; anxiety: Hamilton Anxiety Scale (HAMA) score ≥ 14.
17. Suicidal ideation with or without plan at screening or within 6 months prior to screening (score ≥ 3 on item 3 \[suicide\] of HAMD, or select "Yes" on item 3, 4 or 5 of suicidal ideation subscale of C-SSRS), or have any suicidal behavior in the past 10 years (as assessed by the suicidal ideation subscale of C-SSRS).
18. ECG at screening shows QTcF interval prolongation (QTcF \> 450 ms, QTcF=QT/(RR\^0.33)).
19. AST or ALT \> 2 × the upper limit of normal (ULN), or Cr \> 1.5 × ULN.
20. Known to be human immunodeficiency virus (HIV) antibody positive at screening.
21. Apnea-hypopnea index \[AHI\] or periodic limb movement index \[PLMI\] \> 10 times/hour detected by PSG monitoring during the run-in period.
22. Unable to avoid vaccination within 1 month prior to screening.
23. Enrolled in another clinical trial and used any investigational drug within 1 month or 5 half-lives (whichever is longer) prior to the run-in period, or participation in another investigational trial at the same time during this trial.
24. Previously participated in any clinical trial of YZJ-1139; or treated with other orexin receptor antagonists of appropriate amount and sufficient duration and who, in the opinion of the investigator, have failed treatment due to efficacy or safety.
25. Pregnant or lactating women.
26. Have other conditions that make the subject unsuitable for participation in the clinical study in the opinion of the investigator.
Minimum Eligible Age

18 Years

Maximum Eligible Age

65 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

No

Sponsors

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Shanghai Haiyan Pharmaceutical Technology Co., Ltd.

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Locations

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Peking University People's Hospital

Beijing, , China

Site Status RECRUITING

ChengDu Second People's Hospital

Chengdu, , China

Site Status RECRUITING

ChongQing Traditional Chinese Medicine Hospital

Chongqing, , China

Site Status RECRUITING

Deyang People's Hospital

Deyang, , China

Site Status RECRUITING

The First Affiliated Hospital of Jinan University (Guangzhou Overseas Chinese Hospital)

Guangzhou, , China

Site Status RECRUITING

The First Affiliated Hospital of Shandong First Medical University (Qianfoshan Hospital)

Jinan, , China

Site Status RECRUITING

The Second Affiliated Hospital Of NanChang University

Nanchang, , China

Site Status RECRUITING

The First Affiliated Hospital of Ningbo University

Ningbo, , China

Site Status RECRUITING

ShengJing Hospital Of China Medical University

Shenyang, , China

Site Status RECRUITING

The Third Hospital of Hebei Medical University

Shijiazhuang, , China

Site Status RECRUITING

SuZhou GuangJi Hospital

Suzhou, , China

Site Status RECRUITING

The Second Affiliated Hospital of Soochow University

Suzhou, , China

Site Status RECRUITING

Tianjin Anding Hospital

Tianjin, , China

Site Status RECRUITING

Wuhan No.1 Hospital

Wuhan, , China

Site Status RECRUITING

Yan'an University Xianyang Hospital

Yan’an, , China

Site Status RECRUITING

The Second Affiliated Hospital of Zhengzhou University

Zhengzhou, , China

Site Status RECRUITING

Countries

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China

Facility Contacts

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fang han

Role: primary

13511074278

jian wang

Role: primary

13689063972

chenyu li

Role: primary

18983744422

ping liu

Role: primary

15982902050

jiyang pan

Role: primary

13380095658

jiyou tang

Role: primary

15866635908

lijun xu

Role: primary

18970907115

yunxin ji

Role: primary

13857422531

Xiao li

Role: primary

18940256863

hanqiao wang

Role: primary

18533112218

yansong liu

Role: primary

19951316780

chunfeng liu

Role: primary

13606210609

xingjun zhang

Role: primary

13034336931

junhua mei

Role: primary

18995635558

qiaorong xu

Role: primary

13809100163

chunling liu

Role: primary

13298425452

Other Identifiers

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YZJ-1139-3-02

Identifier Type: -

Identifier Source: org_study_id

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