A First-in-human Study to Learn How Safe BAY 3713372 is and How it Works in Participants With MTAP-deleted Solid Tumors

NCT ID: NCT06914128

Last Updated: 2025-11-10

Study Results

Results pending

The study team has not published outcome measurements, participant flow, or safety data for this trial yet. Check back later for updates.

Basic Information

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Recruitment Status

RECRUITING

Clinical Phase

PHASE1/PHASE2

Total Enrollment

370 participants

Study Classification

INTERVENTIONAL

Study Start Date

2025-03-21

Study Completion Date

2029-06-17

Brief Summary

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The study treatment, BAY 3713372, is under development to treat MTAP (methylthioadenosine phosphorylase)-deleted solid tumors. It is thought to work by blocking the protein arginine N-methyltransferase 5 (PRMT5). This may kill the MTAP-deleted cancer cells while sparing the normal cells.

The main objective of this first-in-human study is to learn how safe BAY 3713372 is, how the body processes it, and how well it works in people with MTAP-deleted solid tumors.

For this, the researchers will study and analyze:

* the number of participants who have adverse events (AEs) after receiving different doses of BAY 3713372 and the AE's severity.
* the number of participants who experience dose-limiting toxicities (DLTs) after receiving different doses of BAY 3713372, the DLT's severity and how often they happened. A DLT is a pre-defined medical problem caused by a specific dose of a drug that is too severe to continue using that dose.
* the total amount of BAY 3713372 in participants' blood (also called AUC) over time after single and multiple doses.
* the highest level of BAY 3713372 in participants' blood (also called Cmax) after single and multiple doses.

Other than the main objective, researchers will also check for the number of participants who show a response to treatment and how long they live without the cancer getting worse.

The study participants will take part in one of the seven distinct groups or "intervention cohorts" of the study. The study will start with a dose escalation phase where distinct groups of participants will receive different doses of BAY 3713372 alone to find the dose that is deemed safe and works best for the participants. When this dose has been found, a larger number of participants will receive BAY 3713372 alone or with other treatments in a dose expansion phase.

Participants may take the study treatment as long as they benefit from the treatment without any severe medical problems.

Participants will visit the study site:

* at least twice before the treatment starts
* multiple times when they start taking the treatment
* once after 30 days of receiving the last dose and every 9 weeks after that until the cancer worsens, or the participant stops for any other reason

During the study, the doctors and their study team will:

* check participants' health by performing tests such as blood and urine tests, and checking heart health using an electrocardiogram
* check if the participants' cancer has grown and/or spread using computed tomography (CT) or magnetic resonance imaging (MRI) and, if needed, bone scan
* take tumor samples

The study doctors and their team will contact the participants every 3 months until 2 years after the last participant's last dose or the end of the study to learn about the participant's health.

Detailed Description

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Conditions

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MTAP-deleted Solid Tumors

Keywords

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Solid Tumors Non-small cell lung cancer NSCLC Pancreatic adenocarcinoma PDAC

Study Design

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Allocation Method

NON_RANDOMIZED

Intervention Model

SEQUENTIAL

Primary Study Purpose

TREATMENT

Blinding Strategy

NONE

Study Groups

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Dose Escalation (Intervention Cohort 1)

For the escalation part, different dose levels of BAY 3713372 administered as monotherapy are planned.

Group Type EXPERIMENTAL

BAY 3713372

Intervention Type DRUG

Daily oral administration

Backfill cohorts in Intervention Cohort 1 (Dose Escalation)

Backfill cohorts may be initiated concurrently with dose escalation cohorts to generate additional safety, pharmacokinetic, and pharmacodynamic data to facilitate the selection of the optimal doses for use in further development.

Group Type EXPERIMENTAL

BAY 3713372

Intervention Type DRUG

Daily oral administration

Dose Expansion (Intervention Cohort 1)

Dose expansion with BAY 3713372 monotherapy in selected participants with MTAP-deleted solid tumors.

Group Type EXPERIMENTAL

BAY 3713372

Intervention Type DRUG

Daily oral administration

Dose Expansion (Intervention Cohort 2)

Dose expansion with BAY 3713372 monotherapy in participants with MTAP-deleted non-small cell lung cancer (NSCLC).

Group Type EXPERIMENTAL

BAY 3713372

Intervention Type DRUG

Daily oral administration

Dose Expansion (Intervention Cohort 3)

Dose expansion with BAY 3713372 in combination with other treatments in participants with MTAP-deleted NSCLC.

Group Type EXPERIMENTAL

BAY 3713372

Intervention Type DRUG

Daily oral administration

Dose Expansion (Intervention Cohort 4)

Dose expansion with BAY 3713372 in combination with other treatments in participants with MTAP-deleted NSCLC.

Group Type EXPERIMENTAL

BAY 3713372

Intervention Type DRUG

Daily oral administration

Dose Expansion (Intervention Cohort 5)

Dose expansion with BAY 3713372 monotherapy in participants with MTAP-deleted pancreatic ductal adenocarcinoma (PDAC).

Group Type EXPERIMENTAL

BAY 3713372

Intervention Type DRUG

Daily oral administration

Dose Expansion (Intervention Cohort 6)

Dose expansion with BAY 3713372 in combination with other treatments in participants with MTAP-deleted PDAC.

Group Type EXPERIMENTAL

BAY 3713372

Intervention Type DRUG

Daily oral administration

Interventions

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BAY 3713372

Daily oral administration

Intervention Type DRUG

Eligibility Criteria

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Inclusion Criteria

* Participant must be ≥ 18 years old of age, or the legal age of consent in the jurisdiction of the country in which the study takes place, at the time of signing the informed consent.
* At least one measurable lesion that would qualify as target lesion by Response Evaluation Criteria in Solid Tumors, Version 1.1 (RECIST 1.1).
* Homozygous MTAP-deletion identified through molecular testing from a locally certified laboratory.
* Eastern Cooperative Oncology Group (ECOG) performance status of 0 or 1.

Exclusion Criteria

* Previous additional cancer else than the one evaluated in this study within the past 2 years except for basal or squamous cell carcinoma of the skin, carcinoma in situ of the cervix, superficial bladder tumors, localized prostate cancer or other tumors that in the opinion of the investigator, are considered cured or not immediately life-threatening, and will not interfere with the scientific goals of this study.
* A marked prolongation of QT/QTc interval at screening (e.g., repeated demonstration of a QTc interval \>450 ms). Participants with permanent pacemakers (i.e., a paced rhythm) may be eligible after discussion with the sponsor.
* Cardiac history comprising:

* History of congestive heart failure Class \>II according to the New York Heart Association Functional Classification.
* Myocardial infarction less than 6 months before the start of study intervention.
* Serious cardiac arrhythmias requiring treatment or any clinically important abnormalities in rhythm, conduction or morphology on resting ECG with the exception of atrial fibrillation which is well-controlled and requires only digoxin or beta blockers.
* Unstable angina within 4 weeks before start of study intervention.
Minimum Eligible Age

18 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

No

Sponsors

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Bayer

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Locations

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Sarah Cannon Research Institute at HCA HealthONE Presbyterian St. Luke's

Denver, Colorado, United States

Site Status RECRUITING

Sarah Cannon Research Institute at Florida Cancer Specialists- Lake Nona

Orlando, Florida, United States

Site Status RECRUITING

START | Midwest

Grand Rapids, Michigan, United States

Site Status RECRUITING

SCRI Oncology Partners

Nashville, Tennessee, United States

Site Status RECRUITING

NEXT Dallas - Oncology Department

Irving, Texas, United States

Site Status RECRUITING

START | San Antonio

San Antonio, Texas, United States

Site Status RECRUITING

Chris O'Brien Lifehouse

Camperdown, New South Wales, Australia

Site Status RECRUITING

Concord Repatriation General Hospital (CRGH) (Concord Hospital) - Concord Cancer Centre

Concord, New South Wales, Australia

Site Status NOT_YET_RECRUITING

Calvary Mater Hospital Newcastle

Waratah, New South Wales, Australia

Site Status NOT_YET_RECRUITING

Northern Hospital

Epping, Victoria, Australia

Site Status NOT_YET_RECRUITING

Ghent University Hospital | Drug Research Unit Department

Ghent, , Belgium

Site Status NOT_YET_RECRUITING

Centre Hospitalier Universitaire (CHU) de Liege - Domaine Universitaire du Sart Tilman - Medical Oncology

Liège, , Belgium

Site Status NOT_YET_RECRUITING

Beijing Cancer Hospital - Oncology Department

Beijing, Beijing Municipality, China

Site Status NOT_YET_RECRUITING

Tongji Hosp. of Tongji Med Coll, Huazhong Uni of Sci & Tech.

Wuhan, Hubei, China

Site Status NOT_YET_RECRUITING

Masarykova Univerzita - Masarykuv Onkologicky Ustav (MOU) - Klinika Komplexni Onkologicke Pece (KKOP)

Brno, , Czechia

Site Status NOT_YET_RECRUITING

Fakultní Nemocnice Olomouc

Olomouc, , Czechia

Site Status NOT_YET_RECRUITING

Rigshospitalet - Kræftbehandling

Copenhagen, , Denmark

Site Status NOT_YET_RECRUITING

Odense University Hospital - Oncology Department

Odense C, , Denmark

Site Status NOT_YET_RECRUITING

Fondazione IRCCS Istituto Nazionale dei Tumori - S. C. Oncologia Medica 1

Milan, , Italy

Site Status NOT_YET_RECRUITING

Fondazione Policlinico Universitario Agostino Gemelli IRCCS - UOC Fase I

Roma, , Italy

Site Status NOT_YET_RECRUITING

Humanitas Mirasole S.p.A. - Oncologia Medica ed Ematologia

Rozzano, , Italy

Site Status NOT_YET_RECRUITING

Shizuoka Cancer Center

Sunto, Shizuoka, Japan

Site Status NOT_YET_RECRUITING

National Cancer Center Hospital

Chuo-ku, Tokyo, Japan

Site Status NOT_YET_RECRUITING

The Cancer Institute Hospital of JFCR

Koto-ku, Tokyo, Japan

Site Status NOT_YET_RECRUITING

Nederlands Kanker Instituut

Amsterdam, , Netherlands

Site Status NOT_YET_RECRUITING

Erasmus Medisch Centrum

Rotterdam, , Netherlands

Site Status NOT_YET_RECRUITING

National University Hospital Medical Centre

Singapore, , Singapore

Site Status RECRUITING

National Cancer Center Singapore - Oncology Department

Singapore, , Singapore

Site Status RECRUITING

Hospital Hm Nou Delfos - Oncologia

Barcelona, , Spain

Site Status NOT_YET_RECRUITING

Hospital Universitari Vall d'Hebron- Oncology Service

Barcelona, , Spain

Site Status NOT_YET_RECRUITING

Hospital San Pedro

Logroño, , Spain

Site Status NOT_YET_RECRUITING

The START Center for Cancer Care - Mardrid-Fundacion Jimenez Diaz (START Madrid-FJD)

Madrid, , Spain

Site Status NOT_YET_RECRUITING

Hospital Universitario Virgen De La Victoria - Oncology

Málaga, , Spain

Site Status NOT_YET_RECRUITING

NEXT Oncology- Next Madrid

Pozuelo de Alarcón, , Spain

Site Status NOT_YET_RECRUITING

Instituto de Investigacion Sanitaria (INCLIVA) (Institute of Health Research Hospital Clinic of Valencia)

Valencia, , Spain

Site Status NOT_YET_RECRUITING

Sahlgrenska Universitetssjukhuset - Klinisk prövningsenhet Fas I/FIH

Gothenburg, , Sweden

Site Status NOT_YET_RECRUITING

Karolinska Universitetssjukhuset - Fas I-enheten Solna CKC

Stockholm, , Sweden

Site Status NOT_YET_RECRUITING

The Royal Marsden NHS Foundation Trust | Sutton - Oak Foundation Drug Development Unit

London, Greater London, United Kingdom

Site Status NOT_YET_RECRUITING

The Christie NHS Foundation Trust | Christie Hospital - Experimental Cancer Medicine Team

Manchester, , United Kingdom

Site Status NOT_YET_RECRUITING

Countries

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United States Australia Belgium China Czechia Denmark Italy Japan Netherlands Singapore Spain Sweden United Kingdom

Central Contacts

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Bayer Clinical Trials Contact

Role: CONTACT

Phone: (+)1-888-84 22937

Email: [email protected]

Related Links

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https://clinicaltrials.bayer.com/study/22931

Click here to find further information and, after study completion, the study results according to Bayer's transparency standards.

Other Identifiers

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2025-520623-24-00

Identifier Type: REGISTRY

Identifier Source: secondary_id

22931

Identifier Type: -

Identifier Source: org_study_id