Safety, Tolerability, and Pharmacokinetics of Lumateperone Long-Acting Injectable Formulations in Patients With Schizophrenia or Schizoaffective Disorder

NCT ID: NCT06627413

Last Updated: 2025-03-24

Study Results

Results pending

The study team has not published outcome measurements, participant flow, or safety data for this trial yet. Check back later for updates.

Basic Information

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Recruitment Status

RECRUITING

Clinical Phase

PHASE1

Total Enrollment

72 participants

Study Classification

INTERVENTIONAL

Study Start Date

2024-08-23

Study Completion Date

2026-03-31

Brief Summary

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Study ITI-007-037 is a Phase 1b, open-label study to evaluate the safety, tolerability, and PK of lumateperone long-acting injectable (LAI) formulations after a single intramuscular injection in patients with stale schizophrenia or schizoaffective disorder.

Detailed Description

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Conditions

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Schizophrenia or Schizoaffective

Study Design

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Allocation Method

RANDOMIZED

Intervention Model

PARALLEL

This study includes 3 sequential study parts (Parts A, B and C). Part A consists of 4 cohorts (Cohorts 1 to 4), Part B of up to 3 cohorts (Cohorts 5 to 7), and Part C of up to 2 cohorts (Cohorts 8 and 9). Within each study part, cohorts may be enrolled in parallel.
Primary Study Purpose

TREATMENT

Blinding Strategy

NONE

Study Groups

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Cohort 1

Lumateperone 42 mg once daily for 5 days following by a single IM dose of lumateperone 100 mg LAI formulation X500-E2 after a 5-day washout

Group Type EXPERIMENTAL

Lumateperone Capsule

Intervention Type DRUG

Lumateperone 42 mg capsule, oral administration

Lumateperone LAI

Intervention Type DRUG

Lumateperone LAI X500-E2 IM injection

Cohort 2

Lumateperone 42 mg once daily for 5 days following by a single IM dose of lumateperone 100 mg LAI formulation X500-E3 after a 5-day washout

Group Type EXPERIMENTAL

Lumateperone Capsule

Intervention Type DRUG

Lumateperone 42 mg capsule, oral administration

Lumateperone LAI

Intervention Type DRUG

Lumateperone LAI X500-E3 IM injection

Cohort 3

Lumateperone 42 mg once daily for 5 days following by a single IM dose of lumateperone 100 mg LAI formulation X500-X2 after a 5-day washout

Group Type EXPERIMENTAL

Lumateperone Capsule

Intervention Type DRUG

Lumateperone 42 mg capsule, oral administration

Lumateperone LAI

Intervention Type DRUG

Lumateperone LAI X500-X2 IM injection

Cohort 4

Lumateperone 42 mg once daily for 5 days following by a single IM dose of lumateperone 100 mg LAI formulation X500-X5 after a 5-day washout

Group Type EXPERIMENTAL

Lumateperone Capsule

Intervention Type DRUG

Lumateperone 42 mg capsule, oral administration

Lumateperone LAI

Intervention Type DRUG

Lumateperone LAI X500-X5 IM injection

Cohort 5

Lumateperone 42 mg once daily for 5 days following by a single IM dose (\> 100 mg) of lumateperone LAI formulation (chosen from Part A) after a 5-day washout

Group Type EXPERIMENTAL

Lumateperone Capsule

Intervention Type DRUG

Lumateperone 42 mg capsule, oral administration

Lumateperone LAI

Intervention Type DRUG

Lumateperone LAI (X500-E2 or X500-E3 or X500-X2 or X500-X5) IM injection

Cohort 6

Lumateperone 42 mg once daily for 5 days following by a single IM dose (\> 100 mg) of lumateperone LAI formulation (chosen from Part A) after a 5-day washout

Group Type EXPERIMENTAL

Lumateperone Capsule

Intervention Type DRUG

Lumateperone 42 mg capsule, oral administration

Lumateperone LAI

Intervention Type DRUG

Lumateperone LAI (X500-E2 or X500-E3 or X500-X2 or X500-X5) IM injection

Cohort 7

Lumateperone 42 mg once daily for 5 days following by a single IM dose (\> 100 mg) of lumateperone LAI formulation (chosen from Part A) after a 5-day washout

Group Type EXPERIMENTAL

Lumateperone Capsule

Intervention Type DRUG

Lumateperone 42 mg capsule, oral administration

Lumateperone LAI

Intervention Type DRUG

Lumateperone LAI (X500-E2 or X500-E3 or X500-X2 or X500-X5) IM injection

Cohort 8

Lumateperone 42 mg once daily for 5 days following by a single IM dose (\> dose in Part B) of lumateperone LAI formulation (chosen from Part B) after a 5-day washout

Group Type EXPERIMENTAL

Lumateperone Capsule

Intervention Type DRUG

Lumateperone 42 mg capsule, oral administration

Lumateperone LAI

Intervention Type DRUG

Lumateperone LAI (X500-E2 or X500-E3 or X500-X2 or X500-X5) IM injection

Cohort 9

Lumateperone 42 mg once daily for 5 days following by a single IM dose (\> dose in Part B) of lumateperone LAI formulation (chosen from Part B) after a 5-day washout

Group Type EXPERIMENTAL

Lumateperone Capsule

Intervention Type DRUG

Lumateperone 42 mg capsule, oral administration

Lumateperone LAI

Intervention Type DRUG

Lumateperone LAI (X500-E2 or X500-E3 or X500-X2 or X500-X5) IM injection

Interventions

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Lumateperone Capsule

Lumateperone 42 mg capsule, oral administration

Intervention Type DRUG

Lumateperone LAI

Lumateperone LAI X500-E2 IM injection

Intervention Type DRUG

Lumateperone LAI

Lumateperone LAI X500-E3 IM injection

Intervention Type DRUG

Lumateperone LAI

Lumateperone LAI X500-X2 IM injection

Intervention Type DRUG

Lumateperone LAI

Lumateperone LAI X500-X5 IM injection

Intervention Type DRUG

Lumateperone LAI

Lumateperone LAI (X500-E2 or X500-E3 or X500-X2 or X500-X5) IM injection

Intervention Type DRUG

Eligibility Criteria

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Inclusion Criteria

* Male or female patients between 18 and 55 years of age, inclusive;
* Clinical diagnosis of schizophrenia or schizoaffective disorder according to Diagnostic and Statistical Manual of Mental Disorders (DSM-5);
* Clinically stable and free from acute exacerbation of psychosis for at least 3 months prior to Screening;
* Clinical Global Impression - Severity (CGI-S) score ≤ 3 at Screening and prior to dosing on Day 1;
* Body mass index (BMI) between 18.0 and 38.0 kg/m2, inclusive at Screening, and a minimum body weight of 50 kg at Screening.

Exclusion Criteria

* History of psychiatric condition other than schizophrenia that, in the Investigator's opinion, may be detrimental to participation in the study;
* Any suicidal ideation or wish to be dead within the past 6 months of Screening, any suicide attempt within the past 2 years prior to Screening, or any current concern for the patient's safety based on the Columbia-Suicide Severity Rating Scale (C-SSRS) (excluding self-injurious, non-suicidal behavior), and/or Investigator assessment that the patient is a safety risk to him/herself or others;
* Clinically significant abnormality within 2 years of Screening that in the Investigator's opinion may place the patient at risk or interfere with study outcome variables;
* Has a QT interval corrected for heart rate using Fridericia formula \> 450 msec in males or \> 470 msec in females, or evidence of clinically significant bundle branch blocks on ECG at Screening.
Minimum Eligible Age

18 Years

Maximum Eligible Age

55 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

No

Sponsors

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Intra-Cellular Therapies, Inc.

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Locations

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Clinical Site 2

Los Alamitos, California, United States

Site Status RECRUITING

Clinical Site 3

Atlanta, Georgia, United States

Site Status RECRUITING

Clinical Site 4

Decatur, Georgia, United States

Site Status RECRUITING

Clinical Site 1

Marlton, New Jersey, United States

Site Status RECRUITING

Countries

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United States

Central Contacts

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ITI Clinical Trials

Role: CONTACT

6464409333

Facility Contacts

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Clinical Site 2

Role: primary

Clinical Site 3

Role: primary

Clinical Site 4

Role: primary

Clinical Site 1

Role: primary

Other Identifiers

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ITI-007-037

Identifier Type: -

Identifier Source: org_study_id

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