A Phase 2 Study of AMG 193 in Participants With MTAP-deleted Advanced NSCLC (MTAPESTRY 201)

NCT ID: NCT06593522

Last Updated: 2025-12-12

Study Results

Results pending

The study team has not published outcome measurements, participant flow, or safety data for this trial yet. Check back later for updates.

Basic Information

Get a concise snapshot of the trial, including recruitment status, study phase, enrollment targets, and key timeline milestones.

Recruitment Status

RECRUITING

Clinical Phase

PHASE2

Total Enrollment

200 participants

Study Classification

INTERVENTIONAL

Study Start Date

2024-12-26

Study Completion Date

2030-11-29

Brief Summary

Review the sponsor-provided synopsis that highlights what the study is about and why it is being conducted.

The main objective of the study is to characterize safety and efficacy of 2 dose levels of AMG 193 by investigator, and to evaluate AMG 193 monotherapy efficacy by Blinded Independent Central Review (BICR).

Detailed Description

Dive into the extended narrative that explains the scientific background, objectives, and procedures in greater depth.

Conditions

See the medical conditions and disease areas that this research is targeting or investigating.

MTAP-deleted NSCLC

Study Design

Understand how the trial is structured, including allocation methods, masking strategies, primary purpose, and other design elements.

Allocation Method

RANDOMIZED

Intervention Model

SEQUENTIAL

Primary Study Purpose

TREATMENT

Blinding Strategy

NONE

Study Groups

Review each arm or cohort in the study, along with the interventions and objectives associated with them.

Part 1: Dose Evaluation

Participants will be randomized to receive one of 2 active dose levels of AMG 193 orally (PO) daily (QD) in 28 days cycles. Part 1 of the study will determine the recommended phase 2 dose (RP2D).

Group Type EXPERIMENTAL

AMG 193

Intervention Type DRUG

Film-coated tablet

Part 2: Dose Expansion

Participants will receive AMG 193 PO QD in 28-day cycles at the RP2D.

Group Type EXPERIMENTAL

AMG 193

Intervention Type DRUG

Film-coated tablet

Interventions

Learn about the drugs, procedures, or behavioral strategies being tested and how they are applied within this trial.

AMG 193

Film-coated tablet

Intervention Type DRUG

Eligibility Criteria

Check the participation requirements, including inclusion and exclusion rules, age limits, and whether healthy volunteers are accepted.

Inclusion Criteria

* Histologically or cytologically confirmed metastatic or unresectable locally advanced MTAP-deleted (Homozygous deletion of MTAP) NSCLC
* Participants will have received and progressed or experienced disease recurrence on or after receiving at least 1 prior systemic therapy for locally advanced and unresectable or metastatic disease.
* Either an archival tissue sample or an archival block must be available.
* Life expectancy of greater than 3 months, in the opinion of the investigator.
* Participants who have had brain metastases and have been appropriately treated with radiation therapy or surgery ending at least 14 days before study day 1 are eligible.
* Participants with untreated asymptomatic brain metastases smaller or equal to 2 cm in size (per lesion if more than one) and not requiring corticosteroid treatment are eligible.

Exclusion Criteria

Disease Related

• Tumors harboring the following mutations amenable to targeted therapies: epidermal growth factor receptor (EGFR), ALK receptor tyrosine kinase (ALK), ROS proto-oncogene 1 (ROS1), neurotrophic tyrosine receptor kinase (NTRK), MET proto-oncogene (MET), B-Raf proto-oncogene (BRAF), RET proto-oncogene (RET), Human epidermal growth factor receptor 2 (HER2/ERBB2), KRAS proto-oncogene G12C (KRAS G12C).

Other Medical Conditions

* Major surgery within 28 days of study day 1.
* Untreated symptomatic central nervous system (CNS) metastatic disease regardless of size or asymptomatic brain metastases greater than 2 cm per lesion.
Minimum Eligible Age

18 Years

Maximum Eligible Age

99 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

No

Sponsors

Meet the organizations funding or collaborating on the study and learn about their roles.

Amgen

INDUSTRY

Sponsor Role lead

Responsible Party

Identify the individual or organization who holds primary responsibility for the study information submitted to regulators.

Responsibility Role SPONSOR

Principal Investigators

Learn about the lead researchers overseeing the trial and their institutional affiliations.

MD

Role: STUDY_DIRECTOR

Amgen

Locations

Explore where the study is taking place and check the recruitment status at each participating site.

City of Hope National Medical Center

Duarte, California, United States

Site Status RECRUITING

City of Hope Orange County Lennar Foundation Cancer Center

Duarte, California, United States

Site Status RECRUITING

Cedars-Sinai Medical Center

Los Angeles, California, United States

Site Status RECRUITING

Valkyrie Clinical Trials

Los Angeles, California, United States

Site Status RECRUITING

University of California Los Angeles

Los Angeles, California, United States

Site Status RECRUITING

Rocky Mountain Cancer Centers

Denver, Colorado, United States

Site Status RECRUITING

Eastern Connecticut Hematology and Oncology Associates

Norwich, Connecticut, United States

Site Status RECRUITING

Hartford HealthCare Cancer Institute - Manchester

Plainville, Connecticut, United States

Site Status RECRUITING

Medstar Georgetown University Hospital

Washington D.C., District of Columbia, United States

Site Status RECRUITING

Our Lady of the Lake Cancer Institute

Baton Rouge, Louisiana, United States

Site Status RECRUITING

Trinity Health Saint Joseph Mercy Ann Arbor

Ann Arbor, Michigan, United States

Site Status RECRUITING

Cancer and Hematology Centers of Western Michigan

Grand Rapids, Michigan, United States

Site Status RECRUITING

Sarah Cannon Research Institute Oncology Partners

Nashville, Tennessee, United States

Site Status RECRUITING

United States Oncology Regulatory Affairs Corporate Office

Nashville, Tennessee, United States

Site Status RECRUITING

Texas Oncology Central/South Texas

Austin, Texas, United States

Site Status RECRUITING

Sarah Cannon Research Institute

Dallas, Texas, United States

Site Status RECRUITING

Texas Oncology - Dallas Fort Worth

Dallas, Texas, United States

Site Status RECRUITING

US Oncology Research Investigational Products Center

Irving, Texas, United States

Site Status RECRUITING

Texas Oncology Northeast Texas

Tyler, Texas, United States

Site Status RECRUITING

Virginia Cancer Specialists PC

Fairfax, Virginia, United States

Site Status RECRUITING

GenesisCare -North Shore Oncology

St Leonards, New South Wales, Australia

Site Status RECRUITING

Calvary Mater Newcastle Hospital

Waratah, New South Wales, Australia

Site Status RECRUITING

Mater Hospital Brisbane

South Brisbane, Queensland, Australia

Site Status RECRUITING

Cancer Research South Australia

Adelaide, South Australia, Australia

Site Status RECRUITING

Núcleo de Oncologia da Bahia

Salvador, Estado de Bahia, Brazil

Site Status RECRUITING

Liga Norte-Riograndense Contra O Cancer

Natal, Rio Grande do Norte, Brazil

Site Status RECRUITING

Hospital Sao Lucas da Pontificia Universidade Catolica do Rio Grande do Sul

Porto Alegre, Rio Grande do Sul, Brazil

Site Status RECRUITING

Hospital Nossa Senhora da Conceicao

Porto Alegre, Rio Grande do Sul, Brazil

Site Status RECRUITING

Fundacao Pio Xii Barretos

Barretos, São Paulo, Brazil

Site Status RECRUITING

Fund Fac Reg Med Sao Jose Rio Preto

São José do Rio Preto, São Paulo, Brazil

Site Status RECRUITING

Instituto do Cancer Estado SP Icesp

São Paulo, São Paulo, Brazil

Site Status RECRUITING

Fundacao Antonio Prudente - Hosp AC Camargo

São Paulo, São Paulo, Brazil

Site Status RECRUITING

Instituto de Educacao Pesquisa e Gestao em Saude

Rio de Janeiro, , Brazil

Site Status RECRUITING

Centro Paulista de Oncologia

São Paulo, , Brazil

Site Status RECRUITING

Cross Cancer Institute

Edmonton, Alberta, Canada

Site Status RECRUITING

William Osler Health System - Brampton Civic Hospital

Brampton, Ontario, Canada

Site Status RECRUITING

London Health Sciences Centre

London, Ontario, Canada

Site Status RECRUITING

Princess Margaret Cancer Centre

Toronto, Ontario, Canada

Site Status RECRUITING

McGill University Health Centre Glen Site

Montreal, Quebec, Canada

Site Status RECRUITING

Beijing Cancer Hospital

Beijing, Beijing Municipality, China

Site Status RECRUITING

Mengchao Hepatobiliary Hospital of Fujian Medical University

Fuzhou, Fujian, China

Site Status RECRUITING

Henan Cancer Hospital

Zhengzhou, Henan, China

Site Status RECRUITING

The First Affiliated Hospital of Zhengzhou University

Zhengzhou, Henan, China

Site Status RECRUITING

Union Hospital Tongji Medical College Huazhong University of Science and Technology

Wuhan, Hubei, China

Site Status RECRUITING

The Second Xiangya Hospital of Central South University

Changsha, Hunan, China

Site Status RECRUITING

Jilin Cancer Hospital

Changchun, Jilin, China

Site Status RECRUITING

Jinan Central Hospital

Jinan, Shandong, China

Site Status RECRUITING

Shanghai East Hospital

Shanghai, Shanghai Municipality, China

Site Status RECRUITING

West China Hospital Sichuan University

Chengdu, Sichuan, China

Site Status RECRUITING

The First Affiliated Hospital Zhejiang University School Of Medicine

Hangzhou, Zhejiang, China

Site Status RECRUITING

Zhejiang Cancer Hospital

Hangzhou, Zhejiang, China

Site Status RECRUITING

Beijing Cancer Hospital

Beijing, , China

Site Status RECRUITING

Beijing Chest Hospital, Capital Medical University

Beijing, , China

Site Status RECRUITING

Masarykuv onkologicky ustav

Brno, , Czechia

Site Status RECRUITING

Fakultni nemocnice Olomouc

Olomouc, , Czechia

Site Status RECRUITING

Vseobecna fakultni nemocnice v Praze

Prague, , Czechia

Site Status RECRUITING

Fakultni Thomayerova nemocnice

Prague, , Czechia

Site Status RECRUITING

Queen Mary Hospital, The University of Hong Kong

Hong Kong, , Hong Kong

Site Status RECRUITING

Prince of Wales Hospital, Chinese University of Hong Kong

Shatin, New Territories, , Hong Kong

Site Status RECRUITING

Aichi Cancer Center

Nagoya, Aichi-ken, Japan

Site Status RECRUITING

National Cancer Center Hospital East

Kashiwa-shi, Chiba, Japan

Site Status RECRUITING

Shizuoka Cancer Center

Sunto-gun, Shizuoka, Japan

Site Status RECRUITING

National Cancer Center Hospital

Chuo-ku, Tokyo, Japan

Site Status RECRUITING

The Cancer Institute Hospital of Japanese Foundation for Cancer Research

Koto-ku, Tokyo, Japan

Site Status RECRUITING

Wakayama Medical University Hospital

Wakayama, Wakayama, Japan

Site Status RECRUITING

Pauls Stradins Clinical University Hospital

Riga, , Latvia

Site Status RECRUITING

Riga East Clinical University Hospital

Riga, , Latvia

Site Status RECRUITING

Nederlands Kanker Instituut Antoni van Leeuwenhoekziekenhuis

Amsterdam, , Netherlands

Site Status RECRUITING

Sint Jansdal Ziekenhuis

Harderwijk, , Netherlands

Site Status RECRUITING

Erasmus Medisch Centrum

Rotterdam, , Netherlands

Site Status RECRUITING

Unidade Local de Saude de Braga, EPE

Braga, , Portugal

Site Status RECRUITING

Fundacao Champalimaud

Lisbon, , Portugal

Site Status RECRUITING

Hospital Cuf porto

Porto, , Portugal

Site Status RECRUITING

Instituto Portugues de Oncologia do Porto Francisco Gentil, EPE

Porto, , Portugal

Site Status RECRUITING

National University Hospital

Singapore, , Singapore

Site Status RECRUITING

National Cancer Centre Singapore

Singapore, , Singapore

Site Status RECRUITING

Cha Bundang Medical Center, Cha University

Seongnam-si, Gyeonggi-do, , South Korea

Site Status RECRUITING

Severance Hospital Yonsei University Health System

Seoul, , South Korea

Site Status RECRUITING

Ajou University Hospital

Suwon-si Gyeonggi-do, , South Korea

Site Status RECRUITING

The Catholic University of Korea St Vincents Hospital

Suwon-si, Gyeonggi-do, , South Korea

Site Status RECRUITING

Universitaetsspital Basel

Basel, , Switzerland

Site Status RECRUITING

Hopitaux Universitaires de Geneve

Geneva, , Switzerland

Site Status RECRUITING

Kantonsspital Sankt Gallen

Sankt Gallen, , Switzerland

Site Status RECRUITING

Taichung Veterans General Hospital

Taichung, , Taiwan

Site Status RECRUITING

National Cheng Kung University Hospital

Tainan, , Taiwan

Site Status RECRUITING

National Taiwan University Hospital

Taipei, , Taiwan

Site Status RECRUITING

Adana Sehir Egitim ve Arastirma Hastanesi

Adana, , Turkey (Türkiye)

Site Status RECRUITING

Gazi Universitesi Saglik Arastirma ve Uygulama Merkezi Gazi Hastanesi

Ankara, , Turkey (Türkiye)

Site Status RECRUITING

Ankara Bilkent Sehir Hastanesi

Ankara, , Turkey (Türkiye)

Site Status RECRUITING

Memorial Bahcelievler Hastanesi

Istanbul, , Turkey (Türkiye)

Site Status RECRUITING

Bagcilar Medipol Mega Universite Hastanesi

Istanbul, , Turkey (Türkiye)

Site Status RECRUITING

Countries

Review the countries where the study has at least one active or historical site.

United States Australia Brazil Canada China Czechia Hong Kong Japan Latvia Netherlands Portugal Singapore South Korea Switzerland Taiwan Turkey (Türkiye)

Central Contacts

Reach out to these primary contacts for questions about participation or study logistics.

Amgen Call Center

Role: CONTACT

866-572-6436

Related Links

Access external resources that provide additional context or updates about the study.

http://www.amgentrials.com

AmgenTrials clinical trials website

Other Identifiers

Review additional registry numbers or institutional identifiers associated with this trial.

20230153

Identifier Type: -

Identifier Source: org_study_id

More Related Trials

Additional clinical trials that may be relevant based on similarity analysis.

Etirinotecan Pegol (NKTR-102) in NSCLC
NCT01773109 COMPLETED PHASE2