A Drug-drug Interaction Study Evaluating the Perpetrator Potential of LY4100511 (DC-853) on Midazolam, Repaglinide, Digoxin, Rosuvastatin in Healthy Participants

NCT ID: NCT06503679

Last Updated: 2025-01-24

Study Results

Results pending

The study team has not published outcome measurements, participant flow, or safety data for this trial yet. Check back later for updates.

Basic Information

Get a concise snapshot of the trial, including recruitment status, study phase, enrollment targets, and key timeline milestones.

Recruitment Status

COMPLETED

Clinical Phase

PHASE1

Total Enrollment

49 participants

Study Classification

INTERVENTIONAL

Study Start Date

2024-07-16

Study Completion Date

2024-12-31

Brief Summary

Review the sponsor-provided synopsis that highlights what the study is about and why it is being conducted.

The main purpose of this study is to assess the safety and tolerability and pharmacokinetics of LY4100511 (DC-853) when administered alone or in the presence of cytochrome P450 substrates in healthy participants.

Detailed Description

Dive into the extended narrative that explains the scientific background, objectives, and procedures in greater depth.

Conditions

See the medical conditions and disease areas that this research is targeting or investigating.

Healthy

Study Design

Understand how the trial is structured, including allocation methods, masking strategies, primary purpose, and other design elements.

Allocation Method

NON_RANDOMIZED

Intervention Model

PARALLEL

Primary Study Purpose

BASIC_SCIENCE

Blinding Strategy

NONE

Study Groups

Review each arm or cohort in the study, along with the interventions and objectives associated with them.

LY4100511 Dose 1 + Midazolam + Repaglinide (Cohort 1)

Participants will receive an oral dose 1 of LY4100511 and single dose of midazolam and repaglinide.

Group Type EXPERIMENTAL

LY4100511 (DC-853) Dose 1

Intervention Type DRUG

Administered orally

Midazolam

Intervention Type DRUG

Administered orally

Repaglinide

Intervention Type DRUG

Administered orally

LY4100511 Dose 2 + Midazolam + Repaglinide (Cohort 2)

Participants will receive up to an oral dose 2 of LY4100511 and single dose of midazolam and repaglinide. Dosing will not proceed until a satisfactory review of the safety and tolerability data from lower dose level is performed.

Group Type EXPERIMENTAL

LY4100511 (DC-853) Dose 2

Intervention Type DRUG

Administered orally

Midazolam

Intervention Type DRUG

Administered orally

Repaglinide

Intervention Type DRUG

Administered orally

LY4100511 Dose 3 + Digoxin and Rosuvastatin (Cohort 3)

Participants will recive an oral dose 3 of LY4100511 and single dose of digoxin and rosuvastatin.

Group Type EXPERIMENTAL

LY4100511 (DC-853) Dose 3

Intervention Type DRUG

Administered orally

Digoxin

Intervention Type DRUG

Administered orally

Rosuvastatin

Intervention Type DRUG

Administered orally

Interventions

Learn about the drugs, procedures, or behavioral strategies being tested and how they are applied within this trial.

LY4100511 (DC-853) Dose 1

Administered orally

Intervention Type DRUG

LY4100511 (DC-853) Dose 2

Administered orally

Intervention Type DRUG

LY4100511 (DC-853) Dose 3

Administered orally

Intervention Type DRUG

Midazolam

Administered orally

Intervention Type DRUG

Repaglinide

Administered orally

Intervention Type DRUG

Digoxin

Administered orally

Intervention Type DRUG

Rosuvastatin

Administered orally

Intervention Type DRUG

Eligibility Criteria

Check the participation requirements, including inclusion and exclusion rules, age limits, and whether healthy volunteers are accepted.

Inclusion Criteria

* Females must be of childbearing potential
* Males must agree to use contraception
* Have body mass index (BMI) between 18.0 and 32.0 kilogram/square meter (kg/m²), inclusive, and a body weight of greater than or equal to 50 kg.
* In good health, as determined by no clinically significant findings from medical history, 12-lead ECG and vital signs measurements, and clincial laboratory evaluations (congentical nonhemolytic hyperbilirubinemia) at screening and check-in, and from the physical examination at check-in as assessed by the investigator.

Exclusion Criteria

* Have a 12-lead ECG abnormality that, in the opinion of the investigator,

* increases the risks associated with participating in the study
* may confound ECG data analysis
* a QTCF \>450 msec for males, or \>470 msec for females

* short PR interval \<120 msec or PR interval \>220 msec
* second or third degree atrioventricular block
* intraventricular conduction delay with QRS \>120 msec
* complete right bundle branch block
* left bundle branch block, or
* Wolff Parkinson-White syndrome.
* Have had current or recent acute infection
* Show evidence of active or latent tuberculosis (TB)
* Had any surgical procedures within 12 weeks prior to screening or any planned surgical procedure scheduled to occur during the study.
* Have a history or presence of multiple or severe allergies, or an anaphylactic reaction to prescription or non prescription drugs.
* Are immunocompromised
* Presence of active suicidal ideation or positive suicide behavior using baseline/screening version of the C-SSRS
Minimum Eligible Age

18 Years

Maximum Eligible Age

55 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

Yes

Sponsors

Meet the organizations funding or collaborating on the study and learn about their roles.

DICE Therapeutics, Inc., a wholly owned subsidiary of Eli Lilly and Company

INDUSTRY

Sponsor Role lead

Responsible Party

Identify the individual or organization who holds primary responsibility for the study information submitted to regulators.

Responsibility Role SPONSOR

Principal Investigators

Learn about the lead researchers overseeing the trial and their institutional affiliations.

Call 1-877-CTLILLY (1-877-285-4559) or 1-317-615-4559 Mon - Fri 9 AM - 5 PM Eastern time (UTC/GMT - 5 hours, EST)

Role: STUDY_DIRECTOR

Eli Lilly and Company

Locations

Explore where the study is taking place and check the recruitment status at each participating site.

Fortrea Clinical Research Unit

Dallas, Texas, United States

Site Status

Countries

Review the countries where the study has at least one active or historical site.

United States

Other Identifiers

Review additional registry numbers or institutional identifiers associated with this trial.

J5C-MC-FOAF, DC-853104

Identifier Type: OTHER

Identifier Source: secondary_id

27110

Identifier Type: -

Identifier Source: org_study_id

More Related Trials

Additional clinical trials that may be relevant based on similarity analysis.

Transporter Cocktail Mutual Interaction
NCT02854527 COMPLETED PHASE1