A Drug-Drug Interaction Study of Orforglipron (LY3502970) in Healthy Overweight and Obese Participants

NCT ID: NCT06186622

Last Updated: 2024-07-22

Study Results

Results pending

The study team has not published outcome measurements, participant flow, or safety data for this trial yet. Check back later for updates.

Basic Information

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Recruitment Status

COMPLETED

Clinical Phase

PHASE1

Total Enrollment

50 participants

Study Classification

INTERVENTIONAL

Study Start Date

2024-01-02

Study Completion Date

2024-07-10

Brief Summary

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The main purpose of this study is to determine effect of orforglipron capsule formulation on the amount of digoxin, rosuvastatin, acetaminophen, midazolam, and simvastatin (each given alone and together with orforglipron) that enters the bloodstream and how long it takes the body to eliminate them when administered orally in healthy overweight and obese participants. In addition, the effect of the orforglipron tablet on the amount of simvastatin that enters the bloodstream and how long it takes the body to eliminate it will be evaluated.

The study will also assess the effect of sodium bicarbonate when administered alone with simvastatin versus orforglipron capsule containing sodium bicarbonate administered with simvastatin. The safety and tolerability of orforglipron and information about any side effects experienced will be collected.

Study will be conducted in two parts, with part 1 and 2 lasting up to approximately 23 and 24 weeks each, including the screening period.

Detailed Description

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Conditions

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Healthy Obese Overweight

Study Design

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Allocation Method

NON_RANDOMIZED

Intervention Model

SEQUENTIAL

Primary Study Purpose

BASIC_SCIENCE

Blinding Strategy

NONE

Study Groups

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Orforglipron (Part 1)

Participants will receive Orforglipron capsule and tablet formulation with Simvastatin, Digoxin, Rosuvastatin, Acetaminophen, Midazolam and Sodium Bicarbonate administered orally.

Group Type EXPERIMENTAL

Orforglipron

Intervention Type DRUG

Administered orally.

Simvastatin

Intervention Type DRUG

Administered orally.

Digoxin

Intervention Type DRUG

Administered orally.

Rosuvastatin

Intervention Type DRUG

Administered orally.

Acetaminophen

Intervention Type DRUG

Administered orally.

Midazolam

Intervention Type DRUG

Administered orally.

Sodium Bicarbonate

Intervention Type DRUG

Administered orally.

Orforglipron (Part 2)

Participants will receive Orforglipron capsule and tablet formulation with Simvastatin, Digoxin and Sodium Bicarbonate administered orally.

Group Type EXPERIMENTAL

Orforglipron

Intervention Type DRUG

Administered orally.

Simvastatin

Intervention Type DRUG

Administered orally.

Digoxin

Intervention Type DRUG

Administered orally.

Sodium Bicarbonate

Intervention Type DRUG

Administered orally.

Interventions

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Orforglipron

Administered orally.

Intervention Type DRUG

Simvastatin

Administered orally.

Intervention Type DRUG

Digoxin

Administered orally.

Intervention Type DRUG

Rosuvastatin

Administered orally.

Intervention Type DRUG

Acetaminophen

Administered orally.

Intervention Type DRUG

Midazolam

Administered orally.

Intervention Type DRUG

Sodium Bicarbonate

Administered orally.

Intervention Type DRUG

Other Intervention Names

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LY3502970

Eligibility Criteria

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Inclusion Criteria

* Participants who are overtly healthy as determined by medical history and physical examination.
* Have body mass index (BMI) equal to or greater than 27 kilograms per meter squared (kg/m²), inclusive, at screening.
* Have an estimated glomerular filtration rate equal to or greater than 60 milliliters per minute (mL/min).
* Males and females who agree to follow contraceptive requirements, or women not of childbearing potential (WNOCBP).
* Have venous access sufficient to allow for blood sampling.

Exclusion Criteria

* Have any type of diabetes with hemoglobin A1c (HbA1c) level of 6.5 percent (%) or greater.
* Have significant history of or currently have Major Depressive Disorder or psychiatric disorder within the last 2 years.
* Obesity induced by other endocrine disorders, such as Cushing's syndrome or Prader-Willi syndrome.
* Have known clinically significant gastric emptying abnormality.
* Have undergone bariatric surgery (for example: Lap-Band, Gastric Bypass)
* Have a known self or family history (first-degree relative) of multiple endocrine neoplasia type 2A or type 2B, thyroid C-cell hyperplasia, or any form of thyroid cancer.
* Have an abnormal 12-lead electrocardiogram (ECG) at screening.
* Have significant previous or current history of comorbidities capable of significantly altering the absorption, metabolism, or elimination of drug.
* Participants must not be currently participating in or completed a clinical trial within the last 90 days.
* Have a known allergy or hypersensitivity to midazolam, simvastatin, rosuvastatin, or digoxin.
Minimum Eligible Age

18 Years

Maximum Eligible Age

70 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

Yes

Sponsors

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Eli Lilly and Company

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Principal Investigators

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Call 1-877-CTLILLY (1-877-285-4559) or 1-317-615-4559 Mon - Fri 9 AM - 5 PM Eastern time (UTC/GMT - 5 hours, EST)

Role: STUDY_DIRECTOR

Eli Lilly and Company

Locations

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Fortrea Clinical Research Unit Inc.

Daytona Beach, Florida, United States

Site Status

Fortrea Clinical Research Unit Inc.

Dallas, Texas, United States

Site Status

Countries

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United States

Other Identifiers

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J2A-MC-GZPG

Identifier Type: OTHER

Identifier Source: secondary_id

18631

Identifier Type: -

Identifier Source: org_study_id

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