A Study to Evaluate the Safety, Tolerability, Pharmacokinetics and Clinical Activity of GSK5733584 for Injection in Participants With Advanced Solid Tumors

NCT ID: NCT06431594

Last Updated: 2025-06-25

Study Results

Results pending

The study team has not published outcome measurements, participant flow, or safety data for this trial yet. Check back later for updates.

Basic Information

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Recruitment Status

RECRUITING

Clinical Phase

PHASE1

Total Enrollment

385 participants

Study Classification

INTERVENTIONAL

Study Start Date

2024-07-02

Study Completion Date

2027-09-20

Brief Summary

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The goal of this study is to assess the safety and tolerability of GSK5733584. The study will also see how the levels of GSK5733584 change over time at different dose amount.

Detailed Description

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Conditions

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Solid Tumors Neoplasms

Study Design

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Allocation Method

RANDOMIZED

Intervention Model

SEQUENTIAL

Primary Study Purpose

TREATMENT

Blinding Strategy

NONE

Study Groups

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Part 1: Dose Escalation

Participants with advanced solid tumors who are refractory or intolerant to established standard therapies

Group Type EXPERIMENTAL

GSK5733584

Intervention Type DRUG

GSK5733584 will be administered

Part 2: Dose Expansion

Participants with platinum-resistant ovarian cancer (PROC) and endometrial cancer (EC)

Group Type EXPERIMENTAL

GSK5733584

Intervention Type DRUG

GSK5733584 will be administered

Interventions

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GSK5733584

GSK5733584 will be administered

Intervention Type DRUG

Eligibility Criteria

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Inclusion Criteria

* Males or females aged 18 years or older (≥18 years).
* Participants with pathologically confirmed advanced solid tumor (who have failed or are intolerant to standard of care).
* PROC cohort

1. Histologically documented, advanced (metastatic and/or unresectable) high-grade serous/endometrioid ovarian, primary peritoneal, or fallopian tube cancer.
2. Must have received or are intolerant to 1 but no more than 3 lines of prior systemic therapy.
3. Platinum-resistant disease, defined as progression or relapse within 6 months after the completion of platinum-based therapy.
4. Must have had prior bevacizumab if the participant was considered a candidate for this regimen and the regimen is locally available.
5. Participants with known Folate receptor-α (FR-α) expressing tumors must have received mirvetuximab soravtasine if the participants was considered a candidate for this regimen and the regimen is locally available.
6. Participants with known Breast cancer susceptibility gene (BRCA) mutated tumors should have received a Poly adenosine diphosphate-ribose polymerase (PARP) inhibitor if the participant was considered a candidate for this regimen and the regimen is locally available.
* Endometrial cancer cohort

1. Histologically documented, advanced (metastatic and/or unresectable) or recurrent endometrial cancer.
2. Must have received or are intolerant to 1 but no more than 3 lines of prior systemic therapy.
3. Must have had prior platinum and PD(L)-1 inhibitor (in same regimen or in separate regimens), if considered a candidate for this regimen and the regimen is locally available.
4. All epithelial histologies are permitted including carcinosarcoma.
* Participants have at least one target lesion as assessed per the RECIST 1.1
* Tumor tissue from a newly obtained biopsy or archival tumor tissue is required for retrospective detection of B7 homolog 4 (B7-H4) expression by Immunohistochemistry (IHC) in central laboratory and other biomarker analysis. Tissue from a newly obtained biopsy is preferred. If a newly obtained biopsy is not feasible, archival tumor tissue within 2 years prior to the first dose of study drug is acceptable.
* Eastern Cooperative Oncology Group Performance Status (ECOG PS) score of 0 to 2 and no deterioration within 2 weeks before the first dose.
* Have a life expectancy of at least 12 weeks.

Exclusion Criteria

* Have received any of B7-H4-targeted therapies.
* Have received any of cytotoxic chemotherapy drugs, anti-tumor traditional Chinese medicines or other anti-tumor drugs within 28 days prior to the first dose of study drug; or need to continue these drugs during the study.
* Have received locoregional radiation therapy within 2 weeks prior to the first dose of study drug; more than 30% of bone marrow irradiation or wide-field radiation therapy within 4 weeks prior to the first dose of study treatment.
* Presence of pleural/abdominal effusion/ascites requiring clinical intervention; presence of pericardial effusion
* Major surgery within 28 days prior to the first dose of study treatment.
* Evidence of brain metastasis unless asymptomatic.
* Has inadequate bone marrow reserve or hepatic/renal functions.
* Mean Fridericia-corrected QT interval (QTcF) \> 470 millisecond (msec) on resting ECG.
* Evidence of current clinically significant arrhythmias or ECG abnormalities
* Risk factors of prolonged QTc or arrhythmia events,
* Left ventricular ejection fraction (LVEF) \< 50%.
* Have severe, uncontrolled or active cardiovascular disorders, serious or poorly controlled hypertension, clinically significant bleeding symptoms or serious arteriovenous thromboembolic events
* Any evidence of current Interstitial lung disease (ILD) or pneumonitis or a prior history of ILD or pneumonitis requiring high-dose systemic glucocorticoids.
* Have received prior therapy with topoisomerase inhibitors or topoisomerase inhibitor Antibody-drug conjugate (ADCs)
* PROC

1. Primary platinum refractory disease defined as those who have progressed on or within 12 weeks of last dose of first line platinum therapy not permitted.
2. Non-epithelial carcinoma, clear-cell, mucinous, germ-cell, low-grade serous, or low-grade endometrioid carcinoma not permitted.
* Endometrial cancer a. Mesenchymal tumors of the uterus (uterine sarcomas) not permitted.
Minimum Eligible Age

18 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

No

Sponsors

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GlaxoSmithKline

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Locations

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GSK Investigational Site

Lake Mary, Florida, United States

Site Status RECRUITING

GSK Investigational Site

Fairway, Kansas, United States

Site Status RECRUITING

GSK Investigational Site

Boston, Massachusetts, United States

Site Status RECRUITING

GSK Investigational Site

Boston, Massachusetts, United States

Site Status RECRUITING

GSK Investigational Site

Detroit, Michigan, United States

Site Status RECRUITING

GSK Investigational Site

Grand Rapids, Michigan, United States

Site Status RECRUITING

GSK Investigational Site

Nashville, Tennessee, United States

Site Status RECRUITING

GSK Investigational Site

Dallas, Texas, United States

Site Status RECRUITING

GSK Investigational Site

West Valley City, Utah, United States

Site Status RECRUITING

GSK Investigational Site

Cipoletti Rio Negro, , Argentina

Site Status RECRUITING

GSK Investigational Site

Ciudad de Buenos Aires, , Argentina

Site Status RECRUITING

GSK Investigational Site

Rosario, , Argentina

Site Status RECRUITING

GSK Investigational Site

Blacktown, New South Wales, Australia

Site Status RECRUITING

GSK Investigational Site

Macquarie University, New South Wales, Australia

Site Status RECRUITING

GSK Investigational Site

Leuven, , Belgium

Site Status RECRUITING

GSK Investigational Site

Ottawa, Ontario, Canada

Site Status RECRUITING

GSK Investigational Site

Toronto, Ontario, Canada

Site Status RECRUITING

GSK Investigational Site

Montreal, Quebec, Canada

Site Status RECRUITING

GSK Investigational Site

Helsinki, , Finland

Site Status RECRUITING

GSK Investigational Site

Helsinki, , Finland

Site Status RECRUITING

GSK Investigational Site

Tampere, , Finland

Site Status RECRUITING

GSK Investigational Site

Lyon, , France

Site Status RECRUITING

GSK Investigational Site

Saint-Herblain, , France

Site Status RECRUITING

GSK Investigational Site

Villejuif, , France

Site Status RECRUITING

GSK Investigational Site

Roma, , Italy

Site Status RECRUITING

GSK Investigational Site

Rozzano MI, , Italy

Site Status RECRUITING

GSK Investigational Site

Saitama, , Japan

Site Status RECRUITING

GSK Investigational Site

Shizuoka, , Japan

Site Status RECRUITING

GSK Investigational Site

Tokyo, , Japan

Site Status RECRUITING

GSK Investigational Site

Amsterdam, , Netherlands

Site Status RECRUITING

GSK Investigational Site

Gyeonggi-do, , South Korea

Site Status RECRUITING

GSK Investigational Site

Seoul, , South Korea

Site Status RECRUITING

GSK Investigational Site

Seoul, , South Korea

Site Status RECRUITING

GSK Investigational Site

Seoul, , South Korea

Site Status RECRUITING

GSK Investigational Site

Barcelona, , Spain

Site Status RECRUITING

GSK Investigational Site

Córdoba, , Spain

Site Status RECRUITING

GSK Investigational Site

Girona, , Spain

Site Status RECRUITING

GSK Investigational Site

Madrid, , Spain

Site Status RECRUITING

GSK Investigational Site

Madrid, , Spain

Site Status RECRUITING

GSK Investigational Site

Madrid, , Spain

Site Status RECRUITING

GSK Investigational Site

Madrid, , Spain

Site Status RECRUITING

GSK Investigational Site

Pozuelo de AlarcOn Madr, , Spain

Site Status RECRUITING

GSK Investigational Site

Stockholm, , Sweden

Site Status RECRUITING

GSK Investigational Site

Uppsala, , Sweden

Site Status RECRUITING

GSK Investigational Site

Cambridge, , United Kingdom

Site Status RECRUITING

GSK Investigational Site

London, , United Kingdom

Site Status RECRUITING

GSK Investigational Site

London, , United Kingdom

Site Status RECRUITING

Countries

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United States Argentina Australia Belgium Canada Finland France Italy Japan Netherlands South Korea Spain Sweden United Kingdom

Central Contacts

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US GSK Clinical Trials Call Center

Role: CONTACT

877-379-3718

EU GSK Clinical Trials Call Center

Role: CONTACT

+44 (0) 20 89904466

Facility Contacts

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US GSK Clinical Trials Call Center

Role: primary

877-379-3718

EU GSK Clinical Trials Call Centre

Role: backup

+44 (0) 20 8990 4466

US GSK Clinical Trials Call Center

Role: primary

877-379-3718

EU GSK Clinical Trials Call Centre

Role: backup

+44 (0) 20 8990 4466

US GSK Clinical Trials Call Center

Role: primary

877-379-3718

EU GSK Clinical Trials Call Centre

Role: backup

+44 (0) 20 8990 4466

US GSK Clinical Trials Call Center

Role: primary

877-379-3718

EU GSK Clinical Trials Call Centre

Role: backup

+44 (0) 20 8990 4466

US GSK Clinical Trials Call Center

Role: primary

877-379-3718

EU GSK Clinical Trials Call Centre

Role: backup

+44 (0) 20 8990 4466

US GSK Clinical Trials Call Center

Role: primary

877-379-3718

EU GSK Clinical Trials Call Centre

Role: backup

+44 (0) 20 8990 4466

US GSK Clinical Trials Call Center

Role: primary

877-379-3718

EU GSK Clinical Trials Call Centre

Role: backup

+44 (0) 20 8990 4466

US GSK Clinical Trials Call Center

Role: primary

877-379-3718

EU GSK Clinical Trials Call Centre

Role: backup

+44 (0) 20 8990 4466

US GSK Clinical Trials Call Center

Role: primary

877-379-3718

EU GSK Clinical Trials Call Centre

Role: backup

+44 (0) 20 8990 4466

US GSK Clinical Trials Call Center

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877-379-3718

EU GSK Clinical Trials Call Centre

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+44 (0) 20 8990 4466

US GSK Clinical Trials Call Center

Role: primary

877-379-3718

EU GSK Clinical Trials Call Centre

Role: backup

+44 (0) 20 8990 4466

US GSK Clinical Trials Call Center

Role: primary

877-379-3718

EU GSK Clinical Trials Call Centre

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+44 (0) 20 8990 4466

US GSK Clinical Trials Call Center

Role: primary

877-379-3718

EU GSK Clinical Trials Call Centre

Role: backup

+44 (0) 20 8990 4466

US GSK Clinical Trials Call Center

Role: primary

877-379-3718

EU GSK Clinical Trials Call Centre

Role: backup

+44 (0) 20 8990 4466

US GSK Clinical Trials Call Center

Role: primary

877-379-3718

EU GSK Clinical Trials Call Centre

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+44 (0) 20 8990 4466

US GSK Clinical Trials Call Center

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877-379-3718

EU GSK Clinical Trials Call Centre

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US GSK Clinical Trials Call Center

Role: primary

877-379-3718

EU GSK Clinical Trials Call Centre

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+44 (0) 20 8990 4466

US GSK Clinical Trials Call Center

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877-379-3718

EU GSK Clinical Trials Call Centre

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+44 (0) 20 8990 4466

US GSK Clinical Trials Call Center

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877-379-3718

EU GSK Clinical Trials Call Centre

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+44 (0) 20 8990 4466

US GSK Clinical Trials Call Center

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877-379-3718

EU GSK Clinical Trials Call Centre

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US GSK Clinical Trials Call Center

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877-379-3718

EU GSK Clinical Trials Call Centre

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US GSK Clinical Trials Call Center

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877-379-3718

EU GSK Clinical Trials Call Centre

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US GSK Clinical Trials Call Center

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877-379-3718

EU GSK Clinical Trials Call Centre

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US GSK Clinical Trials Call Center

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877-379-3718

EU GSK Clinical Trials Call Centre

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US GSK Clinical Trials Call Center

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877-379-3718

EU GSK Clinical Trials Call Centre

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US GSK Clinical Trials Call Center

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877-379-3718

EU GSK Clinical Trials Call Centre

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877-379-3718

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US GSK Clinical Trials Call Center

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877-379-3718

EU GSK Clinical Trials Call Centre

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US GSK Clinical Trials Call Center

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877-379-3718

EU GSK Clinical Trials Call Centre

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US GSK Clinical Trials Call Center

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877-379-3718

EU GSK Clinical Trials Call Centre

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US GSK Clinical Trials Call Center

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877-379-3718

EU GSK Clinical Trials Call Centre

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US GSK Clinical Trials Call Center

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877-379-3718

EU GSK Clinical Trials Call Centre

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US GSK Clinical Trials Call Center

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877-379-3718

EU GSK Clinical Trials Call Centre

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US GSK Clinical Trials Call Center

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877-379-3718

EU GSK Clinical Trials Call Centre

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US GSK Clinical Trials Call Center

Role: primary

877-379-3718

EU GSK Clinical Trials Call Centre

Role: backup

+44 (0) 20 8990 4466

US GSK Clinical Trials Call Center

Role: primary

877-379-3718

EU GSK Clinical Trials Call Centre

Role: backup

+44 (0) 20 8990 4466

US GSK Clinical Trials Call Center

Role: primary

877-379-3718

EU GSK Clinical Trials Call Centre

Role: backup

+44 (0) 20 8990 4466

US GSK Clinical Trials Call Center

Role: primary

877-379-3718

EU GSK Clinical Trials Call Centre

Role: backup

+44 (0) 20 8990 4466

US GSK Clinical Trials Call Center

Role: primary

877-379-3718

EU GSK Clinical Trials Call Centre

Role: backup

+44 (0) 20 8990 4466

US GSK Clinical Trials Call Center

Role: primary

877-379-3718

EU GSK Clinical Trials Call Centre

Role: backup

+44 (0) 20 8990 4466

US GSK Clinical Trials Call Center

Role: primary

877-379-3718

EU GSK Clinical Trials Call Centre

Role: backup

+44 (0) 20 8990 4466

US GSK Clinical Trials Call Center

Role: primary

877-379-3718

EU GSK Clinical Trials Call Centre

Role: backup

+44 (0) 20 8990 4466

US GSK Clinical Trials Call Center

Role: primary

877-379-3718

EU GSK Clinical Trials Call Centre

Role: backup

+44 (0) 20 8990 4466

US GSK Clinical Trials Call Center

Role: primary

877-379-3718

EU GSK Clinical Trials Call Centre

Role: backup

+44 (0) 20 8990 4466

US GSK Clinical Trials Call Center

Role: primary

877-379-3718

EU GSK Clinical Trials Call Centre

Role: backup

+44 (0) 20 8990 4466

US GSK Clinical Trials Call Center

Role: primary

877-379-3718

EU GSK Clinical Trials Call Centre

Role: backup

+44 (0) 20 8990 4466

US GSK Clinical Trials Call Center

Role: primary

877-379-3718

EU GSK Clinical Trials Call Centre

Role: backup

+44 (0) 20 8990 4466

Other Identifiers

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2024-513860-25

Identifier Type: REGISTRY

Identifier Source: secondary_id

222730

Identifier Type: -

Identifier Source: org_study_id

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