A Study to Investigate the Efficacy and Safety of Dato-DXd With or Without Osimertinib Compared With Platinum Based Doublet Chemotherapy in Participants With EGFR-Mutated Locally Advanced or Metastatic Non-Small Cell Lung Cancer

NCT ID: NCT06417814

Last Updated: 2026-01-09

Study Results

Results pending

The study team has not published outcome measurements, participant flow, or safety data for this trial yet. Check back later for updates.

Basic Information

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Recruitment Status

RECRUITING

Clinical Phase

PHASE3

Total Enrollment

744 participants

Study Classification

INTERVENTIONAL

Study Start Date

2024-10-04

Study Completion Date

2028-09-27

Brief Summary

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This study will assess the effect of Dato-DXd in combination with osimertinib or Dato-DXd monotherapy versus platinum-based doublet chemotherapy in terms of progression-free survival (PFS).

Detailed Description

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This is a Phase III, open-label, 3-arm, multicenter study assessing the effects of Dato-DXd in combination with osimertinib or Dato-DXd monotherapy versus platinum-based doublet chemotherapy in participants with epidermal growth factor receptor gene mutation (EGFRm) locally advanced or metastatic non-small cell lung cancer (NSCLC) whose disease has progressed on prior osimertinib treatment.

Participants will be randomized in a 1:1:1 ratio to one of the following intervention groups:

1. Dato-DXd + osimertinib combination therapy
2. Dato-DXd monotherapy
3. Platinum-based doublet chemotherapy

Participants will receive study intervention until Response Evaluation Criteria in Solid Tumors, Version 1.1 (RECIST v1.1) -defined radiological progression by the investigator, unacceptable toxicity, or other discontinuation criterion is met.

After study intervention discontinuation, all participants will undergo an end of treatment (EoT) visit within 35 days of discontinuation and will be followed up for safety assessments 28 (+ 7) days after their last dose of study intervention.

Conditions

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Metastatic Non-small Cell Lung Cancer

Study Design

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Allocation Method

RANDOMIZED

Intervention Model

PARALLEL

Primary Study Purpose

TREATMENT

Blinding Strategy

NONE

Study Groups

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Group 1: Dato-DXd + Osimertinib Combination Therapy

Participants will receive Dato-DXd 6 milligrams per kilogram (mg/kg) as intravenous (IV) infusion every 3 weeks (Q3W) on Day 1 of every 21-day cycle, and osimertinib 80 milligrams (mg) once daily (QD) orally, until RECIST v1.1-defined radiological progression by investigator, unacceptable toxicity, or other discontinuation criterion is met.

Group Type EXPERIMENTAL

Dato-DXd

Intervention Type DRUG

Dato-DXd will be administered as IV infusion.

Osimertinib

Intervention Type DRUG

Osimertinib will be administered orally.

Group 2: Dato-DXd Monotherapy

Participants will receive Dato-DXd 6 mg/kg as IV infusion Q3W on Day 1 of every 21-day cycle, until RECIST v1.1-defined radiological progression by investigator, unacceptable toxicity, or other discontinuation criterion is met.

Group Type EXPERIMENTAL

Dato-DXd

Intervention Type DRUG

Dato-DXd will be administered as IV infusion.

Group 3: Platinum-based Doublet Chemotherapy

Participants will receive pemetrexed 500 milligrams per meter square (mg/m2) in combination with carboplatin (AUC5) or cisplatin 75 mg/m2 as IV infusion Q3W for 4 cycles followed by pemetrexed maintenance 500 mg/m2 as IV infusion Q3W, until RECIST v1.1-defined radiological progression by investigator, unacceptable toxicity, or another discontinuation criterion is met.

Group Type EXPERIMENTAL

Pemetrexed

Intervention Type DRUG

Pemetrexed will be administered as IV infusion.

Carboplatin

Intervention Type DRUG

Carboplatin will be administered as IV infusion.

Cisplatin

Intervention Type DRUG

Cisplatin will be administered as IV infusion.

Interventions

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Dato-DXd

Dato-DXd will be administered as IV infusion.

Intervention Type DRUG

Osimertinib

Osimertinib will be administered orally.

Intervention Type DRUG

Pemetrexed

Pemetrexed will be administered as IV infusion.

Intervention Type DRUG

Carboplatin

Carboplatin will be administered as IV infusion.

Intervention Type DRUG

Cisplatin

Cisplatin will be administered as IV infusion.

Intervention Type DRUG

Other Intervention Names

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DS-1062a Tagrisso AZD9291

Eligibility Criteria

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Inclusion Criteria

* Histologically or cytologically confirmed non-squamous NSCLC.
* Must have evidence of documented pre-existing EGFRm information (EGFRm known to be associated with (epidermal growth factor receptor \[EGFR\] tyrosine kinase inhibitor \[TKis\] sensitivity \[Ex19del, L858R, G719X, S768I, or L861Q\], either alone or in combination with other EGFR mutations, which may include T790M).
* Documented extra-cranial radiologic progression on prior osimertinib monotherapy (as most recent line of treatment) in the adjuvant, locally advanced, or metastatic setting.
* Less than or equal to (\<=2) prior lines of EGFR TKIs (osimertinib is the only permitted prior third generation EGFR TKI).
* At least one lesion, not previously irradiated, that qualifies as a RECIST v1.1 TL at baseline and can be accurately measured at baseline.
* World Health Organization (WHO)/Eastern Cooperative Oncology Group (ECOG) performance status of 0 or 1.
* Adequate bone marrow reserve and organ function within 7 days before randomization.

Exclusion Criteria

* Use of chemotherapy, vascular endothelial growth factor inhibitor, immunotherapy or any anti-cancer therapy in the metastatic setting. Platinum-based chemotherapy in non-metastatic setting within 12 months prior to randomization.
* History of another primary malignancy except for malignancy treated with curative intent with no known active disease within 2 years before the first dose of study intervention.
* Any evidence of severe or uncontrolled systemic diseases, including, but not limited to active bleeding diseases, active infection, active ILD/pneumonitis, cardiac disease.
* Has significant third-space fluid retention (example \[eg.\], ascites or pleural effusion) as judged by the investigator and is not amenable for required repeated drainage.
* History of non-infectious ILD/pneumonitis including radiation pneumonitis that required steroids or drug-induced ILD, has current ILD/pneumonitis, or has suspected ILD/pneumonitis that cannot be ruled out by imaging at screening.
* Has severe pulmonary function compromise resulting from intercurrent pulmonary illnesses.
* Unstable spinal cord compression and/or unstable brain metastases.
* Participants with symptomatic brain metastases (including leptomeningeal involvement).
* Clinically significant corneal disease.
* Uncontrolled infection requiring systemic antibiotics, antivirals, or antifungals, suspected infections or inability to rule out infections. Use of systemic antibiotics within 14 days of randomization.
* Has known human immunodeficiency virus (HIV) infection that is not well controlled.
Minimum Eligible Age

18 Years

Maximum Eligible Age

130 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

No

Sponsors

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Daiichi Sankyo

INDUSTRY

Sponsor Role collaborator

AstraZeneca

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Locations

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Research Site

Fayetteville, Arkansas, United States

Site Status RECRUITING

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Duarte, California, United States

Site Status NOT_YET_RECRUITING

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Fountain Valley, California, United States

Site Status RECRUITING

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La Jolla, California, United States

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Los Angeles, California, United States

Site Status NOT_YET_RECRUITING

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San Diego, California, United States

Site Status NOT_YET_RECRUITING

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Colorado Springs, Colorado, United States

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Fort Collins, Colorado, United States

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Gainesville, Florida, United States

Site Status NOT_YET_RECRUITING

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Jacksonville, Florida, United States

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Athens, Georgia, United States

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Chicago, Illinois, United States

Site Status NOT_YET_RECRUITING

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Evanston, Illinois, United States

Site Status NOT_YET_RECRUITING

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Louisville, Kentucky, United States

Site Status NOT_YET_RECRUITING

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Baltimore, Maryland, United States

Site Status NOT_YET_RECRUITING

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Bethesda, Maryland, United States

Site Status RECRUITING

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Boston, Massachusetts, United States

Site Status NOT_YET_RECRUITING

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Boston, Massachusetts, United States

Site Status NOT_YET_RECRUITING

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Detroit, Michigan, United States

Site Status RECRUITING

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Kansas City, Missouri, United States

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Omaha, Nebraska, United States

Site Status RECRUITING

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Morristown, New Jersey, United States

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Northfield, New Jersey, United States

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New York, New York, United States

Site Status SUSPENDED

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New York, New York, United States

Site Status RECRUITING

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The Bronx, New York, United States

Site Status RECRUITING

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Maumee, Ohio, United States

Site Status RECRUITING

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Philadelphia, Pennsylvania, United States

Site Status NOT_YET_RECRUITING

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Pittsburgh, Pennsylvania, United States

Site Status RECRUITING

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Chattanooga, Tennessee, United States

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Nashville, Tennessee, United States

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Fairfax, Virginia, United States

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Seattle, Washington, United States

Site Status WITHDRAWN

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Fitzroy, , Australia

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Heidelberg, , Australia

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Kogarah, , Australia

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Liverpool, , Australia

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Nedlands, , Australia

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Port Macquarie, , Australia

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St Leonards, , Australia

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Westmead, , Australia

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Woodville, , Australia

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Woolloongabba, , Australia

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Charleroi, , Belgium

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Edegem, , Belgium

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Ghent, , Belgium

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Hasselt, , Belgium

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Jette, , Belgium

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La Louvière, , Belgium

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Leuven, , Belgium

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Namur, , Belgium

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Roeselare, , Belgium

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Barretos, , Brazil

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Betim, , Brazil

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Blumenau, , Brazil

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Florianópolis, , Brazil

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Itajaí, , Brazil

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Pelotas, , Brazil

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Porto Alegre, , Brazil

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Porto Alegre, , Brazil

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Porto Alegre, , Brazil

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Rio de Janeiro, , Brazil

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Rio de Janeiro, , Brazil

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Rio de Janeiro, , Brazil

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São Paulo, , Brazil

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São Paulo, , Brazil

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Brampton, Ontario, Canada

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Newmarket, Ontario, Canada

Site Status WITHDRAWN

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Toronto, Ontario, Canada

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Toronto, Ontario, Canada

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Montreal, Quebec, Canada

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Québec, Quebec, Canada

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Baoding, , China

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Beijing, , China

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Beijing, , China

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Beijing, , China

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Beijing, , China

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Beijing, , China

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Beijing, , China

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Beijing, , China

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Bengbu, , China

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Changchun, , China

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Changchun, , China

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Changsha, , China

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Chengdu, , China

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Deyang, , China

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Ganzhou, , China

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Guangzhou, , China

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Hangzhou, , China

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Hangzhou, , China

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Hefei, , China

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Hengyang, , China

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Huaian, , China

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Jinan, , China

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Linyi, , China

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Luoyang, , China

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Luzhou, , China

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Nanchang, , China

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Nanjing, , China

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Shanghai, , China

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Shantou, , China

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Shenyang, , China

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Shenyang, , China

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Tianjin, , China

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Tianjin, , China

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Weifang, , China

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Wuhan, , China

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Zhengzhou, , China

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Zhengzhou, , China

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Zhengzhou, , China

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Angers, , France

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Avignon, , France

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Bordeaux, , France

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Caen, , France

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Lille, , France

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Montpellier, , France

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Nantes, , France

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Paris, , France

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Paris, , France

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Pessac, , France

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Quimper, , France

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Toulon Armees, , France

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Toulouse, , France

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Tours, , France

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Villejuif, , France

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Berlin, , Germany

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Berlin-Zehlendorf, , Germany

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Bonn, , Germany

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Essen, , Germany

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Georgsmarienhütte, , Germany

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Giessen, , Germany

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Großhansdorf, , Germany

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Hamburg, , Germany

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Hamburg, , Germany

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Heidelberg, , Germany

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Kempten, , Germany

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Löwenstein, , Germany

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Nuremberg, , Germany

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Oldenburg, , Germany

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Athens, , Greece

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Athens, , Greece

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Athens, , Greece

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Athens, , Greece

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Heraklion, , Greece

Site Status NOT_YET_RECRUITING

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Thessaloniki, , Greece

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Thessaloniki, , Greece

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Thessaloniki, , Greece

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Thessaloniki, , Greece

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Hong Kong, , Hong Kong

Site Status NOT_YET_RECRUITING

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Hong Kong, , Hong Kong

Site Status NOT_YET_RECRUITING

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Hong Kong, , Hong Kong

Site Status NOT_YET_RECRUITING

Research Site

Shatin, , Hong Kong

Site Status NOT_YET_RECRUITING

Research Site

Amravati, , India

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Bhubaneswar, , India

Site Status NOT_YET_RECRUITING

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Hyderabad, , India

Site Status RECRUITING

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Kolhāpur, , India

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Mumbai, , India

Site Status NOT_YET_RECRUITING

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Mysuru, , India

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Research Site

Namakkal, , India

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Research Site

Pune, , India

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Research Site

Raipur, , India

Site Status COMPLETED

Research Site

Rajasthan, , India

Site Status RECRUITING

Research Site

Ranchi, , India

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Research Site

Thane, , India

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Trivandrum, , India

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Varanasi, , India

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Research Site

Beersheba, , Israel

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Haifa, , Israel

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Haifa, , Israel

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Jerusalem, , Israel

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Jerusalem, , Israel

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Kfar Saba, , Israel

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Petah Tikva, , Israel

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Ramat Gan, , Israel

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Tel Aviv, , Israel

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Bari, , Italy

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Milan, , Italy

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Misterbianco, , Italy

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Monza, , Italy

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Napoli, , Italy

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Orbassano, , Italy

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Padua, , Italy

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Parma, , Italy

Site Status NOT_YET_RECRUITING

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Perugia, , Italy

Site Status RECRUITING

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Roma, , Italy

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Rozzano, , Italy

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Verona, , Italy

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Bunkyō City, , Japan

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Bunkyō City, , Japan

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Fukuoka, , Japan

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Hiroshima, , Japan

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Iruma-Gun, , Japan

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Iwakuni-shi, , Japan

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Kobe, , Japan

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Kōtoku, , Japan

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Kumamoto, , Japan

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Kyoto, , Japan

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Matsuyama, , Japan

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Nagoya, , Japan

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Nagoya, , Japan

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Niigata, , Japan

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Osaka, , Japan

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Osaka, , Japan

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Ōsaka-sayama, , Japan

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Sendai, , Japan

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Sunto-gun, , Japan

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Toyoake-shi, , Japan

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Utsunomiya, , Japan

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Wakayama, , Japan

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Yokohama, , Japan

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Yokohama, , Japan

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Alor Star, , Malaysia

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Cheras, , Malaysia

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Johor Bahru, , Malaysia

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Kuala Lumpur, , Malaysia

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Kuala Selangor, , Malaysia

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Kuching, , Malaysia

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Perai, , Malaysia

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Petaling Jaya, , Malaysia

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Amersfoort, , Netherlands

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Harderwijk, , Netherlands

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Rotterdam, , Netherlands

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Zutphen, , Netherlands

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Bacolod, , Philippines

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Cebu City, , Philippines

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Davao City, , Philippines

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Manila, , Philippines

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Quezon, , Philippines

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Quezon, , Philippines

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San Juan City, , Philippines

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Katowice, , Poland

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Krakow, , Poland

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Lodz, , Poland

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Olsztyn, , Poland

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Poznan, , Poland

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Braga, , Portugal

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Lisbon, , Portugal

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Loures, , Portugal

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Porto, , Portugal

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Porto, , Portugal

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Craiova, , Romania

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Craiova, , Romania

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Singapore, , Singapore

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Singapore, , Singapore

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Singapore, , Singapore

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Busan, , South Korea

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Chungcheongbuk-do, , South Korea

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Goyang-si, , South Korea

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Gyeonggi-do, , South Korea

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Jinju, , South Korea

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Seoul, , South Korea

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Seoul, , South Korea

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Seoul, , South Korea

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Seoul, , South Korea

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Seoul, , South Korea

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Suwon, , South Korea

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A Coruña, , Spain

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Barakaldo, , Spain

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Barcelona, , Spain

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Barcelona, , Spain

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El Palmar, , Spain

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L'Hospitalet de Llobregat, , Spain

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Madrid, , Spain

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Madrid, , Spain

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Majadahonda, , Spain

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Málaga, , Spain

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Oviedo, , Spain

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Palma de Mallorca, , Spain

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Pamplona, , Spain

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Santander, , Spain

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Santiago de Compostela-Coruña, , Spain

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Seville, , Spain

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Valencia, , Spain

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Valencia, , Spain

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Valladolid, , Spain

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Changhua, , Taiwan

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Kaohsiung City, , Taiwan

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New Taipei City, , Taiwan

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Taichung, , Taiwan

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Taichung, , Taiwan

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Tainan, , Taiwan

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Tainan, , Taiwan

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Taipei, , Taiwan

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Taipei, , Taiwan

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Taipei, , Taiwan

Site Status RECRUITING

Research Site

Bangkok, , Thailand

Site Status RECRUITING

Research Site

Bangkok, , Thailand

Site Status RECRUITING

Research Site

Bangkok, , Thailand

Site Status RECRUITING

Research Site

Chiang Mai, , Thailand

Site Status RECRUITING

Research Site

Hat Yai, , Thailand

Site Status RECRUITING

Research Site

Khon Kaen, , Thailand

Site Status RECRUITING

Research Site

Pathum Thani, , Thailand

Site Status RECRUITING

Research Site

Birmingham, , United Kingdom

Site Status RECRUITING

Research Site

Cambridge, , United Kingdom

Site Status RECRUITING

Research Site

Glasgow, , United Kingdom

Site Status RECRUITING

Research Site

Leicester, , United Kingdom

Site Status RECRUITING

Research Site

London, , United Kingdom

Site Status RECRUITING

Research Site

Manchester, , United Kingdom

Site Status RECRUITING

Research Site

Middlesbrough, , United Kingdom

Site Status RECRUITING

Research Site

Hanoi, , Vietnam

Site Status NOT_YET_RECRUITING

Countries

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United States Australia Belgium Brazil Canada China France Germany Greece Hong Kong India Israel Italy Japan Malaysia Netherlands Philippines Poland Portugal Romania Singapore South Korea Spain Taiwan Thailand United Kingdom Vietnam

Central Contacts

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AstraZeneca Clinical Study Information Center

Role: CONTACT

1-877-240-9479

References

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Tan DS, Nadal E, Cheema P, Wu YL, Ahn MJ, Tanizaki J, Grainger E, Nizialek E, Forcina A, van der Gronde T, Yu HA. TROPION-Lung15: a randomized phase III study of osimertinib combined with datopotamab deruxtecan (Dato-DXd) or Dato-DXd alone versus platinum-doublet chemotherapy in patients with EGFR-mutated advanced non-small cell lung cancer and whose disease has progressed on prior osimertinib. Ther Adv Med Oncol. 2025 Dec 23;17:17588359251385410. doi: 10.1177/17588359251385410. eCollection 2025.

Reference Type DERIVED
PMID: 41466843 (View on PubMed)

Other Identifiers

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2024-511362-37-00

Identifier Type: REGISTRY

Identifier Source: secondary_id

D516KC00001

Identifier Type: -

Identifier Source: org_study_id

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