Saruparib (AZD5305) Plus Camizestrant Compared With CDK4/6 Inhibitor Plus Endocrine Therapy or Plus Camizestrant in HR-Positive, HER2-Negative (IHC 0, 1+, 2+/ ISH Non-amplified), BRCA1, BRCA2, or PALB2m Advanced Breast Cancer

NCT ID: NCT06380751

Last Updated: 2026-02-10

Study Results

Results pending

The study team has not published outcome measurements, participant flow, or safety data for this trial yet. Check back later for updates.

Basic Information

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Recruitment Status

RECRUITING

Clinical Phase

PHASE3

Total Enrollment

500 participants

Study Classification

INTERVENTIONAL

Study Start Date

2024-08-01

Study Completion Date

2030-10-18

Brief Summary

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The primary objective of the study is to measure efficacy of saruparib (AZD5305) plus camizestrant compared with physician's choice CDK4/6i plus ET in patients with BRCA1, BRCA2, or PALB2m, HR-positive, HER2-negative (defined as IHC 0, 1+, 2+/ ISH non-amplified) advanced breast cancer

Detailed Description

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Approximately 2,620 participants will be screened to achieve approximately 500 participants randomised to study intervention.

Participants will be randomised in a 2:2:1 ratio to one of the following intervention groups:

* Arm 1: saruparib (AZD5305) plus camizestrant
* Arm 2: Physician's choice CDK4/6i plus physician's choice ET
* Arm 3: Physician's choice CDK4/6i plus camizestrant Treatment continues until BICR-confirmed disease progression, unacceptable toxicity occurs, or the participant withdraws consent.

Conditions

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Advanced Breast Cancer

Study Design

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Allocation Method

RANDOMIZED

Intervention Model

PARALLEL

Primary Study Purpose

TREATMENT

Blinding Strategy

NONE

Open label

Study Groups

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Arm 1: saruparib (AZD5305) plus camizestrant

participants will receive saruparib (AZD5305) orally and camizestrant orally

Group Type EXPERIMENTAL

Saruparib (AZD5305)

Intervention Type DRUG

Saruparib (AZD5305) is a potent and selective inhibitor of PARP1, with minimal effect on PARP2.

Camizestrant

Intervention Type DRUG

Camizestrant (AZD9833) is an orally bioavailable, next generation SERD with non-clinical and clinical activity in both ESR1 mutant and wild type settings .

Arm 2: Physician's choice CDK4/6i plus physician's choice ET

agents are indicated below and should follow local guidelines:

* Physician's Choice CDK4/6i:

* abemaciclib orally, or
* ribociclib orally, or
* palbociclib orally.
* Physician's Choice ET:

* fulvestrant intramuscularly, or
* One of the following AIs:

* letrozole orally, or
* anastrozole orally, or
* exemestane orally

Group Type ACTIVE_COMPARATOR

Abemaciclib

Intervention Type DRUG

CDK4/6 Inhibitor

Ribociclib

Intervention Type DRUG

CDK4/6 Inhibitor

Palbociclib

Intervention Type DRUG

CDK 4/6 Inhibitor

Fulvestrant

Intervention Type DRUG

Endocrine Therapy

Letrozole

Intervention Type DRUG

Endorcine Therapy

Anastrozole

Intervention Type DRUG

Endocrine Therapy

Exemestane

Intervention Type DRUG

Endocrine Therapy

Arm 3: Physician's choice CDK4/6i plus camizestrant

participants will receive camizestrant orally. Agents for CDK4/6i treatment are indicated above and should follow local guidelines

Group Type EXPERIMENTAL

Camizestrant

Intervention Type DRUG

Camizestrant (AZD9833) is an orally bioavailable, next generation SERD with non-clinical and clinical activity in both ESR1 mutant and wild type settings .

Abemaciclib

Intervention Type DRUG

CDK4/6 Inhibitor

Ribociclib

Intervention Type DRUG

CDK4/6 Inhibitor

Palbociclib

Intervention Type DRUG

CDK 4/6 Inhibitor

Interventions

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Saruparib (AZD5305)

Saruparib (AZD5305) is a potent and selective inhibitor of PARP1, with minimal effect on PARP2.

Intervention Type DRUG

Camizestrant

Camizestrant (AZD9833) is an orally bioavailable, next generation SERD with non-clinical and clinical activity in both ESR1 mutant and wild type settings .

Intervention Type DRUG

Abemaciclib

CDK4/6 Inhibitor

Intervention Type DRUG

Ribociclib

CDK4/6 Inhibitor

Intervention Type DRUG

Palbociclib

CDK 4/6 Inhibitor

Intervention Type DRUG

Fulvestrant

Endocrine Therapy

Intervention Type DRUG

Letrozole

Endorcine Therapy

Intervention Type DRUG

Anastrozole

Endocrine Therapy

Intervention Type DRUG

Exemestane

Endocrine Therapy

Intervention Type DRUG

Eligibility Criteria

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Inclusion Criteria

* Adult females, pre/peri-menopausal and/or post-menopausal, and adult males
* Histologically or cytologically documented diagnosis of HR-positive, HER2-negative breast cancer
* Advanced breast cancer with either locally advanced disease not amenable to curative treatment or metastatic disease
* ECOG performance status of 0 or 1 with no deterioration over the previous 2 weeks
* FFPE tumour tissue from each participant
* Documented germline tumour loss of function mutation in BRCA1, BRCA2, or PALB2
* Adequate organ and marrow function

Exclusion Criteria

* Participants with history of MDS/AML or with features suggestive of MDS/AML
* Participants with any known predisposition to bleeding
* Any history of persisting severe cytopenia
* Any evidence of severe or uncontrolled systemic diseases or active uncontrolled infections
* Refractory nausea and vomiting, chronic GI disease, inability to swallow the formulated product, or previous significant bowel resection
* History of another primary malignancy
* Persistent toxicities (CTCAE Grade ≥ 2) caused by previous anti-cancer therapy excluding alopecia
* Spinal cord compression, brain metastases, carcinomatous meningitis, or leptomeningeal disease
* Evidence of active and uncontrolled hepatitis B and/or hepatitis C
* Evidence of active and uncontrolled HIV infection
* Active tuberculosis infection
* Cardiac criteria, including history of arrythmia and cardiovascular disease
* Concurrent exogenous reproductive hormone therapy or non-topical hormonal therapy for non-cancer-related conditions
* Major surgical procedure or significant traumatic injury within 4 weeks of the first dose of study intervention or an anticipated need for major surgery during the study
* Palliative radiotherapy with a limited field of radiation within 2 weeks or with wide field of radiation or to more than 30% of the bone marrow within 4 weeks before the first dose of study treatment
* Prior treatment with systemic anti-cancer therapy for locoregionally recurrent or metastatic disease is not permitted, apart from treatment with ET up to 28 days before randomisation
* Prior treatment within 28 days with blood product support or growth factor support
* Any systemic concurrent anti-cancer treatment
* Concomitant use of the following types of medications or herbal supplements within 21 days or at least 5 half-lives of randomisation:

1. Strong and moderate CYP3A4 inducers/inhibitors
2. Sensitive CYP2B6 substrates
3. Substrates of CYP2C9 and/or CYP2C19 which have a narrow therapeutic index, eg, warfarin (and other coumarin-derived vitamin K antagonist anticoagulants) and phenytoin.
* Concomitant use of drugs that are known to prolong QT and have a known risk of TdP
* Systemic use of atropine

1. Disease progression ≤ 84 days following the last dose of neo-adjuvant or adjuvant chemotherapy
2. Disease progression ≤ 1 year (365 days) from the last dose of treatment with a PARPi and/or platinum agent for early breast cancer
3. Disease progression ≤ 1 year (365 days) from the last dose with a CDK4/6i in the adjuvant setting
4. Disease progression ≤ 1 year (365 days) from the last dose of an oral SERD including camizestrant.
Minimum Eligible Age

18 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

No

Sponsors

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AstraZeneca

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Locations

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Research Site

Gilbert, Arizona, United States

Site Status RECRUITING

Research Site

Fountain Valley, California, United States

Site Status RECRUITING

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Glendale, California, United States

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Los Angeles, California, United States

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Newport Beach, California, United States

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Aurora, Colorado, United States

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Grand Junction, Colorado, United States

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Hollywood, Florida, United States

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Jacksonville, Florida, United States

Site Status NOT_YET_RECRUITING

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Orlando, Florida, United States

Site Status WITHDRAWN

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Chicago, Illinois, United States

Site Status RECRUITING

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Evanston, Illinois, United States

Site Status NOT_YET_RECRUITING

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Park Ridge, Illinois, United States

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Urbana, Illinois, United States

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Winfield, Illinois, United States

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Indianapolis, Indiana, United States

Site Status WITHDRAWN

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Louisville, Kentucky, United States

Site Status WITHDRAWN

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Silver Spring, Maryland, United States

Site Status RECRUITING

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Silver Spring, Maryland, United States

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Boston, Massachusetts, United States

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Dearborn, Michigan, United States

Site Status WITHDRAWN

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Detroit, Michigan, United States

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Royal Oak, Michigan, United States

Site Status WITHDRAWN

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Royal Oak, Michigan, United States

Site Status NOT_YET_RECRUITING

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Rochester, Minnesota, United States

Site Status NOT_YET_RECRUITING

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Springfield, Missouri, United States

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Camden, New Jersey, United States

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New Brunswick, New Jersey, United States

Site Status WITHDRAWN

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Brooklyn, New York, United States

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Mineola, New York, United States

Site Status RECRUITING

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New Hyde Park, New York, United States

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New York, New York, United States

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New York, New York, United States

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New York, New York, United States

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Shirley, New York, United States

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Stony Brook, New York, United States

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The Bronx, New York, United States

Site Status WITHDRAWN

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Westbury, New York, United States

Site Status WITHDRAWN

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Hershey, Pennsylvania, United States

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Philadelphia, Pennsylvania, United States

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Pittsburgh, Pennsylvania, United States

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West Columbia, South Carolina, United States

Site Status WITHDRAWN

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Chattanooga, Tennessee, United States

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Nashville, Tennessee, United States

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Houston, Texas, United States

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Houston, Texas, United States

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Houston, Texas, United States

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Norfolk, Virginia, United States

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Tacoma, Washington, United States

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Morgantown, West Virginia, United States

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Milwaukee, Wisconsin, United States

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Ciudad Autónoma Buenos Aires, , Argentina

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Ciudad de Buenos Aires, , Argentina

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Ciudad de Buenos Aires, , Argentina

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Córdoba, , Argentina

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Rosario, , Argentina

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Salta, , Argentina

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San Miguel de Tucumán, , Argentina

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Darlinghurst, , Australia

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Darlinghurst, , Australia

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Malvern, , Australia

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Melbourne, , Australia

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Graz, , Austria

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Innsbruck, , Austria

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Linz, , Austria

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Vienna, , Austria

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Cachoeira de Itapemirim, , Brazil

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Curitiba, , Brazil

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Fortaleza, , Brazil

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Goiânia, , Brazil

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Jaú, , Brazil

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Porto Alegre, , Brazil

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Ribeirão Preto, , Brazil

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Salvador, , Brazil

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São Paulo, , Brazil

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São Paulo, , Brazil

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Plovdiv, , Bulgaria

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Sofia, , Bulgaria

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Stara Zagora, , Bulgaria

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Vratsa, , Bulgaria

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Toronto, Ontario, Canada

Site Status NOT_YET_RECRUITING

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Greenfield Park, Quebec, Canada

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Montreal, Quebec, Canada

Site Status NOT_YET_RECRUITING

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Montreal, Quebec, Canada

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Montreal, Quebec, Canada

Site Status NOT_YET_RECRUITING

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Saskatoon, Saskatchewan, Canada

Site Status NOT_YET_RECRUITING

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Toronto, , Canada

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Providencia, , Chile

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Recoleta, , Chile

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Santiago, , Chile

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Talca, , Chile

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Viña del Mar, , Chile

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Beijing, , China

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Bengbu, , China

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Changchun, , China

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Changchun, , China

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Changsha, , China

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Changsha, , China

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Chengdu, , China

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Chengdu, , China

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Chongqing, , China

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Foshan, , China

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Fuzhou, , China

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Guangzhou, , China

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Guangzhou, , China

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Guangzhou, , China

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Hangzhou, , China

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Hangzhou, , China

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Harbin, , China

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Hefei, , China

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Hohhot, , China

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Jining, , China

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Kunming, , China

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Liuchow, , China

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Luoyang, , China

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Nanchang, , China

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Nanchang, , China

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Nanjing, , China

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Shandong, , China

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Shanghai, , China

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Shanghai, , China

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Shenyang, , China

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Shijiazhuang, , China

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Tianjin, , China

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Weifang, , China

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Wuhan, , China

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Wuhan, , China

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Wuhan, , China

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Xi'an, , China

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Xi'an, , China

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Xiamen, , China

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Xiangfan, , China

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Xinxiang, , China

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Zhengzhou, , China

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Brno, , Czechia

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Hořovice, , Czechia

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Hradec Králové, , Czechia

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Olomouc, , Czechia

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Prague, , Czechia

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Prague, , Czechia

Site Status NOT_YET_RECRUITING

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Angers, , France

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Besançon, , France

Site Status SUSPENDED

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Lille, , France

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Lyon, , France

Site Status NOT_YET_RECRUITING

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Marseille, , France

Site Status NOT_YET_RECRUITING

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Paris, , France

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Rouen, , France

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Saint-Herblain, , France

Site Status NOT_YET_RECRUITING

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Toulouse, , France

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Villejuif, , France

Site Status SUSPENDED

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Aachen, , Germany

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Augsburg, , Germany

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Berlin, , Germany

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Cologne, , Germany

Site Status WITHDRAWN

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Dessau, , Germany

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Düsseldorf, , Germany

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Erlangen, , Germany

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Göttingen, , Germany

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Hamburg, , Germany

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Hanover, , Germany

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Heidelberg, , Germany

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Kiel, , Germany

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Leipzig, , Germany

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Ludwigsburg, , Germany

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München, , Germany

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Münster, , Germany

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Hong Kong, , Hong Kong

Site Status NOT_YET_RECRUITING

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Hong Kong, , Hong Kong

Site Status NOT_YET_RECRUITING

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Budapest, , Hungary

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Budapest, , Hungary

Site Status RECRUITING

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Budapest, , Hungary

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Debrecen, , Hungary

Site Status NOT_YET_RECRUITING

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Miskolc, , Hungary

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Zalaegerszeg, , Hungary

Site Status NOT_YET_RECRUITING

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Delhi, , India

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Kolkata, , India

Site Status WITHDRAWN

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Lucknow, , India

Site Status WITHDRAWN

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Mumbai, , India

Site Status NOT_YET_RECRUITING

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Mumbai, , India

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Mysuru, , India

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Nagpur, , India

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Nashik, , India

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New Delhi, , India

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Surat, , India

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Thiruvananthapuram, , India

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Jerusalem, , Israel

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Jerusalem, , Israel

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Petah Tikva, , Israel

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Ramat Gan, , Israel

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Tel Aviv, , Israel

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Bergamo, , Italy

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Bologna, , Italy

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Milan, , Italy

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Milan, , Italy

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Modena, , Italy

Site Status WITHDRAWN

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Napoli, , Italy

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Padua, , Italy

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Reggio Emilia, , Italy

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Rome, , Italy

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Rozzano, , Italy

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Chiba, , Japan

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Hidaka-shi, , Japan

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Hirakata-shi, , Japan

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Isehara-shi, , Japan

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Kagoshima, , Japan

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Kashiwa, , Japan

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Kōtoku, , Japan

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Kumamoto, , Japan

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Kyoto, , Japan

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Matsuyama, , Japan

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Nagoya, , Japan

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Nagoya, , Japan

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Nagoya, , Japan

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Osaka, , Japan

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Ota-shi, , Japan

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Sapporo, , Japan

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Sendai, , Japan

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Shinagawa-ku, , Japan

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Suita-shi, , Japan

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Sunto-gun, , Japan

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Takasaki-shi, , Japan

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Tsu, , Japan

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Yokohama, , Japan

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Bandar Puncak Alam, , Malaysia

Site Status NOT_YET_RECRUITING

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Johor Bahru, , Malaysia

Site Status NOT_YET_RECRUITING

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Kuala Lumpur, , Malaysia

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Kuala Selangor, , Malaysia

Site Status NOT_YET_RECRUITING

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Malacca, , Malaysia

Site Status NOT_YET_RECRUITING

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Bellavista, , Peru

Site Status NOT_YET_RECRUITING

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Jesus Maria, Lima, , Peru

Site Status NOT_YET_RECRUITING

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Lima, , Peru

Site Status NOT_YET_RECRUITING

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Lima, , Peru

Site Status NOT_YET_RECRUITING

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Biała Podlaska, , Poland

Site Status WITHDRAWN

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Lodz, , Poland

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Lublin, , Poland

Site Status NOT_YET_RECRUITING

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Poznan, , Poland

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Warsaw, , Poland

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Coimbra, , Portugal

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Lisbon, , Portugal

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Lisbon, , Portugal

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Matosinhos Municipality, , Portugal

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Porto, , Portugal

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Vila Real, , Portugal

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San Juan, , Puerto Rico

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Daegu, , South Korea

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Seongnam-si, , South Korea

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Seoul, , South Korea

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Seoul, , South Korea

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Seoul, , South Korea

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Seoul, , South Korea

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Seoul, , South Korea

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Seoul, , South Korea

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Barcelona, , Spain

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Cáceres, , Spain

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Granada, , Spain

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L'Hospitalet de Llobregat, , Spain

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Madrid, , Spain

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Madrid, , Spain

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Málaga, , Spain

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Pamplona, , Spain

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Seville, , Spain

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Valencia, , Spain

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New Taipei City, , Taiwan

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Taichung, , Taiwan

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Tainan, , Taiwan

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Taipei, , Taiwan

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Taipei, , Taiwan

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Taipei, , Taiwan

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Taoyuan District, , Taiwan

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Bangkok, , Thailand

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Bangkok, , Thailand

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Dusit, , Thailand

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Hat Yai, , Thailand

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Ratchathewi, , Thailand

Site Status RECRUITING

Research Site

Ratchathewi, , Thailand

Site Status NOT_YET_RECRUITING

Research Site

Adapazarı, , Turkey (Türkiye)

Site Status RECRUITING

Research Site

Altındağ-Ankara, , Turkey (Türkiye)

Site Status RECRUITING

Research Site

Çankaya, , Turkey (Türkiye)

Site Status WITHDRAWN

Research Site

Istanbul, , Turkey (Türkiye)

Site Status RECRUITING

Research Site

Kayseri, , Turkey (Türkiye)

Site Status RECRUITING

Research Site

Cambridge, , United Kingdom

Site Status RECRUITING

Research Site

Guildford, , United Kingdom

Site Status RECRUITING

Research Site

London, , United Kingdom

Site Status RECRUITING

Research Site

Manchester, , United Kingdom

Site Status RECRUITING

Research Site

Oxford, , United Kingdom

Site Status WITHDRAWN

Research Site

Swansea, , United Kingdom

Site Status SUSPENDED

Research Site

Taunton, , United Kingdom

Site Status RECRUITING

Research Site

Truro, , United Kingdom

Site Status RECRUITING

Countries

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United States Argentina Australia Austria Brazil Bulgaria Canada Chile China Czechia France Germany Hong Kong Hungary India Israel Italy Japan Malaysia Peru Poland Portugal Puerto Rico South Korea Spain Taiwan Thailand Turkey (Türkiye) United Kingdom

Central Contacts

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AstraZeneca Clinical Study Information Center

Role: CONTACT

1-877-240-9479

Other Identifiers

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D9722C00001

Identifier Type: -

Identifier Source: org_study_id

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