Phase III, Open-label, Study of First-line Dato-DXd in Combination With Rilvegostomig for Advanced Non-squamous NSCLC With High PD-L1 Expression (TC ≥ 50%) and Without Actionable Genomic Alterations

NCT ID: NCT06357533

Last Updated: 2025-10-27

Study Results

Results pending

The study team has not published outcome measurements, participant flow, or safety data for this trial yet. Check back later for updates.

Basic Information

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Recruitment Status

RECRUITING

Clinical Phase

PHASE3

Total Enrollment

675 participants

Study Classification

INTERVENTIONAL

Study Start Date

2024-04-11

Study Completion Date

2030-05-24

Brief Summary

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The purpose of this study is to evaluate efficacy and safety of Dato-DXd in combination with rilvegostomig or rilvegostomig monotherapy compared with pembrolizumab monotherapy as a first line therapy in participants with locally advanced or metastatic non-squamous NSCLC with high PD-L1 expression (TC ≥ 50%) and without actionable genomic alterations.

Detailed Description

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This is a Phase III, randomized, open-label, Global Study of Datopotamab Deruxtecan (Dato-DXd) in Combination With Rilvegostomig or Rilvegostomig monotherapy versus Pembrolizumab monotherapy for the first-line treatment of participants with locally-advanced or metastatic non-squamous NSCLC with high PD-L1 expression (TC ≥ 50%) and without actionable genomic alterations.

Conditions

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Non-Small Cell Lung Cancer

Study Design

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Allocation Method

RANDOMIZED

Intervention Model

PARALLEL

Parallel Assignment
Primary Study Purpose

TREATMENT

Blinding Strategy

SINGLE

Outcome Assessors
Open-label, sponsor-blinded

Study Groups

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Arm 1: Datopotamab Deruxtecan in Combination With Rilvegostomig

Participants in the Datopotamab Deruxtecan (Dato-DXd) in combination with Rilvegostomig group will receive Dato-DXd plus rilvegostomig as intravenous (IV) infusion every 3 weeks (Q3W) on Day 1 of each 21-day cycle.

Group Type EXPERIMENTAL

Datopotamab Deruxtecan

Intervention Type DRUG

Datopotamab Deruxtecan IV (intravenous)

Rilvegostomig

Intervention Type DRUG

Rilvegostomig IV (intravenous)

Arm 2: Rilvegostomig Monotherapy

Participants in the rilvegostomig monotherapy group will receive rilvegostomig as intravenous (IV) infusion every 3 weeks (Q3W) on Day 1 of each 21-day cycle.

Group Type EXPERIMENTAL

Rilvegostomig

Intervention Type DRUG

Rilvegostomig IV (intravenous)

Arm 3: Pembrolizumab Monotherapy

Participants in the pembrolizumab group will receive pembrolizumab as intravenous (IV) infusion every 3 weeks (Q3W) on Day 1 of each 21-day cycle.

Group Type ACTIVE_COMPARATOR

Pembrolizumab

Intervention Type DRUG

Pembrolizumab IV (intravenous)

Interventions

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Datopotamab Deruxtecan

Datopotamab Deruxtecan IV (intravenous)

Intervention Type DRUG

Rilvegostomig

Rilvegostomig IV (intravenous)

Intervention Type DRUG

Pembrolizumab

Pembrolizumab IV (intravenous)

Intervention Type DRUG

Other Intervention Names

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Dato-DXd AZD2936 KEYTRUDA

Eligibility Criteria

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Inclusion Criteria

* Histologically or cytologically documented non-squamous NSCLC.
* Stage IIIB or IIIC or Stage IV metastatic NSCLC (according to Edition 8 of the AJCC staging manual) not amenable to curative surgery or definitive chemoradiation.
* Absence of sensitising EGFR mutations, and ALK and ROS1 rearrangements, and absence of documented local test result for any other known genomic alteration for which there are locally approved and available targeted first-line therapies.
* Must provide tumor sample to determine PD-L1 status, TROP2 status and other biomarkers.
* Known tumour PD-L1 expression status defined as TC ≥ 50%
* At least one lesion, not previously irradiated that qualifies as a RECIST 1.1 target lesion at baseline
* ECOG performance status of 0 or 1
* Adequate bone marrow reserve and organ function within 7 days before the first dose of study intervention

Exclusion Criteria

* Prior systemic therapy for advanced/metastatic NSCLC.
* Squamous cell histology, or predominantly squamous cell histology NSCLC; mixed small cell lung cancer; NSCLC histology, sarcomatoid variant.
* History of another primary malignancy within 3 years
* Active or prior documented autoimmune or inflammatory disorders (with exceptions)
* Any evidence of severe or uncontrolled systemic diseases, including, but not limited to active bleeding diseases, active infection, active ILD/pneumonitis, cardiac disease.
* Has clinically significant third-space fluid retention (for example pleural effusion) and is not amenable for repeated drainage.
* History of non-infectious ILD/pneumonitis that required steroids, has current ILD/pneumonitis, or has suspected ILD/pneumonitis that cannot be ruled out by imaging at screening
* Has significant pulmonary function compromise, as determined by the investigator
* Spinal cord compression, or brain metastases unless participant treated and no longer symptomatic, radiologically stable, and who require no treatment with corticosteroids or anticonvulsants.
* History of leptomeningeal carcinomatosis
* Known clinically significant corneal disease
* Active infection with TB, HBV, HCV, Hepatitis A, or known HIV infection that is not well controlled
* History of active primary immunodeficiency
Minimum Eligible Age

18 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

No

Sponsors

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Daiichi Sankyo

INDUSTRY

Sponsor Role collaborator

AstraZeneca

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Principal Investigators

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Suresh S. Ramalingam, MD

Role: PRINCIPAL_INVESTIGATOR

Emory University, Atlanta, Georgia, United States of America.

Locations

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Research Site

Anchorage, Alaska, United States

Site Status RECRUITING

Research Site

Tucson, Arizona, United States

Site Status RECRUITING

Research Site

Little Rock, Arkansas, United States

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Springdale, Arkansas, United States

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Anaheim, California, United States

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Beverly Hills, California, United States

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Fountain Valley, California, United States

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Newport Beach, California, United States

Site Status NOT_YET_RECRUITING

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Clermont, Florida, United States

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Gainesville, Florida, United States

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Miami Beach, Florida, United States

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Orange City, Florida, United States

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Orlando, Florida, United States

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Orlando, Florida, United States

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West Palm Beach, Florida, United States

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Atlanta, Georgia, United States

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Atlanta, Georgia, United States

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Atlanta, Georgia, United States

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Atlanta, Georgia, United States

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Hinsdale, Illinois, United States

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Noblesville, Indiana, United States

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Annapolis, Maryland, United States

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Boston, Massachusetts, United States

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Boston, Massachusetts, United States

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Dearborn, Michigan, United States

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Farmington Hills, Michigan, United States

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Grand Rapids, Michigan, United States

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Traverse City, Michigan, United States

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Hattiesburg, Mississippi, United States

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Kansas City, Missouri, United States

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Bozeman, Montana, United States

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Grand Island, Nebraska, United States

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Omaha, Nebraska, United States

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Las Vegas, Nevada, United States

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Reno, Nevada, United States

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Voorhees Township, New Jersey, United States

Site Status SUSPENDED

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Stony Brook, New York, United States

Site Status RECRUITING

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Greenville, North Carolina, United States

Site Status NOT_YET_RECRUITING

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Salisbury, North Carolina, United States

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Cincinnati, Ohio, United States

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Columbus, Ohio, United States

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Perrysburg, Ohio, United States

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Portland, Oregon, United States

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Greenville, South Carolina, United States

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Sioux Falls, South Dakota, United States

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Chattanooga, Tennessee, United States

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Knoxville, Tennessee, United States

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Fort Worth, Texas, United States

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Houston, Texas, United States

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Houston, Texas, United States

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Houston, Texas, United States

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Kingwood, Texas, United States

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Odessa, Texas, United States

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Fort Belvoir, Virginia, United States

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Leesburg, Virginia, United States

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Richmond, Virginia, United States

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Tacoma, Washington, United States

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Vancouver, Washington, United States

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Wenatchee, Washington, United States

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Birtinya, , Australia

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Blacktown, , Australia

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Clayton, , Australia

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Gosford, , Australia

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Melbourne, , Australia

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South Brisbane, , Australia

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Southport, , Australia

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Wodonga, , Australia

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Innsbruck, , Austria

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Krems, , Austria

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Linz, , Austria

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Rankweil, , Austria

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Vienna, , Austria

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Vienna, , Austria

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Wels, , Austria

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Anderlecht, , Belgium

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Hasselt, , Belgium

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La Louvière, , Belgium

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Liège, , Belgium

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Barretos, , Brazil

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Curitiba, , Brazil

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Florianópolis, , Brazil

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Ipatinga, , Brazil

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Natal, , Brazil

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Porto Alegre, , Brazil

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Rio de Janeiro, , Brazil

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Santa Maria, , Brazil

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São Paulo, , Brazil

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Taubaté, , Brazil

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Vancouver, British Columbia, Canada

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Winnipeg, Manitoba, Canada

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St. John's, Newfoundland and Labrador, Canada

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London, Ontario, Canada

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Newmarket, Ontario, Canada

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Oshawa, Ontario, Canada

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Toronto, Ontario, Canada

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Lévis, Quebec, Canada

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Montreal, Quebec, Canada

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Montreal, Quebec, Canada

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Montreal, Quebec, Canada

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Rimouski, Quebec, Canada

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Trois-Rivières, Quebec, Canada

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Saskatoon, Saskatchewan, Canada

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Chicoutimi, , Canada

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Beijing, , China

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Beijing, , China

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Changsha, , China

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Chengdu, , China

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Chengdu, , China

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Chongqing, , China

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Fuzhou, , China

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Guangzhou, , China

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Hangzhou, , China

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Hangzhou, , China

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Hangzhou, , China

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Harbin, , China

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Hefei, , China

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Hefei, , China

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Jinan, , China

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Jining, , China

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Kunming, , China

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Lanzhou, , China

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Linhai, , China

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Linyi, , China

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Nanjing, , China

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Nanning, , China

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Nanning, , China

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Shanghai, , China

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Shanghai, , China

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Shanghai, , China

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Shenyang, , China

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Taiyuan, , China

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Tianjin, , China

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Wenzhou, , China

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Wuhan, , China

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Wuhan, , China

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Wuhan, , China

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Wuhan, , China

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Xi'an, , China

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Yangzhou, , China

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Zhengzhou, , China

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Zhengzhou, , China

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Berlin, , Germany

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Bonn, , Germany

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Düsseldorf, , Germany

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Essen, , Germany

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Freiburg im Breisgau, , Germany

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Gauting, , Germany

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Georgsmarienhütte, , Germany

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Gera, , Germany

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Gütersloh, , Germany

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Hamburg, , Germany

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Hamburg, , Germany

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Heidelberg, , Germany

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Kempten, , Germany

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Koblenz, , Germany

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Ludwigsburg, , Germany

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München, , Germany

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Nuremberg, , Germany

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Potsdam, , Germany

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Ravensburg, , Germany

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Budapest, , Hungary

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Gyöngyös, , Hungary

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Gyöngyös - Mátraháza, , Hungary

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Győr, , Hungary

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Gyula, , Hungary

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Kecskemét, , Hungary

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Salgótarján, , Hungary

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Szekszárd, , Hungary

Site Status NOT_YET_RECRUITING

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Székesfehérvár, , Hungary

Site Status NOT_YET_RECRUITING

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Törökbálint, , Hungary

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Chennai, , India

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Dwārka, , India

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Jaipur, , India

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Kolkata, , India

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Marg Jaipur, , India

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Nagpur, , India

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Nashik, , India

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New Delhi, , India

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New Delhi, , India

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Thiruvananthapuram, , India

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Bergamo, , Italy

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Genoa, , Italy

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Milan, , Italy

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Milan, , Italy

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Monza, , Italy

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Padua, , Italy

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Pavia, , Italy

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Ravenna, , Italy

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Roma, , Italy

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Rozzano, , Italy

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Bunkyō City, , Japan

Site Status NOT_YET_RECRUITING

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Bunkyō City, , Japan

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Fukuoka, , Japan

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Fukuoka, , Japan

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Hidaka-shi, , Japan

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Hirakata-shi, , Japan

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Hirosaki-shi, , Japan

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Hiroshima, , Japan

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Kanazawa, , Japan

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Kashiwa, , Japan

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Kawasaki-shi, , Japan

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Kumamoto, , Japan

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Nagoya, , Japan

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Niigata, , Japan

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Okayama, , Japan

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Osaka, , Japan

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Osakasayama-shi, , Japan

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Sagamihara-shi, , Japan

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Sapporo, , Japan

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Takaoka-shi, , Japan

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Takatsuki-shi, , Japan

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Tokushima, , Japan

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Tokyo, , Japan

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Utsunomiya, , Japan

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Yokohama, , Japan

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Olsztyn, , Poland

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Poznan, , Poland

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Przemyśl, , Poland

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Warsaw, , Poland

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Warsaw, , Poland

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San Juan, , Puerto Rico

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Changwon, , South Korea

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Incheon, , South Korea

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Seongnam-si, , South Korea

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Seoul, , South Korea

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Seoul, , South Korea

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Suwon, , South Korea

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Suwon, , South Korea

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Alicante, , Spain

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Barcelona, , Spain

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Barcelona, , Spain

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Jerez de la Frontera, , Spain

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Reus,Tarragona, , Spain

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Salamanca, , Spain

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Kaohsiung City, , Taiwan

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New Taipei City, , Taiwan

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Taichung, , Taiwan

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Taichung, , Taiwan

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Tainan City, , Taiwan

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Taipei, , Taiwan

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Taipei, , Taiwan

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Taipei, , Taiwan

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Taipei, , Taiwan

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Taoyuan District, , Taiwan

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Bangkok, , Thailand

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Hat Yai, , Thailand

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Muang, , Thailand

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Mueang, , Thailand

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Mueang, , Thailand

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Adapazarı, , Turkey (Türkiye)

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Ankara, , Turkey (Türkiye)

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Ankara, , Turkey (Türkiye)

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Antalya, , Turkey (Türkiye)

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Diyarbakır, , Turkey (Türkiye)

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Istanbul, , Turkey (Türkiye)

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Istanbul, , Turkey (Türkiye)

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Cheltenham, , United Kingdom

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Inverness, , United Kingdom

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London, , United Kingdom

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London, , United Kingdom

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London, , United Kingdom

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Preston, , United Kingdom

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Truro, , United Kingdom

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Da Nang, , Vietnam

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Hanoi, , Vietnam

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Hà Nội, , Vietnam

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Ho Chi Minh City, , Vietnam

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Ho Chi Minh City, , Vietnam

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Huế, , Vietnam

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Vinh, , Vietnam

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Vĩnh Yên, , Vietnam

Site Status NOT_YET_RECRUITING

Countries

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United States Australia Austria Belgium Brazil Canada China Germany Hungary India Italy Japan Poland Puerto Rico South Korea Spain Taiwan Thailand Turkey (Türkiye) United Kingdom Vietnam

Central Contacts

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AstraZeneca Clinical Study Information Center

Role: CONTACT

1-877-240-9479

Other Identifiers

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2023-505077-32-00

Identifier Type: REGISTRY

Identifier Source: secondary_id

D7632C00001

Identifier Type: -

Identifier Source: org_study_id

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