Evaluate the Safety, Tolerability, Pharmacokinetics, and Preliminary Efficacy of ICP-248 as Monotherapy or in Combination With Anti-CD20 Monoclonal Antibody in Mature B-cell Malignancies

NCT ID: NCT06351527

Last Updated: 2025-06-19

Study Results

Results pending

The study team has not published outcome measurements, participant flow, or safety data for this trial yet. Check back later for updates.

Basic Information

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Recruitment Status

RECRUITING

Clinical Phase

PHASE1

Total Enrollment

78 participants

Study Classification

INTERVENTIONAL

Study Start Date

2024-04-23

Study Completion Date

2027-10-25

Brief Summary

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Evaluate the Safety, Tolerability, Pharmacokinetics and Preliminary Efficacy of ICP-248 as monotherapy or in combination with anti-CD20 monoclonal antibody in Mature B-cell Malignancies

Detailed Description

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Conditions

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Mature B-cell Malignancies

Study Design

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Allocation Method

NON_RANDOMIZED

Intervention Model

SINGLE_GROUP

Primary Study Purpose

TREATMENT

Blinding Strategy

NONE

Study Groups

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Dose-Escalation Cohort - CLL/SLL and MCL

Participants will receive ICP-248 daily from an initial dose of 5/10 mg to the target dose. Cycles will comprise 28 days.

Group Type EXPERIMENTAL

ICP-248

Intervention Type DRUG

ICP-248 will be administered orally once daily at escalated doses (starting dose 5/10 mg, maximum 150 mg).

Dose-Expansion Cohort A - CLL/SLL

Participants will receive ICP-248 daily from an initial dose of 5/10 mg to the target dose and obinutuzumab for 6 cycles. Cycles will comprise 28 days.

Group Type EXPERIMENTAL

ICP-248

Intervention Type DRUG

ICP-248 will be administered orally once daily at escalated doses (starting dose 5/10 mg, maximum 150 mg).

Obinutuzumab (G)

Intervention Type DRUG

Obinutuzumab will be administered by IV infusion at a dose of 100 mg or 1000 mg, depending on splitting rules, at Cycle 1, Day 1 (if 100 mg was received on Day 1, 900 mg will be administered on Cycle 1, Day 2); 1000 mg at Cycle 1, Day 8 and Day 15; 1000 mg at Day 1 for all subsequent cycles until the end of Cycle 6.

Dose-Expansion Cohort B - MCL

Participants will receive ICP-248 daily from an initial dose of 5/10 mg to the target dose. Cycles will comprise 28 days.

Group Type EXPERIMENTAL

ICP-248

Intervention Type DRUG

ICP-248 will be administered orally once daily at escalated doses (starting dose 5/10 mg, maximum 150 mg).

Dose-Expansion Cohort C - MCL

Participants will receive ICP-248 daily from an initial dose of 5/10 mg to the target dose and Rituximab for 18 cycles. Cycles will comprise 28 days.

Group Type EXPERIMENTAL

ICP-248

Intervention Type DRUG

ICP-248 will be administered orally once daily at escalated doses (starting dose 5/10 mg, maximum 150 mg).

Rituximab (R)

Intervention Type DRUG

Rituximab will be administered by IV infusion at a dose of 375 milligrams per square meter (mg/m\^2) at Day 1 per week for 4 weeks during cycle 1, then on day 1 of cycles 3-8, and thereafter once every other cycle up to 2 years.

Interventions

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ICP-248

ICP-248 will be administered orally once daily at escalated doses (starting dose 5/10 mg, maximum 150 mg).

Intervention Type DRUG

Obinutuzumab (G)

Obinutuzumab will be administered by IV infusion at a dose of 100 mg or 1000 mg, depending on splitting rules, at Cycle 1, Day 1 (if 100 mg was received on Day 1, 900 mg will be administered on Cycle 1, Day 2); 1000 mg at Cycle 1, Day 8 and Day 15; 1000 mg at Day 1 for all subsequent cycles until the end of Cycle 6.

Intervention Type DRUG

Rituximab (R)

Rituximab will be administered by IV infusion at a dose of 375 milligrams per square meter (mg/m\^2) at Day 1 per week for 4 weeks during cycle 1, then on day 1 of cycles 3-8, and thereafter once every other cycle up to 2 years.

Intervention Type DRUG

Eligibility Criteria

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Exclusion Criteria

1. Known central nervous system involvement by lymphoma/leukemia.
2. Known or suspected history of Richter's transformation.
3. Prior autologous stem cell transplant (unless ≥ 3 months since transplant); or prior chimeric cell therapy (unless ≥ 3 months since cell infusion).
4. A history of allogeneic stem cell transplantation.
5. An interval of less than 5 half-lives from the last dose of a strong CYP3A or CYP2C8 inhibitor or inducer (chemical agent, herbal medicine and dietary supplement) to the first dose of the investigational product, or a plan to use concurrently medications, dietary supplements or food (e.g., grapefruit or grapefruit juice) with strong CYP3A or CYP2C8 inhibitory or inductive effect during study participation
6. Presence of active infection that currently requires intravenous systemic anti-infective therapy.
7. History of immunodeficiency, including a positive human immunodeficiency virus (HIV) antibody test.
8. History of significant cardiovascular disease
9. Patients with previous or concomitant central nervous system disorders
10. Grade 2 or above toxicity due to prior anti-cancer therapy at screening
11. Known alcohol or drug dependence
12. Unable to swallow tablets or presence of disease significantly affecting gastrointestinal function such as malabsorption syndrome, resection of the stomach or small bowel, bariatric surgery procedures, symptomatic inflammatory bowel disease, or partial or complete bowel obstruction.
Minimum Eligible Age

18 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

No

Sponsors

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InnoCare Pharma Inc.

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Locations

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BRCR Medical Center

Plantation, Florida, United States

Site Status RECRUITING

Clinical Research Alliance

Westbury, New York, United States

Site Status RECRUITING

Pan American Center for Oncology Trials

San Juan, , Puerto Rico

Site Status RECRUITING

CNE CCOHTPC of Cherkasy Regional Council

Cherkasy, , Ukraine

Site Status RECRUITING

CNE"City Clin Hosp#4"of Dnipro City Council

Dnipro, , Ukraine

Site Status RECRUITING

Medical Center of Limited Liability Company Arensia Exploratory Medicine

Kyiv, , Ukraine

Site Status RECRUITING

Med Center 'Ok!Clinic+' of International Institute of Clinical Trials LLC

Kyiv, , Ukraine

Site Status RECRUITING

SI Institute of Blood Pathology and Transfusion Medicine of AMSU

Lviv, , Ukraine

Site Status RECRUITING

Countries

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United States Puerto Rico Ukraine

Central Contacts

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Study Director

Role: CONTACT

609-524-1106

Facility Contacts

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BRCR Medical Center

Role: primary

Clinical Research Alliance

Role: primary

Pan American Center for Oncology Trials

Role: primary

CNE CCOHTPC of Cherkasy Regional Council

Role: primary

CNE CCOHTPC of Cherkasy Regional Council

Role: primary

Medical Center of Limited Liability Company Arensia Explorator

Role: primary

Med Center 'Ok!Clinic+' of International Institute of Clinical

Role: primary

SI Institute of Blood Pathology and Transfusion Medicine of AM

Role: primary

Other Identifiers

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ICP-CL-01202

Identifier Type: -

Identifier Source: org_study_id

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