Evaluate The Efficacy, Safety, Pharmacokinetics And Pharmacodynamics Of EVER001

NCT ID: NCT05800873

Last Updated: 2025-05-31

Study Results

Results pending

The study team has not published outcome measurements, participant flow, or safety data for this trial yet. Check back later for updates.

Basic Information

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Recruitment Status

RECRUITING

Clinical Phase

PHASE1

Total Enrollment

30 participants

Study Classification

INTERVENTIONAL

Study Start Date

2023-05-15

Study Completion Date

2026-09-15

Brief Summary

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EVER001 is a highly selective, oral, reversable, covalent Bruton tyrosine kinase (BTK) inhibitor with high selectivity over other kinases, which is being developed to treat proteinuric glomerular diseases.

The overall aim of the study is to evaluate the efficacy, safety, pharmacokinetics and pharmacodynamics of EVER001 in subjects with selected proteinuric glomerular diseases. The first targeted disease is primary membranous nephropathy.

Detailed Description

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Conditions

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Primary Membranous Nephropathy

Study Design

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Allocation Method

NON_RANDOMIZED

Intervention Model

SINGLE_GROUP

Primary Study Purpose

TREATMENT

Blinding Strategy

NONE

Study Groups

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EVER001 100mg

EVER001 100mg QD for 4 weeks, followed by EVER001 100mg BID for 32 weeks.

Group Type EXPERIMENTAL

EVER001

Intervention Type DRUG

A highly selective, oral, reversable, covalent Bruton tyrosine kinase (BTK) inhibitor with high selectivity over other kinases.

EVER001 200mg

EVER001 200mg BID for 36 weeks.

Group Type EXPERIMENTAL

EVER001

Intervention Type DRUG

A highly selective, oral, reversable, covalent Bruton tyrosine kinase (BTK) inhibitor with high selectivity over other kinases.

Interventions

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EVER001

A highly selective, oral, reversable, covalent Bruton tyrosine kinase (BTK) inhibitor with high selectivity over other kinases.

Intervention Type DRUG

EVER001

A highly selective, oral, reversable, covalent Bruton tyrosine kinase (BTK) inhibitor with high selectivity over other kinases.

Intervention Type DRUG

Eligibility Criteria

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Inclusion Criteria

1. Having clinical diagnosis of primary membranous nephropathy, as verified by biopsy.
2. Have positive anti-PLA2R autoantibody test results \> 20 relative units (RU)/ml.
3. During screening at least one testing of proteinuria must be \>3.5 g/24h.
4. Have nephrotic range proteinuria for at least 8 weeks prior to Day 1 and no improvement (\<50% reduction) despite supportive therapy of ACE inhibitor or ARB unless contraindicated, for patients who have two tests of proteinuria during screening ≥8.0g/24h, the duration of nephrotic range proteinuria for at least 8 weeks is not required.

Exclusion Criteria

1. Non-primary membranous nephropathy or other condition affecting the kidney.
2. eGFR at screening \< 45 mL/min/1.73m2 or kidney function not stable .
3. Uncontrolled hypertension .
4. Serum albumin level at screening # 25g/l.
5. Have received: B-cell targeted therapy except rituximab at any time;Rituximab and the biosimilars within 2 years (participants with rituximab treatment between 1 and 2 years prior to Day 1 are eligible if there is documented evidence of B-cell repopulation to \>90% of Lower Limits of Normal Range.); Cyclophosphamide or Chlorambucil within 180 days;other immunosuppressive/immunomodulatory agents within 90 days;greater than 30mg/day prednisone or equivalence within 30 days.
6. Acute or chronic infection,including positivity of tuberculosis infection test.
7. Positive serology for TP,HIV, HBV, or HCV.
8. Lab testing abnormality as: WBC\< 3000/mm³, Lymphocyte \< 1000/ mm³, neutrophil \<1500/mm³, Hb \< 80g/L, Platelet count \<100×10e9/ L, Prothrombin time\>1.5×ULN, Activated partial thromboplastin time ≥1.5×ULN, Aspartate aminotransferase (AST) and alanine aminotransferase (ALT) ≥ 1.5×ULN, alkaline phosphatase and bilirubin \>1.5×ULN.
9. Judged by the investigator that the participant is unlikely to comply with study procedures, restrictions, and requirements.
Minimum Eligible Age

18 Years

Maximum Eligible Age

75 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

No

Sponsors

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Everest Medicines (China) Co.,Ltd.

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Locations

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The Second Xiangya Hospital Of Central South University

Changsha, Changsha, China

Site Status RECRUITING

The First Affiliated Hospital of PLA Army Medical University

Chongqing, Chongqing Municipality, China

Site Status RECRUITING

The Third Affiliated Hospital,Sun Yat Sen University

Guangzhou, Guangdong, China

Site Status RECRUITING

Peking University Shenzhen Hospital

Shenzhen, Guangdong, China

Site Status RECRUITING

The Second Affiliated Hospital of Harbin Medical University

Harbin, Harbin, China

Site Status RECRUITING

Xiangya Third Hospital, Central South University

Changsha, Hunan, China

Site Status RECRUITING

The First Affiliated Hospital of Baotou Medical College

Baotou, Inner Mongolia, China

Site Status RECRUITING

Zhongda Hospital Southeast University

Nanjing, Jiangsu, China

Site Status RECRUITING

The Second Affiliated Hospital of Soochow University

Suzhou, Jiangsu, China

Site Status RECRUITING

The Second Affiliated Hospital of Nanchang University

Nanchang, Jiangxi, China

Site Status RECRUITING

Ruijin Hospital, Shanghai Jiaotong University School of Medicine

Shanghai, Shanghai Municipality, China

Site Status RECRUITING

The First Affiliated Hospital of Medical college of Xi'an Jiaotong University

Xian, Shanxi, China

Site Status RECRUITING

Sichuan Province People's Hospital

Chengdu, Sichuan, China

Site Status RECRUITING

Second Hospital of Shanxi Medical University

Shanxi, Taiyuan, China

Site Status RECRUITING

The Second Affiliated Hospital of Zhejiang University School of Medicine

Hangzhou, Zhejiang, China

Site Status RECRUITING

Zhejiang Provincial People's Hospital

Hangzhou, Zhejiang, China

Site Status RECRUITING

The first affliated hospital of NingBo university

Ningbo, Zhejiang, China

Site Status RECRUITING

Taizhou Hospital of Zhejiang Province

Taizhou, Zhejiang, China

Site Status RECRUITING

Peking University First Hospital

Beijing, , China

Site Status RECRUITING

Countries

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China

Central Contacts

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Lixia Wang

Role: CONTACT

00862180123250

Facility Contacts

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Liu Hong

Role: primary

Zhao Hong Wen

Role: primary

Peng Hui

Role: primary

Xiong Zu Ying

Role: primary

Du Xuan Yi

Role: primary

Zhang Hao

Role: primary

Wang Cai Li

Role: primary

Liu Bi Cheng

Role: primary

Zeng Ying

Role: primary

Xu Cheng Yun

Role: primary

Zhang Wen

Role: primary

Lu Wan Hong

Role: primary

Chen Xiu Ling

Role: primary

Wang Li Hua

Role: primary

Ma Kun Ling

Role: primary

Li Yi Wen

Role: primary

Huang Jian Cheng

Role: primary

Xu Guang Biao

Role: primary

Minghui Zhao

Role: primary

Other Identifiers

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ES108001

Identifier Type: -

Identifier Source: org_study_id

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