ZN-c3 in Adult Participants With Metastatic Colorectal Cancer

NCT ID: NCT05743036

Last Updated: 2025-08-08

Study Results

Results pending

The study team has not published outcome measurements, participant flow, or safety data for this trial yet. Check back later for updates.

Basic Information

Get a concise snapshot of the trial, including recruitment status, study phase, enrollment targets, and key timeline milestones.

Recruitment Status

TERMINATED

Clinical Phase

PHASE1

Total Enrollment

44 participants

Study Classification

INTERVENTIONAL

Study Start Date

2023-02-27

Study Completion Date

2025-07-09

Brief Summary

Review the sponsor-provided synopsis that highlights what the study is about and why it is being conducted.

The purpose of this study is to evaluate the safety, tolerability, and potential clinical benefits of ZN-c3 administered in combination with encorafenib and cetuximab in adult participants with metastatic BRAF V600E mutant colorectal cancer previously treated with one or two treatment regimens.

Detailed Description

Dive into the extended narrative that explains the scientific background, objectives, and procedures in greater depth.

Conditions

See the medical conditions and disease areas that this research is targeting or investigating.

Metastatic Colorectal Cancer

Study Design

Understand how the trial is structured, including allocation methods, masking strategies, primary purpose, and other design elements.

Allocation Method

RANDOMIZED

Intervention Model

SEQUENTIAL

Primary Study Purpose

TREATMENT

Blinding Strategy

NONE

Study Groups

Review each arm or cohort in the study, along with the interventions and objectives associated with them.

Dose Escalation

Participants will receive different doses of ZN-c3 in combination with different doses of Encorafenib and a fixed dose of Cetuximab

Group Type EXPERIMENTAL

ZN-c3

Intervention Type DRUG

ZN-c3 tablet by mouth, in combination with encorafenib

Encorafenib

Intervention Type DRUG

Encorafenib capsule by mouth, in combination with ZN-c3

Cetuximab

Intervention Type DRUG

Infusion

Dose Expansion

Participants will receive recommended dose of ZN-c3 and encorafenib as determined in dose escalation phase in combination with cetuximab

Group Type EXPERIMENTAL

ZN-c3

Intervention Type DRUG

ZN-c3 tablet by mouth, in combination with encorafenib

Encorafenib

Intervention Type DRUG

Encorafenib capsule by mouth, in combination with ZN-c3

Cetuximab

Intervention Type DRUG

Infusion

Interventions

Learn about the drugs, procedures, or behavioral strategies being tested and how they are applied within this trial.

ZN-c3

ZN-c3 tablet by mouth, in combination with encorafenib

Intervention Type DRUG

Encorafenib

Encorafenib capsule by mouth, in combination with ZN-c3

Intervention Type DRUG

Cetuximab

Infusion

Intervention Type DRUG

Other Intervention Names

Discover alternative or legacy names that may be used to describe the listed interventions across different sources.

BRAFTOVI® ERBITUX®

Eligibility Criteria

Check the participation requirements, including inclusion and exclusion rules, age limits, and whether healthy volunteers are accepted.

Inclusion Criteria

* Histologically or cytologically confirmed metastatic Stage IV colorectal adenocarcinoma.
* Documented evidence of a BRAF V600E mutation in tumor tissue or blood
* Presence of measurable disease per RECIST version 1.1 guidelines.
* Disease progression after 1 or 2 previous systemic regimens for metastatic disease
* Adequate bone marrow function
* Adequate hepatic and renal function

Exclusion Criteria

* Documented clinical disease progression or radiographic disease progression during the screening period
* Leptomeningeal disease.
* Symptomatic brain metastasis.
* Presence of acute or chronic pancreatitis.
* Unable to swallow, retain, and absorb oral medications.
* Clinically significant cardiovascular diseases
* Evidence of active noninfectious pneumonitis.
* Evidence of active and uncontrolled bacterial or viral infection, within 2 weeks prior to start of any of the study interventions
* Participants with known positivity for HIV
* Active hepatitis B or hepatitis C infection
* Concurrent or previous other malignancy within 2 years of study entry
* Has had an allogeneic tissue/solid organ transplant
* Pregnant or females of childbearing potential who have a positive β-hCG laboratory test result within 14 days prior to enrollment or is breastfeeding
Minimum Eligible Age

18 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

No

Sponsors

Meet the organizations funding or collaborating on the study and learn about their roles.

Pfizer

INDUSTRY

Sponsor Role collaborator

K-Group, Beta, Inc., a wholly owned subsidiary of Zentalis Pharmaceuticals, Inc

INDUSTRY

Sponsor Role lead

Responsible Party

Identify the individual or organization who holds primary responsibility for the study information submitted to regulators.

Responsibility Role SPONSOR

Locations

Explore where the study is taking place and check the recruitment status at each participating site.

USC Norris Comprehensive Cancer Center

Los Angeles, California, United States

Site Status

Alliance for Multispecialty Research, LLC

Merriam, Kansas, United States

Site Status

University of Texas MD Anderson Cancer Center

Houston, Texas, United States

Site Status

The Queen Elizabeth Hospital

Woodville South, South Australia, Australia

Site Status

Peter MacCallum Cancer Centre

Melbourne, Victoria, Australia

Site Status

Hämatologie- Onkologie im Zentrum MVZ GmbH

Augsburg, Bavaria, Germany

Site Status

Klinikum der Universität München Großhadern

Munich, Bavaria, Germany

Site Status

Muenchen Klinik Neuperlach, Klinik fuer Haematologie und Onkologie

Munich, Bavaria, Germany

Site Status

Institut für Klinisch Onkologische Forschung

Frankfurt am Main, Hesse, Germany

Site Status

DRK Kliniken Berlin - Köpenick

Berlin, State of Berlin, Germany

Site Status

Semmelweis University-Department of Internal Medicine and Oncology

Budapest, Budapest, Hungary

Site Status

Clinexpert Kft. Bugat Pal Korhaz

Gyöngyös, , Hungary

Site Status

Istituto Nazionale Tumori IRCCS Fondazione Pascale

Napoli, Campania, Italy

Site Status

IRCCS Casa Sollievo della Sofferenza

San Giovanni Rotondo, Foggia, Italy

Site Status

Istituto Europeo di Oncologia

Milan, Milano, Italy

Site Status

ASST Grande Ospedale Metropolitano Niguarda

Milan, Milano, Italy

Site Status

AOUI Verona

Verona, Veneto, Italy

Site Status

Szpital Uniwersytecki w Krakowie

Krakow, Lesser Poland Voivodeship, Poland

Site Status

Szpital Specjalistyczny im. Ludwika Rydygiera w Krakowie

Krakow, Lesser Poland Voivodeship, Poland

Site Status

Narodowy Instytut Onkologii im. Marii Sklodowskiej-Curie - Panstwowy Instytut Badawczy w Warszawie

Warsaw, Masovian Voivodeship, Poland

Site Status

Opolskie Centrum Onkologii w Opolu im. prof. Tadeusza Koszarowskiego

Opole, Opole Voivodeship, Poland

Site Status

Hospital Universitari Vall d'Hebron

Barcelona, Barcelona, Spain

Site Status

Parc de Salut Mar - Hospital del Mar

Barcelona, Catalonia, Spain

Site Status

Hospital Universitario Reina Sofia

Córdoba, Cordoba, Spain

Site Status

Hospital Universitario La Paz

Madrid, Madrid, Spain

Site Status

Hospital Universitario Puerta de Hierro Majadahonda

Madrid, Madrid, Spain

Site Status

Fundación Instituto Valenciano de Oncología

Valencia, Valenciana, Comunitat, Spain

Site Status

Countries

Review the countries where the study has at least one active or historical site.

United States Australia Germany Hungary Italy Poland Spain

Other Identifiers

Review additional registry numbers or institutional identifiers associated with this trial.

Z0011001

Identifier Type: OTHER

Identifier Source: secondary_id

ZN-c3-016

Identifier Type: -

Identifier Source: org_study_id

More Related Trials

Additional clinical trials that may be relevant based on similarity analysis.

Cetuximab for Elderly Patients With mCRC
NCT01718808 TERMINATED PHASE2