Strategies and Treatments for Respiratory Infections & Viral Emergencies (STRIVE): Shionogi Protease Inhibitor (Ensitrelvir)

NCT ID: NCT05605093

Last Updated: 2025-11-17

Study Results

Results pending

The study team has not published outcome measurements, participant flow, or safety data for this trial yet. Check back later for updates.

Basic Information

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Recruitment Status

TERMINATED

Clinical Phase

PHASE3

Total Enrollment

602 participants

Study Classification

INTERVENTIONAL

Study Start Date

2022-12-23

Study Completion Date

2025-10-28

Brief Summary

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Treatments are needed to improve outcomes among patients hospitalized for COVID-19, including direct-acting antiviral (DAA) agents to mitigate the pathology driven by ongoing viral replication. This trial will evaluate S-217622 (ensitrelvir), an anti-SARS-CoV2 3C-like protease inhibitor (PI) developed by Shionogi \&; Co. Ltd.

The study design is a randomized, placebo-controlled, multi-center international clinical trial that will evaluate the clinical efficacy of ensitrelvir when given in addition to standard of care (SOC) for inpatients with COVID-19. The SOC will be determined by local established guidelines and may include additional DAA (e.g., remdesivir) and immunomodulatory treatment strategies. Certain SOC treatments will be pre-specified prior to randomization.

Detailed Description

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Conditions

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COVID-19

Study Design

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Allocation Method

RANDOMIZED

Intervention Model

PARALLEL

Primary Study Purpose

TREATMENT

Blinding Strategy

DOUBLE

Participants Investigators

Study Groups

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S-217622 (ensitrelvir) plus standard of care (SOC)

Study investigational agent (ensitrelvir) will be administered as oral tablets with dosing of 375mg (3 tabs) once on Day 0 and 125mg (1 tab) once daily on Days 1-4. All participants will receive the full 5-day course, including those who are discharged from hospitalization prior to Day 4.

Group Type EXPERIMENTAL

Shionogi Protease Inhibitor (S-217622)

Intervention Type DRUG

S-217622 (ensitrelvir) is an oral anti-SARS-CoV2 PI that does not require ritonavir co-administration The dose is 375/125 (375 mg on Day 0, followed by 125 mg daily on Days 1-4).

placebo plus standard of care (SOC)

Study investigational placebo will be administered as oral tablets with dosing of 375mg (3 tabs) once on Day 0 and 125mg (1 tab) once daily on Days 1-4. All participants will receive the full 5-day course, including those who are discharged from hospitalization prior to Day 4.

Group Type PLACEBO_COMPARATOR

placebo

Intervention Type DRUG

Placebo is an oral tablet administered once (3 tabs) on Day 0 and once (1 tab) daily on days 1-4, 5-day course.

Interventions

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Shionogi Protease Inhibitor (S-217622)

S-217622 (ensitrelvir) is an oral anti-SARS-CoV2 PI that does not require ritonavir co-administration The dose is 375/125 (375 mg on Day 0, followed by 125 mg daily on Days 1-4).

Intervention Type DRUG

placebo

Placebo is an oral tablet administered once (3 tabs) on Day 0 and once (1 tab) daily on days 1-4, 5-day course.

Intervention Type DRUG

Other Intervention Names

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ensitrelvir

Eligibility Criteria

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Inclusion Criteria

* Age ≥18 years.
* Informed consent for trial participation.
* Hospital admission (or boarding in an emergency department or other area awaiting hospital admission) with signs and/or symptoms of a respiratory infection.
* Confirmation of SARS-CoV2 infection by nucleic acid test (NAT) or equivalent non- NAT test \[list of approved tests is in the PIM\] collected within the prior 14 days.
* Onset of symptoms attributable to SARS-CoV2 infection occurred within 14 days before randomization.
* Hospitalized for the management of COVID-19, with signs and/or symptoms suggestive of lower respiratory tract infection.

Exclusion Criteria

* The patient is expected to be discharged from the hospital within the next 24 hours.
* Medical condition other than the acute respiratory infection (and its manifestations) that is likely to result in death within 7 days of randomization.
* Use of a strong CYP3A inducer within 14 days prior to enrollment
* Moribund condition, defined as prior cardiac arrest during this hospitalization and life expectancy less than 48 hours of randomization.
* Patient undergoing comfort care measures only such that treatment focuses on end-of- life symptom management over prolongation of life.
* Expected inability or unwillingness to participate in study procedures.
* In the opinion of the investigator, participation in a trial is not in the best interest of the patient.
* Allergy to investigational agent or vehicle
* Use of a concomitant medication that is contraindicated due to a drug-drug interaction with S-217622
* Moderate to severe hepatic impairment (i.e., Child-Pugh class B or C) or acute liver failure.
* Known estimated glomerular filtration rate (eGRF) \<30 mL/min/1.73m 2
* Continuous renal replacement therapy or chronic dialysis
* Current pregnancy
* Current breastfeeding and unwillingness to defer breastfeeding for 30 days after the last dose of investigational agent.
* Women of child-bearing potential who are unwilling to abstain from sexual intercourse with men or practice appropriate contraception through 30 days from the last dose of the investigational agent.
* Men who are unwilling to abstain from sexual intercourse with women of child- bearing potential or to use barrier contraception through 30 days from the last dose of the investigational agent.
* Inability to take investigational agent in tablet form by mouth.
Minimum Eligible Age

18 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

No

Sponsors

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National Institute of Allergy and Infectious Diseases (NIAID)

NIH

Sponsor Role collaborator

University of Minnesota

OTHER

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Principal Investigators

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Cavan Reilly, PhD

Role: PRINCIPAL_INVESTIGATOR

University of Minnesota

Jason Baker, MD

Role: STUDY_CHAIR

University of Minnesota

Locations

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University of Alabama Birmingham University Hospital (Site 213-002)

Birmingham, Alabama, United States

Site Status

Banner University Medical Center Tucson (Site 206-004)

Tucson, Arizona, United States

Site Status

Southern Arizona VA Healthcare System (Site 074-009)

Tucson, Arizona, United States

Site Status

UCSF Fresno (Site 203-005)

Fresno, California, United States

Site Status

VA Loma Linda Healthcare System (Site 074-017)

Loma Linda, California, United States

Site Status

MemorialCare Health System (Site 066-003

Long Beach, California, United States

Site Status

VA Long Beach Healthcare System (Site 074-026)

Long Beach, California, United States

Site Status

Cedars-Sinai Medical Center (Site 208-002)

Los Angeles, California, United States

Site Status

Ronald Reagan UCLA Medical Center (Site 203-002)

Los Angeles, California, United States

Site Status

VA Northern California Health Care System (Site 074-023)

Mather, California, United States

Site Status

Hoag Memorial Hospital Presbyterian (Site 080-026)

Newport Beach, California, United States

Site Status

Veterans Affairs Palo Alto Health Care System (VAPAHCS) (Site 074-005)

Palo Alto, California, United States

Site Status

UC Davis Health (Site 203-004)

Sacramento, California, United States

Site Status

VA San Diego Healthcare System (Site 074-016)

San Diego, California, United States

Site Status

Zuckerberg San Francisco General Hospital and Trauma Center (Site 213-007)

San Francisco, California, United States

Site Status

UCSF Medical Center at Mount Zion (203-007)

San Francisco, California, United States

Site Status

San Francisco VAMC (Site 074-002)

San Francisco, California, United States

Site Status

University of California San Francisco (Site 203-001)

San Francisco, California, United States

Site Status

Stanford University Hospital & Clinics (Site 203-003)

Stanford, California, United States

Site Status

Lundquist Institute for Biomedical Innovation (Site 066-002)

Torrance, California, United States

Site Status

Rocky Mountain Regional VA Medical Center (Site 074-010)

Aurora, Colorado, United States

Site Status

University of Colorado Hospital (Site 204-001)

Aurora, Colorado, United States

Site Status

Public Health Institute at Denver Health (Site 017-004)

Denver, Colorado, United States

Site Status

Yale University (Site 025-001)

New Haven, Connecticut, United States

Site Status

MedStar Health Research Institute/MedStar Washington Hospital Center (Site 009-021)

Washington D.C., District of Columbia, United States

Site Status

Washington DC VA Medical Center (Site 009-004)

Washington D.C., District of Columbia, United States

Site Status

University of Florida - Gainesville (Site 201-004)

Gainesville, Florida, United States

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Miami VA Healthcare System (Site 074-003)

Miami, Florida, United States

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Orlando VA Medical Center (Site 074-032)

Orlando, Florida, United States

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Tampa General Hospital (032-001)

Tampa, Florida, United States

Site Status

John H. Stroger, Jr. Hospital of Cook County (Site 080-046)

Chicago, Illinois, United States

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University of Illinois at Chicago (Site 008-012)

Chicago, Illinois, United States

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Carle Foundation Hospital (Site 080-049)

Urbana, Illinois, United States

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Lutheran Medical Group (Site 301-010)

Fort Wayne, Indiana, United States

Site Status

The University of Kansas Hospital (Site 080-044)

Kansas City, Kansas, United States

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University of Kentucky (Site 210-004)

Lexington, Kentucky, United States

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NIH Clinical Center (Site 080-043)

Bethesda, Maryland, United States

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Massachusetts General Hospital (202-002)

Boston, Massachusetts, United States

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Beth Israel Deaconess Medical Center (Site 202-001)

Boston, Massachusetts, United States

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Baystate Medical Center (Site 201-001)

Springfield, Massachusetts, United States

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UMass Chan Medical School (Site 080-007)

Worcester, Massachusetts, United States

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VA Ann Arbor Healthcare System (Site 074-028)

Ann Arbor, Michigan, United States

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Henry Ford Health System (Site 014-001)

Detroit, Michigan, United States

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Sinai-Grace Hospital (Site 205-005)

Detroit, Michigan, United States

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Hennepin Healthcare Research Institute (Site 027-001)

Minneapolis, Minnesota, United States

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M Health Fairview University of Minnesota Medical Center (Site 112-001)

Minneapolis, Minnesota, United States

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University of Minnesota

Minneapolis, Minnesota, United States

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Mayo Clinic (Site 054-001)

Rochester, Minnesota, United States

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University of Mississippi Medical Center (Site 202-005)

Jackson, Mississippi, United States

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Washington University School of Medicine (Site 003-001)

St Louis, Missouri, United States

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University of Nebraska Medical Center (Site 080-045)

Omaha, Nebraska, United States

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Dartmouth-Hitchcock Medical Center (301-024)

Lebanon, New Hampshire, United States

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Cooper University Hospital (Site 019-001)

Camden, New Jersey, United States

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Hackensack Meridian Health (Site 301-030)

Hackensack, New Jersey, United States

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New Jersey Medical School Clinical Research Center (028-001)

Newark, New Jersey, United States

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University of New Mexico Hospital (Site 213-008)

Albuquerque, New Mexico, United States

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CHRISTUS - St. Vincent (Site 080-051)

Santa Fe, New Mexico, United States

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NYU Brooklyn (301-033)

Brooklyn, New York, United States

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New York Presbyterian Queens (003-005)

Flushing, New York, United States

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Mount Sinai Queens (Site 081-105)

Long Island City, New York, United States

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NYU Long Island (301-034)

Mineola, New York, United States

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New York University Tisch Hospital (Site 301-013)

New York, New York, United States

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Mount Sinai Medical Center (Site 301-012)

New York, New York, United States

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NYC Health + Hospital Harlem (Site 003-003)

New York, New York, United States

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Weill Cornell Clinical Research Unit (065-001)

New York, New York, United States

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St. Lawrence Health System (Site 301-029)

Potsdam, New York, United States

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Lincoln Medical Center (Site 003-016)

The Bronx, New York, United States

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Montefiore Medical Center - Moses Hospital (Site 206-001)

The Bronx, New York, United States

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Montefiore Medical Center - Weiler campus (Site 206-003)

The Bronx, New York, United States

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James J. Peters VAMC (Site 023-003)

The Bronx, New York, United States

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Duke University Hospital (Site 301-006)

Durham, North Carolina, United States

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Wake Forest Baptist Health (Site 210-001)

Winston-Salem, North Carolina, United States

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University of Cincinnati Medical Center (Site 207-003)

Cincinnati, Ohio, United States

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Cleveland Clinic Foundation (Site 207-001)

Cleveland, Ohio, United States

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Ohio State University Wexner Medical Center (Site 207-004)

Columbus, Ohio, United States

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Portland VA Health Care System (074-024)

Portland, Oregon, United States

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Penn State Health Milton S. Hershey Medical Center (Site 209-002)

Hershey, Pennsylvania, United States

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Rhode Island Hospital (Site 080-036)

Providence, Rhode Island, United States

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The Miriam Hospital (Site 080-039)

Providence, Rhode Island, United States

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Kent County Memorial Hospital (080-048)

Warwick, Rhode Island, United States

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Ralph H. Johnson VA Medical Center (Site 074-015)

Charleston, South Carolina, United States

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Medical University of South Carolina (Site 210-002)

Charleston, South Carolina, United States

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Monument Health Rapid City Hospital (Site 213-005)

Rapid City, South Dakota, United States

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Vanderbilt University Medical Center (Site 212-001)

Nashville, Tennessee, United States

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Hendrick Medical Center (Site 080-014)

Abilene, Texas, United States

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CHRISTUS Spohn Shoreline Hospital (Site 080-001)

Corpus Christi, Texas, United States

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Baylor, Scott and White Health (301-003)

Dallas, Texas, United States

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Parkland Health and Hospital Systems (Site 084-002)

Dallas, Texas, United States

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UT Southwestern Medical Center (Site 084-001)

Dallas, Texas, United States

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Houston Methodist Hospital (Site 301-028)

Houston, Texas, United States

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MEDVAMC (Site 074-006)

Houston, Texas, United States

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University of Texas Health Science Center (Site 203-006)

Houston, Texas, United States

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CHRISTUS Good Shepherd Medical Center (Site 080-031)

Longview, Texas, United States

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UT Health San Antonio (Site 009-022)

San Antonio, Texas, United States

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Intermountain Medical Center (Site 211-001)

Murray, Utah, United States

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University of Utah Health (Site 211-002)

Salt Lake City, Utah, United States

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University of Virginia Health System, University Hospital (Site 210-003)

Charlottesville, Virginia, United States

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Salem VA Medical Center (Site 074-014)

Salem, Virginia, United States

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Harborview Medical Center (208-001)

Seattle, Washington, United States

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Providence (Sacred Heart) (Site 213-004)

Spokane, Washington, United States

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West Virginia University Medicine (301-023)

Morgantown, West Virginia, United States

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William S. Middleton Memorial Veterans Hospital (074-030)

Madison, Wisconsin, United States

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Froedtert Memorial Lutheran Hospital (052-001)

Milwaukee, Wisconsin, United States

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Instituto Medico Platense (Site 611-025)

La Plata, Buenos Aires, Argentina

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Sanatorio Allende (Site 611-030)

Córdoba, Córdoba Province, Argentina

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Clínica Central S.A. (611-028)

Villa Regina, Río Negro Province, Argentina

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Sanatorio Británico S.A. (611-027)

Rosario, Santa Fe Province, Argentina

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CEMIC (Site 611-021)

Buenos Aires, , Argentina

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Hospital Rawson (Site 611-012)

Córdoba, , Argentina

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Sanatorio Medico de Diagnostico y Tratamiento (611-029)

Santa Fe, , Argentina

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South Western Sydney Local Health District, Liverpool (Site 612-063)

Liverpool, New South Wales, Australia

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St. Vincent's Hospital (Site 612-002)

Sydney, New South Wales, Australia

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Westmead Hospital (Site 612-058)

Westmead, New South Wales, Australia

Site Status

Austin Health (612-020)

Heidelberg, Victoria, Australia

Site Status

The Alfred Hospital (Site 612-017)

Melbourne, Victoria, Australia

Site Status

Fundação Universidade Caxias do Sul Hospital Geral (649-218)

Caxias do Sul, Rio Grande do Sul, Brazil

Site Status

Hospital de Clínicas de Porto Alegre (649-101)

Porto Alegre, Rio Grande do Sul, Brazil

Site Status

Sociedade Literária e Caritativa Santo Agostinho - Hospital São José (Site 649-204)

Criciúma, Santa Catarina, Brazil

Site Status

Hospital Nereu Ramos (Site 649-210)

Florianópolis, Santa Catarina, Brazil

Site Status

Unimed Joinville Cooperativa de Trabalho Médico (Site 649-202)

Joinville, Santa Catarina, Brazil

Site Status

Associação Beneficente Hospital Universitário - Universidade de Marília (Site 649-212)

Marília, São Paulo, Brazil

Site Status

Instituto de Infectologia Emílio Ribas - IIER (Site 649-001)

São Paulo, São Paulo, Brazil

Site Status

Real e Benemérita Associação Portuguesa de Beneficência de São Paulo (Site 649-201

São Paulo, São Paulo, Brazil

Site Status

Hospital Alemão Oswaldo Cruz (649-215)

São Paulo, São Paulo, Brazil

Site Status

Associação Beneficente Síria - HCor (Site 649-203)

São Paulo, São Paulo, Brazil

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Hospital SEPACO (649-207)

São Paulo, São Paulo, Brazil

Site Status

Sociedade Beneficente de Senhoras Hospital Sirio-Libanês (Site 649-217)

São Paulo, São Paulo, Brazil

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Aarhus Universitetshospital, Skejby (625-002)

Aarhus, N, Denmark

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Aalborg Hospital (Site 625-005)

Aalborg, , Denmark

Site Status

Rigshospitalet, CHIP (Site 625-006)

Copenhagen, , Denmark

Site Status

Bispebjerg Hospital (Site 625-013)

Copenhagen, , Denmark

Site Status

Herlev/Gentofte Hospital (Site 625-012)

Hellerup, , Denmark

Site Status

Nordsjaellands Hospital, Hillerod (Site 625-009)

Hillerød, , Denmark

Site Status

Hvidovre University Hospital, Department of Infections Diseases (Site 625-001)

Hvidovre, , Denmark

Site Status

Kolding Sygehus, Medicinsk Afdeling (Site 625-011)

Kolding, , Denmark

Site Status

Odense University Hospital (Site 625-004)

Odense, , Denmark

Site Status

Zealand University Hospital Roskilde (Site 625-010)

Roskilde, , Denmark

Site Status

AIDS and Clinical Immunology Research Center (Site 627-201)

Tbilisi, , Georgia

Site Status

Universitätsklinikum Bonn, Medizinische Klinik I, Immunologische Ambulanz (622-010)

Bonn, , Germany

Site Status

Klinik I für Innere Medizin der Universität zu Köln (Site 622-008)

Cologne, , Germany

Site Status

Johann Wolfgang Goethe Univ. Hosp., Infektionsambulanz CRS (622-001)

Frankfurt, , Germany

Site Status

Dept of Critical Care and Pulmonary Medicine, Evangelismos General Hospital (635-020)

Athens, Attica, Greece

Site Status

1st Respiratory Medicine Dept, Athens University Medical School (635-015)

Athens, Attica, Greece

Site Status

3rd Dept of Medicine, Medical School (635-022)

Athens, Attica, Greece

Site Status

Attikon University General Hospital (Site 635-009)

Athens, Attica, Greece

Site Status

Democritus University of Thrace (635-021)

Alexandroupoli, Evros, Greece

Site Status

Fujita Health University Hospital (Site 612-105)

Toyoake, Aichi-ken, Japan

Site Status

Center Hospital of the National Center for Global Health and Medicine (Site 612-101)

Shinjuku-Ku, Tokyo, Japan

Site Status

Rinku General Medical Center (Site 612-107)

Osaka, , Japan

Site Status

Instituto Nacional de Ciencias Medicas y Nutricion Salvador Zubiran (Site 653-001)

Mexico City, Mexico City, Mexico

Site Status

Instituto Nacional de Enfermedades Respiratorias Ismael Cosió Villegas (Site 653-002)

Mexico City, Mexico City, Mexico

Site Status

Hospital General Dr. Aurelio Valdivieso (Site 653-004)

Oaxaca City, OA, Mexico

Site Status

Institute of Human Virology-Nigeria (IHVN) (Site 612-601)

Abuja, Federal Capital Territory, Nigeria

Site Status

Hospital Nacional Hipolito Unanue (651-008)

Lima, , Peru

Site Status

Hospital Nacional Sergio E. Bernales (651-007)

Lima, , Peru

Site Status

Wojewodzki Szpital Zakazny (Site 625-302)

Warsaw, , Poland

Site Status

VA Caribbean Health Care (074-033)

San Juan, PR, Puerto Rico

Site Status

Tan Tock Seng Hospital (Site 612-201)

Singapore, , Singapore

Site Status

Durban International Clinical Research Site (WWH) (652-005)

Durban, KwaZulu-Natal, South Africa

Site Status

Greys Hospital (080-202)

Pietermaritzburg, KwaZulu-Natal, South Africa

Site Status

University of Cape Town (UCT) Lung Institute (Site 080-201)

Cape Town, Western Cape, South Africa

Site Status

Seoul National University Bundang Hospital (Site 612-904)

Seongnam-si, Gyeonggi-do, South Korea

Site Status

Seoul St. Mary's Hospital (Site 612-903)

Seocho, Seoul, South Korea

Site Status

Asan Medical Center (612-901)

Seoul, , South Korea

Site Status

Chung-Ang University Hospital (Site 612-902)

Seoul, , South Korea

Site Status

Hospital Universitari Germans Trias i Pujol (626-003)

Badalona, Barcelona, Spain

Site Status

Hospital del Mar (626-025)

Barcelona, , Spain

Site Status

Hospital Universitari Vall d'Hebron (Site 626-033)

Barcelona, , Spain

Site Status

Hospital Clinic de Barcelona (626-004)

Barcelona, , Spain

Site Status

Hospital General Universitario Gregorio Marañón (Site 626-001)

Madrid, , Spain

Site Status

Hospital Clínico San Carlos (Site 626-017)

Madrid, , Spain

Site Status

Hospital Universitario La Paz (Site 626-012)

Madrid, , Spain

Site Status

University Hospital Zurich (Site 621-201)

Zurich, , Switzerland

Site Status

Chulalongkorn University and The HIV-NAT (Site 613-001)

Bangkok, , Thailand

Site Status

Khon Kaen University, Srinagarind Hospital (Site 613-003)

Khon Kaen, , Thailand

Site Status

MRC/UVRI & LSHTM Uganda Research Unit (634-601)

Entebbe, , Uganda

Site Status

Gulu Regional Referral Hospital (634-603)

Gulu, , Uganda

Site Status

St. Francis Hospital, Nsambya (Site 634-607)

Kampala, , Uganda

Site Status

Lira Regional Referral Hospital (634-605)

Lira, , Uganda

Site Status

Masaka Regional Referral Hospital (634-606)

Masaka, , Uganda

Site Status

Central City Clinical Hospital of Ivano-Frankivsk City Council (Site 627-302)

Ivano-Frankivsk, , Ukraine

Site Status

Treatment and Diagnostic Center ADONIS Plus (627-304)

Kyiv, , Ukraine

Site Status

Hospital #1 of Zhytomyr City Council (627-303)

Zhytomyr, , Ukraine

Site Status

Royal Free Hospital (634-006)

London, , United Kingdom

Site Status

Guy's & St. Thomas' NHS Foundation Trust (Site 634-011)

London, , United Kingdom

Site Status

Royal Victoria Infirmary (Site 634-007)

Newcastle upon Tyne, , United Kingdom

Site Status

Parirenyatwa General Hospital (Site 634-901)

Harare, , Zimbabwe

Site Status

Countries

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United States Argentina Australia Brazil Denmark Georgia Germany Greece Japan Mexico Nigeria Peru Poland Puerto Rico Singapore South Africa South Korea Spain Switzerland Thailand Uganda Ukraine United Kingdom Zimbabwe

Other Identifiers

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S-217622

Identifier Type: -

Identifier Source: org_study_id

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