Study to Compare Bictegravir/Lenacapavir Versus Current Therapy in People With HIV-1 Who Are Successfully Treated With a Complicated Regimen

NCT ID: NCT05502341

Last Updated: 2025-10-14

Study Results

Results pending

The study team has not published outcome measurements, participant flow, or safety data for this trial yet. Check back later for updates.

Basic Information

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Recruitment Status

ACTIVE_NOT_RECRUITING

Clinical Phase

PHASE2/PHASE3

Total Enrollment

689 participants

Study Classification

INTERVENTIONAL

Study Start Date

2022-08-16

Study Completion Date

2028-07-31

Brief Summary

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The goal of this clinical study is to learn more about the effects of switching to the study drugs, bictegravir (BIC) plus lenacapavir (LEN), versus current therapy (Phase 2) and BIC/LEN fixed-dose combination (FDC) versus current therapy (Phase 3) in people living with HIV (PWH).

Detailed Description

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Conditions

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HIV-1-infection

Study Design

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Allocation Method

RANDOMIZED

Intervention Model

PARALLEL

Primary Study Purpose

TREATMENT

Blinding Strategy

NONE

Study Groups

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Phase 2: Bictegravir (BIC) 75 mg + Lenacapavir (LEN) 25 mg

Participants will switch from their stable baseline regimen (SBR) to a regimen of BIC 75 mg + LEN 25 mg. Participants will receive a 2-day loading dose regimen of LEN 600 mg, in addition to the daily doses of BIC 75 mg + LEN 25 mg starting on Day 1 up to the end of randomized treatment (ERT) visit, participants will be treated for at least 24 weeks during the Randomized Period.

Following Randomized Period, the participants will have an option to participate in an Extension Period to receive BIC/LEN 75 mg/50 mg fixed dose combination (FDC).

Group Type EXPERIMENTAL

Bictegravir

Intervention Type DRUG

Tablets administered orally without regard to food

Lenacapavir

Intervention Type DRUG

Tablets administered orally without regard to food

Phase 2: BIC 75 mg + LEN 50 mg

Participants will switch from their SBR to a regimen of BIC 75 mg + LEN 50 mg. Participants will receive a 2-day loading dose regimen of LEN 600 mg, in addition to the daily doses of BIC 75 mg + LEN 50 mg starting on Day 1 up to the ERT visit, participants will be treated for at least 24 weeks during the Randomized Period.

Following Randomized Period, the participants will have an option to participate in an Extension Period to receive BIC/LEN 75 mg/50 mg FDC.

Group Type EXPERIMENTAL

Bictegravir

Intervention Type DRUG

Tablets administered orally without regard to food

Lenacapavir

Intervention Type DRUG

Tablets administered orally without regard to food

Phase 2: Stable Baseline Regimen (SBR)

Participants will continue with their SBR per prescription for up to the ERT visit, participants will be treated for at least 24 weeks during the Randomized Period.

Following Randomized Period, the participants will have an option to participate in an Extension Period to receive BIC/LEN 75 mg/50 mg FDC.

Group Type ACTIVE_COMPARATOR

Stable Baseline Regimen

Intervention Type DRUG

SBR will include a combination of antiretroviral (ARV) regimen. ARV regimen may include the following, except for participants taking a single tablet regimen or taking a complete parenteral regimen (Cabenuva).

* Nucleos(t)ide Reverse Transcriptase Inhibitors:

* Abacavir
* Emtricitabine
* Lamivudine
* Tenofovir alafenamide
* Tenofovir disoproxil fumarate
* Zidovudine
* Non-Nucleosite Reverse Transcriptase Inhibitors:

* Delavirdine
* Efavirenz
* Nevirapine
* Rilpivirine
* Doravirine
* Integrase Inhibitors:

* Bictegravir
* Cabotegravir
* Dolutegravir
* Elvitegravir
* Raltegravir
* Protease Inhibitors:

* Atazanavir
* Darunavir
* Fosamprenavir
* Indinavir
* Lopinavir
* Nelfinavir
* Saquinavir
* Tipranavir
* Chemokine Co-receptor 5 (CCR5) Antagonist:

* Maraviroc
* Fusion Inhibitors:

* Enfuvirtide
* gp120 Attachment Inhibitor:

* Fostemsavir
* Anti-CD4 Monoclonal Antibodies:

* Ibalizumab-uiyk

Phase 3: BIC/LEN 75 mg/50 mg Fixed-dose Combination (FDC)

Participants will switch from their SBR to a regimen of BIC/LEN 75 mg/50 mg FDC. Participants will receive a 2-day loading dose regimen of LEN 600 mg, in addition to the daily doses of BIC/LEN 75 mg/50 mg FDC starting on Day 1 up to the ERT visit, participants will be treated for at least 48 weeks during the Randomized Period.

Following Randomized Period, the participants will have an option to participate in an Extension Period to receive BIC/LEN 75 mg/50 mg FDC.

Group Type EXPERIMENTAL

BIC/LEN FDC

Intervention Type DRUG

Tablets administered orally without regard to food

Phase 3: Stable Baseline Regimen

Participants will continue with their SBR per prescription for up to the ERT visit, participants will be treated for at least 48 weeks during the Randomized Period.

Following Randomized Period, the participants will have an option to participate in an Extension Period to receive BIC/LEN 75 mg/50 mg FDC.

Group Type ACTIVE_COMPARATOR

Stable Baseline Regimen

Intervention Type DRUG

SBR will include a combination of antiretroviral (ARV) regimen. ARV regimen may include the following, except for participants taking a single tablet regimen or taking a complete parenteral regimen (Cabenuva).

* Nucleos(t)ide Reverse Transcriptase Inhibitors:

* Abacavir
* Emtricitabine
* Lamivudine
* Tenofovir alafenamide
* Tenofovir disoproxil fumarate
* Zidovudine
* Non-Nucleosite Reverse Transcriptase Inhibitors:

* Delavirdine
* Efavirenz
* Nevirapine
* Rilpivirine
* Doravirine
* Integrase Inhibitors:

* Bictegravir
* Cabotegravir
* Dolutegravir
* Elvitegravir
* Raltegravir
* Protease Inhibitors:

* Atazanavir
* Darunavir
* Fosamprenavir
* Indinavir
* Lopinavir
* Nelfinavir
* Saquinavir
* Tipranavir
* Chemokine Co-receptor 5 (CCR5) Antagonist:

* Maraviroc
* Fusion Inhibitors:

* Enfuvirtide
* gp120 Attachment Inhibitor:

* Fostemsavir
* Anti-CD4 Monoclonal Antibodies:

* Ibalizumab-uiyk

Interventions

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Bictegravir

Tablets administered orally without regard to food

Intervention Type DRUG

Lenacapavir

Tablets administered orally without regard to food

Intervention Type DRUG

BIC/LEN FDC

Tablets administered orally without regard to food

Intervention Type DRUG

Stable Baseline Regimen

SBR will include a combination of antiretroviral (ARV) regimen. ARV regimen may include the following, except for participants taking a single tablet regimen or taking a complete parenteral regimen (Cabenuva).

* Nucleos(t)ide Reverse Transcriptase Inhibitors:

* Abacavir
* Emtricitabine
* Lamivudine
* Tenofovir alafenamide
* Tenofovir disoproxil fumarate
* Zidovudine
* Non-Nucleosite Reverse Transcriptase Inhibitors:

* Delavirdine
* Efavirenz
* Nevirapine
* Rilpivirine
* Doravirine
* Integrase Inhibitors:

* Bictegravir
* Cabotegravir
* Dolutegravir
* Elvitegravir
* Raltegravir
* Protease Inhibitors:

* Atazanavir
* Darunavir
* Fosamprenavir
* Indinavir
* Lopinavir
* Nelfinavir
* Saquinavir
* Tipranavir
* Chemokine Co-receptor 5 (CCR5) Antagonist:

* Maraviroc
* Fusion Inhibitors:

* Enfuvirtide
* gp120 Attachment Inhibitor:

* Fostemsavir
* Anti-CD4 Monoclonal Antibodies:

* Ibalizumab-uiyk

Intervention Type DRUG

Other Intervention Names

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GS-9883 GS-6207

Eligibility Criteria

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Inclusion Criteria

* If plasma HIV-1 RNA measurements in the 6 months prior to screening are available, all levels must be \< 50 copies/mL.
* At least one documented plasma HIV-1 RNA level measured between 6 and 12 months (± 2 months) prior to screening. This and any other HIV-1 RNA measurements documented in this period must be \< 50 copies/mL
* Plasma HIV-1 RNA levels \< 50 copies/mL at screening.
* Currently receiving a complex antiretroviral (ARV) regimen due to previous viral resistance, or intolerance, or contraindication to existing single-tablet regimens (STR), and on this regimen for at least 6 months prior to the screening visit. The criteria to define a complex regimen in this study are as follows:

* A regimen containing a boosted protease inhibitor or a nonnucleos(t)ide reverse transcriptase inhibitor (NRTI) plus at least 1 other third agent (ie, an agent from a class other than NRTIs) (eg, bictegravir/emtricitabine/tenofovir alafenamide (coformulated; Biktarvy®)(BVY) + darunavir/cobicistat, BVY + etravirine), or
* A regimen of ≥ 2 pills/day, or a regimen requiring dosing more than once daily, or
* A regimen containing parenteral agent(s) (excluding a complete long-acting injectable regimen, such as intramuscular cabotegravir plus rilpivirine) as well as oral agents.
* No documented or suspected resistance to bictegravir (BIC).
* Estimated glomerular filtration rate ≥ 15 mL/min according to the Cockcroft-Gault formula for creatinine clearance (CLcr) who are not on renal replacement therapy.

Exclusion Criteria

* Prior use of, or exposure to, lenacapavir (LEN)
* Active tuberculosis infection
* Chronic hepatitis B virus (HBV) infection
Minimum Eligible Age

18 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

No

Sponsors

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Gilead Sciences

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Principal Investigators

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Gilead Study Director

Role: STUDY_DIRECTOR

Gilead Sciences

Locations

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Be Well Medical Center

Berkeley, California, United States

Site Status

Pacific Oaks Medical Group

Beverly Hills, California, United States

Site Status

Ruane Clinical Research Group, Inc

Los Angeles, California, United States

Site Status

Alta Bates Summit Medical Center, Summit Campus, East Bay Advanced Care

Oakland, California, United States

Site Status

Bios Clinical Research

Palm Springs, California, United States

Site Status

University of California San Diego (UCSD)

San Diego, California, United States

Site Status

Lundquist Institute for Biomedical Innovation at Harbor - UCLA Medical Center

Torrance, California, United States

Site Status

The Men's Health Foundation

West Hollywood, California, United States

Site Status

Denver Health Medical Center

Denver, Colorado, United States

Site Status

Yale University; School of Medicine; AIDS Program

New Haven, Connecticut, United States

Site Status

Midland Florida Clinical Research Center, LLC

DeLand, Florida, United States

Site Status

Therafirst Medical Centers

Fort Lauderdale, Florida, United States

Site Status

Gary Richmond, MD, PA, Inc.

Fort Lauderdale, Florida, United States

Site Status

Midway Immunology & Research Center, LLC

Ft. Pierce, Florida, United States

Site Status

Schiff Center for liver Diseases/University of Miami

Miami, Florida, United States

Site Status

Floridian Clinical Research

Miami Lakes, Florida, United States

Site Status

Orlando Immunology Center

Orlando, Florida, United States

Site Status

Therapeutic Concepts, PA

Orlando, Florida, United States

Site Status

Triple O Research Institute PA

West Palm Beach, Florida, United States

Site Status

Atlanta ID Group

Atlanta, Georgia, United States

Site Status

Mercer University School of Medicine

Macon, Georgia, United States

Site Status

Howard Brown Health Center

Chicago, Illinois, United States

Site Status

Kansas City Care Clinic

Kansas City, Missouri, United States

Site Status

Southampton Healthcare, Inc.

St Louis, Missouri, United States

Site Status

Saint Michael's Medical Center

Newark, New Jersey, United States

Site Status

AXCES Research Group

Santa Fe, New Mexico, United States

Site Status

New York Presbyterian Hospital

Flushing, New York, United States

Site Status

Ricky K. Hsu, MD, PC

New York, New York, United States

Site Status

University of North Carolina - Chapel Hill

Chapel Hill, North Carolina, United States

Site Status

East Carolina University

Greenville, North Carolina, United States

Site Status

Philadelphia FIGHT

Philadelphia, Pennsylvania, United States

Site Status

Medical University of South Carolina (MUSC) Research NEXUS

Charleston, South Carolina, United States

Site Status

Central Texas Clinical Research

Austin, Texas, United States

Site Status

St. Hope Foundation

Bellaire, Texas, United States

Site Status

AIDS Arms, Inc., DBA Prism Health North Texas

Dallas, Texas, United States

Site Status

North Texas Infectious Diseases Consultants

Dallas, Texas, United States

Site Status

Texas Centers for Infectious Disease Associates

Fort Worth, Texas, United States

Site Status

Gordon E. Crofoot MD PA

Houston, Texas, United States

Site Status

Diagnostic Clinic of Longview - Center for Clinical Research

Longview, Texas, United States

Site Status

Peter Shalit, MD

Seattle, Washington, United States

Site Status

Hospital General de Agudos J.M Ramon Mejia

Buenos Aires, , Argentina

Site Status

Fundación Huésped

Buenos Aires, , Argentina

Site Status

Helios Salud

Buenos Aires, , Argentina

Site Status

St.Vincent's Hospital Sydney

Darlinghurst, New South Wales, Australia

Site Status

Taylor Square Private Clinic

Darlinghurst, New South Wales, Australia

Site Status

Holdsworth House Medical Practice

Sydney, New South Wales, Australia

Site Status

Alfred Health

Melbourne, Victoria, Australia

Site Status

Chronic Viral Illness Service / McGill University Health Centre (MUHC)

Decarie Montreal, , Canada

Site Status

Clinique Medicale du Quartier Latin

Montreal, , Canada

Site Status

The Ottawa Hospital - General Campus

Ottawa, , Canada

Site Status

ID Clinic

Regina, , Canada

Site Status

Maple Leaf Research

Toronto, , Canada

Site Status

Spectrum Health

Vancouver, , Canada

Site Status

Instituto Dominicano de Estudio Virologicos - IDEV

Santo Domingo, , Dominican Republic

Site Status

CHU Nice-Hôpital l'Archet

Nice, , France

Site Status

Hospital Saint Louis

Paris, , France

Site Status

Groupe Hospitalier Bichat Claude Bernard

Paris, , France

Site Status

Höpital de la Pitié Salpêtrière

Paris, , France

Site Status

zibp Zentrum für Infektiologie Berlin Prenzlauer Berg GmbH

Berlin, , Germany

Site Status

Universitatsklinikum Bonn

Bonn, , Germany

Site Status

Infektio Research GmbH & Co.KG

Frankfurt, , Germany

Site Status

ICH Study Center GmbH & Co. KG

Hamburg, , Germany

Site Status

MVZ München am Goetheplatz

München, , Germany

Site Status

IRCCS Ospedale San Raffaele

Milan, , Italy

Site Status

ASST Fatebenefratelli Sacco

Milan, , Italy

Site Status

Azienda Ospedaliero-Universitaria di Modena

Modena, , Italy

Site Status

Istituto Nazionale Malattie Infettive "Lazzaro Spallanzani" IRCCS

Roma, , Italy

Site Status

ASL Città di Torino

Torino, , Italy

Site Status

National Hospital Organization Nagoya Medical Center

Nagoya, , Japan

Site Status

National Hospital Organization Osaka National Hospital

Osaka, , Japan

Site Status

Center Hospital of the National Center for Global Health and Medicine

Tokyo, , Japan

Site Status

Hope Clinical Research

San Juan, PR, Puerto Rico

Site Status

Proyecto ACTU

San Juan, PR, Puerto Rico

Site Status

Desmond Tutu Health Foundation Clinical Trials Unit

Cape Town, , South Africa

Site Status

Sefako Makgatho Health Sciences University

Ga-Rankuwa, , South Africa

Site Status

Ezintsha

Johannesburg, , South Africa

Site Status

Kyungpook National University Hospital

Daegu, , South Korea

Site Status

Chungnam National University Hospital

Daejeon, , South Korea

Site Status

Yonsei University Severance Hospital

Seoul, , South Korea

Site Status

The Catholic University of Korea Seoul St. Mary's Hospital

Seoul, , South Korea

Site Status

Hospital Clinic Provincial de Barcelona

Barcelona, , Spain

Site Status

Hospital Ramon y Cajal, Madrid

Madrid, , Spain

Site Status

Hospital Clinico San Carlos

Madrid, , Spain

Site Status

Hospital Universitario La Paz

Madrid, , Spain

Site Status

Hospital Universitario Virgen del Rocio

Seville, , Spain

Site Status

Kaohsiung Medical University Chung-Ho Memorial Hospital

Kaohsiung City, , Taiwan

Site Status

Kaohsiung Medical University Chung-Ho Memorial Hospital

Kaohsiung City, , Taiwan

Site Status

Far Eastern Memorial Hospital

New Taipei City, , Taiwan

Site Status

Taoyuan General Hospital

Taoyuan, , Taiwan

Site Status

Department of HIV & Sexual Medicine

Birmingham, , United Kingdom

Site Status

Brighton and Sussex University Hospitals NHS Trust

Brighton, , United Kingdom

Site Status

Barts Health NHS Trust

London, , United Kingdom

Site Status

HIV medicine and infectious diseases

London, , United Kingdom

Site Status

St.Stephen's AIDS Trust, Clinical Trials Unit, 1st Floor, St.Stephen's Centre

London, , United Kingdom

Site Status

Countries

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United States Argentina Australia Canada Dominican Republic France Germany Italy Japan Puerto Rico South Africa South Korea Spain Taiwan United Kingdom

Related Links

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Other Identifiers

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2022-500929-33

Identifier Type: OTHER

Identifier Source: secondary_id

DOH-27-052023-8574

Identifier Type: OTHER

Identifier Source: secondary_id

jRCT2051230168

Identifier Type: OTHER

Identifier Source: secondary_id

GS-US-621-6289

Identifier Type: -

Identifier Source: org_study_id

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