A Study to Evaluate KIN-3248 in Participants With Advanced Tumors Harboring FGFR2 and//or FGFR3 Gene Alterations

NCT ID: NCT05242822

Last Updated: 2025-05-07

Study Results

Results pending

The study team has not published outcome measurements, participant flow, or safety data for this trial yet. Check back later for updates.

Basic Information

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Recruitment Status

TERMINATED

Clinical Phase

PHASE1

Total Enrollment

54 participants

Study Classification

INTERVENTIONAL

Study Start Date

2022-03-29

Study Completion Date

2024-10-03

Brief Summary

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The purpose of this study is to evaluate the safety, tolerability, pharmacokinetics (PK), and preliminary efficacy of KIN-3248, an oral small molecule FGFR inhibitor, in adults with advanced tumors harboring FGFR2 and/or FGFR3 gene alterations.

Detailed Description

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This is a two-part, open label, multi-center, dose escalation and dose expansion study in participants with advanced tumors harboring FGFR2 and/or FGFR3 gene alterations.

Part A (dose escalation) is aimed at evaluating the safety, tolerability, pharmacokinetics (PK), and pharmacodynamics (PD) of KIN-3248, and determining the maximum tolerated dose (MTD) of daily dosing of KIN-3248.

Part B (dose expansion) may open once either the MTD and/or a biologically active dose of KIN-3248 is identified. Part B is aimed at evaluating the safety and efficacy of KIN-3248 at the recommended dose and schedule in participants with cancers harboring FGFR2 and/or FGFR3 gene alterations, including intrahepatic cholangiocarcinoma (ICC), urothelial cancer (UC), and other solid tumors.

Conditions

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Solid Tumor, Adult Intrahepatic Cholangiocarcinoma Urothelial Carcinoma

Study Design

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Allocation Method

NON_RANDOMIZED

Intervention Model

SEQUENTIAL

Primary Study Purpose

TREATMENT

Blinding Strategy

NONE

Study Groups

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Part A - dose escalation

Dose escalation of KIN-3248 in patients with solid tumors

Group Type EXPERIMENTAL

KIN-3248

Intervention Type DRUG

KIN-3248 will be administered orally once daily in 28-day cycles

Part B - dose expansion

Dose expansion evaluating the recommended dose and schedule of KIN-3248 identified from Part A

Group Type EXPERIMENTAL

KIN-3248

Intervention Type DRUG

KIN-3248 will be administered orally once daily in 28-day cycles

Interventions

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KIN-3248

KIN-3248 will be administered orally once daily in 28-day cycles

Intervention Type DRUG

Eligibility Criteria

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Inclusion Criteria

* Provide written informed consent prior to initiation of any study-specific procedures
* Advanced stage solid tumor
* Known FGFR2 and/or FGFR3 gene alteration, as confirmed by previous genomic analysis of tumor tissue or ctDNA
* Measurable or evaluable disease according to RECIST v1.1
* ECOG performance status 0 or 1
* Adequate organ function, as measured by laboratory values (criteria listed in protocol)
* Able to swallow, retain, and absorb oral medications

Exclusion Criteria

* Known clinically-active or clinically-progressive brain metastases from non-brain tumors
* History and/or current evidence of abnormal calcium-phosphorous homeostasis, ectopic mineralization or calcification, or corneal or retinal disorder/keratopathy
* GI tract disease causing an inability to take oral medication, malabsorption syndrome, requirement for intravenous alimentation, or uncontrolled inflammatory GI disease
* Active, uncontrolled bacterial, fungal, or viral infection
* Women who are lactating or breastfeeding, or pregnant
Minimum Eligible Age

18 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

No

Sponsors

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Kinnate Biopharma

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Locations

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Mayo Clinic Arizona

Phoenix, Arizona, United States

Site Status

UC San Diego Moores Cancer Center

La Jolla, California, United States

Site Status

Mayo Clinic Florida

Jacksonville, Florida, United States

Site Status

Sarah Cannon Research Institute - Lake Nona

Orlando, Florida, United States

Site Status

Massachusetts General Hospital

Boston, Massachusetts, United States

Site Status

START Midwest

Grand Rapids, Michigan, United States

Site Status

Mayo Clinic Rochester

Rochester, Minnesota, United States

Site Status

NYU Langone Cancer Center

New York, New York, United States

Site Status

Fox Chase Cancer Center

Philadelphia, Pennsylvania, United States

Site Status

Sarah Cannon Research Institute

Nashville, Tennessee, United States

Site Status

MD Anderson Cancer Center

Houston, Texas, United States

Site Status

University of Wisconsin Carbone Cancer Center

Madison, Wisconsin, United States

Site Status

Beijing Cancer Hospital

Beijing, Haidian District, China

Site Status

Rigshospitalet (Copenhagen University Hospital) - Finsencentret - Onkologisk Klinik

Copenhagen, , Denmark

Site Status

Seoul National University Hospital (SNUH)

Seoul, , South Korea

Site Status

Severance Hospital Yonsei University Health System

Seoul, , South Korea

Site Status

Samsung Medical Center

Seoul, , South Korea

Site Status

START (Fundacion Jimenez Diaz)

Madrid, Madrid, Spain

Site Status

National Taiwan University Hospital

Taipei, Taiwan, Taiwan

Site Status

Kaohsiung Medical University Hospital

Kaohsiung City, , Taiwan

Site Status

Veterans General Hospital - Taipei

Taipei, , Taiwan

Site Status

Countries

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United States China Denmark South Korea Spain Taiwan

Other Identifiers

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KN-4802

Identifier Type: -

Identifier Source: org_study_id

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