A Clinical Trial of GSK3640254 + Dolutegravir (DTG) in Human Immunodeficiency Virus-1 Infected Treatment-naive Adults

NCT ID: NCT04900038

Last Updated: 2023-12-14

Study Results

Results available

Outcome measurements, participant flow, baseline characteristics, and adverse events have been published for this study.

View full results

Basic Information

Get a concise snapshot of the trial, including recruitment status, study phase, enrollment targets, and key timeline milestones.

Recruitment Status

TERMINATED

Clinical Phase

PHASE2

Total Enrollment

85 participants

Study Classification

INTERVENTIONAL

Study Start Date

2021-08-18

Study Completion Date

2023-05-11

Brief Summary

Review the sponsor-provided synopsis that highlights what the study is about and why it is being conducted.

The purpose of this study was to evaluate the efficacy of GSK3640254 + DTG relative to lamivudine (3TC) + DTG in treatment-naïve adult participants living with human immunodeficiency virus (HIV)-1. The participants were randomized to one of the three doses of blinded GSK3640254 (100, 150, or 200 milligrams \[mgs\]) or a reference arm of blinded 3TC-each in combination with open label DTG.

Detailed Description

Dive into the extended narrative that explains the scientific background, objectives, and procedures in greater depth.

Conditions

See the medical conditions and disease areas that this research is targeting or investigating.

HIV Infections

Keywords

Explore important study keywords that can help with search, categorization, and topic discovery.

Human immunodeficiency virus-1 GSK3640254 Dolutegravir Lamivudine Treatment-naive

Study Design

Understand how the trial is structured, including allocation methods, masking strategies, primary purpose, and other design elements.

Allocation Method

RANDOMIZED

Intervention Model

PARALLEL

This is a randomized, parallel-group study.
Primary Study Purpose

TREATMENT

Blinding Strategy

DOUBLE

Participants Investigators
The dose level of GSK3640254 in each of the treatment arms containing GSK3640254 was blinded to the research participants and all study personnel during the study through the Week 24 primary endpoint.

Study Groups

Review each arm or cohort in the study, along with the interventions and objectives associated with them.

GSK3640254 100 mg + Dolutegravir (DTG) 50 mg

Participants with human immunodeficiency virus type 1 (HIV-1) orally received low dose (100 mg) GSK3640254 tablet blinded and 50 mg DTG unblinded. Each participant received one tablet per day of each intervention up to Week 24.

Group Type EXPERIMENTAL

GSK3640254

Intervention Type DRUG

GSK3640254 was available as 25 mg or 100 mg tablets administered orally.

Dolutegravir

Intervention Type DRUG

DTG was available as 50 mg tablets administered orally.

GSK3640254 150 mg + DTG 50 mg

Participants with HIV-1 orally received medium dose (150 mg) GSK3640254 tablet blinded and 50 mg DTG unblinded. Each participant received one tablet per day of each intervention up to Week 24.

Group Type EXPERIMENTAL

GSK3640254

Intervention Type DRUG

GSK3640254 was available as 25 mg or 100 mg tablets administered orally.

Dolutegravir

Intervention Type DRUG

DTG was available as 50 mg tablets administered orally.

GSK3640254 200 mg + DTG 50 mg

Participants with HIV-1 orally received high dose (200 mg) GSK3640254 tablet blinded and 50 mg DTG unblinded. Each participant received one tablet per day of each intervention up to Week 24.

Group Type EXPERIMENTAL

GSK3640254

Intervention Type DRUG

GSK3640254 was available as 25 mg or 100 mg tablets administered orally.

Dolutegravir

Intervention Type DRUG

DTG was available as 50 mg tablets administered orally.

DTG 50 mg + Lamivudine (3TC) 300 mg

Participants with HIV-1 orally received unblinded 50 mg DTG one tablet and blinded 300 mg 3TC. Each participant received one capsule per day of each intervention up to Week 24.

Group Type ACTIVE_COMPARATOR

Dolutegravir

Intervention Type DRUG

DTG was available as 50 mg tablets administered orally.

Lamivudine capsules

Intervention Type DRUG

3TC was available as 300 mg capsules administered orally as a blinded treatment.

Lamivudine tablets

Intervention Type DRUG

3TC was available as 300 mg tablets administered orally as an unblinded treatment.

Interventions

Learn about the drugs, procedures, or behavioral strategies being tested and how they are applied within this trial.

GSK3640254

GSK3640254 was available as 25 mg or 100 mg tablets administered orally.

Intervention Type DRUG

Dolutegravir

DTG was available as 50 mg tablets administered orally.

Intervention Type DRUG

Lamivudine capsules

3TC was available as 300 mg capsules administered orally as a blinded treatment.

Intervention Type DRUG

Lamivudine tablets

3TC was available as 300 mg tablets administered orally as an unblinded treatment.

Intervention Type DRUG

Eligibility Criteria

Check the participation requirements, including inclusion and exclusion rules, age limits, and whether healthy volunteers are accepted.

Inclusion Criteria

* Treatment-naive, defined as no anti-retrovirals (ARVs) (in combination or monotherapy) received after a known diagnosis of HIV-1 infection.
* Documented HIV infection and Screening plasma HIV-1 RNA greater than or equal to (\>=)1000 c/mL.
* Screening CD4+ T-cell count \>=250 cells per millimeter\^3 (cells/cubic millimeter).
* Body weight \>=50.0 kilograms (kg) (110 pounds \[lbs.\]) for men and \>=45.0 kg (99 lbs.) for women and body mass index (BMI) \>18.5 kilograms per meter\^2 (kg/meter square). Calculations will utilize sex assigned at birth.

Exclusion Criteria

* Any evidence of an active Centers for Disease Control and Prevention (CDC) Stage 3 disease \[CDC, 2014\], except cutaneous Kaposi's sarcoma not requiring systemic therapy.
* Presence of primary HIV infection, evidenced by acute retroviral syndrome (example \[e.g.\], fever, malaise, fatigue, etc.) and/or evidence of recent (within 3 months) documented viremia without antibody production and/or evidence of recent (within 3 months) documented seroconversion.
* Unstable liver disease (as defined by any of the following: presence of ascites, encephalopathy, coagulopathy, hypoalbuminemia, esophageal or gastric varices, or persistent jaundice or cirrhosis), known biliary abnormalities (with the exception of Gilbert's syndrome or asymptomatic gallstones or otherwise stable chronic liver disease per investigator assessment);
* History of ongoing or clinically relevant hepatitis within the previous 6 months.
* Any history of significant underlying psychiatric disorder.
* Any history of major depressive disorder with or without suicidal features, or anxiety disorders, that required medical intervention (pharmacologic or not) such as hospitalization or other inpatient treatment and/or chronic (\>6 months) outpatient treatment.
* A pre-existing condition, in the opinion of the Investigator or Medical Monitor, that could interfere with normal gastrointestinal anatomy or motility (e.g., gastroesophageal reflux disease \[GERD\], gastric ulcers, gastritis, inflammatory bowel disease), hepatic and/or renal function, or with the absorption, metabolism, and/or excretion of the study interventions or render the participant unable to take oral study treatment.
* Familial or personal history of long QT syndrome or sudden cardiac death.
* Active treatment for a viral infection other than HIV-1, such as Hepatitis B, with an agent that is active against HIV-1 (were known to be infected with HIV-1 after treatment for Hepatitis B was completed).
* Participants who require concomitant medications known to be associated with a prolonged corrected QT (QTc) interval.
* Exposure to an experimental drug, human blood product, monoclonal antibody, or vaccine (which does not have emergency, conditional, or standard market authorization) within 28 days prior to the first dose of study treatment.
Minimum Eligible Age

18 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

No

Sponsors

Meet the organizations funding or collaborating on the study and learn about their roles.

Syneos Health

OTHER

Sponsor Role collaborator

ViiV Healthcare

INDUSTRY

Sponsor Role lead

Responsible Party

Identify the individual or organization who holds primary responsibility for the study information submitted to regulators.

Responsibility Role SPONSOR

Principal Investigators

Learn about the lead researchers overseeing the trial and their institutional affiliations.

GSK Clinical Trials

Role: STUDY_DIRECTOR

ViiV Healthcare

Locations

Explore where the study is taking place and check the recruitment status at each participating site.

GSK Investigational Site

Bakersfield, California, United States

Site Status

GSK Investigational Site

Palm Springs, California, United States

Site Status

GSK Investigational Site

Denver, Colorado, United States

Site Status

GSK Investigational Site

Ft. Pierce, Florida, United States

Site Status

GSK Investigational Site

Miami, Florida, United States

Site Status

GSK Investigational Site

Orlando, Florida, United States

Site Status

GSK Investigational Site

Kansas City, Missouri, United States

Site Status

GSK Investigational Site

Omaha, Nebraska, United States

Site Status

GSK Investigational Site

Ciudad Autónoma de Buenos Aires, Buenos Aires, Argentina

Site Status

GSK Investigational Site

Buenos Aires, , Argentina

Site Status

GSK Investigational Site

Buenos Aires, , Argentina

Site Status

GSK Investigational Site

Montreal, Quebec, Canada

Site Status

GSK Investigational Site

Montreal, Quebec, Canada

Site Status

GSK Investigational Site

Paris, , France

Site Status

GSK Investigational Site

Tourcoing, , France

Site Status

GSK Investigational Site

Frankfurt am Main, Hesse, Germany

Site Status

GSK Investigational Site

Cologne, North Rhine-Westphalia, Germany

Site Status

GSK Investigational Site

Berlin, , Germany

Site Status

GSK Investigational Site

Hamburg, , Germany

Site Status

GSK Investigational Site

Bergamo, Lombardy, Italy

Site Status

GSK Investigational Site

Milan, Lombardy, Italy

Site Status

GSK Investigational Site

Porto, , Portugal

Site Status

GSK Investigational Site

Vila Nova de Gaia, , Portugal

Site Status

GSK Investigational Site

San Juan, , Puerto Rico

Site Status

GSK Investigational Site

Durban, , South Africa

Site Status

GSK Investigational Site

Johannesburg, , South Africa

Site Status

GSK Investigational Site

Parow, , South Africa

Site Status

GSK Investigational Site

Vosloorus Ext 2, , South Africa

Site Status

GSK Investigational Site

Barcelona, , Spain

Site Status

GSK Investigational Site

Barcelona, , Spain

Site Status

GSK Investigational Site

Barcelona, , Spain

Site Status

GSK Investigational Site

Bilbao, , Spain

Site Status

GSK Investigational Site

Elche, , Spain

Site Status

GSK Investigational Site

La Laguna-Tenerife, , Spain

Site Status

GSK Investigational Site

Madrid, , Spain

Site Status

GSK Investigational Site

Madrid, , Spain

Site Status

GSK Investigational Site

Madrid, , Spain

Site Status

GSK Investigational Site

Madrid, , Spain

Site Status

GSK Investigational Site

Madrid, , Spain

Site Status

GSK Investigational Site

Murcia, , Spain

Site Status

GSK Investigational Site

Palma de Mallorca, , Spain

Site Status

GSK Investigational Site

Sant Boi de Llobregat, , Spain

Site Status

GSK Investigational Site

Valencia, , Spain

Site Status

GSK Investigational Site

Vigo, , Spain

Site Status

Countries

Review the countries where the study has at least one active or historical site.

United States Argentina Canada France Germany Italy Portugal Puerto Rico South Africa Spain

Provided Documents

Download supplemental materials such as informed consent forms, study protocols, or participant manuals.

Document Type: Study Protocol

View Document

Document Type: Statistical Analysis Plan

View Document

Other Identifiers

Review additional registry numbers or institutional identifiers associated with this trial.

212483

Identifier Type: -

Identifier Source: org_study_id