First-in-Human Study of Orally Administered GS-441524 for COVID-19

NCT ID: NCT04859244

Last Updated: 2021-08-10

Study Results

Results pending

The study team has not published outcome measurements, participant flow, or safety data for this trial yet. Check back later for updates.

Basic Information

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Recruitment Status

COMPLETED

Clinical Phase

PHASE1

Total Enrollment

1 participants

Study Classification

INTERVENTIONAL

Study Start Date

2021-01-01

Study Completion Date

2021-08-01

Brief Summary

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This is a two-part study is to evaluate the multi-day safety, tolerability, and pharmacokinetics (PK) of orally administered GS-441524 in a healthy human volunteer.

Detailed Description

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Part 1: 750 mg GS-441524 administered once daily (QD) for 7 days. Part 2: 750 mg GS-441524 administered three times daily (TID) for 3 days.

Conditions

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COVID-19

Study Design

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Allocation Method

NON_RANDOMIZED

Intervention Model

CROSSOVER

Primary Study Purpose

TREATMENT

Blinding Strategy

NONE

Study Groups

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Part 1: GS-441524 (QD, 7 days)

750 mg GS-441524 administered QD for 7 days

Group Type EXPERIMENTAL

GS-441524

Intervention Type DRUG

750 mg administered as a solution

Part 2: GS-441524 (TID, 3 days)

750 mg GS-441524 administered TID for 3 days

Group Type EXPERIMENTAL

GS-441524

Intervention Type DRUG

750 mg administered as a solution

Interventions

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GS-441524

750 mg administered as a solution

Intervention Type DRUG

Other Intervention Names

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Parent nucleoside of remdesivir

Eligibility Criteria

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Inclusion Criteria

* Willing and able to provide written informed consent
* Negative pregnancy test at screening and prior to dosing
* Minimum body weight of 50 kg and body mass index (BMI) of 18-32 kg/m2

Exclusion Criteria

* Use of other investigational drugs within 28 days of dosing
* Positive pregnancy test
* Abuse of alcohol or drugs
* Other clinically significant medical conditions or laboratory abnormalities
Minimum Eligible Age

18 Years

Eligible Sex

FEMALE

Accepts Healthy Volunteers

Yes

Sponsors

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Copycat Sciences LLC

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Principal Investigators

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Victoria Yan

Role: PRINCIPAL_INVESTIGATOR

Copycat Sciences

Locations

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Copycat Sciences Study Site

Houston, Texas, United States

Site Status

Countries

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United States

References

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Humeniuk R, Mathias A, Cao H, Osinusi A, Shen G, Chng E, Ling J, Vu A, German P. Safety, Tolerability, and Pharmacokinetics of Remdesivir, An Antiviral for Treatment of COVID-19, in Healthy Subjects. Clin Transl Sci. 2020 Sep;13(5):896-906. doi: 10.1111/cts.12840. Epub 2020 Aug 5.

Reference Type BACKGROUND
PMID: 32589775 (View on PubMed)

Tempestilli M, Caputi P, Avataneo V, Notari S, Forini O, Scorzolini L, Marchioni L, Ascoli Bartoli T, Castilletti C, Lalle E, Capobianchi MR, Nicastri E, D'Avolio A, Ippolito G, Agrati C; COVID 19 INMI Study Group. Pharmacokinetics of remdesivir and GS-441524 in two critically ill patients who recovered from COVID-19. J Antimicrob Chemother. 2020 Oct 1;75(10):2977-2980. doi: 10.1093/jac/dkaa239.

Reference Type BACKGROUND
PMID: 32607555 (View on PubMed)

Davis MR, Pham CU, Cies JJ. Remdesivir and GS-441524 plasma concentrations in patients with end-stage renal disease on haemodialysis. J Antimicrob Chemother. 2021 Feb 11;76(3):822-825. doi: 10.1093/jac/dkaa472. No abstract available.

Reference Type BACKGROUND
PMID: 33152758 (View on PubMed)

Yan VC, Muller FL. Advantages of the Parent Nucleoside GS-441524 over Remdesivir for Covid-19 Treatment. ACS Med Chem Lett. 2020 Jun 23;11(7):1361-1366. doi: 10.1021/acsmedchemlett.0c00316. eCollection 2020 Jul 9.

Reference Type BACKGROUND
PMID: 32665809 (View on PubMed)

Study Documents

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Document Type: Individual Participant Data Set

Supplementary Table 1: Blood chemistry (CBC, CMP) results. Supplementary Table 2: Plasma concentrations of GS-441524 at indicated timepoints.

View Document

Related Links

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https://osf.io/am5s8/

Preliminary results

Other Identifiers

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CC-2021-001

Identifier Type: -

Identifier Source: org_study_id

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