Study of IDE397 in Participants With Solid Tumors Harboring MTAP Deletion

NCT ID: NCT04794699

Last Updated: 2025-11-12

Study Results

Results pending

The study team has not published outcome measurements, participant flow, or safety data for this trial yet. Check back later for updates.

Basic Information

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Recruitment Status

RECRUITING

Clinical Phase

PHASE1

Total Enrollment

180 participants

Study Classification

INTERVENTIONAL

Study Start Date

2021-04-14

Study Completion Date

2027-03-30

Brief Summary

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This is a Phase 1, open-label, multicenter, dose escalation and expansion study of the safety, PK, PD, and preliminary anti-tumor activity of IDE397 as a single agent and in combination with other anticancer agents including taxanes (docetaxel, paclitaxel), or sacituzumab govitecan (SG), in adult patients with selected advanced or metastatic MTAP-deleted advanced solid tumors who are unresponsive to standard of care therapy. IDE397 is a small molecule inhibitor of methionine adenosyltransferase 2 alpha (MAT2A).

Detailed Description

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Conditions

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Solid Tumor

Keywords

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MAT2A 9p21 CDKN2A MTAP Solid Tumors PRMT5 SAM Synthetic Lethality Inhibitor MTAP deletion CDKN2A deletion MAT2A Inhibitor Advanced solid tumors Lung Cancer Bladder Cancer Squamous NSCLC Urothelial Cancer Non small cell Docetaxel Paclitaxel Sacituzumab govitecan Trodelvy

Study Design

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Allocation Method

NON_RANDOMIZED

Intervention Model

PARALLEL

Primary Study Purpose

TREATMENT

Blinding Strategy

NONE

Study Groups

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Part 1: Dose Escalation Monotherapy (Solid Tumors)

Group Type EXPERIMENTAL

IDE397

Intervention Type DRUG

IDE397 dosed orally

Part 2: Monotherapy Dose Expansion (NSCLC, EG and Urothelial)

Group Type EXPERIMENTAL

IDE397

Intervention Type DRUG

IDE397 dosed orally

Part 3: Combination Dose Escalation with docetaxel or paclitaxel (NSCLC, EG and Urothelial)

Group Type EXPERIMENTAL

IDE397

Intervention Type DRUG

IDE397 dosed orally

Docetaxel

Intervention Type DRUG

Intravenous infusion

Paclitaxel

Intervention Type DRUG

Intravenous infusion

Part 4: Combination Dose Expansion with docetaxel or paclitaxel (NSCLC, EG and Urothelial)

Group Type EXPERIMENTAL

IDE397

Intervention Type DRUG

IDE397 dosed orally

Docetaxel

Intervention Type DRUG

Intravenous infusion

Paclitaxel

Intervention Type DRUG

Intravenous infusion

Part 5: Combination Dose Escalation with sacituzumab govitecan (SG) (Urothelial)

Group Type EXPERIMENTAL

IDE397

Intervention Type DRUG

IDE397 dosed orally

Sacituzumab govitecan

Intervention Type DRUG

Intravenous infusion

Part 6: Combination Dose Expansion with sacituzumab govitecan (SG) (Urothelial)

Group Type EXPERIMENTAL

IDE397

Intervention Type DRUG

IDE397 dosed orally

Sacituzumab govitecan

Intervention Type DRUG

Intravenous infusion

Interventions

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IDE397

IDE397 dosed orally

Intervention Type DRUG

Docetaxel

Intravenous infusion

Intervention Type DRUG

Paclitaxel

Intravenous infusion

Intervention Type DRUG

Sacituzumab govitecan

Intravenous infusion

Intervention Type DRUG

Eligibility Criteria

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Inclusion Criteria

* Participant must be at least 18 years of age
* Advanced or metastatic solid tumor that has progressed on at least one prior line of treatment or is intolerant to additional effective standard therapy
* Have evidence of homozygous loss of MTAP or MTAP deletion
* Willing to undergo paired fresh biopsy (pre- and post-treatment) procedure. Exceptions may be made for feasibility and safety concerns
* Measurable disease
* ECOG performance status \<= 1
* Adequate organ function
* Able to swallow and retain orally administered study treatment
* Recovery from acute effects of prior therapy
* Able to comply with contraceptive/barrier requirements

Exclusion Criteria

* Known symptomatic brain metastases
* Known primary CNS malignancy
* Current active liver or biliary disease
* Impairment of gastrointestinal (GI) function
* Active uncontrolled infection
* Clinically significant cardiac abnormalities
* Previous treatment with a MAT2A inhibitor and / or PRMT inhibitor or sacituzumab govitecan
* Systemic anti-cancer therapy or major surgery within 4 weeks prior to study entry
* Radiation therapy within 2 weeks prior to study entry
* Prior irradiation to \>25% of the bone marrow
* Current use or anticipated need for food or drugs that are known strong CYP3A4/5 inhibitors or inducers
* Currently receiving another investigational study drug.
* Known or suspected hypersensitivity to IDE397/excipients or components
Minimum Eligible Age

18 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

No

Sponsors

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IDEAYA Biosciences

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Principal Investigators

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Jasgit Sachdev, MD

Role: STUDY_DIRECTOR

IDEAYA Biosciences

Locations

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Honor Health Research Institute

Scottsdale, Arizona, United States

Site Status COMPLETED

Rockefeller Cancer Institute

Little Rock, Arkansas, United States

Site Status RECRUITING

City of Hope

Duarte, California, United States

Site Status RECRUITING

Hoag Memorial Hospital

Newport Beach, California, United States

Site Status RECRUITING

Providence Medical Group

Santa Rosa, California, United States

Site Status WITHDRAWN

Advent Health

Celebration, Florida, United States

Site Status WITHDRAWN

Orlando Health Cancer Institute

Orlando, Florida, United States

Site Status RECRUITING

Indiana University Health Hospital

Indianapolis, Indiana, United States

Site Status COMPLETED

Markey Cancer Center

Lexington, Kentucky, United States

Site Status WITHDRAWN

Sidney Kimmel Comprehensive Cancer Center at Johns Hopkins

Baltimore, Maryland, United States

Site Status RECRUITING

Dana Farber Cancer Institute

Boston, Massachusetts, United States

Site Status RECRUITING

Barbara Ann Karmanos Cancer Institute

Detroit, Michigan, United States

Site Status WITHDRAWN

Columbia University Medical Center - Herbert Irving Pavilion

New York, New York, United States

Site Status RECRUITING

Weill Cornell Medical College

New York, New York, United States

Site Status COMPLETED

Stephenson Cancer Center

Oklahoma City, Oklahoma, United States

Site Status RECRUITING

LifeSpan - Brown University

Providence, Rhode Island, United States

Site Status COMPLETED

Sarah Cannon Research Institute

Nashville, Tennessee, United States

Site Status RECRUITING

MD Anderson

Houston, Texas, United States

Site Status RECRUITING

Next Oncology

San Antonio, Texas, United States

Site Status COMPLETED

Swedish Cancer Institute

Seattle, Washington, United States

Site Status RECRUITING

The Kinghorn Cancer Centre, St Vincent's Health Network Sydney

Darlinghurst, New South Wales, Australia

Site Status RECRUITING

Southern Oncology Clinical Research Unit

Bedford Park, South Australia, Australia

Site Status COMPLETED

Institut Bergonie

Bordeaux, Bordeaux Cedex, France

Site Status RECRUITING

Institut Claudius Regaud - IUCT-Oncopole

Toulouse, Cedex 9, France

Site Status RECRUITING

Hôpital Timone

Marseille, Marseille, France

Site Status RECRUITING

Centre Eugène Marquis

Rennes, , France

Site Status RECRUITING

Universitaetsklinikum Hamburg-Eppendorf (UKE)

Hamburg, , Germany

Site Status RECRUITING

National Cancer Center

Goyang-si, Gyeonggi-do, South Korea

Site Status RECRUITING

CHA University - Bundang Medical Center

Seongnam-si, Gyeonggi-do, South Korea

Site Status RECRUITING

Chungbuk National University Hospital

Cheongju-si, North Chungcheong, South Korea

Site Status RECRUITING

Sevrance Hospital

Seoul, , South Korea

Site Status RECRUITING

Asan Medical Center

Seoul, , South Korea

Site Status RECRUITING

Vall Hebron Institute of Oncology

Barcelona, , Spain

Site Status RECRUITING

Hospital Universitario 12 de Octubre (H12O)

Madrid, , Spain

Site Status RECRUITING

START Madrid-HM - Centro Integral Oncológico Clara Campal (CIOCC)

Madrid, , Spain

Site Status RECRUITING

NEXT Madrid, Universitary Hospital QuironSAlud

Madrid, , Spain

Site Status RECRUITING

Instituto Valenciano de Oncología (IVO)

Valencia, , Spain

Site Status RECRUITING

National Cheng Kung University Hospital

Tainan, Tainan, Taiwan

Site Status RECRUITING

National Taiwan University Hospital

Taipei, Taipei, Taiwan

Site Status RECRUITING

Countries

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United States Australia France Germany South Korea Spain Taiwan

Central Contacts

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IDEAYA Clinical Trials

Role: CONTACT

Phone: 855-433-2246

Email: [email protected]

Facility Contacts

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Maroof Khan Zafar

Role: primary

New Patient Services

Role: primary

Estefania Bobe Cortes

Role: primary

Carol Goldener

Role: primary

Kailene Sullivan

Role: primary

Benjamin Herzberg, MD

Role: primary

Christina Seunath

Role: primary

askSARAH

Role: primary

Jordi Rodon, MD

Role: primary

Jia Liu

Role: primary

Antoine Italiano

Role: primary

Carlos Gomez-Roca

Role: primary

Laurent Greillier

Role: primary

Thibault De la Motte Rouge

Role: primary

Frank Knauer

Role: primary

Ji-Youn Han

Role: primary

Joo-Hang Kim

Role: primary

Ki Hyeong Lee

Role: primary

Hye Ryun Kim

Role: primary

Changmin Choi

Role: primary

Montserrat Pequera Juvany

Role: primary

Elisa Lorente

Role: primary

Marta Benitez

Role: primary

Jorge Mercado

Role: primary

Laura Bailach

Role: primary

Ya-Zong Hsu

Role: primary

Chia-Chi Lin

Role: primary

Other Identifiers

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IDE397-001

Identifier Type: -

Identifier Source: org_study_id