First-in-Human Study of EOS100850 (Inupadenant) in Patients with Cancer

NCT ID: NCT03873883

Last Updated: 2024-09-19

Study Results

Results pending

The study team has not published outcome measurements, participant flow, or safety data for this trial yet. Check back later for updates.

Basic Information

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Recruitment Status

COMPLETED

Clinical Phase

PHASE1

Total Enrollment

119 participants

Study Classification

INTERVENTIONAL

Study Start Date

2019-02-05

Study Completion Date

2024-05-28

Brief Summary

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Multicenter, open-label, dose-escalation Phase I/Ib clinical study to evaluate the safety and tolerability, the MTD/RP2D, pharmacokinetics (PK), pharmacodynamics (PD), and antitumor activity of EOS100850 (Inupadenant) as a Single Agent and in Combination with Pembrolizumab and/or Chemotherapy in Participants with Advanced Cancers.

Detailed Description

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Conditions

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Solid Tumor, Adult

Study Design

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Allocation Method

NON_RANDOMIZED

Intervention Model

SEQUENTIAL

Primary Study Purpose

TREATMENT

Blinding Strategy

NONE

Study Groups

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1A Dose escalation EOS100850

Dose Escalation- EOS100850 Monotherapy: to confirm RP2D

Group Type EXPERIMENTAL

EOS100850

Intervention Type DRUG

Oral administration

1B Dose escalation EOS100850 and Pembrolizumab

EOS100850 and Pembrolizumab Combination Therapy: to confirm RP2D as combination

Group Type EXPERIMENTAL

EOS100850

Intervention Type DRUG

Oral administration

Pembrolizumab

Intervention Type DRUG

IV Infusion

2A Dose Expansion- EOS100850

Dose Expansion - EOS100850 Monotherapy: to explore safety, PK, PD, and antitumor activity of inupadenant as monotherapy

Group Type EXPERIMENTAL

EOS100850

Intervention Type DRUG

Oral administration

2B Dose Expansion - EOS100850 and Pembrolizumab

Dose Expansion - EOS100850 and Pembrolizumab Combination Therapy: to explore safety, PK, PD, and antitumor activity of inupadenant in combination with pembrolizumab in melanoma and CRPC patients

Group Type EXPERIMENTAL

EOS100850

Intervention Type DRUG

Oral administration

Pembrolizumab

Intervention Type DRUG

IV Infusion

2D Dose expansion - EOS100850 and Chemotherapy in TNBC

Dose expansion - EOS100850 and Chemotherapy Combination: to explore safety, PK, PD, and antitumor activity of inupadenant in combination with chemotherapy SOC carboplatin and paclitaxel in patients with TNBC

Group Type EXPERIMENTAL

EOS100850

Intervention Type DRUG

Oral administration

Chemotherapy

Intervention Type DRUG

Standard of Care IV Infusion

3 EOS100850 in BMK-H participants

Dose expansion - EOS100850 Monotherapy : to evaluate the safety, PD, and antitumor activity of inupadenant as monotherapy at the mono-RP2D in BMK-H participants in 4 disease-specific cohorts: NSCLC; HNSCC; EC; and other forms of cancer

Group Type EXPERIMENTAL

EOS100850

Intervention Type DRUG

Oral administration

Interventions

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EOS100850

Oral administration

Intervention Type DRUG

Pembrolizumab

IV Infusion

Intervention Type DRUG

Chemotherapy

Standard of Care IV Infusion

Intervention Type DRUG

Other Intervention Names

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Inupadenant Keytruda MK-3475 carboplatin and paclitaxel

Eligibility Criteria

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Inclusion Criteria

* Women and men ≥18 years of age with Eastern Cooperative Oncology Group (ECOG) performance status of 0 or 1
* Subject with histologically or cytologically confirmed advanced solid tumor for whom no standard treatment is further available.
* At least 4 weeks since any previous treatment for cancer
* Subject must consent to pretreatment and on treatment tumor biopsies
* Adequate organ and marrow function

Exclusion Criteria

* Patients with primary brain tumors or primary tumors with central nervous system metastases as only location of disease. Controlled brain metastases are permitted
* Participants with second/other active cancers requiring current treatment
* Uncontrolled/significant heart disease
* Known History of chronic hepatitis, Positive test for Hepatitis B virus surface antigen or Hepatitis C antibody (except participants with liver cancer) or Human Immunodeficiency Virus/Acquired Immunodeficiency Syndrome(HIV/AIDS)
* Active/uncontrolled autoimmune disease
* Active infection
Minimum Eligible Age

18 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

No

Sponsors

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iTeos Belgium SA

INDUSTRY

Sponsor Role collaborator

Merck Sharp & Dohme LLC

INDUSTRY

Sponsor Role collaborator

iTeos Therapeutics

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Principal Investigators

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Iteos Clinical Trials

Role: STUDY_DIRECTOR

iTeos Belgium SA

Locations

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Karmanos Cancer Institute

Michigan Center, Michigan, United States

Site Status

John Theurer Cancer Center, Hackensack University Medical Center

Hackensack, New Jersey, United States

Site Status

University of Texas Health Science Center at San Antonio

San Antonio, Texas, United States

Site Status

Hospital GZA Sint-Augustinus

Wilrijk, Antwerpen, Belgium

Site Status

Institut Jules Bordet

Anderlecht, Brussels Capital, Belgium

Site Status

UCL Saint-Luc

Brussels, Brussels Capital, Belgium

Site Status

UZ Ghent

Ghent, East-Flanders, Belgium

Site Status

Centre de Lutte Contre le Cancer (CLCC) - Universite de Lyon - Centre Leon-Berard

Lyon, , France

Site Status

Centre Hospitalier Universitaire de Poitiers - Hopital la Miletrie- Pôle Régional de Cancérologie

Poitiers, , France

Site Status

Centre de Lutte Contre le Cancer - Institut de Cancerologie de l'Ouest - Rene Gauducheau

Saint-Herblain, , France

Site Status

Gustave Roussy

Villejuif, , France

Site Status

Yonsei University Severance Hospital

Seoul, , South Korea

Site Status

Samsung Medical Center

Seoul, , South Korea

Site Status

St Mary's Hospital, The Catholic University of Korea

Seoul, , South Korea

Site Status

Hospital del Mar

Barcelona, , Spain

Site Status

START Madrid-HM CIOCC Hospital Universitario HM Sanchinarro

Madrid, , Spain

Site Status

Universidad de Navarra - Clinica Universitaria de Navarra

Pamplona, , Spain

Site Status

Onkologikoa

San Sebastián, , Spain

Site Status

The Royal Marsden NHS Foundation Trust - Royal Marsden Hospital

Sutton, , United Kingdom

Site Status

Countries

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United States Belgium France South Korea Spain United Kingdom

Other Identifiers

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2018-003173-10

Identifier Type: EUDRACT_NUMBER

Identifier Source: secondary_id

Keynote A45

Identifier Type: OTHER

Identifier Source: secondary_id

IO-001

Identifier Type: -

Identifier Source: org_study_id

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