A Study to Compare Bioavailability of Naloxone Nasal Spray, Naloxone Hydrochloride (HCl) Intravenous (IV) and Intramuscular Injection (IM) in Healthy Volunteers

NCT ID: NCT03827642

Last Updated: 2019-02-01

Study Results

Results pending

The study team has not published outcome measurements, participant flow, or safety data for this trial yet. Check back later for updates.

Basic Information

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Recruitment Status

COMPLETED

Clinical Phase

PHASE1

Total Enrollment

24 participants

Study Classification

INTERVENTIONAL

Study Start Date

2018-04-23

Study Completion Date

2018-05-06

Brief Summary

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The main objective of this study was to compare the bioavailability of two test formulations of Naloxone Nasal Spray with the reference formulations of Naloxone HCl IV and IM injection under fasted conditions.

Detailed Description

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Conditions

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Healthy Volunteer

Study Design

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Allocation Method

RANDOMIZED

Intervention Model

CROSSOVER

Primary Study Purpose

TREATMENT

Blinding Strategy

NONE

Study Groups

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Cohort 1: Treatment Sequence A-D-C-B

Participants received Treatment A on Day 1 of Period 1, Treatment D on Day 1 of Period 2, Treatment C on Day 1 of Period 3 and Treatment B on Day 1 of Period 4.

Group Type EXPERIMENTAL

Treatment A: Naloxone Nasal Spray

Intervention Type DRUG

Participants received naloxone nasal spray following a 10 hour fast.

Treatment B: Naloxone Nasal Spray

Intervention Type DRUG

Participants received naloxone nasal spray following a 10 hour fast.

Treatment C: Naloxone HCl Intravenous (IV) Injection

Intervention Type DRUG

Participants received naloxone HCl IV injection following a 10 hour fast.

Treatment D: Naloxone HCl Intramuscular (IM) Injection

Intervention Type DRUG

Participants received naloxone HCl IM injection following a 10 hour fast.

Cohort 2: Treatment Sequence B-C-D-A

Participants received Treatment B on Day 1 of Period 1, Treatment C on Day 1 of Period 2, Treatment D on Day 1 of Period 3 and Treatment A on Day 1 of Period 4.

Group Type EXPERIMENTAL

Treatment A: Naloxone Nasal Spray

Intervention Type DRUG

Participants received naloxone nasal spray following a 10 hour fast.

Treatment B: Naloxone Nasal Spray

Intervention Type DRUG

Participants received naloxone nasal spray following a 10 hour fast.

Treatment C: Naloxone HCl Intravenous (IV) Injection

Intervention Type DRUG

Participants received naloxone HCl IV injection following a 10 hour fast.

Treatment D: Naloxone HCl Intramuscular (IM) Injection

Intervention Type DRUG

Participants received naloxone HCl IM injection following a 10 hour fast.

Cohort 3: Treatment Sequence C-A-B-D

Participants received Treatment C on Day 1 of Period 1, Treatment A on Day 1 of Period 2, Treatment B on Day 1 of Period 3 and Treatment D on Day 1 of Period 4.

Group Type EXPERIMENTAL

Treatment A: Naloxone Nasal Spray

Intervention Type DRUG

Participants received naloxone nasal spray following a 10 hour fast.

Treatment B: Naloxone Nasal Spray

Intervention Type DRUG

Participants received naloxone nasal spray following a 10 hour fast.

Treatment C: Naloxone HCl Intravenous (IV) Injection

Intervention Type DRUG

Participants received naloxone HCl IV injection following a 10 hour fast.

Treatment D: Naloxone HCl Intramuscular (IM) Injection

Intervention Type DRUG

Participants received naloxone HCl IM injection following a 10 hour fast.

Cohort 4: Treatment Sequence D-B-A-C

Participants received Treatment D on Day 1 of Period 1, Treatment B on Day 1 of Period 2, Treatment A on Day 1 of Period 3 and Treatment C on Day 1 of Period 4.

Group Type EXPERIMENTAL

Treatment A: Naloxone Nasal Spray

Intervention Type DRUG

Participants received naloxone nasal spray following a 10 hour fast.

Treatment B: Naloxone Nasal Spray

Intervention Type DRUG

Participants received naloxone nasal spray following a 10 hour fast.

Treatment C: Naloxone HCl Intravenous (IV) Injection

Intervention Type DRUG

Participants received naloxone HCl IV injection following a 10 hour fast.

Treatment D: Naloxone HCl Intramuscular (IM) Injection

Intervention Type DRUG

Participants received naloxone HCl IM injection following a 10 hour fast.

Interventions

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Treatment A: Naloxone Nasal Spray

Participants received naloxone nasal spray following a 10 hour fast.

Intervention Type DRUG

Treatment B: Naloxone Nasal Spray

Participants received naloxone nasal spray following a 10 hour fast.

Intervention Type DRUG

Treatment C: Naloxone HCl Intravenous (IV) Injection

Participants received naloxone HCl IV injection following a 10 hour fast.

Intervention Type DRUG

Treatment D: Naloxone HCl Intramuscular (IM) Injection

Participants received naloxone HCl IM injection following a 10 hour fast.

Intervention Type DRUG

Eligibility Criteria

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Inclusion Criteria

* A minimum body weight of 50 kg. Body mass index (BMI) between 18.0 and 32.0 kg/m2
* A seated blood pressure between 90 and 140 mmHg systolic/50 and 90 mmHg diastolic
* Female subjects had a negative serum β human chorionic gonadotropin (β-hCG) pregnancy test at screening

Exclusion Criteria

* A known allergy or history of significant adverse reaction to naloxone, other opioids or related compounds, or to any of the excipients
* Any documented clinically significant infection, injury, or illness within 1 month prior to screening
* An active malignancy of any type, or had been diagnosed with cancer within 5 years prior to screening
* A documented history of alcohol or drug abuse/dependence/misuse or narcotic analgesic abuse/dependence/misuse within 2 years prior to screening
* A positive urine test result for alcohol, drugs, or cotinine at screening or check-in
* A condition that the investigator believed would have interfered with the ability to provide informed consent or comply with study instructions, or that could confound the interpretation of the study results or put the subject at undue risk
* Used any opioids for 30 days prior to Day 1
* Required treatment with monoamine oxidase inhibitors (MAOIs) within 30 days prior to Day 1 and during the study.
* Presence of an ongoing upper respiratory infection, rhinitis, rhinorrhea, or nasal congestions
Minimum Eligible Age

18 Years

Maximum Eligible Age

45 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

Yes

Sponsors

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INSYS Therapeutics Inc

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Principal Investigators

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Giovanni DeCastro

Role: STUDY_DIRECTOR

INSYS Therapeutics Inc

Locations

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Worldwide Clinical Trials

San Antonio, Texas, United States

Site Status

Countries

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United States

Other Identifiers

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INS012-18-119

Identifier Type: -

Identifier Source: org_study_id

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