Exploratory Bioavailability of Fentanyl Sublingual Spray Under Fasting Conditions

NCT ID: NCT02138396

Last Updated: 2014-12-12

Study Results

Results pending

The study team has not published outcome measurements, participant flow, or safety data for this trial yet. Check back later for updates.

Basic Information

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Recruitment Status

COMPLETED

Clinical Phase

NA

Total Enrollment

12 participants

Study Classification

INTERVENTIONAL

Study Start Date

2014-01-31

Study Completion Date

2014-01-31

Brief Summary

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The objective of this study is to compare the rate of absorption and bioavailability of fentanyl sublingual spray 400 mcg to fentanyl citrate 100 mcg by intramuscular injection.

Detailed Description

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Conditions

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Bioavailability

Study Design

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Allocation Method

RANDOMIZED

Intervention Model

CROSSOVER

Primary Study Purpose

BASIC_SCIENCE

Blinding Strategy

NONE

Study Groups

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FSS first, then FCI

At each of two treatment visits participants fast for 10 hours before dosing, and receive naltrexone before and after dosing. Participants in this group receive a single dose of fentanyl sublingual spray (FSS) at the first visit. After a washout period of at least seven days, they receive a single intramuscular fentanyl citrate injection (FCI) at the second treatment visit.

Group Type EXPERIMENTAL

Fentanyl Sublingual Spray (FSS)

Intervention Type DRUG

A single dose of fentanyl, 400 mcg per sublingual spray

Fentanyl Citrate Injection (FCI)

Intervention Type DRUG

A single dose of fentanyl citrate, 100 mcg per intramuscular injection

Naltrexone

Intervention Type DRUG

Naltrexone is provided as a 50 mg tablet before and after product dosing to minimize unacceptable adverse effects of fentanyl.

FCI first, then FSS

At each of two treatment visits participants fast for 10 hours before dosing, and receive naltrexone before and after dosing. Participants in this group receive a single intramuscular fentanyl citrate injection (FCI) at the first visit. After a washout period of at least seven days, they receive a single dose of fentanyl sublingual spray (FSS) at the second treatment visit.

Group Type EXPERIMENTAL

Fentanyl Sublingual Spray (FSS)

Intervention Type DRUG

A single dose of fentanyl, 400 mcg per sublingual spray

Fentanyl Citrate Injection (FCI)

Intervention Type DRUG

A single dose of fentanyl citrate, 100 mcg per intramuscular injection

Naltrexone

Intervention Type DRUG

Naltrexone is provided as a 50 mg tablet before and after product dosing to minimize unacceptable adverse effects of fentanyl.

Interventions

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Fentanyl Sublingual Spray (FSS)

A single dose of fentanyl, 400 mcg per sublingual spray

Intervention Type DRUG

Fentanyl Citrate Injection (FCI)

A single dose of fentanyl citrate, 100 mcg per intramuscular injection

Intervention Type DRUG

Naltrexone

Naltrexone is provided as a 50 mg tablet before and after product dosing to minimize unacceptable adverse effects of fentanyl.

Intervention Type DRUG

Other Intervention Names

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Subsys®

Eligibility Criteria

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Inclusion Criteria

* Meets protocol-specified criteria for qualification and contraception
* Good access to veins on both sides
* Willing and able to remain confined in the study unit for the entire duration of each treatment period and comply with restrictions related food, drink and medications
* Voluntarily consents to participate and provides written informed consent prior to any protocol-specific procedures

Exclusion Criteria

* Intolerance to venipuncture or injections
* Presence or history of oral disease, irritation or piercings
* Allergy or adverse response to fentanyl, naltrexone, or related drugs
* Tattoos, scarring, or other skin abnormality at planned injection sites
* History or current use of over-the-counter medications, dietary supplements, or drugs (including nicotine and alcohol) outside protocol-specified parameters
* Signs, symptoms or history of any condition that, per protocol or in the opinion of the investigator, might compromise: 1) the safety or well-being of the participant or study staff; 2) the safety or well-being of the participant's offspring (such as through pregnancy or breast-feeding); 3) the analysis of results
Minimum Eligible Age

18 Years

Maximum Eligible Age

55 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

Yes

Sponsors

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INSYS Therapeutics Inc

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Principal Investigators

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George J Atiee, MD

Role: PRINCIPAL_INVESTIGATOR

Worldwide Clinical Trials Early Phase Services, LLC

Locations

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Worldwide Clinical Trials Early Phase Services, LLC

San Antonio, Texas, United States

Site Status

Countries

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United States

Other Identifiers

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INS-13-019

Identifier Type: -

Identifier Source: org_study_id