A Study to Assess Efficacy and Safety of GLPG1972/S201086 in Participants With Knee Osteoarthritis

NCT ID: NCT03595618

Last Updated: 2021-07-28

Study Results

Results available

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Basic Information

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Recruitment Status

COMPLETED

Clinical Phase

PHASE2

Total Enrollment

932 participants

Study Classification

INTERVENTIONAL

Study Start Date

2018-08-14

Study Completion Date

2020-07-14

Brief Summary

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This study is a phase 2, 52-week international, multi-regional, multi-center, randomized, double-blind, placebo-controlled dose-ranging study for the treatment of osteoarthritis.

Detailed Description

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Conditions

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Osteoarthritis

Study Design

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Allocation Method

RANDOMIZED

Intervention Model

PARALLEL

Primary Study Purpose

TREATMENT

Blinding Strategy

QUADRUPLE

Participants Caregivers Investigators Outcome Assessors

Study Groups

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GLPG1972 75 mg

Participants received 1 film-coated tablet of GLPG1972 75 mg and 3 GLPG1972 matching placebo tablets, orally once daily for 52 weeks.

Group Type EXPERIMENTAL

GLPG1972

Intervention Type DRUG

Film-coated tablets of GLPG1972 for oral use.

Placebo

Intervention Type DRUG

Film-coated tablets of matching placebo for oral use.

GLPG1972 150 mg

Participants received 2 film-coated tablets of GLPG1972 75 mg (total dose 150 mg) and 2 GLPG1972 matching placebo tablets, orally once daily for 52 weeks.

Group Type EXPERIMENTAL

GLPG1972

Intervention Type DRUG

Film-coated tablets of GLPG1972 for oral use.

Placebo

Intervention Type DRUG

Film-coated tablets of matching placebo for oral use.

GLPG1972 300 mg

Participants received 4 film-coated tablets of GLPG1972 75 mg (total dose 300 mg), orally once daily for 52 weeks.

Group Type EXPERIMENTAL

GLPG1972

Intervention Type DRUG

Film-coated tablets of GLPG1972 for oral use.

Placebo

Participants received 4 film-coated tablets of GLPG1972 matching placebo, orally once daily for 52 weeks.

Group Type PLACEBO_COMPARATOR

Placebo

Intervention Type DRUG

Film-coated tablets of matching placebo for oral use.

Interventions

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GLPG1972

Film-coated tablets of GLPG1972 for oral use.

Intervention Type DRUG

Placebo

Film-coated tablets of matching placebo for oral use.

Intervention Type DRUG

Eligibility Criteria

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Inclusion Criteria

* Male participants or female participants of non-childbearing potential and not breastfeeding.
* Body weight \> 40 kg, body mass index (BMI) \< 40 kg/m\^2.
* Diagnosed for knee osteoarthritis based on clinical and radiological criteria of the American College of Rheumatology.
* History of knee pain for at least 6 months and on the majority of days (\> 50%) during the preceding month.
* Symptom severity defined by a pain ≥ 40 mm and ≤ 90 mm on visual analogue scale (VAS, 100 mm) at screening and inclusion visits.
* Documented need for symptomatic as needed-treatment for osteoarthritis (OA) in the target knee with systemic non-steroidal anti-inflammatory drugs (NSAIDs) and/or other analgesics

Exclusion Criteria

* Severe clinical knee malalignment according to the investigator.
* Knee prosthesis already implanted (\< 1 year) or not well-tolerated (contralateral side).
* Knee prosthesis already foreseen within the study period (whichever side).
* Hip prosthesis recently implanted (\< 1 year) or foreseen within the study period (whichever side).
* Previous osteotomy on the inferior limbs (whichever side).
* Surgical operation on the target knee within the 12 months prior to the screening visit or planned during the study.
* Diagnostic arthroscopy of the target knee within the 6 months prior to the screening visit or planned during the study.
* Other pathologies affecting the target knee.
* Any contraindication to magnetic resonance imaging (MRI) including the inability to undergo a knee MRI exam because of inability to fit in the scanner or knee coil.
Minimum Eligible Age

40 Years

Maximum Eligible Age

75 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

No

Sponsors

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Institut de Recherches Internationales Servier

OTHER

Sponsor Role collaborator

Galapagos NV

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Principal Investigators

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Galapagos Study Director

Role: STUDY_DIRECTOR

Galapagos NV

Locations

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Central Research Associates, Inc.

Birmingham, Alabama, United States

Site Status

Achieve Clinical Research, LLC

Birmingham, Alabama, United States

Site Status

Elite Clinical Studies

Phoenix, Arizona, United States

Site Status

Hope Research Institute, LLC - Arizona

Phoenix, Arizona, United States

Site Status

Arizona Research Center

Phoenix, Arizona, United States

Site Status

Clinical Research Consortium Arizona

Tempe, Arizona, United States

Site Status

Samy Metyas MD, Inc - Covina Arthritis Clinic

Covina, California, United States

Site Status

TriWest Research Associates, LLC

El Cajon, California, United States

Site Status

BioSolutions Clinical Research Center

La Mesa, California, United States

Site Status

The Helm Center for Pain Management

Laguna Hills, California, United States

Site Status

Stanford University

Palo Alto, California, United States

Site Status

Artemis Institute for Clinical Research - San Diego

San Diego, California, United States

Site Status

Artemis Institute for Clinical Research - San Marcos

San Marcos, California, United States

Site Status

Encompass Clinical Research

Spring Valley, California, United States

Site Status

Center for Musculoskeletal Care - Yale Medicine

New Haven, Connecticut, United States

Site Status

Avail Clinical Research, LLC

DeLand, Florida, United States

Site Status

Clinical Physiology Associates Clinical Study Center

Fort Myers, Florida, United States

Site Status

Health Awareness, Inc

Jupiter, Florida, United States

Site Status

Bioclinica Research

Orlando, Florida, United States

Site Status

Stedman Clinical Trials, LLC

Tampa, Florida, United States

Site Status

Compass Research, LLC

The Villages, Florida, United States

Site Status

Injury Care Research, LLC

Boise, Idaho, United States

Site Status

Millennium Pain Center - Bloomington

Bloomington, Illinois, United States

Site Status

Northwestern University

Chicago, Illinois, United States

Site Status

Medisphere Medical Research Center

Evansville, Indiana, United States

Site Status

University of Kansas Medical Center

Kansas City, Kansas, United States

Site Status

Phoenix Medical Reasearch

Prairie Village, Kansas, United States

Site Status

Central Kentucky Research Associates, Inc.

Lexington, Kentucky, United States

Site Status

Medpharmics

Metairie, Louisiana, United States

Site Status

The Center for Rheumatology and Bone Research

Wheaton, Maryland, United States

Site Status

Tufts Medical Center

Boston, Massachusetts, United States

Site Status

Clinical Research Consortium Nevada

Las Vegas, Nevada, United States

Site Status

NY Scientific

Brooklyn, New York, United States

Site Status

Rochester Clinical Research, Inc.

Rochester, New York, United States

Site Status

Upstate Clinical Research Associates

Williamsville, New York, United States

Site Status

Lillestol Research, LCC

Fargo, North Dakota, United States

Site Status

Optimed Research, LTD

Columbus, Ohio, United States

Site Status

Altoona Center for Clinical Research

Duncansville, Pennsylvania, United States

Site Status

Pioneer Research Solutions Inc.

Houston, Texas, United States

Site Status

Diagnostics Research Group

San Antonio, Texas, United States

Site Status

Advanced Clinical Research

West Jordan, Utah, United States

Site Status

Charlottesville Medical Research Center, LCC

Charlottesville, Virginia, United States

Site Status

Health Research of Hampton Roads, Inc. - Newport News

Newport News, Virginia, United States

Site Status

Clinical Research Associates of Tidewater

Norfolk, Virginia, United States

Site Status

Countries

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United States

References

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Chen L, Huang FL, Tang Q, Zhao ZK, Ye ZY, Liang JH. Targeted therapy for knee osteoarthritis: From basic to clinics. Medicine (Baltimore). 2025 Aug 15;104(33):e43686. doi: 10.1097/MD.0000000000043686.

Reference Type DERIVED
PMID: 40826764 (View on PubMed)

Schnitzer T, Pueyo M, Deckx H, van der Aar E, Bernard K, Hatch S, van der Stoep M, Grankov S, Phung D, Imbert O, Chimits D, Muller K, Hochberg MC, Bliddal H, Wirth W, Eckstein F, Conaghan PG. Evaluation of S201086/GLPG1972, an ADAMTS-5 inhibitor, for the treatment of knee osteoarthritis in ROCCELLA: a phase 2 randomized clinical trial. Osteoarthritis Cartilage. 2023 Jul;31(7):985-994. doi: 10.1016/j.joca.2023.04.001. Epub 2023 Apr 13.

Reference Type DERIVED
PMID: 37059327 (View on PubMed)

Brebion F, Gosmini R, Deprez P, Varin M, Peixoto C, Alvey L, Jary H, Bienvenu N, Triballeau N, Blanque R, Cottereaux C, Christophe T, Vandervoort N, Mollat P, Touitou R, Leonard P, De Ceuninck F, Botez I, Monjardet A, van der Aar E, Amantini D. Discovery of GLPG1972/S201086, a Potent, Selective, and Orally Bioavailable ADAMTS-5 Inhibitor for the Treatment of Osteoarthritis. J Med Chem. 2021 Mar 25;64(6):2937-2952. doi: 10.1021/acs.jmedchem.0c02008. Epub 2021 Mar 15.

Reference Type DERIVED
PMID: 33719441 (View on PubMed)

Provided Documents

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Document Type: Study Protocol

View Document

Document Type: Statistical Analysis Plan

View Document

Other Identifiers

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2017-004581-10

Identifier Type: EUDRACT_NUMBER

Identifier Source: secondary_id

U1111-1205-0321

Identifier Type: OTHER

Identifier Source: secondary_id

GLPG1972-CL-201

Identifier Type: -

Identifier Source: org_study_id

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