Study to Evaluate the Safety, Tolerate, Pharmacokinetics and Preliminary Efficacy of CYH33

NCT ID: NCT03544905

Last Updated: 2025-04-22

Study Results

Results pending

The study team has not published outcome measurements, participant flow, or safety data for this trial yet. Check back later for updates.

Basic Information

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Recruitment Status

COMPLETED

Clinical Phase

PHASE1

Total Enrollment

206 participants

Study Classification

INTERVENTIONAL

Study Start Date

2018-07-05

Study Completion Date

2024-12-04

Brief Summary

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This study is a Multi-center, Open-label, single arm, Dose Escalation and Dose Extension Phase 1 Study to Evaluate the Safety , Tolerability, Pharmacokinetics and Preliminary Efficacy of CYH33 in Advanced Solid Tumors Patients.

Detailed Description

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This study includes Phase Ia and Phase Ib.

In the dose climbing part of phase Ia, the safety, tolerance and pharmacokinetics characteristics of CYH33 in patients with advanced solid tumors who failed to receive standard treatment, did not tolerate or did not have standard treatment at present will be observed to determine MTD; Before determining MTD, select safe and highly reliable and effective dose levels for simultaneous expansion. Phase Ia dose expansion includes patients with advanced solid tumors who have failed to undergo standard treatment, who are intolerant of PIK3CA gene mutation, or who do not have standard treatment at present, to further evaluate safety, tolerance and initial efficacy.

In Phase Ib, the safety and preliminary efficacy of CYH33 on patients with advanced breast cancer, ovarian cancer, endometrial cancer, cervical cancer, head and neck squamous cell carcinoma, esophageal and gastroesophageal junction squamous cell carcinoma, ovarian clear cell carcinoma and other solid tumors with PIK3CA gene mutation who have failed, are intolerant or do not have standard treatment at present will be evaluated.

Conditions

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Advanced Solid Tumors

Study Design

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Allocation Method

NA

Intervention Model

SINGLE_GROUP

Primary Study Purpose

TREATMENT

Blinding Strategy

NONE

Study Groups

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Dose escalation study of CYH33

To determine the maximum tolerated dose (MTD) of CYH33

Group Type EXPERIMENTAL

CYH33 for tablet

Intervention Type DRUG

1mg; 5mg; 10mg; 20mg; 30mg; 50mg; 75mg; 100mg; 130mg; 160mg; 200mg; 240mgBID or QD(Decided by SMC accroding to the safty and PK data)

Interventions

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CYH33 for tablet

1mg; 5mg; 10mg; 20mg; 30mg; 50mg; 75mg; 100mg; 130mg; 160mg; 200mg; 240mgBID or QD(Decided by SMC accroding to the safty and PK data)

Intervention Type DRUG

Eligibility Criteria

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Inclusion Criteria

* main inclusion:

1. Evidence of a personally signed informed consent document;
2. Male and/or female subjects above the ages of 18 years;
3. Locally advanced or metastatic solid tumor patients who have failed or relapsed on current standard of care for Phase 1a;
4. Subject may provide Tumor tissue section(at least 8 pieces) if they agree;
5. ECOG performance score 0-1;
6. Life expectancy ≥ 12 weeks;
7. At least 1 measurable target lesion on the baseline scan as per RECIST 1.1

Exclusion Criteria

* main criteria:

1. prior received anti-tumor treatment, including anticancer drugs for the treatment within 28 days of first dose of study treatment;
2. Prior or concomitant other malignant tumor;
Minimum Eligible Age

18 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

No

Sponsors

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Haihe Biopharma Co., Ltd.

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Principal Investigators

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Ruihua Xu, M.D

Role: PRINCIPAL_INVESTIGATOR

Sun Yat-sen University

Locations

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Anhui Provincial Hospital

Hefei, Anhui, China

Site Status

Lu'an People's Hospital

Lu'an, Anhui, China

Site Status

Lu'an Hospital of Traditional Chinese Medicine

Lu'an, Anhui, China

Site Status

Beijing Cancer Hospital

Beijing, Beijing Municipality, China

Site Status

Chongqing Cancer Hospital

Chongqing, Chongqing Municipality, China

Site Status

Xiang'an Hospital of Xiamen University

Xiamen, Fujian, China

Site Status

Dongguan People's Hospital

Dongguan, Guangdong, China

Site Status

The First Affiliated Hospital, Sun Yat-sen University

Guangzhou, Guangdong, China

Site Status

Sun Yat-sen Memorial Hospital, Sun Yat-sen University

Guangzhou, Guangdong, China

Site Status

Sun Yat-sen University Cancer Center

Guangzhou, Guangdong, China

Site Status

Yuebei People's Hospital

Shaoguan, Guangdong, China

Site Status

Shenzhen Hospital of Cancer Hospital, Chinese Academy of Medical Sciences

Shenzhen, Guangdong, China

Site Status

Liuzhou Workers Hospital

Liuzhou, Guangxi, China

Site Status

Affiliated Tumor Hospital of Guangxi Medical University

Nanning, Guangxi, China

Site Status

Harbin Medical University Cancer Hospital

Harbin, Heilongjiang, China

Site Status

Anyang Cancer Hospital

Anyang, Henan, China

Site Status

Nanyang First People's Hospital

Nanyang, Henan, China

Site Status

The First Affiliated Hospital of Nanyang Medical College

Nanyang, Henan, China

Site Status

Henan Cancer Hospital

Zhengzhou, Henan, China

Site Status

Zhongnan Hospital of Wuhan University

Wuhan, Hubei, China

Site Status

Hunan Cancer Hospital

Changsha, Hunan, China

Site Status

Hunan Province Directly Affiliated Traditional Chinese Medicine Hospital

Zhuzhou, Hunan, China

Site Status

Liaoning Cancer Hospital

Shenyang, Liaoning, China

Site Status

Qilu Hospital of Shandong University

Jinan, Shandong, China

Site Status

Zhongshan Hospital Fudan University

Shanghai, Shanghai Municipality, China

Site Status

Obstetrics and Gynecology Hospital of Fudan University

Shanghai, Shanghai Municipality, China

Site Status

Tianjin Medical University Cancer Institute & Hospital

Tianjin, Tianjin Municipality, China

Site Status

The First Affiliated Hospital of Dali University

Dali, Yunnan, China

Site Status

The First Affiliated Hospital, Zhejiang University School of Medicine

Hangzhou, Zhejiang, China

Site Status

Zhejiang Cancer Hospital

Hangzhou, Zhejiang, China

Site Status

Countries

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China

Other Identifiers

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CYH33-101

Identifier Type: -

Identifier Source: org_study_id

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