A Study of Molidustat for Correction of Renal Anemia in Non-dialysis Subjects

NCT ID: NCT03350321

Last Updated: 2021-01-29

Study Results

Results pending

The study team has not published outcome measurements, participant flow, or safety data for this trial yet. Check back later for updates.

Basic Information

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Recruitment Status

COMPLETED

Clinical Phase

PHASE3

Total Enrollment

162 participants

Study Classification

INTERVENTIONAL

Study Start Date

2017-12-12

Study Completion Date

2019-10-11

Brief Summary

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The purpose of this study is to evaluate the efficacy and safety of molidustat in non-dialysis subjects with renal anemia who are not treated with Erythropoiesis-Stimulating Agents (ESAs).

Detailed Description

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Conditions

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Anemia Renal Insufficiency, Chronic

Study Design

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Allocation Method

RANDOMIZED

Intervention Model

PARALLEL

Primary Study Purpose

TREATMENT

Blinding Strategy

NONE

Study Groups

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Molidustat (BAY85-3934)

Molidustat group

Group Type EXPERIMENTAL

Molidustat (BAY85-3934)

Intervention Type DRUG

Starting dose of molidustat once daily (OD) will be titrated based on the subject's Hb (Hemoglobin) response

Darbepoetin alfa

Darbepoetin alfa group

Group Type ACTIVE_COMPARATOR

Darbepoetin alfa

Intervention Type DRUG

Starting dose of darbepoetin alfa once every 2 weeks will be titrated based on the subject's Hb (Hemoglobin) response

Interventions

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Molidustat (BAY85-3934)

Starting dose of molidustat once daily (OD) will be titrated based on the subject's Hb (Hemoglobin) response

Intervention Type DRUG

Darbepoetin alfa

Starting dose of darbepoetin alfa once every 2 weeks will be titrated based on the subject's Hb (Hemoglobin) response

Intervention Type DRUG

Eligibility Criteria

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Inclusion Criteria

* Subjects with estimated glomerular filtration rate (eGFR)\< 60 mL/min/1.73m\^2 (Chronic kidney disease \[CKD\] stages 3 to 5)
* Body weight \> 40 and ≤ 160 kg at screening
* Male or female subject ≥ 20 years of age at screening
* Not on dialysis and not expected to start dialysis during the study period
* Not treated with ESAs and/or HIF-PH inhibitors within 8 weeks prior to randomization
* Mean of the last 2 central laboratory Hb levels during the screening period must be ≥ 8.0 and \< 11.0 g/dL (2 measurements must be taken ≥ 2 days apart and the difference between the 2 measurements must be \< 1.2 g/dL) and the last measurements must be taken within 14 days prior to randomization
* Ferritin ≥ 50 ng/mL at screening

Exclusion Criteria

* New York Heart Association (NYHA) Class III or IV congestive heart failure
* History of cardio- (cerebro-) vascular events (e.g., unstable angina, myocardial infarction, stroke, pulmonary thromboembolism, and acute limb ischemia) within 6 months prior to randomization
* Sustained and poorly controlled arterial hypertension (defined as systolic BP≥ 180mmHg or diastolic BP ≥ 110mmHg) or hypotension (defined as systolic BP \< 90mmHg) at randomization
* Proliferative choroidal or retinal disease, such as neovascular age-related macular degeneration or proliferative diabetic retinopathy requiring invasive treatment (e.g., intraocular injections or laser photocoagulation)
Minimum Eligible Age

20 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

No

Sponsors

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Bayer

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Locations

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Kainan Hospital

Yatomi, Aichi-ken, Japan

Site Status

Seikeikai New Tokyo Heart Clinic

Matsudo, Chiba, Japan

Site Status

Ehime Prefectural Central Hospital

Matsuyama, Ehime, Japan

Site Status

Saiseikai Matsuyama Hospital

Matsuyama, Ehime, Japan

Site Status

Iizuka Hospital

Iizuka, Fukuoka, Japan

Site Status

Kokura Memorial Hospital

Kitakyushu, Fukuoka, Japan

Site Status

Steel Memorial Yawata Hospital

Kitakyushu, Fukuoka, Japan

Site Status

National Fukuoka-Higashi Medical Center

Koga, Fukuoka, Japan

Site Status

Kurume University Hospital

Kurume, Fukuoka, Japan

Site Status

St.Mary's Hospital

Kurume, Fukuoka, Japan

Site Status

Matsunami Health Promotion Clinic

Hashima-gun, Gifu, Japan

Site Status

Gifu Prefectural Tajimi Hospital

Tajimi, Gifu, Japan

Site Status

Mazda Hospital of Mazda Motor Corporation

Aki-gun, Hiroshima, Japan

Site Status

Nippon Kokan Fukuyama Hospital

Fukuyama, Hiroshima, Japan

Site Status

Teine Keijinkai Clinic

Sapporo, Hokkaido, Japan

Site Status

Kobe City Medical Center General Hospital

Kobe, Hyōgo, Japan

Site Status

National Hospital Organization Kobe Medical Center

Kobe, Hyōgo, Japan

Site Status

National hospital Organization Mito Medical Center

Higashiibaraki, Ibaraki, Japan

Site Status

Mito Kyodo General Hospital

Mito, Ibaraki, Japan

Site Status

KenAiKai medical corporation Akiyama clinic

Takamatsu, Kagawa-ken, Japan

Site Status

Ikeda Hospital

Kanoya, Kagoshima-ken, Japan

Site Status

Fujisawa City Hospital

Fujisawa, Kanagawa, Japan

Site Status

Koukan Clinic

Kawasaki, Kanagawa, Japan

Site Status

Showa University Fujigaoka Hospital

Yokohama, Kanagawa, Japan

Site Status

Yokosuka Kyosai Hospital

Yokosuka, Kanagawa, Japan

Site Status

Arao Municipal Hospital

Arao, Kumamoto, Japan

Site Status

Kumamoto Rosai Hospital

Yatsushiro, Kumamoto, Japan

Site Status

Uji-Tokushukai Medical Center

Uji, Kyoto, Japan

Site Status

JCHO Yokkaichi Hazu Medical Center

Yokkaichi, Mie-ken, Japan

Site Status

Japanese Red Cross Ishinomaki Hospital

Ishinomaki, Miyagi, Japan

Site Status

Asama Nanroku Komoro Medical Center

Komoro, Nagano, Japan

Site Status

Niigata Prefectural Shibata Hospital

Shibata, Niigata, Japan

Site Status

Okinawa prefectural Chubu Hospital

Uruma, Okinawa, Japan

Site Status

Osaka Saiseikai Senri Hospital

Suita, Osaka, Japan

Site Status

Osaka Pref. Saiseikai Tondabayashi Hospital

Tondabayashi, Osaka, Japan

Site Status

Kitasato University Medical Center

Kitamoto, Saitama, Japan

Site Status

Iwata City Hospital

Iwata, Shizuoka, Japan

Site Status

Toshima Hospital

Itabashi-ku, Tokyo, Japan

Site Status

Nihon University Itabashi Hospital

Itabashi-ku, Tokyo, Japan

Site Status

Showa University Koto Toyosu Hospital

Koto-ku, Tokyo, Japan

Site Status

National Hospital Organization Tokyo Medical Center

Meguro-ku, Tokyo, Japan

Site Status

University of Yamanashi Hospital

Chūō, Yamanashi, Japan

Site Status

Fukui Prefectural Hospital

Fukui, , Japan

Site Status

National Hospital Organization Kyushu Medical Center

Fukuoka, , Japan

Site Status

Kyushu University Hospital

Fukuoka, , Japan

Site Status

Fukuoka University Hospital

Fukuoka, , Japan

Site Status

Fukushima Medical University Hospital

Fukushima, , Japan

Site Status

Asahi University Hospital

Gifu, , Japan

Site Status

National Hospital Organization Kochi National Hospital

Kochi, , Japan

Site Status

Nara Prefecture General Medical Center

Nara, , Japan

Site Status

Kitano Hospital

Osaka, , Japan

Site Status

National Hospital Organization Osaka National Hospital

Osaka, , Japan

Site Status

Osaka Red Cross Hospital

Osaka, , Japan

Site Status

Nippon Life Hospital

Osaka, , Japan

Site Status

Chibune Clinic

Osaka, , Japan

Site Status

Osaka General Medical Center

Osaka, , Japan

Site Status

Social Corporation Keigakukai Minamiosaka Hospital

Osaka, , Japan

Site Status

Japanese Red Cross Oita Hospital

Ōita, , Japan

Site Status

Shizuoka Saiseikai General Hospital

Shizuoka, , Japan

Site Status

Suruga Clinic

Shizuoka, , Japan

Site Status

Wakayama Medical University Hospital

Wakayama, , Japan

Site Status

Countries

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Japan

References

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Yamamoto H, Yamada T, Miyazaki K, Yamashita T, Kato T, Ohara K, Nakamura Y, Akizawa T. Treatment satisfaction with molidustat in CKD-related anemia in non-dialysis patients: a post-hoc analysis of two clinical trials. Clin Exp Nephrol. 2023 Aug;27(8):651-659. doi: 10.1007/s10157-023-02353-x. Epub 2023 Apr 24.

Reference Type DERIVED
PMID: 37095342 (View on PubMed)

Natale P, Palmer SC, Jaure A, Hodson EM, Ruospo M, Cooper TE, Hahn D, Saglimbene VM, Craig JC, Strippoli GF. Hypoxia-inducible factor stabilisers for the anaemia of chronic kidney disease. Cochrane Database Syst Rev. 2022 Aug 25;8(8):CD013751. doi: 10.1002/14651858.CD013751.pub2.

Reference Type DERIVED
PMID: 36005278 (View on PubMed)

Yamamoto H, Taguchi M, Matsuda Y, Iekushi K, Yamada T, Akizawa T. Molidustat for the treatment of renal anaemia in patients with non-dialysis-dependent chronic kidney disease: design and rationale of two phase III studies. BMJ Open. 2019 Jun 14;9(6):e026704. doi: 10.1136/bmjopen-2018-026704.

Reference Type DERIVED
PMID: 31203242 (View on PubMed)

Related Links

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http://clinicaltrials.bayer.com/

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Other Identifiers

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19349

Identifier Type: -

Identifier Source: org_study_id

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