A Phase 1/2 Study of INCB001158 in Combination With Chemotherapy in Subjects With Solid Tumors

NCT ID: NCT03314935

Last Updated: 2025-08-12

Study Results

Results available

Outcome measurements, participant flow, baseline characteristics, and adverse events have been published for this study.

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Basic Information

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Recruitment Status

COMPLETED

Clinical Phase

PHASE1/PHASE2

Total Enrollment

149 participants

Study Classification

INTERVENTIONAL

Study Start Date

2017-11-21

Study Completion Date

2022-11-28

Brief Summary

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The purpose of this open-label nonrandomized Phase 1/2 study is to evaluate INCB001158 in combination with chemotherapy in participants with advanced/metastatic solid tumors.

Detailed Description

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Conditions

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Biliary Tract Cancer (BTC) Colorectal Cancer (CRC) Endometrial Cancer Gastroesophageal Cancer (GC) Ovarian Cancer Solid Tumors

Study Design

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Allocation Method

NON_RANDOMIZED

Intervention Model

SINGLE_GROUP

Primary Study Purpose

TREATMENT

Blinding Strategy

NONE

Study Groups

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Treatment Group A

INCB001158 + FOLFOX

Group Type EXPERIMENTAL

INCB001158

Intervention Type DRUG

Phase 1: INCB001158 administered orally twice daily at the protocol-defined dose. Phase 2: INCB001158 administered orally twice daily at the recommended dose from Phase 1.

Oxaliplatin

Intervention Type DRUG

Oxaliplatin administered intravenously at the protocol-defined dose and schedule.

Leucovorin

Intervention Type DRUG

Leucovorin at the protocol-defined dose and regimen.

5-Fluorouracil

Intervention Type DRUG

5-Fluorouracil at the protocol-defined dose and regimen.

Treatment Group B

INCB001158 + gemcitabine/cisplatin

Group Type EXPERIMENTAL

INCB001158

Intervention Type DRUG

Phase 1: INCB001158 administered orally twice daily at the protocol-defined dose. Phase 2: INCB001158 administered orally twice daily at the recommended dose from Phase 1.

Gemcitabine

Intervention Type DRUG

Gemcitabine at the protocol-defined dose and regimen.

Cisplatin

Intervention Type DRUG

Cisplatin at the protocol-defined dose and regimen.

Treatment Group C

INCB001158 + paclitaxel

Group Type EXPERIMENTAL

INCB001158

Intervention Type DRUG

Phase 1: INCB001158 administered orally twice daily at the protocol-defined dose. Phase 2: INCB001158 administered orally twice daily at the recommended dose from Phase 1.

Paclitaxel

Intervention Type DRUG

Paclitaxel at the protocol-defined dose and regimen.

Interventions

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INCB001158

Phase 1: INCB001158 administered orally twice daily at the protocol-defined dose. Phase 2: INCB001158 administered orally twice daily at the recommended dose from Phase 1.

Intervention Type DRUG

Oxaliplatin

Oxaliplatin administered intravenously at the protocol-defined dose and schedule.

Intervention Type DRUG

Leucovorin

Leucovorin at the protocol-defined dose and regimen.

Intervention Type DRUG

5-Fluorouracil

5-Fluorouracil at the protocol-defined dose and regimen.

Intervention Type DRUG

Gemcitabine

Gemcitabine at the protocol-defined dose and regimen.

Intervention Type DRUG

Cisplatin

Cisplatin at the protocol-defined dose and regimen.

Intervention Type DRUG

Paclitaxel

Paclitaxel at the protocol-defined dose and regimen.

Intervention Type DRUG

Other Intervention Names

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Arginase inhibitor

Eligibility Criteria

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Inclusion Criteria

* Histologically or cytologically confirmed diagnosis of selected advanced or metastatic solid tumors.
* Presence of measurable disease per RECIST v1.1.
* Eastern Cooperative Oncology Group (ECOG) performance status of 0 or 1.
* Baseline archival tumor specimen available or willingness to undergo a pretreatment tumor biopsy to obtain the specimen.
* Resolution of treatment-related toxicities.
* Adequate hepatic, renal, cardiac, and hematologic function.
* Additional cohort-specific criteria may apply.

Exclusion Criteria

* Subjects who participated in any other study in which receipt of an investigational study drug or device occurred within 28 days or 5 half-lives (whichever is longer) prior to first dose.
* Has received a prior monoclonal antibody within 4 weeks or 5 half-lives (whichever is shorter) before administration of study drug.
* Has had prior chemotherapy or targeted small molecule therapy within 2 weeks before administration of study treatment.
* Has received prior approved radiotherapy within 14 days of study therapy.
* Has had known additional malignancy that is progressing or requires active treatment, or history of other malignancy within 2 years of study entry.
* Has an active autoimmune disease that has required systemic treatment in past 2 years.
* Has an active infection requiring systemic therapy.
* Has known active CNS metastases and/or carcinomatous meningitis.
* Women who are pregnant or breastfeeding.
Minimum Eligible Age

18 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

No

Sponsors

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Incyte Corporation

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Principal Investigators

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Lance Leopold, MD

Role: STUDY_DIRECTOR

Incyte Corporation

Locations

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University of Alabama

Birmingham, Alabama, United States

Site Status

USA Mitchell Cancer Center

Mobile, Alabama, United States

Site Status

UC Davis - Comprehensive Cancer Centre

Sacramento, California, United States

Site Status

Northwest Georgia Oncology Centers

Marietta, Georgia, United States

Site Status

The University of Texas MD Anderson Cancer Center

Houston, Texas, United States

Site Status

START San Antonio

San Antonio, Texas, United States

Site Status

Grand Hopital de Charleroi - Department of Medical Oncology

Brussels, , Belgium

Site Status

Institut Jules Bordet - Clinical Trials Conduct Unit

Brussels, , Belgium

Site Status

UCL Cancer Institute

London, , United Kingdom

Site Status

The Christie NHS Foundation Trust

Manchester, , United Kingdom

Site Status

Countries

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United States Belgium United Kingdom

References

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Aden D, Sureka N, Zaheer S, Chaurasia JK, Zaheer S. Metabolic Reprogramming in Cancer: Implications for Immunosuppressive Microenvironment. Immunology. 2025 Jan;174(1):30-72. doi: 10.1111/imm.13871. Epub 2024 Oct 27.

Reference Type DERIVED
PMID: 39462179 (View on PubMed)

Provided Documents

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Document Type: Study Protocol

View Document

Document Type: Statistical Analysis Plan

View Document

Other Identifiers

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2017-002904-29

Identifier Type: EUDRACT_NUMBER

Identifier Source: secondary_id

INCB 01158-203

Identifier Type: -

Identifier Source: org_study_id

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