Safety, Tolerability and Pharmacokinetics of ONC1-0013B in Patients With Progressive Metastatic Castration-resistant Prostate Cancer

NCT ID: NCT03074032

Last Updated: 2017-07-11

Study Results

Results pending

The study team has not published outcome measurements, participant flow, or safety data for this trial yet. Check back later for updates.

Basic Information

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Recruitment Status

COMPLETED

Clinical Phase

PHASE1

Total Enrollment

17 participants

Study Classification

INTERVENTIONAL

Study Start Date

2014-06-30

Study Completion Date

2017-04-30

Brief Summary

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This is a PhaseI, open-label study, Dose-Escalation Study, where tolerated doses will be escalated to the next doses with the safety, tolerability, and PK being evaluated in metastatic castration-resistant prostate cancer (mCRPC) patients. Tumor assessment and PSA values will be evaluated during the study as an additional point.

Detailed Description

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Conditions

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Metastatic Castration-Resistant Prostate Cancer (mCRPC)

Study Design

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Allocation Method

NON_RANDOMIZED

Intervention Model

SINGLE_GROUP

Single Group Assignment
Primary Study Purpose

TREATMENT

Blinding Strategy

NONE

Study Groups

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ONC1-0013B 40 mg

ONC1-0013B 40 mg per os daily

Group Type EXPERIMENTAL

ONC1-0013B

Intervention Type DRUG

ONC1-0013B per os daily

ONC1-0013B 80 mg

ONC1-0013B 80 mg per os daily

Group Type EXPERIMENTAL

ONC1-0013B

Intervention Type DRUG

ONC1-0013B per os daily

ONC1-0013B 160 mg

ONC1-0013B 160 mg per os daily

Group Type EXPERIMENTAL

ONC1-0013B

Intervention Type DRUG

ONC1-0013B per os daily

ONC1-0013B 320 mg

ONC1-0013B 320 mg per os daily

Group Type EXPERIMENTAL

ONC1-0013B

Intervention Type DRUG

ONC1-0013B per os daily

Interventions

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ONC1-0013B

ONC1-0013B per os daily

Intervention Type DRUG

Eligibility Criteria

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Inclusion Criteria

1. Men aged 18 years and older.
2. Histologically confirmed diagnosis of prostate cancer
3. Castrate level of testosterone in blood serum \< 1,7 nmol/l or \< 50 ng/dl
4. PSA level at screening \> 2 ng/ml
5. Progression of metastatic CRPC after the chemical castration with gonadotropin-releasing hormone (GnRH) analogue or after the chemical castration and subsequent chemotherapy.
6. The patient's ECOG performance status of 0 - 2
7. Patients previously treated with docetaxel chemotherapy should have received 2 or less prior lines of chemotherapy for mCRPC
8. The expected survival time of not less than 12 weeks

Exclusion Criteria

1. Prior anticancer therapy:

* Treatment with chemotherapeutic agents or radiotherapy within 4 weeks prior to screening or preserved toxicities of ≥ II grade according to CTCAE scale, related to prior anticancer therapy (excluding alopecia)
* Prior antiandrogen therapy: flutamide within 4 weeks prior to screening or bicalutamide within 6 weeks prior to screening
* Exposure to bisphosphonates is allowed only if the treatment started prior to screening
2. Clinically significant cardiovascular system diseases:
3. Clinically significant central nervous system diseases:
4. History of other significant concomitant diseases which, in the Investigator's opinion, may cause a disease recurrence (i.e. uncontrolled diabetes mellitus)
5. Prior or concomitant therapy:

* Exposure to drugs which may cause a convulsive state within 4 weeks prior to screening
* Exposure to treatment with characteristics of CYP3A4 or CYP2D6 inhibitors within 4 weeks prior to screening
* Exposure to treatment relating to the Class I risk of QT-interval prolongation; exposure to treatment relating to the Class II risk of QT-interval prolongation is allowed if the patient have received not less than 5 half-life periods of flat-dosed treatment
Minimum Eligible Age

18 Years

Eligible Sex

MALE

Accepts Healthy Volunteers

No

Sponsors

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Avionco LLC

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Locations

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Research Institute of Urology and Interventional Radiology n.a. N.A. Lopatkin (branch of FSBI NMRRC of the Ministry of Health of the Russian Federation)

Moscow, , Russia

Site Status

Medical Radiological Research Center n.a. A.F. Tsyb (branch of FSBI NMRRC of the Ministry of Health of the Russian Federation)

Obninsk, , Russia

Site Status

Countries

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Russia

Other Identifiers

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ONC-ONC10013B-01

Identifier Type: -

Identifier Source: org_study_id

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