A Study to Assess the Relative Bioavailability And Food Effect of a Tablet Formulation of GDC-0276 in Healthy Participants

NCT ID: NCT02856152

Last Updated: 2018-02-19

Study Results

Results pending

The study team has not published outcome measurements, participant flow, or safety data for this trial yet. Check back later for updates.

Basic Information

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Recruitment Status

WITHDRAWN

Clinical Phase

PHASE1

Study Classification

INTERVENTIONAL

Study Start Date

2016-06-30

Study Completion Date

2016-11-30

Brief Summary

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This open-label, randomized, 4-way crossover study in healthy participants will determine the relative bioavailability of the tablet formulation relative to the capsule formulation and the effect of a high-fat and low-fat meal on the relative bioavailability of the tablet formulation.

Detailed Description

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Conditions

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Healthy Volunteer

Study Design

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Allocation Method

RANDOMIZED

Intervention Model

CROSSOVER

Primary Study Purpose

BASIC_SCIENCE

Blinding Strategy

NONE

Study Groups

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Treatment A Then B Then D Then C

Treatment A: a single dose of three 90-mg capsules of GDC-0276 administered orally after at least an 8-hour fast. Treatment B: a single dose of three 90-mg tablets GDC-0276 administered orally after at least an 8-hour fast. Treatment C: a single dose of three 90-mg tablets of GDC-0276 administered orally within 30 minutes of eating a standardized FDA high-fat meal. Treatment D: a single dose of three 90-mg tablets of GDC-0276 administered orally within 30 minutes of eating a standardized low-fat meal. Participants will receive Treatment A on Day 1 of first intervention period, followed by Treatment B on Day 1 of second intervention period, followed by Treatment D on Day 1 of third intervention period, and then Treatment C on Day 1 of fourth intervention period. A washout period of 6 days will be maintained between each intervention period.

Group Type EXPERIMENTAL

GDC-0276 capsule

Intervention Type DRUG

Three 90 milligram \[mg\] capsules of GDC-0276 administered orally.

GDC-0276 tablets

Intervention Type DRUG

Three 90 mg GDC-0276 tablets administered orally.

Treatment B, Then C, Then A, Then D

Treatment A: a single dose of three 90-mg capsules of GDC-0276 administered orally after at least an 8-hour fast. Treatment B: a single dose of three 90-mg tablets GDC-0276 administered orally after at least an 8-hour fast. Treatment C: a single dose of three 90-mg tablets of GDC-0276 administered orally within 30 minutes of eating a standardized FDA high-fat meal. Treatment D: a single dose of three 90-mg tablets of GDC-0276 administered orally within 30 minutes of eating a standardized low-fat meal. Participants will receive Treatment B on Day 1 of first intervention period, followed by Treatment C on Day 1 of second intervention period, followed by Treatment A on Day 1 of third intervention period, and then Treatment D on Day 1 of fourth intervention period. A washout period of 6 days will be maintained between each intervention period.

Group Type EXPERIMENTAL

GDC-0276 capsule

Intervention Type DRUG

Three 90 milligram \[mg\] capsules of GDC-0276 administered orally.

GDC-0276 tablets

Intervention Type DRUG

Three 90 mg GDC-0276 tablets administered orally.

Treatment C, Then D, Then B, Then A

Treatment A: a single dose of three 90-mg capsules of GDC-0276 administered orally after at least an 8-hour fast. Treatment B: a single dose of three 90-mg tablets GDC-0276 administered orally after at least an 8-hour fast. Treatment C: a single dose of three 90-mg tablets of GDC-0276 administered orally within 30 minutes of eating a standardized FDA high-fat meal. Treatment D: a single dose of three 90-mg tablets of GDC-0276 administered orally within 30 minutes of eating a standardized low-fat meal. Participants will receive Treatment C on Day 1 of first intervention period, followed by Treatment D on Day 1 of second intervention period, followed by Treatment B on Day 1 of third intervention period, and then Treatment A on Day 1 of fourth intervention period. A washout period of 6 days will be maintained between each intervention period.

Group Type EXPERIMENTAL

GDC-0276 capsule

Intervention Type DRUG

Three 90 milligram \[mg\] capsules of GDC-0276 administered orally.

GDC-0276 tablets

Intervention Type DRUG

Three 90 mg GDC-0276 tablets administered orally.

Treatment D, Then A, Then C, Then B

Treatment A: a single dose of three 90-mg capsules of GDC-0276 administered orally after at least an 8-hour fast. Treatment B: a single dose of three 90-mg tablets GDC-0276 administered orally after at least an 8-hour fast. Treatment C: a single dose of three 90-mg tablets of GDC-0276 administered orally within 30 minutes of eating a standardized FDA high-fat meal. Treatment D: a single dose of three 90-mg tablets of GDC-0276 administered orally within 30 minutes of eating a standardized low-fat meal. Participants will receive Treatment D on Day 1 of first intervention period, followed by Treatment A on Day 1 of second intervention period, followed by Treatment C on Day 1 of third intervention period, and then Treatment B on Day 1 of fourth intervention period. A washout period of 6 days will be maintained between each intervention period.

Group Type EXPERIMENTAL

GDC-0276 capsule

Intervention Type DRUG

Three 90 milligram \[mg\] capsules of GDC-0276 administered orally.

GDC-0276 tablets

Intervention Type DRUG

Three 90 mg GDC-0276 tablets administered orally.

Interventions

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GDC-0276 capsule

Three 90 milligram \[mg\] capsules of GDC-0276 administered orally.

Intervention Type DRUG

GDC-0276 tablets

Three 90 mg GDC-0276 tablets administered orally.

Intervention Type DRUG

Eligibility Criteria

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Inclusion Criteria

* Body mass index within the range 18.0 to 32.0 kilograms per meter squared (kg/m\^2), inclusive, and a minimum weight of 50.0 kg
* Male participants of reproductive potential must be and willing to continue using medically acceptable contraception and must avoid sperm donation from screening and for at least 90 days after the last study drug administration

Exclusion Criteria

* Self-reported substance or alcohol dependence (excluding nicotine and caffeine) within the past 2 years, and/or participants who have ever been in a substance or alcohol rehabilitation program to treat their substance or alcohol dependence
* Have used any prescription or over-the-counter (OTC) medication or supplement within 14 days or 5 times the elimination half-life (whichever is longer) before Day -1 until the end of their participation in the study
* Have used any vaccine within 7 days before GDC-0276 administration
* Female participants with a positive serum or urine pregnancy test or are breast feeding
* Donation or loss of more than 500 milliliter (mL) whole blood within 3 months preceding entry into the treatment period
* Blood transfusion within 30 days preceding entry into the treatment period
Minimum Eligible Age

18 Years

Maximum Eligible Age

55 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

Yes

Sponsors

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Genentech, Inc.

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Principal Investigators

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Clinical Trials

Role: STUDY_DIRECTOR

Hoffmann-La Roche

Locations

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Quotient Clinical Ltd, Clinical Research Unit

Nottingham, , United Kingdom

Site Status

Countries

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United Kingdom

Other Identifiers

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2016-001572-30

Identifier Type: EUDRACT_NUMBER

Identifier Source: secondary_id

GX29841

Identifier Type: -

Identifier Source: org_study_id

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