Effect of Food on PC14586 in Healthy Volunteers and the PK of PC14586 in Healthy Japanese Volunteers

NCT ID: NCT05249348

Last Updated: 2024-11-13

Study Results

Results pending

The study team has not published outcome measurements, participant flow, or safety data for this trial yet. Check back later for updates.

Basic Information

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Recruitment Status

COMPLETED

Clinical Phase

PHASE1

Total Enrollment

34 participants

Study Classification

INTERVENTIONAL

Study Start Date

2021-12-20

Study Completion Date

2022-06-09

Brief Summary

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This is a 2-part Phase 1 cross-over study to assess the effects of food on the pharmacokinetics of PC14586 in healthy volunteers. The pharmacokinetics of PC14586 at a clinically relevant dose in Japanese participants will also be studied.

Detailed Description

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PC14586 is a first-in-class, oral, small molecule p53 reactivator that is selective for the p53 Y220C mutation. This Phase 1 trial will be conducted in 2 parts (Part 1 - pilot and Part 2 - pivotal) to assess the pharmacokinetics of PC14586 in healthy volunteers including Japanese participants.

Conditions

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Healthy Volunteers

Study Design

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Allocation Method

RANDOMIZED

Intervention Model

CROSSOVER

Single-dose crossover study one dose with food and one dose without food.
Primary Study Purpose

OTHER

Blinding Strategy

NONE

Study Groups

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Part 1 Sequence A

Period 1 will be fed, then washout, then Period 2 will be fasted.

Group Type EXPERIMENTAL

PC14586

Intervention Type DRUG

An oral dose of PC14586 will be used in Arms A and B (Part 1) and a different dose will be used for Arms C and D and the Japanese cohort (Part 2).

Part 1 Sequence B

Period 1 will be fasted, then washout, then Period 2 will be fed.

Group Type EXPERIMENTAL

PC14586

Intervention Type DRUG

An oral dose of PC14586 will be used in Arms A and B (Part 1) and a different dose will be used for Arms C and D and the Japanese cohort (Part 2).

Part 2 Sequence C

Period 1 will be fed, then washout, then Period 2 will be fasted. A different dose of PC14586 will be tested.

Group Type EXPERIMENTAL

PC14586

Intervention Type DRUG

An oral dose of PC14586 will be used in Arms A and B (Part 1) and a different dose will be used for Arms C and D and the Japanese cohort (Part 2).

Part 2 Sequence D

Period 1 will be fasted, then washout, then Period 2 will be fed. A different dose of PC14586 will be tested.

Group Type EXPERIMENTAL

PC14586

Intervention Type DRUG

An oral dose of PC14586 will be used in Arms A and B (Part 1) and a different dose will be used for Arms C and D and the Japanese cohort (Part 2).

Part 2 Japanese Cohort

6 Japanese participants will be administered a single dose of PC14586.

Group Type EXPERIMENTAL

PC14586

Intervention Type DRUG

An oral dose of PC14586 will be used in Arms A and B (Part 1) and a different dose will be used for Arms C and D and the Japanese cohort (Part 2).

Interventions

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PC14586

An oral dose of PC14586 will be used in Arms A and B (Part 1) and a different dose will be used for Arms C and D and the Japanese cohort (Part 2).

Intervention Type DRUG

Eligibility Criteria

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Inclusion Criteria

* Healthy, non-smoking male and female Caucasian/ non-Asian or Japanese human volunteers
* 18 to 55 years of age
* Able to swallow tablets.


* Japanese and born in Japan (1st generation)
* The parents and grandparents of the participant are ethnically Japanese and born in Japan
* Has undergone no significant change in lifestyle since leaving Japan
* Has lived \< 10 years outside of Japan

Exclusion Criteria

* Clinically significant medical history as determined by the PI.
* Any disorder that would interfere with the absorption, distribution, metabolism or excretion of drugs.
* A p53 Y220C mutation.
* Blood pressure \>140 mm systolic or \>90 diastolic.
* Smoked or used other nicotine-containing products during the previous 3 months.
* History of alcohol and/or illicit drug abuse within the previous 5 years.
* Hepatitis B surface antigen (HBsAg), Hepatitis C antibody or human immunodeficiency virus (HIV).
* Positive blood test for ethanol.
* Positive urine drug test.
* Pregnancy or breastfeeding.
* Unwilling to avoid use of alcohol or alcohol-containing foods, medications or beverages, within 48 hours prior to admission until discharge from the clinical site.
* Has donated blood within 2 months prior to admission.
* Has used over-the-counter (OTC) medications (including vitamins), prescription medications or herbal remedies from 14 days prior to admission.
* Has used an investigational drug within 30 days prior to Screening.
Minimum Eligible Age

18 Years

Maximum Eligible Age

55 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

Yes

Sponsors

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PMV Pharmaceuticals, Inc

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Locations

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Parexel Early Phase Clinical Unit - Los Angeles

Glendale, California, United States

Site Status

Countries

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United States

Other Identifiers

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262612

Identifier Type: OTHER

Identifier Source: secondary_id

PMV-586-102

Identifier Type: -

Identifier Source: org_study_id

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