Activity & Safety Study of KX2-391 Ointment in Participants With Actinic Keratosis on the Face or Scalp

NCT ID: NCT02838628

Last Updated: 2021-04-14

Study Results

Results available

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Basic Information

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Recruitment Status

COMPLETED

Clinical Phase

PHASE2

Total Enrollment

168 participants

Study Classification

INTERVENTIONAL

Study Start Date

2016-04-11

Study Completion Date

2017-12-22

Brief Summary

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In this study, the activity, safety, and pharmacokinetics (PK) of KX2-391 Ointment was evaluated in adult participants with a clinical diagnosis of stable, clinically typical actinic keratosis (AK) on the face or scalp.

Detailed Description

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This study was an open-label, multicenter, activity, safety, tolerability, and PK study of KX2-391 Ointment administered topically to the face or scalp of participants with AK.

The study consists of Screening, Treatment, and Follow-up Periods. Eligible participants were received 3 or 5 consecutive days of topical treatment, applied at the study site. Blood samples for PK analysis were collected. Activity (lesion counts) and safety evaluations were performed.

Conditions

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Actinic Keratosis

Study Design

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Allocation Method

NON_RANDOMIZED

Intervention Model

PARALLEL

Primary Study Purpose

TREATMENT

Blinding Strategy

NONE

Study Groups

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KX2-391 50 mg (Days 1 to 5)

Participants were applied 50 milligrams (mg) of KX2-391 Ointment 1% topically on face or scalp in 25 centimeter square (cm\^2) treatment area, once daily for 5 consecutive days.

Group Type EXPERIMENTAL

50 mg of KX2-391 Ointment 1%

Intervention Type DRUG

Dose: 50 mg; Route of administration: Topical

KX2-391 50 mg (Days 1 to 3)

Participants were applied 50 mg of KX2-391 Ointment 1% topically on face or scalp in 25 cm\^2 treatment area, once daily for 3 consecutive days.

Group Type EXPERIMENTAL

50 mg of KX2-391 Ointment 1%

Intervention Type DRUG

Dose: 50 mg; Route of administration: Topical

Interventions

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50 mg of KX2-391 Ointment 1%

Dose: 50 mg; Route of administration: Topical

Intervention Type DRUG

50 mg of KX2-391 Ointment 1%

Dose: 50 mg; Route of administration: Topical

Intervention Type DRUG

Eligibility Criteria

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Inclusion Criteria

1. Males and females ≥18 years old
2. Clinical diagnosis of stable, clinically typical actinic keratosis
3. A define treatment area on the face or scalp
4. Females must be postmenopausal, surgically sterile or otherwise incapable of pregnancy for at least 1 year; or must be using highly effective contraception for at least 90 days prior to treatment with KX2-391 Ointment
5. Males who have not had a vasectomy must agree to use barrier contraception
6. Participants who in the judgment of the Investigator, are in good general health
7. Willing to avoid excessive sun exposure
8. Able to comprehend and are willing to sign an informed consent form (ICF)

Exclusion Criteria

1. Clinically atypical and/or rapidly changing AK lesions on the treatment area
2. Malignancy within 5 years prior to Screening except basal or squamous cell carcinoma not on the treatment area that were treated with curative intent and are without recurrence
3. Used any of retinoids at the most 90 days before Visit 1 glucocorticosteroids and methotrexate or other anti-metabolites within, at the most 28 days, before Visit 1
4. Used any topical therapies, treatments, or surgical or destructive modalities on the treatment area within, at the most 90 days, before Visit 1
5. Currently, or has experienced cutaneous malignancy, sunburn or body art on the treatment area within, at the most 180 days, before Visit 1
6. A history of sensitivity and/or allergy to any of the ingredients in the study medication
7. A skin disease or condition that, in the opinion of the Investigator, might interfere with the study conduct or evaluations, or which exposes the participant to an unacceptable risk by study participation
8. Other significant uncontrolled or unstable medical diseases or conditions that, in the opinion of the Investigator, would expose the participant to unacceptable risk by study participation
9. Females who are pregnant or nursing
10. Participated in an investigational drug trial during which an investigational study medication was administered within 14 days or 5 half-lives of the investigational product, whichever is longer, before dosing.
Minimum Eligible Age

18 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

No

Sponsors

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Athenex, Inc.

INDUSTRY

Sponsor Role collaborator

Almirall, S.A.

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Principal Investigators

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Jane Fang, MD

Role: STUDY_CHAIR

Kinex Pharmaceuticals Inc.

Locations

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Center for Dermatology Clinical Research

Fremont, California, United States

Site Status

eStudy Site

La Mesa, California, United States

Site Status

Palmtree Clinical Research, Inc.

Palm Springs, California, United States

Site Status

Horizons Clinical Research Center

Denver, Colorado, United States

Site Status

Clinical Research of South Florida

Coral Gables, Florida, United States

Site Status

International Dermatology Research

Miami, Florida, United States

Site Status

Compass Research

Orlando, Florida, United States

Site Status

Forward Clinical Trials, Inc.

Tampa, Florida, United States

Site Status

Palm Beach Research Center

West Palm Beach, Florida, United States

Site Status

Minnesota Clinical Study Center

Fridley, Minnesota, United States

Site Status

Dermatology and Laser Center of Charleston

Charleston, South Carolina, United States

Site Status

Institute of Clinical Research - Tennessee, LLC

Murfreesboro, Tennessee, United States

Site Status

J&S Studies, Inc.

College Station, Texas, United States

Site Status

The Center for Skin Research

Houston, Texas, United States

Site Status

Clinical Trials of Texas, Inc.

San Antonio, Texas, United States

Site Status

Dermatology Clinical Research Center

San Antonio, Texas, United States

Site Status

Countries

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United States

References

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Kempers S, DuBois J, Forman S, Poon A, Cutler E, Wang H, Cutler D, Fang J, Kwan R. Tirbanibulin Ointment 1% as a Novel Treatment for Actinic Keratosis: Phase 1 and 2 Results. J Drugs Dermatol. 2020 Nov 1;19(11):1093-1100. doi: 10.36849/JDD.2020.5576.

Reference Type DERIVED
PMID: 33196758 (View on PubMed)

Provided Documents

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Document Type: Study Protocol

View Document

Document Type: Statistical Analysis Plan

View Document

Other Identifiers

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U1111-1173-5677

Identifier Type: OTHER

Identifier Source: secondary_id

KX01-AK-002

Identifier Type: -

Identifier Source: org_study_id

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