DS-3201b in Participants With Lymphomas

NCT ID: NCT02732275

Last Updated: 2025-02-07

Study Results

Results pending

The study team has not published outcome measurements, participant flow, or safety data for this trial yet. Check back later for updates.

Basic Information

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Recruitment Status

ACTIVE_NOT_RECRUITING

Clinical Phase

PHASE1

Total Enrollment

100 participants

Study Classification

INTERVENTIONAL

Study Start Date

2016-03-31

Study Completion Date

2026-12-31

Brief Summary

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DS-3201b is an experimental drug that is being investigated in clinical research.

Adults with non-Hodgkin lymphoma (NHL) may be able to join this study if their disease has come back after remission or is not responding to current treatment

This study has three parts. The Dose Escalation part is designed is to find the safe dose of DS-3201b that adults with advanced NHL can tolerate. The Dose Expansion phase will determine how effective DS-3201b is for rare types of NH and collect additional safety data. Last, the Drug-Drug Interaction (DDI) Cohort (US Only) will evaluate the effect of DS-3201b on the pharmacokinetics (PK) of midazolam and digoxin when co-administered to patients with NHL

Detailed Description

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Conditions

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Lymphoma, Malignant Non-hodgkin Lymphoma

Study Design

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Allocation Method

NA

Intervention Model

SINGLE_GROUP

Primary Study Purpose

TREATMENT

Blinding Strategy

NONE

Study Groups

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Dose Escalation - DS-3201b

Dose escalation is to identify the recommended phase 2 dose of DS-3201b guided by the modified continuous reassessment method using a Bayesian logistic regression model following escalation.

Group Type EXPERIMENTAL

DS-3201b

Intervention Type DRUG

DS-3201 to be administered orally once daily in each 28-day cycle.

Dose Expansion - DS-3201b

Part 2 is a dose expansion to examine the safety and efficacy of DS-3201b.

Group Type EXPERIMENTAL

DS-3201b

Intervention Type DRUG

DS-3201 to be administered orally once daily in each 28-day cycle at the recommended dose for expansion.

Interventions

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DS-3201b

DS-3201 to be administered orally once daily in each 28-day cycle.

Intervention Type DRUG

DS-3201b

DS-3201 to be administered orally once daily in each 28-day cycle at the recommended dose for expansion.

Intervention Type DRUG

Eligibility Criteria

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Inclusion Criteria

* Has hematocytological or pathological diagnosis of non- Hodgkin's lymphoma (NHL)
* Has relapsed from or is refractory to standard treatment or no standard treatment is available
* Is the age of majority in their country (18 in the US and 20 in Japan) at the time of informed consent
* Has Eastern Cooperative Oncology Group (ECOG) performance status 0 or 1
* Has at least one evaluable lesion site (not applicable for the DDI cohort)
* Has preserved organ function based on baseline laboratory data at screening tests
* If of reproductive potential, agrees to avoid harvesting ova or sperm, and to use a protocol-defined form of contraception or avoid intercourse, during and upon completion of the study, and for at least 3 months after the last dose of study drug
* Tumor biopsy collections:

1. willing to provide archived or fresh tumor tissue samples that are sufficient for comprehensive genomic and/or proteomic analyses at baseline
2. \[US only\] willing to provide fresh on-treatment tumor biopsy if deemed acceptable risk by the investigator

\[Japan only\] fresh on-treatment tumor biopsy should be performed if deemed acceptable risk by the investigator
3. willing to provide optional fresh end-of-treatment biopsy

For ATL subjects:

* Has a positive test result for human T-lymphotropic virus type I antibody
* Has ATL subtype classified as acute, lymphomatous, or chronic with poor prognostic factor
* Has diagnosis of relapse (including relapse after partial remission \[PR\]) or treatment-resistant ATL at the time of informed consent after prior treatment with at least 1 anti-cancer medication regimen

Exclusion Criteria

* Has been diagnosed with protocol-defined cutaneous T-cell lymphoma or T-cell leukemia. For DDI cohort, CTCL is not exclusionary.
* Has a history or presence of central nervous system (CNS) involvement
* Has a medical history, complication or other malignancy considered inappropriate for participation in the study, or a serious physical or psychiatric disease, the risk of which may be increased by participation in the study
* Has received drugs or other treatments not allowed by the protocol
* History of treatment with other enhancer of zeste (EZH) inhibitors
* Has had allogeneic hematopoietic stem cell transplantation (HTCP) within 90 days before scheduled dosing on Cycle 1 Day 1
* Is pregnant or breastfeeding
* Is otherwise deemed ineligible to participate by the investigator or sub-investigator

DDI Cohort Only:

* Has received following medications within 14 days prior to study drug administration
* Any CYP3A inhibitors/inducers including weak CYP3A inhibitors/inducers, and P-gp inhibitors, midazolam as well as digoxin
Minimum Eligible Age

18 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

No

Sponsors

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Daiichi Sankyo

INDUSTRY

Sponsor Role collaborator

Daiichi Sankyo Co., Ltd.

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Principal Investigators

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Global Clinical Leader, MD

Role: STUDY_DIRECTOR

Daiichi Sankyo

Locations

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City of Hope National Medical center

Duarte, California, United States

Site Status

Yale University

New Haven, Connecticut, United States

Site Status

Emory University

Atlanta, Georgia, United States

Site Status

Dana-Farber Cancer Institute

Boston, Massachusetts, United States

Site Status

Hackensack University Medical Center

Hackensack, New Jersey, United States

Site Status

Weill Cornell Medicine

New York, New York, United States

Site Status

Memorial Sloan Kettering Cancer Center

New York, New York, United States

Site Status

Duke University Medical Center

Durham, North Carolina, United States

Site Status

The Ohio State University Wexner Medical Center and James Cancer Hospital

Columbus, Ohio, United States

Site Status

Thomas Jefferson University

Philadelphia, Pennsylvania, United States

Site Status

Nagoya City University Hospital

Nagoya, Aichi-ken, Japan

Site Status

National Cancer Center Hospital East

Kahiwa-shi, Chiba, Japan

Site Status

Iwate Medical University Hospital

Morioka, Iwate, Japan

Site Status

Imamura General Hospital

Kagoshima, Kagoshima-ken, Japan

Site Status

Kagoshima University Hospital

Kagoshima, Kagoshima-ken, Japan

Site Status

Kumamoto University Hosipital

Kumamoto, Kumamoto, Japan

Site Status

Nagasaki University Hospital

Nagasaki, Nagasaki, Japan

Site Status

University of the Ryukyus Hospital

Nakagami-gun, Okinawa, Japan

Site Status

The Institute of Medical Science, The University of Tokyo

Minato-ku, Tokyo, Japan

Site Status

National Cancer Center Hospital

Chūōku, Toyko, Japan

Site Status

Countries

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United States Japan

References

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Maruyama D, Jacobsen E, Porcu P, Allen P, Ishitsuka K, Kusumoto S, Narita T, Tobinai K, Foss F, Tsukasaki K, Feldman T, Imaizumi Y, Izutsu K, Morishima S, Yamauchi N, Yuda J, Brammer JE, Kawamata T, Ruan J, Nosaka K, Utsunomiya A, Wang J, Zain J, Kakurai Y, Yamauchi H, Hizukuri Y, Biserna N, Tachibana M, Inoue A, Horwitz SM. Valemetostat monotherapy in patients with relapsed or refractory non-Hodgkin lymphoma: a first-in-human, multicentre, open-label, single-arm, phase 1 study. Lancet Oncol. 2024 Dec;25(12):1589-1601. doi: 10.1016/S1470-2045(24)00502-3. Epub 2024 Oct 29.

Reference Type DERIVED
PMID: 39486432 (View on PubMed)

Other Identifiers

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163173

Identifier Type: REGISTRY

Identifier Source: secondary_id

DS3201-A-J101

Identifier Type: -

Identifier Source: org_study_id

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