An Exploratory Study Investigating Safety, Tolerability and Pharmacokinetics of Ascending Doses of Lu AE04621 in Parkinson Disease Patients

NCT ID: NCT02649608

Last Updated: 2021-02-24

Study Results

Results available

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Basic Information

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Recruitment Status

COMPLETED

Clinical Phase

PHASE1

Total Enrollment

15 participants

Study Classification

INTERVENTIONAL

Study Start Date

2016-01-31

Study Completion Date

2016-12-31

Brief Summary

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To evaluate the safety, tolerability, pharmacokinetics, and efficacy of the Lu AE04621 and metabolite after ascending oral doses of Lu AE04621 in patients with Parkinson's Disease.

Detailed Description

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The study comprised 5 cohorts (Cohorts 1 to 5), with each cohort consisting of 3 patients with Parkinson's disease (men and/or women). Each patient will be treated for 3 or 4 days, with increasing dose each day.

Dosing regimen will be decided at a dosing conferences. Dose levels can be increased, maintained or reduced both between cohorts but also within same cohort. The results are presented by dose level and reflect the actual doses administered.

A follow-up safety visit was scheduled approximately 7 days after the last dose of IMP.

Conditions

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Parkinson Disease

Study Design

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Allocation Method

NON_RANDOMIZED

Intervention Model

SINGLE_GROUP

The study comprised 5 cohorts (Cohorts 1 to 5), with each cohort consisting of 3 patients (men and/or women). The dosing regimen planned for Cohort 1 was a dose of 0.2 mg Lu AE04621 on Day 1 followed by a dose of 0.4 mg Lu AE04621 on Day 2, and a dose of 0.6 mg Lu AE04621 on Day 3. • The dosing regimen planned for Cohort 2 was 0.4 mg Lu AE04621 on Day 1 followed by a dose of 0.6 mg Lu AE04621 on Day 2, and a dose of 0.8 mg Lu AE04621 on Day 3. The dosing regimen planned for Cohort 3 was 0.2 mg Lu AE04621 on Day 1 followed by a dose of 0.4 mg Lu AE04621 on Day 2, a dose of 0.6 mg Lu AE04621 on Day 3, and a dose of 1.0 mg Lu AE04621 on Day 4. The dosing regimen planned for Cohorts 4 and 5 was 0.2 mg Lu AE04621 on Day 1 followed by a dose of 0.4 mg Lu AE04621 on Day 2, a dose of 0.6 mg Lu AE04621 on Day 3, and a dose of 1.2 mg Lu AE04621 on Day 4. The results are presented by dose groups and are based on the actual doses administered.
Primary Study Purpose

TREATMENT

Blinding Strategy

NONE

Study Groups

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0.04 mg Lu AE04621

Patients having received a dose of 0.04 mg, independent of which Cohort they belong to.

Group Type EXPERIMENTAL

0.04 mg Lu AE04621

Intervention Type DRUG

0.04 mg dose group

0.08 mg Lu AE04621

Patients having received a dose of 0.08 mg, independent of which Cohort they belong to.

Group Type EXPERIMENTAL

0.08 mg Lu AE04621

Intervention Type DRUG

0.08mg dose group

0.2 mg Lu AE04621

Patients having received a dose of 0.2 mg, independent of which Cohort they belong to.

Group Type EXPERIMENTAL

0.2 mg Lu AE04621

Intervention Type DRUG

0.2 mg dose group

0.4 mg Lu AE04621

Patients having received a dose of 1.2 mg, independent of which Cohort they belong to.

Group Type EXPERIMENTAL

0.4 mg Lu AE04621

Intervention Type DRUG

0.4 mg dose group

0.6 mg Lu AE04621

Patients having received a dose of 0.6 mg, independent of which Cohort they belong to.

Group Type EXPERIMENTAL

0.6 mg Lu AE04621

Intervention Type DRUG

0.6 mg dose group

0.8 mg Lu AE04621

Patients having received a dose of 0.8 mg, independent of which Cohort they belong to.

Group Type EXPERIMENTAL

0.8 mg Lu AE04621

Intervention Type DRUG

0.8 mg dose group

1.0 mg Lu AE04621

Patients having received a dose of 1.0 mg, independent of which Cohort they belong to.

Group Type EXPERIMENTAL

1.0 mg Lu AE04621

Intervention Type DRUG

1.0 mg dose group

1.2 mg Lu AE04621

Patients having received a dose of 1.2 mg, independent of which Cohort they belong to.

Group Type EXPERIMENTAL

1.2 mg Lu AE04621

Intervention Type DRUG

1.2 mg dose group

Interventions

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0.04 mg Lu AE04621

0.04 mg dose group

Intervention Type DRUG

0.08 mg Lu AE04621

0.08mg dose group

Intervention Type DRUG

0.2 mg Lu AE04621

0.2 mg dose group

Intervention Type DRUG

0.4 mg Lu AE04621

0.4 mg dose group

Intervention Type DRUG

0.6 mg Lu AE04621

0.6 mg dose group

Intervention Type DRUG

0.8 mg Lu AE04621

0.8 mg dose group

Intervention Type DRUG

1.0 mg Lu AE04621

1.0 mg dose group

Intervention Type DRUG

1.2 mg Lu AE04621

1.2 mg dose group

Intervention Type DRUG

Eligibility Criteria

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Inclusion Criteria

* The patient is diagnosed with idiopathic Parkinson Disease (consistent with the UK Parkinson's Disease Society Brain Bank Criteria for the Diagnosis of PD).
* The patient's Hoehn and Yahr Staging score is ≤ 3 in the "ON" state.
* The patient experiences motor fluctuations with at least 2.5 hours of "OFF" periods in the awake time and has predictable morning "OFF" episodes, which have been consistent within the past 4 weeks.
* The patient currently has a good response to L-DOPA and has been receiving a stable dose of L-DOPA (≥3 doses per day of standard L-DOPA or ≥3 doses per day of Carbidopa and L-DOPA, Extended-Release Capsules) during at least four weeks prior to screening.

Exclusion Criteria

* The patient has cognitive impairment, defined as a Mini Mental State Examination(MMSE) score ≤ 26 at the Screening Visit.
* The patient has severe disabling dyskinesia
* The patient takes or has taken disallowed recent or concomitant medication (CYP2D6 inhibitors, CYP 3A4 substrate, Dopamine agonists, 5 HT3 antagonists, Anti-viral (Amantadine))
Minimum Eligible Age

45 Years

Maximum Eligible Age

75 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

No

Sponsors

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H. Lundbeck A/S

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Principal Investigators

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Email contact via H. Lundbeck A/S

Role: STUDY_DIRECTOR

[email protected]

Locations

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US1251

Hallandale, Florida, United States

Site Status

US1126

Orlando, Florida, United States

Site Status

US1352

Chicago, Illinois, United States

Site Status

US1084

Detroit, Michigan, United States

Site Status

Countries

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United States

Other Identifiers

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16779A

Identifier Type: -

Identifier Source: org_study_id

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