A Study of Ramucirumab (LY3009806) in Combination With Erlotinib in Previously Untreated Participants With EGFR Mutation-Positive Metastatic NSCLC (RELAY)

NCT ID: NCT02411448

Last Updated: 2026-01-16

Study Results

Results available

Outcome measurements, participant flow, baseline characteristics, and adverse events have been published for this study.

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Basic Information

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Recruitment Status

ACTIVE_NOT_RECRUITING

Clinical Phase

PHASE3

Total Enrollment

545 participants

Study Classification

INTERVENTIONAL

Study Start Date

2015-05-06

Study Completion Date

2026-12-31

Brief Summary

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The main purpose of this study is to evaluate the efficacy and safety of ramucirumab in combination with erlotinib as compared to placebo in combination with erlotinib in previously untreated participants with stage IV non-small cell lung cancer (NSCLC) harboring an activating epidermal growth factor receptor (EGFR) mutation (Exon 19-Del and Exon 21 L858R). Safety and tolerability of ramucirumab in combination with erlotinib will be assessed in Part A before proceeding to Part B.

The purpose of Part C is to determine the efficacy and safety of ramucirumab in combination with gefitinib in previously untreated East Asian participants with EGFR mutation-positive metastatic NSCLC and of ramucirumab in combination with osimertinib in those participants whose disease progressed on ramucirumab and gefitinib and that have T790M - positive metastatic NSCLC.

Detailed Description

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Conditions

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Metastatic Non-Small Cell Lung Cancer

Study Design

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Allocation Method

RANDOMIZED

Intervention Model

PARALLEL

Primary Study Purpose

TREATMENT

Blinding Strategy

DOUBLE

Participants Investigators

Study Groups

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Ramucirumab + Erlotinib

Part A: 10 milligrams per kilogram (mg/kg) ramucirumab administered every 2 weeks intravenously (IV) in combination with 150 mg erlotinib daily orally.

Participants may continue to receive treatment until discontinuation criteria are met.

Part B: 10 mg/kg ramucirumab administered every 2 weeks IV in combination with 150 mg erlotinib daily orally. Participants may continue to receive treatment until discontinuation criteria are met.

Group Type EXPERIMENTAL

Ramucirumab

Intervention Type DRUG

Administered IV.

Erlotinib

Intervention Type DRUG

Administered orally.

Placebo + Erlotinib

Part B: Placebo administered every 2 weeks IV in combination with 150 mg erlotinib daily orally.

Participants may continue to receive treatment until discontinuation criteria are met.

Group Type PLACEBO_COMPARATOR

Placebo

Intervention Type DRUG

Administered IV.

Erlotinib

Intervention Type DRUG

Administered orally.

Ramucirumab + Gefitinib or Osimertinib

Part C: 10 mg/kg ramucirumab administered every 2 weeks intravenously (IV) + 250 mg Gefitinib or 80 mg Osimertinib daily orally.

* Ramucirumab and gefitinib administered during period 1.
* Ramucirumab and osimertinib administered during period 2.

Group Type EXPERIMENTAL

Ramucirumab

Intervention Type DRUG

Administered IV.

Gefitinib

Intervention Type DRUG

Administered orally.

Osimertinib

Intervention Type DRUG

Administered orally.

Interventions

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Ramucirumab

Administered IV.

Intervention Type DRUG

Placebo

Administered IV.

Intervention Type DRUG

Erlotinib

Administered orally.

Intervention Type DRUG

Gefitinib

Administered orally.

Intervention Type DRUG

Osimertinib

Administered orally.

Intervention Type DRUG

Other Intervention Names

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LY3009806

Eligibility Criteria

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Inclusion Criteria

* Cytologically or histologically confirmed diagnosis of Stage IV NSCLC as defined by the American Joint Committee on Cancer Staging Criteria for Lung Cancer (AJCC 7th edition 2009).
* Eligible for first-line treatment with erlotinib based on documented evidence of tumor harboring an activating EGFR mutation \[exon 19 deletion or exon 21 (L858R) substitution mutation\].
* Mandatory provision of adequate archived stage IV NSCLC tissue samples or tissue samples other than stage IV NSCLC may be acceptable (optional for part C).
* At least one measurable lesion.
* Life expectancy of at least 3 months.

Exclusion Criteria

* Known T790M EGFR mutation (not applicable for Part C Period 2).
* Known leptomeningeal carcinomatosis, uncontrolled/unstable spinal cord compression, or brain metastases.
* Serious illness or medical condition.
* Ongoing treatment with CYP3A4 inducers or strong inhibitors.
* Ongoing therapy with nonsteroidal anti-inflammatory drugs for more than 2 months.
* History of gross hemoptysis.
* Significant bleeding disorders.
* Radiologically documented evidence of major blood vessel invasion or encasement by cancer.
* Radiographic evidence of intratumor cavitation.
* History of gastrointestinal perforation within last 6 months.
* History of bowel obstruction, inflammatory enteropathy or extensive intestinal resection.
* History of any arterial thrombotic event within 6 months prior to enrollment.
* The participant has any known significant ophthalmologic abnormalities of the surface of the eye.
Minimum Eligible Age

18 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

No

Sponsors

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Eli Lilly and Company

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Principal Investigators

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Call 1-877-CTLILLY (1-877-285-4559) or 1-317-615-4559 Mon - Fri 9 AM - 5 PM Eastern time (UTC/GMT - 5 hours, EST)

Role: STUDY_DIRECTOR

Eli Lilly and Company

Locations

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UCLA Hematology/Oncology - Santa Monica

Los Angeles, California, United States

Site Status

St. Charles Health System

Denver, Colorado, United States

Site Status

The Gastroenterology Group, P.C.

Honolulu, Hawaii, United States

Site Status

Cancer Center of Kansas

Wichita, Kansas, United States

Site Status

Queens Medical Associates

Fresh Meadows, New York, United States

Site Status

Levine Cancer Institute

Charlotte, North Carolina, United States

Site Status

AHN Allegheny General Hospital

Pittsburgh, Pennsylvania, United States

Site Status

Cross Cancer Institute

Edmonton, Alberta, Canada

Site Status

Hôpital Arnaud de Villeneuve - CHU Montpellier

Montpellier, Hérault, France

Site Status

Chu Grenoble Alpes

La Tronche, Isère, France

Site Status

Hopital Claude Huriez - CHU de Lille

Lille, Nord, France

Site Status

Centre Hospitalier Universitaire de Poitiers

Poitiers, Vienne, France

Site Status

Hôpital Européen Georges Pompidou

Paris, , France

Site Status

Robert-Bosch-Krankenhaus

Gerlingen, Baden-Wurttemberg, Germany

Site Status

Thoraxklinik Heidelberg gGmbH

Heidelberg, Baden-Wurttemberg, Germany

Site Status

Klinikum Köln-Merheim

Cologne, North Rhine-Westphalia, Germany

Site Status

Klinikum Chemnitz GmbH

Chemnitz, Saxony, Germany

Site Status

Städtisches Krankenhaus Martha-Maria Halle-Dölau gGmbH

Halle, Saxony-Anhalt, Germany

Site Status

LungenClinic Grosshansdorf

Großhansdorf, Schleswig-Holstein, Germany

Site Status

Helios Klinikum Emil von Behring Berlin-Zehlendorf

Berlin, , Germany

Site Status

Sotiria Thoracic Diseases Hospital of Athens

Athens, Attikí, Greece

Site Status

Queen Mary Hospital

Hong Kong, , Hong Kong

Site Status

Queen Elizabeth Hospital

Yau Ma Tei, , Hong Kong

Site Status

Instituto Tumori Giovanni Paolo II

Bari, Apulia, Italy

Site Status

Cro-Irccs

Aviano, Friuli Venezia Giulia, Italy

Site Status

Azienda Sanitaria Ospedaliera S Luigi Gonzaga

Orbassano, Torino, Italy

Site Status

IRCCS - AOU di Bologna

Bologna, , Italy

Site Status

Ospedale San Raffaele

Milan, , Italy

Site Status

Istituto Oncologico Veneto IRCCS

Padua, , Italy

Site Status

Aichi Cancer Center Hospital

Nagoya, Aichi-ken, Japan

Site Status

National Cancer Center Hospital East

Kashiwa, Chiba, Japan

Site Status

Ehime University Hospital

Tōon, Ehime, Japan

Site Status

Kurume University Hospital

Kurume, Fukuoka, Japan

Site Status

National Hospital Organization Asahikawa Medical Center

Asahikawa, Hokkaido, Japan

Site Status

Hyogo Cancer Center

Akashi, Hyōgo, Japan

Site Status

Hyogo Prefectual Amagasaki General Medical Center

Amagashiki, Hyōgo, Japan

Site Status

Himeji Medical Center

Himeji, Hyōgo, Japan

Site Status

Foundation for Biomedical Research and innovation

Kobe, Hyōgo, Japan

Site Status

Kobe City Medical Center General Hospital

Kobe, Hyōgo, Japan

Site Status

Kanazawa University Hospital

Kanazawa, Ishikawa-ken, Japan

Site Status

Kanagawa Cardiovascular and Respiratory Center

Yokohama, Kanagawa, Japan

Site Status

Kanagawa Cancer Center

Yokohama, Kanagawa, Japan

Site Status

Sendai Kousei Hospital

Sendai, Miyagi, Japan

Site Status

Niigata Cancer Center Hospital

Niigata, Niigata, Japan

Site Status

Osaka Habikino Medical Center

Habikino, Osaka, Japan

Site Status

Kansai Medical University Hospital

Hirakata, Osaka, Japan

Site Status

Kishiwada City Hospital

Kishiwada, Osaka, Japan

Site Status

Kindai University Hospital- Osakasayama Campus

Ōsaka-sayama, Osaka, Japan

Site Status

National Hospital Organization Kinki-Chuo Chest Medical Center

Sakai, Osaka, Japan

Site Status

Saitama Prefectural Cancer Center

Ina-machi, Saitama, Japan

Site Status

Shizuoka Cancer Center

Nakatogari, Shizuoka, Japan

Site Status

Tokyo Met Cancer & Infectious Diseases Center Komagome Hp

Bunkyo-ku, Tokyo, Japan

Site Status

National Cancer Center Hospital

Chuo-Ku, Tokyo, Japan

Site Status

Japanese Foundation for Cancer Research

Koto, Tokyo, Japan

Site Status

National Hospital Organization Yamaguchi Ube Medical Center

Ube, Yamaguchi, Japan

Site Status

Chiba University Hospital

Chiba, , Japan

Site Status

National Hospital Organization Kyushu Medical Center

Fukuoka, , Japan

Site Status

National Hospital Organization Kyushu Cancer Center

Fukuoka, , Japan

Site Status

Kyushu University Hospital

Fukuoka, , Japan

Site Status

Kyoto University Hospital

Kyoto, , Japan

Site Status

Nagasaki University Hospital

Nagasaki, , Japan

Site Status

Niigata University Medical & Dental Hospital

Niigata, , Japan

Site Status

Okayama University Hospital

Okayama, , Japan

Site Status

Osaka City General Hospital

Osaka, , Japan

Site Status

Osaka Medical Center for Cancer and Cardiovascular Diseases

Osaka, , Japan

Site Status

Osaka City University Hospital

Osaka, , Japan

Site Status

St. Lukes International Hospital

Tokyo, , Japan

Site Status

Juntendo University Hospital

Tokyo, , Japan

Site Status

Nippon Medical School Hospital

Tokyo, , Japan

Site Status

Wakayama MedicaL University Hospital

Wakayama, , Japan

Site Status

Institutul Oncologic

Bucharest, București, Romania

Site Status

S.C. MedisProf SRL

Cluj-Napoca, Cluj, Romania

Site Status

Chungbuk National University Hospital

Cheongju-si, Chungcheongbuk-do [Chungbuk], South Korea

Site Status

Seoul National University Bundang Hospital

Seongnam, Kyǒnggi-do, South Korea

Site Status

The Catholic University Of Korea St. Vincent's Hospital

Suwon, Kyǒnggi-do, South Korea

Site Status

Ajou University Hospital

Suwon, Kyǒnggi-do, South Korea

Site Status

Gyeongsang National University Hospital

Jinju, Kyǒngsangnam-do, South Korea

Site Status

Asan Medical Center

Seoul, Seoul-teukbyeolsi [Seoul], South Korea

Site Status

Samsung Medical Center

Seoul, Seoul-teukbyeolsi [Seoul], South Korea

Site Status

The Catholic Univ. of Korea Seoul St. Mary's Hospital

Seoul, Seoul-teukbyeolsi [Seoul], South Korea

Site Status

Korea University Guro Hospital

Seoul, Seoul-teukbyeolsi [Seoul], South Korea

Site Status

Ulsan University Hospital

Ulsan, Ulsan-Kwangyǒkshi, South Korea

Site Status

Hospital Universitari Vall d'Hebron

Barcelona, Barcelona [Barcelona], Spain

Site Status

Instituto Catalan de Oncologia - Hospital Duran i Reynals

Hospitalet, Barcelona [Barcelona], Spain

Site Status

Hospital Son Llatzer

Palma, Illes Balears [Islas Baleares], Spain

Site Status

Hospital Universitario Quironsalud Madrid

Pozuelo de Alarcón, Madrid, Spain

Site Status

Hospital Universitario 12 de Octubre

Madrid, Madrid, Comunidad de, Spain

Site Status

Clinica Universitaria De Navarra

Pamplona, Navarre, Spain

Site Status

Hospital Universitario Virgen del Rocio

Seville, , Spain

Site Status

Hospital Universitario Virgen de Valme

Seville, , Spain

Site Status

Hospital Universitari i Politecnic La Fe

Valencia, , Spain

Site Status

Chang Gung Memorial Hospital at Kaohsiung

Kaohsiung Niao Sung Dist, Kaohsiung, Taiwan

Site Status

E-DA Hospital

Kaohsiung City, , Taiwan

Site Status

China Medical University Hospital

Taichung, , Taiwan

Site Status

Taichung Veterans General Hospital

Taichung, , Taiwan

Site Status

National Cheng-Kung University Hospital

Tainan, , Taiwan

Site Status

National Taiwan University Hospital

Taipei, , Taiwan

Site Status

MacKay Memorial Hospital

Taipei, , Taiwan

Site Status

Taipei Veterans General Hospital

Taipei, , Taiwan

Site Status

Ege Universitesi Hastanesi

Bornova, İzmir, Turkey (Türkiye)

Site Status

Baskent University Dr. Turgut Noyan Research and Training Center

Adana, , Turkey (Türkiye)

Site Status

Trakya University

Edirne, , Turkey (Türkiye)

Site Status

İnönü Üniversitesi Turgut Özal Tıp Merkezi Eğitim ve Araştırma Hastanesi

Malatya, , Turkey (Türkiye)

Site Status

Royal Marsden Hospital (Chelsea)

London, Kensington and Chelsea, United Kingdom

Site Status

Charing Cross Hospital

Chelsea, London, United Kingdom

Site Status

City Hospital, Nottingham University Hospitals

Nottingham, Nottinghamshire, United Kingdom

Site Status

Countries

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United States Canada France Germany Greece Hong Kong Italy Japan Romania South Korea Spain Taiwan Turkey (Türkiye) United Kingdom

References

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Nishino K, Seto T, Nishio M, Nishio K, Kasahara K, Satouchi M, Yoh K, Hayashi H, Enatsu S, Matsui T, Varughese SC, Visseren-Grul C, Nakagawa K. RELAY: safety and efficacy of ramucirumab plus erlotinib in elderly Japanese patients with metastatic EGFR-mutated NSCLC. Future Oncol. 2025 Oct;21(24):3197-3206. doi: 10.1080/14796694.2025.2560225. Epub 2025 Sep 25.

Reference Type DERIVED
PMID: 40995949 (View on PubMed)

Nishio M, Seto T, Reck M, Garon EB, Nishio K, Kasahara K, Nishino K, Satouchi M, Yoh K, Hayashi H, Sakai K, Enatsu S, Frimodt-Moller B, Matsui T, Varughese SC, Carlsen M, Visseren-Grul C, Nakagawa K. Final Survival Outcomes With Ramucirumab Plus Erlotinib Versus Placebo Plus Erlotinib in Patients With Untreated EGFR-Mutated Metastatic NSCLC: RELAY Japanese Subset. JTO Clin Res Rep. 2025 Feb 28;6(6):100819. doi: 10.1016/j.jtocrr.2025.100819. eCollection 2025 Jun.

Reference Type DERIVED
PMID: 40458541 (View on PubMed)

Nakagawa K, Garon EB, Seto T, Nishio M, Aix SP, Paz-Ares L, Chiu CH, Park K, Novello S, Nadal E, Nishino K, Yoh K, Shih JY, Chik JYK, Moro-Sibilot D, Puri T, Chacko Varughese S, Frimodt-Moller B, Visseren-Grul C, Reck M. RELAY: Final Overall Survival for Erlotinib Plus Ramucirumab or Placebo in Untreated, EGFR-Mutated Metastatic NSCLC. J Thorac Oncol. 2025 Apr;20(4):487-499. doi: 10.1016/j.jtho.2024.11.032. Epub 2024 Nov 30.

Reference Type DERIVED
PMID: 39622410 (View on PubMed)

Nishio K, Sakai K, Nishio M, Seto T, Visseren-Grul C, Carlsen M, Matsui T, Enatsu S, Nakagawa K. Impact of ramucirumab plus erlotinib on circulating cell-free DNA from patients with untreated metastatic non-small cell lung cancer with EGFR-activating mutations (RELAY phase 3 randomized study). Transl Lung Cancer Res. 2023 Aug 30;12(8):1702-1716. doi: 10.21037/tlcr-22-736. Epub 2023 Aug 10.

Reference Type DERIVED
PMID: 37691865 (View on PubMed)

Garon EB, Reck M, Nishio K, Heymach JV, Nishio M, Novello S, Paz-Ares L, Popat S, Aix SP, Graham H, Butts BD, Visseren-Grul C, Nakagawa K; RELAY study investigators. Ramucirumab plus erlotinib versus placebo plus erlotinib in previously untreated EGFR-mutated metastatic non-small-cell lung cancer (RELAY): exploratory analysis of next-generation sequencing results. ESMO Open. 2023 Aug;8(4):101580. doi: 10.1016/j.esmoop.2023.101580. Epub 2023 Jun 28.

Reference Type DERIVED
PMID: 37390764 (View on PubMed)

Chiu CH, Lin MC, Wei YF, Chang GC, Su WC, Hsia TC, Su J, Wang AK, Jen MH, Puri T, Shih JY. Efficacy and Tolerability of Ramucirumab Plus Erlotinib in Taiwanese Patients with Untreated, Epidermal Growth Factor Receptor-Mutated, Stage IV Non-small Cell Lung Cancer in the RELAY Study. Target Oncol. 2023 Jul;18(4):505-515. doi: 10.1007/s11523-023-00975-5. Epub 2023 Jun 17.

Reference Type DERIVED
PMID: 37329423 (View on PubMed)

Nakagawa K, Garon EB, Gao L, Callies S, Zimmermann A, Walgren R, Visseren-Grul C, Reck M. RELAY, ramucirumab plus erlotinib versus placebo plus erlotinib in untreated EGFR-mutated metastatic non-small cell lung cancer: exposure-response relationship. Cancer Chemother Pharmacol. 2022 Aug;90(2):137-148. doi: 10.1007/s00280-022-04447-x. Epub 2022 Jul 16.

Reference Type DERIVED
PMID: 35841410 (View on PubMed)

Nishio M, Nishio K, Reck M, Garon EB, Imamura F, Kawaguchi T, Yamaguchi H, Ikeda S, Hirano K, Visseren-Grul C, Ceccarelli M, Wijayawardana SR, Zimmermann A, Matsui T, Enatsu S, Nakagawa K. RELAY+: Exploratory Study of Ramucirumab Plus Gefitinib in Untreated Patients With EGFR-Mutated Metastatic NSCLC. JTO Clin Res Rep. 2022 Feb 26;3(4):100303. doi: 10.1016/j.jtocrr.2022.100303. eCollection 2022 Apr.

Reference Type DERIVED
PMID: 35369607 (View on PubMed)

Nadal E, Horinouchi H, Shih JY, Nakagawa K, Reck M, Garon EB, Wei YF, Kollmeier J, Frimodt-Moller B, Barrett E, Lipkovich O, Visseren-Grul C, Novello S. RELAY, Ramucirumab Plus Erlotinib Versus Placebo Plus Erlotinib in Patients with Untreated, Epidermal Growth Factor Receptor Mutation-Positive, Metastatic Non-Small-Cell Lung Cancer: Safety Profile and Manageability. Drug Saf. 2022 Jan;45(1):45-64. doi: 10.1007/s40264-021-01127-2. Epub 2021 Dec 20.

Reference Type DERIVED
PMID: 34928484 (View on PubMed)

Mitani S, Chen Y, Inoue K, Mori J, Gao L, Long A, Wakabayashi S. Clinical Impact of a Shortened Infusion Duration of Ramucirumab in Japanese Patients -A Model-Based Approach. Gan To Kagaku Ryoho. 2021 Nov;48(11):1381-1387.

Reference Type DERIVED
PMID: 34795131 (View on PubMed)

Nakagawa K, Garon EB, Seto T, Nishio M, Ponce Aix S, Paz-Ares L, Chiu CH, Park K, Novello S, Nadal E, Imamura F, Yoh K, Shih JY, Au KH, Moro-Sibilot D, Enatsu S, Zimmermann A, Frimodt-Moller B, Visseren-Grul C, Reck M; RELAY Study Investigators. Ramucirumab plus erlotinib in patients with untreated, EGFR-mutated, advanced non-small-cell lung cancer (RELAY): a randomised, double-blind, placebo-controlled, phase 3 trial. Lancet Oncol. 2019 Dec;20(12):1655-1669. doi: 10.1016/S1470-2045(19)30634-5. Epub 2019 Oct 4.

Reference Type DERIVED
PMID: 31591063 (View on PubMed)

Reck M, Garon EB, Paz-Ares L, Ponce S, Jaime JC, Juan O, Nadal E, Kiura K, Widau RC, He S, Dalal R, Lee P, Nakagawa K. Randomized, Double-Blind Phase Ib/III Study of Erlotinib With Ramucirumab or Placebo in Previously Untreated EGFR-Mutant Metastatic Non-Small-Cell Lung Cancer (RELAY): Phase Ib Results. Clin Lung Cancer. 2018 May;19(3):213-220.e4. doi: 10.1016/j.cllc.2017.11.003. Epub 2017 Nov 21.

Reference Type DERIVED
PMID: 29317191 (View on PubMed)

Garon EB, Reck M, Paz-Ares L, Ponce S, Jaime JC, Juan O, Nadal E, Lee P, Dalal R, Liu J, He S, Treat J, Nakagawa K. Treatment Rationale and Study Design for the RELAY Study: A Multicenter, Randomized, Double-Blind Study of Erlotinib With Ramucirumab or Placebo in Patients With Epidermal Growth Factor Receptor Mutation-Positive Metastatic Non-Small-Cell Lung Cancer. Clin Lung Cancer. 2017 Jan;18(1):96-99. doi: 10.1016/j.cllc.2016.05.023. Epub 2016 Jun 8.

Reference Type DERIVED
PMID: 27894601 (View on PubMed)

Provided Documents

Download supplemental materials such as informed consent forms, study protocols, or participant manuals.

Document Type: Study Protocol: Protocol I4T-MC-JVCY(f)

View Document

Document Type: Study Protocol: Protocol Addendum I4T-MC-JVCY(9)

View Document

Document Type: Statistical Analysis Plan

View Document

Related Links

Access external resources that provide additional context or updates about the study.

https://trials.lillytrialguide.com/en-US/trial/3pxvd64nCo8AmAgMMu6iSo

A Study of Ramucirumab (LY3009806) in Combination With Erlotinib in Participants With EGFR Mutation-Positive Metastatic NSCLC

Other Identifiers

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I4T-MC-JVCY

Identifier Type: OTHER

Identifier Source: secondary_id

2014-004824-22

Identifier Type: EUDRACT_NUMBER

Identifier Source: secondary_id

15540

Identifier Type: -

Identifier Source: org_study_id

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