A Study to Investigate the Safety, Tolerability, and Pharmacokinetics of PF-06649751 in Subjects With Idiopathic Parkinson's Disease

NCT ID: NCT02373072

Last Updated: 2023-09-22

Study Results

Results pending

The study team has not published outcome measurements, participant flow, or safety data for this trial yet. Check back later for updates.

Basic Information

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Recruitment Status

COMPLETED

Clinical Phase

PHASE1

Total Enrollment

18 participants

Study Classification

INTERVENTIONAL

Study Start Date

2015-03-31

Study Completion Date

2016-03-31

Brief Summary

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This is a study with two sequential cohorts, each with three treatment periods. Single doses of PF-06649751 will be tested in this study, starting at a low dose and escalating to a dose projected to be under the current limits for drug concentration. Each cohort will aim to achieve approximately 9 completers. Primary endpoint is safety and tolerability, secondary endpoint is MDS-UPDRS part III.

Detailed Description

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Conditions

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Idiopathic Parkinson Disease

Study Design

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Allocation Method

RANDOMIZED

Intervention Model

PARALLEL

Primary Study Purpose

BASIC_SCIENCE

Blinding Strategy

DOUBLE

Participants Investigators

Study Groups

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Cohort 1

Three single doses over three periods. For each of the three periods, subjects will be crossed-over from placebo or PF-06649751. Each PF-06649751 dose is separated by at least one week.

Group Type EXPERIMENTAL

PF-06649751

Intervention Type DRUG

Subjects completing all three treatment periods will be administered two doses. Doses: 0.75mg, 1.5mg, 3mg, 6mg, 9mg. Tablets in the form of 0.25mg or 1 mg.

Trimethobenzamide Hydrochloride

Intervention Type DRUG

300mg TID, Capsules. Optional in both Cohorts.

Placebo

Intervention Type DRUG

Subjects completing all three treatment periods will be receiving placebo once.

Cohort 2

Three single doses over three periods. For each of the three periods, subjects will be crossed-over from placebo or PF-06649751. Each PF-06649751 dose is separated by at least one week.

Group Type EXPERIMENTAL

PF-06649751

Intervention Type DRUG

Subjects completing all three treatment periods will be administered two doses. Doses: 0.75mg, 1.5mg, 3mg, 6mg, 9mg. Tablets in the form of 0.25mg or 1 mg.

Trimethobenzamide Hydrochloride

Intervention Type DRUG

300mg TID, Capsules. Optional in both Cohorts.

Placebo

Intervention Type DRUG

Subjects completing all three treatment periods will be receiving placebo once.

Interventions

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PF-06649751

Subjects completing all three treatment periods will be administered two doses. Doses: 0.75mg, 1.5mg, 3mg, 6mg, 9mg. Tablets in the form of 0.25mg or 1 mg.

Intervention Type DRUG

Trimethobenzamide Hydrochloride

300mg TID, Capsules. Optional in both Cohorts.

Intervention Type DRUG

Placebo

Subjects completing all three treatment periods will be receiving placebo once.

Intervention Type DRUG

Eligibility Criteria

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Inclusion Criteria

* L-DOPA-responsiveness
* Hoehn \& Yahr Stage II-III inclusive
* Experiencing motor fluctuations
* Stable daily dose of L-DOPA of at least 300 mg
* Females on non-childbearing potential and male subjects

Exclusion Criteria

* History of troublesome dyskinesias
* History of surgical intervention for Parkinson's disease
Minimum Eligible Age

30 Years

Maximum Eligible Age

85 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

No

Sponsors

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Pfizer

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Principal Investigators

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Pfizer CT.gov Call Center

Role: STUDY_DIRECTOR

Pfizer

Locations

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Collaborative Neuroscience Network, LLC.

Long Beach, California, United States

Site Status

MD Clinical

Hallandale, Florida, United States

Site Status

Atlanta Center for Medical Research

Atlanta, Georgia, United States

Site Status

SNBL Clinical Pharmacology Center, Inc.

Baltimore, Maryland, United States

Site Status

Parkinson's Movement Disorder Center of Maryland

Elkridge, Maryland, United States

Site Status

Neurology Consultants of Dallas, PA

Dallas, Texas, United States

Site Status

Walnut Hill Medical Center

Dallas, Texas, United States

Site Status

Pfizer Clinical Research Unit

Brussels, , Belgium

Site Status

Countries

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United States Belgium

References

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Sohur US, Gray DL, Duvvuri S, Zhang Y, Thayer K, Feng G. Phase 1 Parkinson's Disease Studies Show the Dopamine D1/D5 Agonist PF-06649751 is Safe and Well Tolerated. Neurol Ther. 2018 Dec;7(2):307-319. doi: 10.1007/s40120-018-0114-z. Epub 2018 Oct 25.

Reference Type DERIVED
PMID: 30361858 (View on PubMed)

Other Identifiers

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2014-004389-54

Identifier Type: EUDRACT_NUMBER

Identifier Source: secondary_id

B7601009

Identifier Type: -

Identifier Source: org_study_id

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