The Tolerability and Effects of AZD0530 in Individuals With or Without a Family History of Alcoholism

NCT ID: NCT02262026

Last Updated: 2023-02-24

Study Results

Results pending

The study team has not published outcome measurements, participant flow, or safety data for this trial yet. Check back later for updates.

Basic Information

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Recruitment Status

COMPLETED

Clinical Phase

PHASE1

Total Enrollment

49 participants

Study Classification

INTERVENTIONAL

Study Start Date

2014-11-01

Study Completion Date

2019-04-26

Brief Summary

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Functional neuroimaging of alcoholism vulnerability: glutamate, reward, impulsivity, and Pavlovian-to-instrumental transfer (PIT), part II Saracatinib

Detailed Description

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To assess the effect of oral AZ D0530 at various doses on neuroimaging parameters associated with various forms of impulsivity mediated through glutamate-dopamine interactions, as ascertained through functional magnetic resonance imaging. -- --NOTE-- AZD0530 dosage of 50mg was discontinued by manufacturer. Adjustments were made to account for the removal of the 50mg dosage in all arms of the study.

Conditions

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Alcoholism

Study Design

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Allocation Method

RANDOMIZED

Intervention Model

CROSSOVER

Primary Study Purpose

TREATMENT

Blinding Strategy

SINGLE

Participants

Study Groups

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FHP; 125mg AZD0530, then 50mg AZD0530, then placebo

Family History positive for alcoholism will take place in blinded testing of 125 mg, then 50 mg, then placebo separated by 1 week for each test

Group Type EXPERIMENTAL

125 mg AZD0530

Intervention Type DRUG

Randomized to receive 125 mg of AZD0530

50 mg AZD0530

Intervention Type DRUG

Randomized to receive 50 mg of AZD0530

Placebo

Intervention Type DRUG

Placebo

FHP; 125mg AZD0530, then placebo, then 50mg AZD0530

Family History positive for alcoholism will take place in blinded testing of 125 mg, then placebo, then 50mg separated by 1 week for each test

Group Type EXPERIMENTAL

125 mg AZD0530

Intervention Type DRUG

Randomized to receive 125 mg of AZD0530

50 mg AZD0530

Intervention Type DRUG

Randomized to receive 50 mg of AZD0530

Placebo

Intervention Type DRUG

Placebo

FHP; 50mg AZD0530, then 125mg AZD0530, then placebo

Family History positive for alcoholism will take place in blinded testing of 50mg, then 125mg, then placebo separated by 1 week for each test

Group Type EXPERIMENTAL

125 mg AZD0530

Intervention Type DRUG

Randomized to receive 125 mg of AZD0530

50 mg AZD0530

Intervention Type DRUG

Randomized to receive 50 mg of AZD0530

Placebo

Intervention Type DRUG

Placebo

FHP; 50mg AZD0530, then placebo, then 125mg AZD0530

Family History positive for alcoholism will take place in blinded testing of 50mg, then placebo, then 125mg separated by 1 week for each test

Group Type EXPERIMENTAL

125 mg AZD0530

Intervention Type DRUG

Randomized to receive 125 mg of AZD0530

50 mg AZD0530

Intervention Type DRUG

Randomized to receive 50 mg of AZD0530

Placebo

Intervention Type DRUG

Placebo

FHP; placebo, then 50mg AZD0530, then 125mg AZD0530

Family History positive for alcoholism will take place in blinded testing of placebo, then 50 mg, then 125 mg separated by 1 week for each test

Group Type EXPERIMENTAL

125 mg AZD0530

Intervention Type DRUG

Randomized to receive 125 mg of AZD0530

50 mg AZD0530

Intervention Type DRUG

Randomized to receive 50 mg of AZD0530

Placebo

Intervention Type DRUG

Placebo

FHP; placebo, then 125mg AZD0530,then 50mg AZD0530

Family History positive for alcoholism will take place in blinded testing of placebo, then 125 mg, then 50 mg separated by 1 week for each test

Group Type EXPERIMENTAL

125 mg AZD0530

Intervention Type DRUG

Randomized to receive 125 mg of AZD0530

50 mg AZD0530

Intervention Type DRUG

Randomized to receive 50 mg of AZD0530

Placebo

Intervention Type DRUG

Placebo

FHN; 125mg AZD0530, then 50mg AZD0530, then placebo

Family History negative for alcoholism will take place in blinded testing of 125 mg, then 50 mg, then placebo separated by 1 week for each test

Group Type ACTIVE_COMPARATOR

125 mg AZD0530

Intervention Type DRUG

Randomized to receive 125 mg of AZD0530

50 mg AZD0530

Intervention Type DRUG

Randomized to receive 50 mg of AZD0530

Placebo

Intervention Type DRUG

Placebo

FHN; 125mg AZD0530, then placebo, then 50mg AZD0530

Family History negative for alcoholism will take place in blinded testing of 125 mg, then placebo, then 50mg separated by 1 week for each test

Group Type ACTIVE_COMPARATOR

125 mg AZD0530

Intervention Type DRUG

Randomized to receive 125 mg of AZD0530

50 mg AZD0530

Intervention Type DRUG

Randomized to receive 50 mg of AZD0530

Placebo

Intervention Type DRUG

Placebo

FHN; 50mg AZD0530, then 125mg AZD0530, then placebo

Family History negative for alcoholism will take place in blinded testing of 50mg, then 125mg, then placebo separated by 1 week for each test

Group Type ACTIVE_COMPARATOR

125 mg AZD0530

Intervention Type DRUG

Randomized to receive 125 mg of AZD0530

50 mg AZD0530

Intervention Type DRUG

Randomized to receive 50 mg of AZD0530

Placebo

Intervention Type DRUG

Placebo

FHN; 50mg AZD0530, then placebo, then 125mg AZD0530

Family History negative for alcoholism will take place in blinded testing of 50mg, then placebo, then 125mg separated by 1 week for each test

Group Type ACTIVE_COMPARATOR

125 mg AZD0530

Intervention Type DRUG

Randomized to receive 125 mg of AZD0530

50 mg AZD0530

Intervention Type DRUG

Randomized to receive 50 mg of AZD0530

Placebo

Intervention Type DRUG

Placebo

FHN; placebo, then 50mg AZD0530, then 125mg AZD0530

Family History negative for alcoholism will take place in blinded testing of placebo, then 50 mg, then 125 mg separated by 1 week for each test

Group Type ACTIVE_COMPARATOR

125 mg AZD0530

Intervention Type DRUG

Randomized to receive 125 mg of AZD0530

50 mg AZD0530

Intervention Type DRUG

Randomized to receive 50 mg of AZD0530

Placebo

Intervention Type DRUG

Placebo

FHN; placebo, then 125mg AZD0530, then 50mg AZD0530

Family History negative for alcoholism will take place in blinded testing of placebo, then 125 mg, then 50 mg separated by 1 week for each test

Group Type ACTIVE_COMPARATOR

125 mg AZD0530

Intervention Type DRUG

Randomized to receive 125 mg of AZD0530

50 mg AZD0530

Intervention Type DRUG

Randomized to receive 50 mg of AZD0530

Placebo

Intervention Type DRUG

Placebo

Interventions

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125 mg AZD0530

Randomized to receive 125 mg of AZD0530

Intervention Type DRUG

50 mg AZD0530

Randomized to receive 50 mg of AZD0530

Intervention Type DRUG

Placebo

Placebo

Intervention Type DRUG

Other Intervention Names

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saracatinib AZD0530 saracatinib AZD0530

Eligibility Criteria

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Inclusion Criteria

* Clear History of a father having a history of alcoholism, OR a mother AND another 1st or 2nd degree relative having a history of alcoholism, OR no 1st or 2nd degree relatives with alcoholism or substance abuse

Exclusion Criteria

1. Current diagnosis of DSM-IV-TR Axis I disorder, or past diagnosis of any substance use disorder or moderate alcohol use disorder
2. Report of psychotic disorder in a 1ยบ relative
3. Auditory or visual impairment that interferes with test taking
4. History of prenatal exposure to alcohol plus currently meeting criteria for features of fetal alcohol syndrome
5. Not speaking English fluently or being a non-native English speaker, or being educated in a primary language other than English \>grade 1
6. Mental retardation (Full Scale IQ\<70) using 2 WASI subtests for IQ estimate
7. Traumatic brain injury with loss of consciousness \> 30 minutes, or concussion in last 30 days
8. Presence or history of any medical/neurologic illness that may affect brain physiology (e.g., epilepsy, Multiple Sclerosis), including focal brain lesion seen on structural MRI (all structural scans are read by a licensed radiologist)
9. Current pregnancy (all females will be tested with urine screens on the day of MRI and prior to each phase of drug treatment)
10. Positive urine screen for the presence of marijuana, cocaine, opiates or breath screen to detect the presence of alcohol, administered at each lab visit.
11. Inability to comprehend the consent form appropriately
12. Ferromagnetic metal devices, clips or fragments in body (orbital x-ray performed if needed).
13. Current use (within 30 days of screening) of specific psychoactive medications (e.g., typical neuroleptics, narcotic analgesics, antiparkinsonian medications, systemic corticosteroids, or medications with significant central anticholinergic activity, etc.). Current use of warfarin.
14. Current use of the following medications (CYP3A4 substrates whose metabolism may be slowed by AZD0530): carbamazepine, colchicine, cyclosporine, disopyramide, fluticasone, quinidine, vinblastine, vincristine, nifedipine. Patients taking sildenafil, tadalafil, and vardenafil will be advised to stop taking these medications for the duration of the trial. Patients cannot take the following drugs which inhibit the CYP3A4 isoenzyme: cimetidine, cyclosporine, danazol, fluconazole, grapefruit juice, HIV protease inhibitors, itraconazole, ketoconazole, macrolides, miconazole, nefazodone, omeprazole, ritonavir, and verapamil, aromatase inhibitors, docetaxel
15. Neutropenia defined as absolute neutrophils count of \<1,500/microliter.
16. Thrombocytopenia defined as platelet count \<100x103/microliter.
17. AST, ALT, total bilirubin \>1.5 times upper normal; serum creatinine, \>2 time upper normal limit, total bilirubin\>1.5 times ULN; Serum creatinine \>2.0 times ULN.
18. History of interstitial lung disease.
Minimum Eligible Age

18 Years

Maximum Eligible Age

40 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

Yes

Sponsors

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Yale University

OTHER

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Principal Investigators

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Godfrey D Pearlson, MD

Role: PRINCIPAL_INVESTIGATOR

Yale University

Locations

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Hartford Hospital

Hartford, Connecticut, United States

Site Status

Countries

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United States

Provided Documents

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Document Type: Study Protocol and Statistical Analysis Plan

View Document

Document Type: Informed Consent Form

View Document

Other Identifiers

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1503015528

Identifier Type: -

Identifier Source: org_study_id

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