A Phase I Study of 8-week Continuous Treatment With Polyethylene Glycol Loxenatide in Patients With Type 2 Diabetes

NCT ID: NCT01976858

Last Updated: 2013-11-06

Study Results

Results pending

The study team has not published outcome measurements, participant flow, or safety data for this trial yet. Check back later for updates.

Basic Information

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Recruitment Status

COMPLETED

Clinical Phase

PHASE1

Total Enrollment

50 participants

Study Classification

INTERVENTIONAL

Study Start Date

2011-06-30

Study Completion Date

2011-12-31

Brief Summary

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Polyethylene Glycol Loxenatide (PEX168) is a new human glucagon-like peptide 1 (GLP-1) analogue that created on the basis of the Exenatide and modified by polyethylene glycol (PEG).

This study aims to evaluate the PK, PD and safety by 8-week continuous treatment of PEX168.

Detailed Description

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Conditions

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Type 2 Diabetes

Keywords

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PEX168, diabetes, phase I

Study Design

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Allocation Method

RANDOMIZED

Intervention Model

PARALLEL

Primary Study Purpose

TREATMENT

Blinding Strategy

QUADRUPLE

Participants Caregivers Investigators Outcome Assessors

Study Groups

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PEX168 50 microgram

PEX168 50 microgram qw sc. and the medication continued for 8 weeks

Group Type EXPERIMENTAL

PEX168

Intervention Type DRUG

A injection administered subcutaneously

PEX168 100 microgram

PEX168 100 microgram qw sc. and the medication continued for 8 weeks

Group Type EXPERIMENTAL

PEX168

Intervention Type DRUG

A injection administered subcutaneously

PEX168 200 microgram

PEX168 200 microgram qw sc. and the medication continued for 8 weeks

Group Type EXPERIMENTAL

PEX168

Intervention Type DRUG

A injection administered subcutaneously

PEX168 300 microgram

PEX168 300 microgram qw sc. and the medication continued for 8 weeks

Group Type EXPERIMENTAL

PEX168

Intervention Type DRUG

A injection administered subcutaneously

Placebo

Placebo qw sc. and the medication continued for 12 weeks

Group Type PLACEBO_COMPARATOR

PEX168

Intervention Type DRUG

A injection administered subcutaneously

Interventions

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PEX168

A injection administered subcutaneously

Intervention Type DRUG

Other Intervention Names

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Polyethylene Glycol Loxenatide

Eligibility Criteria

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Inclusion Criteria

1. aged 20-65 years old, male or female, diagnosis of type 2 diabetes according to the 1999 WHO criteria more than 3 months.
2. HbA1C 7.0-10.0% and fasting plasma glucose 7.0-10.0 mmol/L after treatment of diet, exercise or a single oral hypoglycemic agents (metformin , glimepiride or pioglitazone).
3. unused insulin within 3 months prior to the enrollment.
4. Body mass index within the range from 19 to 35, and body weight does not changes exceeding 10% in the past 3 months.
5. Normol liver, kidney, heart function.
6. Willing to use physical means of contraception during the trial stage.
7. voluntarily to participate in the study.

Exclusion Criteria

1. 1 diabetes.
2. used GLP-1, GLP-1 analogs or DPP-4 inhibitors in the past 3 months.
3. have diabetic ketoacidosis , diabetic hyperosmolar nonketotic coma patients with a history
4. There is a history of severe hypoglycemia : such as low blood sugar cause drowsiness , unconsciousness , nonsense , and even coma.
5. with severe diabetes complications ( renal , retinal , nerve , vascular disease).
6. has acute and chronic pancreatitis history ;
7. heart failure , unstable angina , severe arrhythmia, patients with a history of myocardial infarction ;
8. There is a history of hypertension and blood pressure is not well controlled : SBP\> 160mmHg and / or DBP\> 95mmHg persons ;
9. severe chronic gastrointestinal disease ( active ulcer nearly six months ) or have been affecting drug absorption in patients treated ;
10. There are obvious blood system diseases ;
11. There are other endocrine system diseases , such as hyperthyroidism , etc. ;
12. with severe trauma or surgery , severe infection ;
13. have mental illness , drug or other substance abuse or alcoholism ( drinking at least 2 times per week , more than 100g each drink ) ;
14. used any drugs that may affect the study , within 3 months before treatment as the subjects participated in any clinical trials ;
15. within the past six months more than 400ml of blood loss (including blood , trauma or other reasons ) ;
16. were receiving steroids or are receiving cancer treatment ;
17. has been prepared during pregnancy or pregnancy test in female patients ;
18. hepatitis B HBeAg , hepatitis C antibody positive , HIV antibody positive , syphilis antibody positive .
19. skin test positive of PEX168;
20. The researchers considered any factors that the subject should not participate in this trial.
Minimum Eligible Age

20 Years

Maximum Eligible Age

65 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

No

Sponsors

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Beijing Tongren Hospital

OTHER

Sponsor Role collaborator

Jiangsu HengRui Medicine Co., Ltd.

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Principal Investigators

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Jinkui Yang, Ph.D, M.D

Role: PRINCIPAL_INVESTIGATOR

Beijing Tongren Hospital

Locations

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Beijing tongren hospital

Beijing, Beijing Municipality, China

Site Status

Countries

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China

Other Identifiers

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PEX168-I-03

Identifier Type: -

Identifier Source: org_study_id