Study to Evaluate the Effect of Single Doses of LX4211 and Canagliflozin on Intestinal Glucose Absorption in Healthy Adult Subjects

NCT ID: NCT01916863

Last Updated: 2013-10-30

Study Results

Results pending

The study team has not published outcome measurements, participant flow, or safety data for this trial yet. Check back later for updates.

Basic Information

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Recruitment Status

COMPLETED

Clinical Phase

PHASE1

Total Enrollment

25 participants

Study Classification

INTERVENTIONAL

Study Start Date

2013-08-31

Brief Summary

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The purpose of this study is to assess the effect of LX4211 and the comparator drug canagliflozin on intestinal glucose absorption and metabolism after a single dose in healthy subjects in comparison to placebo.

Detailed Description

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Conditions

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Healthy Subjects

Study Design

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Allocation Method

RANDOMIZED

Intervention Model

CROSSOVER

Primary Study Purpose

TREATMENT

Blinding Strategy

QUADRUPLE

Participants Caregivers Investigators Outcome Assessors

Study Groups

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LX4211

400 mg of LX4211

Group Type EXPERIMENTAL

LX4211 400 mg

Intervention Type DRUG

canagliflozin 300 mg

Intervention Type DRUG

LX4211 Placebo

Intervention Type DRUG

Canagliflozin

300 mg canagliflozin

Group Type ACTIVE_COMPARATOR

LX4211 400 mg

Intervention Type DRUG

canagliflozin 300 mg

Intervention Type DRUG

LX4211 Placebo

Intervention Type DRUG

Placebo

LX4211 placebo

Group Type PLACEBO_COMPARATOR

LX4211 400 mg

Intervention Type DRUG

canagliflozin 300 mg

Intervention Type DRUG

LX4211 Placebo

Intervention Type DRUG

Interventions

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LX4211 400 mg

Intervention Type DRUG

canagliflozin 300 mg

Intervention Type DRUG

LX4211 Placebo

Intervention Type DRUG

Eligibility Criteria

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Inclusion Criteria

* Adult subjects ≥18 to ≤55 years of age
* Vital signs at Screening in the following ranges: systolic blood pressure, 90-140 mmHg; diastolic blood pressure, 50-90 mmHg; heart rate, 45-100 bpm
* Body mass index (BMI) ≥18 and ≤35 kg/sq m
* Willing and able to provide written informed consent

Exclusion Criteria

* Use of any medication (prescription, over-the-counter, herbal tea, or supplements) within 7 days of dosing
* Use of any investigational agent or study treatment within 30 days of Day -1
* Use of any protein or antibody-based therapeutic agents within 3 months of Screening
* Prior exposure to LX4211 or canagliflozin
* Daily use of \>5 cigarettes or any tobacco products within 6 weeks prior to Screening and while participating in the study
* History of bariatric surgery or any other gastrointestinal surgery that may induce malabsorption
* History of bowel resection, any malabsorptive disorder, severe gastroparesis, any GI procedure for the purpose of weight loss which would slow gastric emptying
* History of any major surgery within 6 months prior to Screening
* History of any hypersensitivity to the inactive components of LX4211, inactive components of canagliflozin, acetaminophen oral solution or any inactive component of acetaminophen liquid preparation
* History of renal disease or significantly abnormal kidney function tests
* History of hepatic disease or significantly abnormal liver function tests
* History of any active infection within 30 days prior to Day -1
* History of alcohol or substance abuse within 2 years prior to Day 1
* History of hepatitis B surface antigen (HBsAg), hepatitis C antibody (HCV Ab), HIV-1 or HIV-2
* Donation or loss of \>500 mL of blood or blood product within 56 days of Day -1
* positive pregnancy test at Screening or Day -1
* Positive urine screen for drugs of abuse at Screening or Day -1
* Positive breath test for alcohol at Screening or Day -1
* Inability or difficulty swallowing whole tablets
* Unable or unwilling to communicate or cooperate with the Investigator
Minimum Eligible Age

18 Years

Maximum Eligible Age

55 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

Yes

Sponsors

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Lexicon Pharmaceuticals

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Principal Investigators

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Paul Strumph, M.D.

Role: STUDY_DIRECTOR

Lexicon Pharmaceuticals, Inc.

Locations

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Lexicon Investigational Site

Chula Vista, California, United States

Site Status

Countries

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United States

References

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Powell DR, Zambrowicz B, Morrow L, Beysen C, Hompesch M, Turner S, Hellerstein M, Banks P, Strumph P, Lapuerta P. Sotagliflozin Decreases Postprandial Glucose and Insulin Concentrations by Delaying Intestinal Glucose Absorption. J Clin Endocrinol Metab. 2020 Apr 1;105(4):e1235-49. doi: 10.1210/clinem/dgz258.

Reference Type DERIVED
PMID: 31837264 (View on PubMed)

Other Identifiers

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LX4211.111

Identifier Type: OTHER

Identifier Source: secondary_id

LX4211.1-111-NRM

Identifier Type: -

Identifier Source: org_study_id