Study of Two Oral Formulations of LX4211 in Patients With Type 2 Diabetes Mellitus

NCT ID: NCT01188863

Last Updated: 2011-03-30

Study Results

Results pending

The study team has not published outcome measurements, participant flow, or safety data for this trial yet. Check back later for updates.

Basic Information

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Recruitment Status

COMPLETED

Clinical Phase

PHASE1

Total Enrollment

15 participants

Study Classification

INTERVENTIONAL

Study Start Date

2010-09-30

Brief Summary

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This protocol is intended to compare the effects of both a solid (tablet) and liquid oral dosage form of LX4211 in subjects with type 2 diabetes mellitus.

Detailed Description

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Conditions

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Type 2 Diabetes Mellitus

Study Design

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Allocation Method

RANDOMIZED

Intervention Model

CROSSOVER

Primary Study Purpose

TREATMENT

Blinding Strategy

NONE

Study Groups

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Solid Oral Dose - 150 mg tablets

Group Type EXPERIMENTAL

300 mg LX4211 (150 mg tablets)

Intervention Type DRUG

Single oral dose of two 150 mg tablets LX4211

Solid Oral Dose - 50 mg tablets

Group Type EXPERIMENTAL

300 mg LX4211 (50 mg tablets)

Intervention Type DRUG

Single oral dose of six 50 mg tablets LX4211

Liquid Oral Dose

Group Type EXPERIMENTAL

300 mg LX4211 (liquid)

Intervention Type DRUG

Single 30 mL dose of liquid oral solution LX4211 (10 mg/mL)

Interventions

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300 mg LX4211 (150 mg tablets)

Single oral dose of two 150 mg tablets LX4211

Intervention Type DRUG

300 mg LX4211 (50 mg tablets)

Single oral dose of six 50 mg tablets LX4211

Intervention Type DRUG

300 mg LX4211 (liquid)

Single 30 mL dose of liquid oral solution LX4211 (10 mg/mL)

Intervention Type DRUG

Eligibility Criteria

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Inclusion Criteria

* Adults aged 18 to 65 years of age
* Males and females of non-childbearing potential
* Diagnosis of type 2 diabetes mellitus for at least 6 months prior to screening
* Fasting plasma glucose ≤240 mg/dL
* Body mass index \<42 kg/sq m
* HbA1c of 7-11%
* C-peptide of ≥1.0 ng/mL
* Ability to provide written informed consent

Exclusion Criteria

* History of type 1 diabetes mellitus, diabetic ketoacidosis, hyperosmolar nonketonic syndrome, incontinence, or nocturia
* Current use of any blood glucose-lowering agent other than metformin
* Exposure to insulin, thiazide, or loop diuretics within 4 weeks prior to screening
* History of HIV, Hepatitis B, or Hepatitis C
* Surgery within 6 months of screening
* Donation or loss of \>400 mL of blood or blood product within 8 weeks prior to start of study
* Use of proteins or antibodies within 12 weeks prior to screening. (Flu shots are allowed.)
* Exposure to any investigational agent or participation in an investigational trial within 30 days of the start of the study
* History of drug or alcohol abuse within 12 months prior to screening.
Minimum Eligible Age

18 Years

Maximum Eligible Age

65 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

No

Sponsors

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Lexicon Pharmaceuticals

INDUSTRY

Sponsor Role lead

Responsible Party

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Lexicon Pharmaceuticals, Inc.

Principal Investigators

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Joel P. Freiman, MD, MPH

Role: STUDY_DIRECTOR

Lexicon Pharmaceuticals, Inc.

Locations

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Lexicon Investigational Site

San Antonio, Texas, United States

Site Status

Countries

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United States

References

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Zambrowicz B, Freiman J, Brown PM, Frazier KS, Turnage A, Bronner J, Ruff D, Shadoan M, Banks P, Mseeh F, Rawlins DB, Goodwin NC, Mabon R, Harrison BA, Wilson A, Sands A, Powell DR. LX4211, a dual SGLT1/SGLT2 inhibitor, improved glycemic control in patients with type 2 diabetes in a randomized, placebo-controlled trial. Clin Pharmacol Ther. 2012 Aug;92(2):158-69. doi: 10.1038/clpt.2012.58. Epub 2012 Jul 4.

Reference Type DERIVED
PMID: 22739142 (View on PubMed)

Other Identifiers

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LX4211.102

Identifier Type: OTHER

Identifier Source: secondary_id

LX4211.1-102-DM

Identifier Type: -

Identifier Source: org_study_id