Study to Evaluate a HIV Drug for the Treatment of HIV Infection

NCT ID: NCT01803074

Last Updated: 2019-11-25

Study Results

Results available

Outcome measurements, participant flow, baseline characteristics, and adverse events have been published for this study.

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Basic Information

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Recruitment Status

COMPLETED

Clinical Phase

PHASE2

Total Enrollment

107 participants

Study Classification

INTERVENTIONAL

Study Start Date

2013-04-04

Study Completion Date

2014-11-29

Brief Summary

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The primary purpose of this study is to study the safety and tolerability of a HIV drug and to evaluate a decrease of HIV-1 virus level in blood after treatments in HIV-1 infected patients

Detailed Description

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Masking: Open-Part B. Double Blind-Parts A and C

Gender: Both female and male participants for Parts A and C. Male participants for Part B.

HIV = Human Immunodeficiency Virus RNA = Ribonucleic acid

Conditions

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Infection, Human Immunodeficiency Virus HIV Infections

Study Design

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Allocation Method

RANDOMIZED

Intervention Model

PARALLEL

Primary Study Purpose

TREATMENT

Blinding Strategy

TRIPLE

Participants Caregivers Investigators

Study Groups

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Part A-Group 1: BMS-955176 (5 mg) or Placebo

BMS-955176 5 mg solution by mouth once daily for 10 days

OR

Placebo matching with BMS-955176 0 mg solution by mouth once daily for 10 days

Group Type EXPERIMENTAL

BMS-955176

Intervention Type DRUG

BMS-955176

Placebo matching with BMS-955176

Intervention Type DRUG

Placebo matching with BMS-955176

Part A-Group 2: BMS-955176 (10 mg) or Placebo

BMS-955176 10 mg solution by mouth once daily for 10 days

OR

Placebo matching with BMS-955176 0 mg solution by mouth once daily for 10 days

Group Type EXPERIMENTAL

BMS-955176

Intervention Type DRUG

BMS-955176

Placebo matching with BMS-955176

Intervention Type DRUG

Placebo matching with BMS-955176

Part A-Group 3: BMS-955176 (20 mg) or Placebo

BMS-955176 20 mg solution by mouth once daily for 10 days

OR

Placebo matching with BMS-955176 0 mg solution by mouth once daily for 10 days

Group Type EXPERIMENTAL

BMS-955176

Intervention Type DRUG

BMS-955176

Placebo matching with BMS-955176

Intervention Type DRUG

Placebo matching with BMS-955176

Part A-Group 4: BMS-955176 (40 mg) or Placebo

BMS-955176 40 mg solution by mouth once daily for 10 days

OR

Placebo matching with BMS-955176 0 mg solution by mouth once daily for 10 days

Group Type EXPERIMENTAL

BMS-955176

Intervention Type DRUG

BMS-955176

Placebo matching with BMS-955176

Intervention Type DRUG

Placebo matching with BMS-955176

Part B-Group 5: BMS-955176 + Atazanavir

BMS-955176 40 mg solution by mouth once daily for 28 days

Atazanavir 2 x 200 mg capsules by mouth once daily for 28 days

Group Type EXPERIMENTAL

BMS-955176

Intervention Type DRUG

BMS-955176

Atazanavir

Intervention Type DRUG

Atazanavir

Part B-Group 6: BMS-955176 + Atazanavir + Ritonavir

BMS-955176 40 mg solution by mouth once daily for 28 days

Atazanavir 1 x 300 mg capsules by mouth once daily for 28 days

Ritonavir 1 x 100 mg tablet by mouth once daily for 28 days

Group Type EXPERIMENTAL

BMS-955176

Intervention Type DRUG

BMS-955176

Atazanavir

Intervention Type DRUG

Atazanavir

Ritonavir

Intervention Type DRUG

Ritonavir

Part B-Group 7: Atazanavir+Ritonavir+Tenofovir+Emtricitabine

Atazanavir 1 x 300 mg capsule by mouth once daily for 28 days

Ritonavir 1 x 100 mg tablet by mouth once daily for 28 days

Tenofovir 1 x 300 mg tablet by mouth once daily for 28 days

Emtricitabine 1 x 200 mg capsule once daily for 28 days

Group Type EXPERIMENTAL

Atazanavir

Intervention Type DRUG

Atazanavir

Ritonavir

Intervention Type DRUG

Ritonavir

Tenofovir

Intervention Type DRUG

Tenofovir

Emtricitabine

Intervention Type DRUG

Emtricitabine

Part C-Group 8: BMS-955176 (40 mg) or Placebo

BMS-955176 40 mg solution by mouth once daily for 10 days

OR

Placebo matching with BMS-955176 0 mg solution by mouth once daily for 10 days

Group Type EXPERIMENTAL

BMS-955176

Intervention Type DRUG

BMS-955176

Placebo matching with BMS-955176

Intervention Type DRUG

Placebo matching with BMS-955176

Part A-Group 9: BMS-955176 (80 mg) or Placebo

BMS-955176 80 mg solution by mouth once daily for 10 days

OR

Placebo matching with BMS-955176 0 mg solution by mouth once daily for 10 days

Group Type EXPERIMENTAL

BMS-955176

Intervention Type DRUG

BMS-955176

Placebo matching with BMS-955176

Intervention Type DRUG

Placebo matching with BMS-955176

Part A-Group 10: BMS-955176 (120 mg) or Placebo

BMS-955176 120 mg solution by mouth once daily for 10 days

OR

Placebo matching with BMS-955176 0 mg solution by mouth once daily for 10 days

Group Type EXPERIMENTAL

BMS-955176

Intervention Type DRUG

BMS-955176

Placebo matching with BMS-955176

Intervention Type DRUG

Placebo matching with BMS-955176

Part A-Group 11 (Optional): BMS-955176 (≤120 mg) or Placebo

BMS-955176 ≤120 mg solution by mouth once daily for 14 days

OR

Placebo matching with BMS-955176 0 mg solution by mouth once daily for 14 days

Group Type EXPERIMENTAL

BMS-955176

Intervention Type DRUG

BMS-955176

Placebo matching with BMS-955176

Intervention Type DRUG

Placebo matching with BMS-955176

Part B-Group 12: BMS-955176 (80 mg) + Atazanavir

BMS-955176 80 mg solution by mouth once daily for 28 days

Atazanavir 2 x 200 mg capsules by mouth once daily for 28 days

Group Type EXPERIMENTAL

BMS-955176

Intervention Type DRUG

BMS-955176

Atazanavir

Intervention Type DRUG

Atazanavir

Part C-Group 13: BMS-955176 (120 mg) or Placebo

BMS-955176 120 mg solution by mouth once daily for 10 days

OR

Placebo matching with BMS-955176 0 mg solution by mouth once daily for 10 days

Group Type EXPERIMENTAL

BMS-955176

Intervention Type DRUG

BMS-955176

Placebo matching with BMS-955176

Intervention Type DRUG

Placebo matching with BMS-955176

Interventions

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BMS-955176

BMS-955176

Intervention Type DRUG

Placebo matching with BMS-955176

Placebo matching with BMS-955176

Intervention Type DRUG

Atazanavir

Atazanavir

Intervention Type DRUG

Ritonavir

Ritonavir

Intervention Type DRUG

Tenofovir

Tenofovir

Intervention Type DRUG

Emtricitabine

Emtricitabine

Intervention Type DRUG

Eligibility Criteria

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Inclusion Criteria

* Age 18-55 years inclusive
* Men and women: (Parts A and C); men only (Part B)
* Women of childbearing potential (WOCBP) must not be pregnant and nursing
* BMI: 18.0-35.0 kg/m2
* Subjects are infected with HIV-1 (clades B or C) and meet following criteria at the screening:

i) Plasma HIV-1 RNA ≥5,000 copies/mL; ii) Antiretroviral treatment naive (defined as \<1 week of ARV treatment) or ART-experienced (protease inhibitor and/or maturation inhibitor naive); iii) Subjects are not eligible for HIV-1 treatment based on the United States Department of Health and Human Services Panel on Antiretroviral Guidelines for Adults and Adolescents or have declined initiation of cART iv) CD4+ lymphocyte measurement ≥200 cells/μL; v) In Parts A and B, all subjects are infected with HIV-1 clade B vi) In Part C, all subjects are infected with HIV-1 clade C

Exclusion Criteria

* History of genotypic and/or phenotypic drug resistance testing showing resistance to protease inhibitors
* Any significant acute or chronic medical illness which is not stable or is not controlled with medication or not consistent with HIV-1 infection
* Receive antiretroviral treatment within 12 weeks prior to screening
* Currently co-infected with hepatitis C or hepatitis B
* Previously received an HIV maturation inhibitor or HIV protease inhibitor
* Current or recent (within 3 months of study drug administration) gastrointestinal disease
* Any major surgery within 4 weeks of study drug administration
* Acute diarrhea lasting ≥1 day, within 3 weeks prior to randomization
* Subjects with history of Gilbert's syndrome
* Subjects previously received an HIV maturation inhibitor or HIV protease inhibitor
* A personal history of clinically relevant cardiac disease, symptomatic or asymptomatic arrhythmias, syncopal episodes, or additional risk factors for torsades de pointes. A personal or family history of long QT syndrome
* Patients who are unwilling to practice adequate infection protection during and after study participation to minimize potential for spread of HIV infection, including HIV which may have developed resistance to HIV maturation inhibitor and/or ATV
* Any gastrointestinal surgery that could impact upon the absorption of study drug
* Smoking \>10 cigarettes per day
* PR ≥210 msec; QRS ≥120 msec; QT ≥500 msec; and QTcF ≥470 msec for women and ≥450 msec for men
* Evidence of second or third degree heart block prior to study drug
* Absolute Neutrophil Count \<(ANC) 0.7 x lower limit of normal (LLN)
* Hemoglobin \<0.8 x LLN
* Alanine aminotransferase (ALT) \>1.25 x upper limit of normal (ULN)
* Aspartate aminotransferase (AST) \>1.25 x ULN
* Total Bilirubin \>1.25 x ULN
* Creatinine clearance \<60 mL/mim
* Positive urine screen for drugs of abuse without a valid prescription (subjects positive for cannabinoids and/or amphetamines will be included)
* Positive blood screen for hepatitis C virus (HCV) RNA, hepatitis B surface antigen (consistent with active or chronic hepatitis B), or HIV-2 antibody
* History of any significant drug allergy
Minimum Eligible Age

18 Years

Maximum Eligible Age

55 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

No

Sponsors

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GlaxoSmithKline

INDUSTRY

Sponsor Role collaborator

ViiV Healthcare

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Principal Investigators

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GSK Clinical Trials

Role: STUDY_DIRECTOR

ViiV Healthcare

Locations

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GSK Investigational Site

Berlin, , Germany

Site Status

Countries

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Germany

References

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Hwang C, Schurmann D, Sobotha C, Boffito M, Sevinsky H, Ray N, Ravindran P, Xiao H, Keicher C, Huser A, Krystal M, Dicker IB, Grasela D, Lataillade M. Antiviral Activity, Safety, and Exposure-Response Relationships of GSK3532795, a Second-Generation Human Immunodeficiency Virus Type 1 Maturation Inhibitor, Administered as Monotherapy or in Combination With Atazanavir With or Without Ritonavir in a Phase 2a Randomized, Dose-Ranging, Controlled Trial (AI468002). Clin Infect Dis. 2017 Aug 1;65(3):442-452. doi: 10.1093/cid/cix239.

Reference Type DERIVED
PMID: 28369211 (View on PubMed)

Related Links

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Other Identifiers

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2012-004124-38

Identifier Type: EUDRACT_NUMBER

Identifier Source: secondary_id

AI468-002

Identifier Type: OTHER

Identifier Source: secondary_id

206739

Identifier Type: -

Identifier Source: org_study_id

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