A Bioequivalence Study of the Fixed Dose Combinations of Saxagliptin/Metformin XR Relative to Co-Administration

NCT ID: NCT01755494

Last Updated: 2013-12-13

Study Results

Results pending

The study team has not published outcome measurements, participant flow, or safety data for this trial yet. Check back later for updates.

Basic Information

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Recruitment Status

COMPLETED

Clinical Phase

PHASE1

Total Enrollment

64 participants

Study Classification

INTERVENTIONAL

Study Start Date

2013-02-28

Study Completion Date

2013-04-30

Brief Summary

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The primary objective of this study is to assess the pharmacokinetic parameters of saxagliptin and metformin in healthy male Chinese subjects.

Detailed Description

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A Single-centre, Randomized, Open-label, Two-period, Cross-over, Bioequivalence Study of the Fixed Dose Combinations of Saxagliptin/Metformin XR Relative to Co-Administration of the Individual Components in two cohorts of Healthy Chinese Subjects under Fed Conditions

Conditions

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Type 2 Diabetes Mellitus(T2DM)

Keywords

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Type 2 diabetes, Saxagliptin, Metformin,Fixed dose combination tablet, Bioequivalence, pharmacokinetic, safety, tolerability

Study Design

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Allocation Method

RANDOMIZED

Intervention Model

CROSSOVER

Primary Study Purpose

BASIC_SCIENCE

Blinding Strategy

NONE

Study Groups

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Lower dose

co-administration of a single oral dose of a 5 mg saxagliptin tablet and a 500 mg metformin XR (Glucophage XR®) tablet vs. single FDC tablet consisting of 5 mg saxagliptin and 500 mg metformin XR (Kombiglyze XR)

Group Type EXPERIMENTAL

Saxagliptin 5 mg

Intervention Type DRUG

Saxagliptin oral tablet 5mg, single dose

Metformin XR 500 mg

Intervention Type DRUG

Metformin XR oral tablet 500 mg, single dose

Komboglyze XR 5/500 mg

Intervention Type DRUG

oral FDC tablet (saxagliptin 5 mg and metformin 500 mg), single dose

Higher dose

co-administration of a single oral dose of a 5 mg saxagliptin tablet and two (2) 500 mg metformin XR (Glucophage XR®) tablets vs. Single FDC tablet consisting of 5 mg saxagliptin and 1000 mg metformin XR (Kombiglyze XR)

Group Type EXPERIMENTAL

Saxagliptin 5 mg

Intervention Type DRUG

Saxagliptin oral tablet 5mg, single dose

Mertformin XR 2 x 500 mg

Intervention Type DRUG

Metformin XR oral tablet 2 x 500 mg, single dose

Komboglyze XR 5/1000 mg

Intervention Type DRUG

oral FDC tablet (saxagliptin 5 mg and metformin 1000 mg), single dose

Interventions

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Saxagliptin 5 mg

Saxagliptin oral tablet 5mg, single dose

Intervention Type DRUG

Metformin XR 500 mg

Metformin XR oral tablet 500 mg, single dose

Intervention Type DRUG

Mertformin XR 2 x 500 mg

Metformin XR oral tablet 2 x 500 mg, single dose

Intervention Type DRUG

Komboglyze XR 5/500 mg

oral FDC tablet (saxagliptin 5 mg and metformin 500 mg), single dose

Intervention Type DRUG

Komboglyze XR 5/1000 mg

oral FDC tablet (saxagliptin 5 mg and metformin 1000 mg), single dose

Intervention Type DRUG

Eligibility Criteria

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Inclusion Criteria

* Chinese ethnicity which is defined as having both parents and 4 grandparents who are Chinese
* Healthy male subjects as determined by no clinically significant deviation from normal in medical history, physical examination, ECGs, and clinical laboratory determinations
* Men, ages 18 to 40 years, inclusive. The age difference among the subjects is within 10 years
* Weigh at least 50 kg and have a body mass index (BMI) between 19 and 24 kg/m2
* Sexually active fertile men must use effective birth control throughout the study and for up to 90 days after the last dose of investigational product if their partners are women of child bearing potential

Exclusion Criteria

* Any significant acute or chronic medical illness
* Current or recent gastrointestinal disease
* Subjects that have lymphocytopenia or thrombocytopenia
* History of autoimmune skin disorder
* Estimatedcreatinine clearance of less than 80 mL/min
Minimum Eligible Age

18 Years

Maximum Eligible Age

40 Years

Eligible Sex

MALE

Accepts Healthy Volunteers

Yes

Sponsors

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Bristol-Myers Squibb

INDUSTRY

Sponsor Role collaborator

AstraZeneca

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Principal Investigators

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Boaz Hirshberg

Role: STUDY_DIRECTOR

Room No.: C3C-718, 1800 Concord Pike, PO Box 15437, Wilmington DE 19850-5437, USA

Haiyan Li

Role: PRINCIPAL_INVESTIGATOR

Peking University Third Hospital (PU3), 49 North Garden Road, Haidian District, Beijing 100191, PR. China

Locations

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Research Site

Beijing, , China

Site Status

Countries

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China

Related Links

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Other Identifiers

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D1681C00001

Identifier Type: -

Identifier Source: org_study_id