Bioequivalence Study of 2.5-mg Saxagliptin and 500-mg Glucophage in Tablets and a Fixed-dose Combination Tablet in Healthy Participants

NCT ID: NCT01068717

Last Updated: 2015-05-12

Study Results

Results available

Outcome measurements, participant flow, baseline characteristics, and adverse events have been published for this study.

View full results

Basic Information

Get a concise snapshot of the trial, including recruitment status, study phase, enrollment targets, and key timeline milestones.

Recruitment Status

COMPLETED

Clinical Phase

PHASE1

Total Enrollment

27 participants

Study Classification

INTERVENTIONAL

Study Start Date

2010-03-31

Study Completion Date

2010-03-31

Brief Summary

Review the sponsor-provided synopsis that highlights what the study is about and why it is being conducted.

To demonstrate the bioequivalence of a 2.5-mg saxagliptin/500-mg metformin fixed-dose combination (FDC) tablet to that of 2.5-mg saxagliptin (Onglyza) and 500-mg metformin (Glucophage, marketed in Canada by Sanofi-Aventis) tablets coadministered to healthy participants in the fasted and fed states.

Detailed Description

Dive into the extended narrative that explains the scientific background, objectives, and procedures in greater depth.

Conditions

See the medical conditions and disease areas that this research is targeting or investigating.

Type 2 Diabetes Mellitus

Study Design

Understand how the trial is structured, including allocation methods, masking strategies, primary purpose, and other design elements.

Allocation Method

RANDOMIZED

Intervention Model

CROSSOVER

Blinding Strategy

NONE

Study Groups

Review each arm or cohort in the study, along with the interventions and objectives associated with them.

Saxagliptin, 2.5 mg + Metformin, 500 mg (fasted state)

Single oral doses of saxagliptin, 2.5 mg, and metformin, 500 mg, administered together as tablets in the fasted state

Group Type OTHER

Saxagliptin, 2.5 mg + Metformin, 500 mg (fasted state)

Intervention Type DRUG

Tablets, oral, 2.5-mg saxagliptin and 500-mg metformin, once daily, 1 week

Saxagliptin, 2.5 mg/Metformin, 500 mg FDC (fasted state)

Single oral dose of a 2.5-mg saxagliptin/500-mg metformin fixed-dose combination (FDC) tablet administered in the fasted state

Group Type OTHER

Saxagliptin, 2.5 mg /Metformin, 500 mg FDC (fasted state)

Intervention Type DRUG

Tablets, oral, 2.5-mg saxagliptin/500-mg metformin fixed-dose combination (FDC), once daily, 1 week

Saxagliptin, 2.5 mg + Metformin, 500 mg (fed state)

Single oral doses of saxagliptin, 2.5 mg, and metformin, 500 mg, administered together as tablets in the fed state

Group Type OTHER

Saxagliptin, 2.5 mg + Metformin, 500 mg (fed state)

Intervention Type DRUG

Tablets, oral, 2.5-mg saxagliptin and 500-mg metformin, once daily, 1 week

Saxagliptin, 2.5 mg/Metformin, 500 mg FDC (fed state)

Single oral dose of saxagliptin, 2.5 mg/metformin, 500 mg, FDC tablet administered in the fed state

Group Type OTHER

Saxagliptin, 2.5 mg /Metformin, 500 mg FDC (fed state)

Intervention Type DRUG

Tablets, oral, 2.5-mg saxagliptin and 500-mg metformin FDC, once daily, 1 week

Interventions

Learn about the drugs, procedures, or behavioral strategies being tested and how they are applied within this trial.

Saxagliptin, 2.5 mg + Metformin, 500 mg (fasted state)

Tablets, oral, 2.5-mg saxagliptin and 500-mg metformin, once daily, 1 week

Intervention Type DRUG

Saxagliptin, 2.5 mg /Metformin, 500 mg FDC (fasted state)

Tablets, oral, 2.5-mg saxagliptin/500-mg metformin fixed-dose combination (FDC), once daily, 1 week

Intervention Type DRUG

Saxagliptin, 2.5 mg + Metformin, 500 mg (fed state)

Tablets, oral, 2.5-mg saxagliptin and 500-mg metformin, once daily, 1 week

Intervention Type DRUG

Saxagliptin, 2.5 mg /Metformin, 500 mg FDC (fed state)

Tablets, oral, 2.5-mg saxagliptin and 500-mg metformin FDC, once daily, 1 week

Intervention Type DRUG

Other Intervention Names

Discover alternative or legacy names that may be used to describe the listed interventions across different sources.

Onglyza™ Glucophage™ Onglyza™ Glucophage™

Eligibility Criteria

Check the participation requirements, including inclusion and exclusion rules, age limits, and whether healthy volunteers are accepted.

Inclusion Criteria

* Men and women, aged 18 to 55 years, inclusive
* Healthy participants as determined by a lack of clinically significant deviation from normal in medical history, physical examination, electrocardiograms, and clinical laboratory determinations
* Body Mass Index of 18 to 32 kg/m\^2, inclusive

Exclusion Criteria

* Any significant acute or chronic medical illness
* Current or recent (within 3 months) gastrointestinal disease
* Any major surgery within 4 weeks of study drug administration
* History of allergy to DPP-4 inhibitors or related compounds
* History of allergy or intolerance to metformin or other similar acting agents
* Previous exposure to saxagliptin
* Exposure to metformin within 3 months pervious to study drug administration
* Estimated creatinine clearance of \<80 mL/min using the Cockcroft Gault formula
Minimum Eligible Age

18 Years

Maximum Eligible Age

55 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

Yes

Sponsors

Meet the organizations funding or collaborating on the study and learn about their roles.

AstraZeneca

INDUSTRY

Sponsor Role lead

Responsible Party

Identify the individual or organization who holds primary responsibility for the study information submitted to regulators.

Responsibility Role SPONSOR

Principal Investigators

Learn about the lead researchers overseeing the trial and their institutional affiliations.

Bristol-Myers Squibb

Role: STUDY_DIRECTOR

Bristol-Myers Squibb

Locations

Explore where the study is taking place and check the recruitment status at each participating site.

Ppd Development, Lp

Austin, Texas, United States

Site Status

Countries

Review the countries where the study has at least one active or historical site.

United States

Related Links

Access external resources that provide additional context or updates about the study.

Other Identifiers

Review additional registry numbers or institutional identifiers associated with this trial.

CV181-118

Identifier Type: -

Identifier Source: org_study_id

More Related Trials

Additional clinical trials that may be relevant based on similarity analysis.

Bioequivalence Study
NCT01874080 COMPLETED PHASE1