Trial Outcomes & Findings for Open-Label Lesinurad Monotherapy Extension Study in Gout (NCT NCT01650246)

NCT ID: NCT01650246

Last Updated: 2016-05-26

Results Overview

Recruitment status

COMPLETED

Study phase

PHASE3

Target enrollment

143 participants

Primary outcome timeframe

Month 1

Results posted on

2016-05-26

Participant Flow

Participant milestones

Participant milestones
Measure
Lesinurad 400 mg
lesinurad 400 mg once daily (qd)
Overall Study
STARTED
143
Overall Study
COMPLETED
0
Overall Study
NOT COMPLETED
143

Reasons for withdrawal

Reasons for withdrawal
Measure
Lesinurad 400 mg
lesinurad 400 mg once daily (qd)
Overall Study
Adverse Event
23
Overall Study
Protocol Violation
5
Overall Study
Sponsor terminated study
53
Overall Study
Lost to Follow-up
5
Overall Study
Withdrawal by Subject
26
Overall Study
Death
1
Overall Study
Lack of Efficacy
30

Baseline Characteristics

Open-Label Lesinurad Monotherapy Extension Study in Gout

Baseline characteristics by cohort

Baseline characteristics by cohort
Measure
Lesinurad 400 mg
n=143 Participants
lesinurad 400 mg once daily (qd)
Age, Continuous
55.1 years
STANDARD_DEVIATION 12.0 • n=93 Participants
Age, Customized
<65 Years
111 Participants
n=93 Participants
Age, Customized
>=65 Years
32 Participants
n=93 Participants
Sex: Female, Male
Female
11 Participants
n=93 Participants
Sex: Female, Male
Male
132 Participants
n=93 Participants
Region of Enrollment
Australia
2 Participants
n=93 Participants
Region of Enrollment
Belgium
9 Participants
n=93 Participants
Region of Enrollment
Canada
6 Participants
n=93 Participants
Region of Enrollment
Germany
6 Participants
n=93 Participants
Region of Enrollment
New Zealand
3 Participants
n=93 Participants
Region of Enrollment
South Africa
16 Participants
n=93 Participants
Region of Enrollment
United States
101 Participants
n=93 Participants

PRIMARY outcome

Timeframe: Month 1

Population: Safety Population

Outcome measures

Outcome measures
Measure
Lesinurad 400 mg
n=143 Participants
lesinurad 400 mg once daily (qd)
Proportion of Subjects With a Serum Urate (sUA) Level That is < 6.0 mg/dL
68 Subjects

PRIMARY outcome

Timeframe: Up to approximately 2 years

Population: Safety Population

Outcome measures

Outcome measures
Measure
Lesinurad 400 mg
n=143 Participants
lesinurad 400 mg once daily (qd)
Incidence of Treatment-emergent Adverse Events (TEAEs)
105 TEAEs

Adverse Events

Lesinurad 400 mg

Serious events: 15 serious events
Other events: 73 other events
Deaths: 0 deaths

Serious adverse events

Serious adverse events
Measure
Lesinurad 400 mg
n=143 participants at risk
lesinurad 400 mg once daily (qd)
Gastrointestinal disorders
Pancreatitis
0.70%
1/143 • Number of events 1
General disorders
Death
0.70%
1/143 • Number of events 1
Infections and infestations
Bursitis infective
0.70%
1/143 • Number of events 1
Infections and infestations
Gastroenteritis salmonella
0.70%
1/143 • Number of events 1
Metabolism and nutrition disorders
Gout
0.70%
1/143 • Number of events 1
Musculoskeletal and connective tissue disorders
Facet joint syndrome
0.70%
1/143 • Number of events 1
Nervous system disorders
Transient ischaemic attack
0.70%
1/143 • Number of events 1
Renal and urinary disorders
Nephrolithiasis
2.1%
3/143 • Number of events 3
Renal and urinary disorders
Renal impairment
0.70%
1/143 • Number of events 1
Renal and urinary disorders
Renal Failure Acute
0.70%
1/143 • Number of events 1
Psychiatric disorders
Depression
0.70%
1/143 • Number of events 1
Psychiatric disorders
Schizoaffective disorder
0.70%
1/143 • Number of events 2
Cardiac disorders
Angina pectoris
0.70%
1/143 • Number of events 1
Cardiac disorders
Atrioventricular clock complete
0.70%
1/143 • Number of events 1
Cardiac disorders
Coronary Artery disease
0.70%
1/143 • Number of events 1
Cardiac disorders
Myocardial infarction
0.70%
1/143 • Number of events 1

Other adverse events

Other adverse events
Measure
Lesinurad 400 mg
n=143 participants at risk
lesinurad 400 mg once daily (qd)
Gastrointestinal disorders
Abdominal pain upper
2.1%
3/143 • Number of events 3
Gastrointestinal disorders
Gastrooesophageal reflux disease
2.1%
3/143 • Number of events 3
Gastrointestinal disorders
Vomiting
2.8%
4/143 • Number of events 7
General disorders
Fatigue
2.8%
4/143 • Number of events 4
General disorders
Pyrexia
2.1%
3/143 • Number of events 3
Infections and infestations
Bronchitis
3.5%
5/143 • Number of events 5
Infections and infestations
Gastroenteritis
4.9%
7/143 • Number of events 8
Infections and infestations
Influenza
2.1%
3/143 • Number of events 3
Infections and infestations
Sinusitis
2.8%
4/143 • Number of events 5
Infections and infestations
Upper respiratory tract infection
9.8%
14/143 • Number of events 15
Infections and infestations
Urinary tract infection
4.9%
7/143 • Number of events 8
Investigations
Blood creatine phosphokinase increased
2.8%
4/143 • Number of events 4
Investigations
Blood creatinine increased
11.2%
16/143 • Number of events 20
Metabolism and nutrition disorders
Hyperlipidaemia
2.1%
3/143 • Number of events 3
Musculoskeletal and connective tissue disorders
Arthralgia
4.2%
6/143 • Number of events 6
Musculoskeletal and connective tissue disorders
Back pain
4.9%
7/143 • Number of events 8
Musculoskeletal and connective tissue disorders
Flank pain
2.1%
3/143 • Number of events 4
Musculoskeletal and connective tissue disorders
Pain in extremity
2.1%
3/143 • Number of events 4
Nervous system disorders
Headache
4.2%
6/143 • Number of events 8
Renal and urinary disorders
Nephrolithiasis
2.1%
3/143 • Number of events 3
Renal and urinary disorders
Renal impairment
2.8%
4/143 • Number of events 4
Respiratory, thoracic and mediastinal disorders
Cough
2.8%
4/143 • Number of events 5
Vascular disorders
Hypertension
7.0%
10/143 • Number of events 10
Infections and infestations
Nasopharyngitis
2.8%
4/143 • Number of events 5

Additional Information

Maple Fung, MD

Ardea Biosciences, Inc.

Phone: 1-858-652-6721

Results disclosure agreements

  • Principal investigator is a sponsor employee Principal Investigator (PI) shall submit a copy of the Publication to Sponsor for review at least 45 days prior to its proposed submission. Sponsor reserves the right to delay any such publication for an additional period of 60 days. Upon Sponsor's request, PI agrees to delete from the proposed publication any Confidential Information. PI agrees not to release any publication without the prior written permission of Sponsor.
  • Publication restrictions are in place

Restriction type: OTHER