A Study to Evaluate the Efficacy and Safety of ALKS 9072 (Also Known as Aripiprazole Lauroxil, ALKS 9070, or ARISTADA) in Subjects With Schizophrenia

NCT ID: NCT01469039

Last Updated: 2019-01-30

Study Results

Results available

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Basic Information

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Recruitment Status

COMPLETED

Clinical Phase

PHASE3

Total Enrollment

623 participants

Study Classification

INTERVENTIONAL

Study Start Date

2011-12-31

Study Completion Date

2014-03-31

Brief Summary

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The study will determine the efficacy of ALKS 9072 (also known as aripiprazole lauroxil or ALKS 9070) for the treatment of schizophrenia in subjects experiencing an acute exacerbation.

Detailed Description

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Conditions

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Schizophrenia

Study Design

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Allocation Method

RANDOMIZED

Intervention Model

PARALLEL

Primary Study Purpose

TREATMENT

Blinding Strategy

QUADRUPLE

Participants Caregivers Investigators Outcome Assessors

Study Groups

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ALKS 9072

Group Type EXPERIMENTAL

ALKS 9072

Intervention Type DRUG

Intramuscular (IM) injection, 441 mg or 882 mg given monthly

Placebo

Group Type PLACEBO_COMPARATOR

Placebo

Intervention Type DRUG

Placebo for IM injection, given monthly

Interventions

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ALKS 9072

Intramuscular (IM) injection, 441 mg or 882 mg given monthly

Intervention Type DRUG

Placebo

Placebo for IM injection, given monthly

Intervention Type DRUG

Eligibility Criteria

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Inclusion Criteria

* Diagnosis of schizophrenia according to DSM-IV-TR criteria
* Has been able to achieve outpatient status for more than 3 months in the past year
* Body mass index (BMI) of 18.5 to 40.0 kg/m2 (inclusive)
* Resides in a stable living situation
* Willing and able to be confined to an inpatient study unit for 2 weeks or longer

Exclusion Criteria

* History of poor or inadequate clinical response to treatment with aripiprazole
* History of treatment resistance
* Known or suspected intolerance of, allergy, or hypersensitivity to aripiprazole, its ingredients, other antipsychotic agent, or INTRALIPID (including peanuts, soy, egg, or glycerol)
* Diagnosis of current substance dependence (including alcohol)
* Pregnant, lactating, or breastfeeding
* Receipt of any antipsychotic medication by IM injection within 60 days before Screening
* Current involuntary hospitalization or incarceration
* Hospitalized for more than 30 days during the 90 days before Screening
Minimum Eligible Age

18 Years

Maximum Eligible Age

70 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

No

Sponsors

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Alkermes, Inc.

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Principal Investigators

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Alkermes Medical Director

Role: STUDY_DIRECTOR

Alkermes, Inc.

Locations

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Alkermes Investigational Site

Little Rock, Arkansas, United States

Site Status

Alkermes Investigational Site

Little Rock, Arkansas, United States

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Alkermes Investigational Site

Springdale, Arkansas, United States

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Cerritos, California, United States

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Alkermes Investigational Site

Garden Grove, California, United States

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Alkermes Investigational Site

La Habra, California, United States

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Alkermes Investigational Site

Oakland, California, United States

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Alkermes Investigational Site

Oceanside, California, United States

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Alkermes Investigational Site

Orange, California, United States

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San Diego, California, United States

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Alkermes Investigational Site

Washington D.C., District of Columbia, United States

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Alkermes Investigational Site

Fort Lauderdale, Florida, United States

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Alkermes Investigational site

Leesburg, Florida, United States

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Alkermes Investigational Site

Atlanta, Georgia, United States

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Alkermes Investigational Site

Chicago, Illinois, United States

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Alkermes Investigational Site

Hoffman Estates, Illinois, United States

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Overland Park, Kansas, United States

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Rockville, Maryland, United States

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Creve Coeur, Missouri, United States

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St Louis, Missouri, United States

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Philadelphia, Pennsylvania, United States

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Charleston, South Carolina, United States

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Austin, Texas, United States

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Austin, Texas, United States

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Alkermes Investigational Site

Dallas, Texas, United States

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Dallas, Texas, United States

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Alkermes Investigational Site

Burgas, , Bulgaria

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Alkermes Investigational Site

Kazanlak, , Bulgaria

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Alkermes Investigational Site

Novi Iskar, , Bulgaria

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Pazardzhik, , Bulgaria

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Pleven, , Bulgaria

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Plovdiv, , Bulgaria

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Radnevo, , Bulgaria

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Rousse, , Bulgaria

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Sofia, , Bulgaria

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Stara Zagora, , Bulgaria

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Targovishte, , Bulgaria

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Veliko Tarnovo, , Bulgaria

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Vratsa, , Bulgaria

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Cheras, , Malaysia

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Johor Bahru, , Malaysia

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Kuala Lumpur, , Malaysia

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Kuching, , Malaysia

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Mariveles, Bataan, Philippines

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Cebu City, , Philippines

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Iloilo City, , Philippines

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Mandaluyong, , Philippines

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Manila, , Philippines

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Pasig, , Philippines

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Oradea, Bihor County, Romania

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Bucharest, , Romania

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Alkermes Investigational Site

Bucharest, , Romania

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Craiova, , Romania

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Iași, , Romania

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Alkermes Investigational Site

Târgu Mureş, , Romania

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Alkermes Investigational Site

Nikol’skoye, Gatchinckiy, Russia

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Alkermes Investigational Site

Staritsa, Orenburg Oblast, Russia

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Alkermes Investigational Site

Talagi, Primorskiy (Maritime) Kray, Russia

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Alkermes Investigational Site

Khot'kovo, Sergievo-Posadskiy, Russia

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Alkermes Investigational Site

Lipetsk, , Russia

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Alkermes Investigational Site

Moscow, , Russia

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Alkermes Investigational Site

Nizhny Novgorod, , Russia

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Alkermes Investigational Site

Rostov-on-Don, , Russia

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Saint Petersburg, , Russia

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Samara, , Russia

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Saratov, , Russia

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Stavropol, , Russia

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Voronezh, , Russia

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Yaroslavl, , Russia

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Alkermes Investigational Site

Jeju City, , South Korea

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Alkermes Investigational Site

Jeollanam-do, , South Korea

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Alkermes Investigational Site

Seoul, , South Korea

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Alkermes Investigational Site

Stepanivka, Kherson Oblast, Ukraine

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Alkermes Investigational Site

Chernihiv, , Ukraine

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Alkermes Investigational Site

Donetsk, , Ukraine

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Alkermes Investigational Site

Kharkiv, , Ukraine

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Kyiv, , Ukraine

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Luhansk, , Ukraine

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Lviv, , Ukraine

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Poltava, , Ukraine

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Simferopol, , Ukraine

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Alkermes Investigational Site

Ternopil, , Ukraine

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Alkermes Investigational Site

Uzhhorod, , Ukraine

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Alkermes Investigational Site

Vinnytsia, , Ukraine

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Countries

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United States Bulgaria Malaysia Philippines Romania Russia South Korea Ukraine

References

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Targum SD, Risinger R, Du Y, Pendergrass JC, Jamal HH, Silverman BL. Effect of patient age on treatment response in a study of the acute exacerbation of psychosis in schizophrenia. Schizophr Res. 2017 Jan;179:64-69. doi: 10.1016/j.schres.2016.09.034. Epub 2016 Oct 1.

Reference Type RESULT
PMID: 27707530 (View on PubMed)

Nasrallah HA, Newcomer JW, Risinger R, Du Y, Zummo J, Bose A, Stankovic S, Silverman BL, Ehrich EW. Effect of Aripiprazole Lauroxil on Metabolic and Endocrine Profiles and Related Safety Considerations Among Patients With Acute Schizophrenia. J Clin Psychiatry. 2016 Nov;77(11):1519-1525. doi: 10.4088/JCP.15m10467.

Reference Type RESULT
PMID: 27574838 (View on PubMed)

Citrome L, Du Y, Risinger R, Stankovic S, Claxton A, Zummo J, Bose A, Silverman BL, Ehrich EW. Effect of aripiprazole lauroxil on agitation and hostility in patients with schizophrenia. Int Clin Psychopharmacol. 2016 Mar;31(2):69-75. doi: 10.1097/YIC.0000000000000106.

Reference Type RESULT
PMID: 26517202 (View on PubMed)

Meltzer HY, Risinger R, Nasrallah HA, Du Y, Zummo J, Corey L, Bose A, Stankovic S, Silverman BL, Ehrich EW. A randomized, double-blind, placebo-controlled trial of aripiprazole lauroxil in acute exacerbation of schizophrenia. J Clin Psychiatry. 2015 Aug;76(8):1085-90. doi: 10.4088/JCP.14m09741.

Reference Type RESULT
PMID: 26114240 (View on PubMed)

Potkin SG, Risinger R, Du Y, Zummo J, Bose A, Silverman B, Stankovic S, Ehrich E. Efficacy and safety of aripiprazole lauroxil in schizophrenic patients presenting with severe psychotic symptoms during an acute exacerbation. Schizophr Res. 2017 Dec;190:115-120. doi: 10.1016/j.schres.2017.03.003. Epub 2017 Mar 23.

Reference Type RESULT
PMID: 28342578 (View on PubMed)

Cameron C, Zummo J, Desai DN, Drake C, Hutton B, Kotb A, Weiden PJ. Aripiprazole Lauroxil Compared with Paliperidone Palmitate in Patients with Schizophrenia: An Indirect Treatment Comparison. Value Health. 2017 Jul-Aug;20(7):876-885. doi: 10.1016/j.jval.2017.03.010. Epub 2017 May 9.

Reference Type RESULT
PMID: 28712616 (View on PubMed)

Citrome L, Risinger R, Cutler AJ, Du Y, Zummo J, Nasrallah HA, Silverman BL. Effect of aripiprazole lauroxil in patients with acute schizophrenia as assessed by the Positive and Negative Syndrome Scale-supportive analyses from a Phase 3 study. CNS Spectr. 2018 Aug;23(4):284-290. doi: 10.1017/S1092852917000396. Epub 2017 Jun 19.

Reference Type RESULT
PMID: 28625204 (View on PubMed)

Hard ML, Mills RJ, Sadler BM, Turncliff RZ, Citrome L. Aripiprazole Lauroxil: Pharmacokinetic Profile of This Long-Acting Injectable Antipsychotic in Persons With Schizophrenia. J Clin Psychopharmacol. 2017 Jun;37(3):289-295. doi: 10.1097/JCP.0000000000000691.

Reference Type RESULT
PMID: 28350572 (View on PubMed)

Cameron C, Zummo J, Desai D, Drake C, Hutton B, Kotb A, Weiden PJ. Efficacy and safety of aripiprazole lauroxil once-monthly versus aripiprazole once-monthly long-acting injectable formulations in patients with acute symptoms of schizophrenia: an indirect comparison of two double-blind placebo-controlled studies. Curr Med Res Opin. 2018 Apr;34(4):725-733. doi: 10.1080/03007995.2017.1410471. Epub 2018 Jan 10.

Reference Type RESULT
PMID: 29179595 (View on PubMed)

Sommi RW, Saklad SR, Weiden PJ, Still D, Wang M, Yagoda S. Initiating Aripiprazole Lauroxil: Post Hoc Analysis of Safety and Tolerability of 1-Day and 21-Day Regimens. J Clin Psychiatry. 2024 Aug 12;85(3):23m15132. doi: 10.4088/JCP.23m15132.

Reference Type DERIVED
PMID: 39145678 (View on PubMed)

McEvoy JP, Risinger R, Mykhnyak S, Du Y, Liu CC, Stanford AD, Weiden PJ. Durability of Therapeutic Response With Long-Term Aripiprazole Lauroxil Treatment Following Successful Resolution of an Acute Episode of Schizophrenia. J Clin Psychiatry. 2017 Sep-Oct;78(8):1103-1109. doi: 10.4088/JCP.17m11625.

Reference Type DERIVED
PMID: 28937706 (View on PubMed)

Related Links

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http://grls.rosminzdrav.ru

Russian clinical trials website

http://www.clinicaltrialsregister.eu

EU Clinical Trials Register; EudraCT number 2012-003445-15

Other Identifiers

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ALK9072-003

Identifier Type: -

Identifier Source: org_study_id

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