Pharmacodynamics, Pharmacokinetics, Safety and Tolerability of Ultra Low Doses of Dapagliflozin in Healthy Subjects

NCT ID: NCT01135446

Last Updated: 2016-10-17

Study Results

Results pending

The study team has not published outcome measurements, participant flow, or safety data for this trial yet. Check back later for updates.

Basic Information

Get a concise snapshot of the trial, including recruitment status, study phase, enrollment targets, and key timeline milestones.

Recruitment Status

COMPLETED

Clinical Phase

PHASE1

Total Enrollment

35 participants

Study Classification

INTERVENTIONAL

Study Start Date

2010-05-31

Study Completion Date

2010-06-30

Brief Summary

Review the sponsor-provided synopsis that highlights what the study is about and why it is being conducted.

The purpose of this study is to evaluate the pharmacodynamics (PD), pharmacokinetics (PK), safety and tolerability following single oral doses of 0.001 mg to 2.5 mg dapagliflozin in healthy subjects.

Detailed Description

Dive into the extended narrative that explains the scientific background, objectives, and procedures in greater depth.

Conditions

See the medical conditions and disease areas that this research is targeting or investigating.

Type 2 Diabetes

Study Design

Understand how the trial is structured, including allocation methods, masking strategies, primary purpose, and other design elements.

Allocation Method

RANDOMIZED

Intervention Model

PARALLEL

Blinding Strategy

NONE

Study Groups

Review each arm or cohort in the study, along with the interventions and objectives associated with them.

dapagliflozin (0.001 mg)

Cohort 1

Group Type EXPERIMENTAL

dapagliflozin

Intervention Type DRUG

Oral Solution, Oral, 0.001 mg, once on Day 1 only, 2 days

dapagliflozin (0.01 mg)

Cohort 2

Group Type EXPERIMENTAL

dapagliflozin

Intervention Type DRUG

Oral Solution, Oral, 0.01 mg, once on Day 1 only, 2 days

dapagliflozin (0.1 mg)

Cohort 3

Group Type EXPERIMENTAL

dapagliflozin

Intervention Type DRUG

Oral Solution, Oral, 0.1 mg, once on Day 1 only, 2 days

dapagliflozin (0.3 mg)

Cohort 4

Group Type EXPERIMENTAL

dapagliflozin

Intervention Type DRUG

Tablets, Oral, 0.3 mg, once on Day 1 only, 2 days

dapagliflozin (1 mg)

Cohort 5

Group Type EXPERIMENTAL

dapagliflozin

Intervention Type DRUG

Tablets, Oral, 1 mg, once on Day 1 only, 2 days

dapagliflozin (2.5 mg)

Cohort 6

Group Type EXPERIMENTAL

dapagliflozin

Intervention Type DRUG

Tablets, Oral, 2.5 mg, once on Day 1 only, 2 days

Interventions

Learn about the drugs, procedures, or behavioral strategies being tested and how they are applied within this trial.

dapagliflozin

Oral Solution, Oral, 0.001 mg, once on Day 1 only, 2 days

Intervention Type DRUG

dapagliflozin

Oral Solution, Oral, 0.01 mg, once on Day 1 only, 2 days

Intervention Type DRUG

dapagliflozin

Oral Solution, Oral, 0.1 mg, once on Day 1 only, 2 days

Intervention Type DRUG

dapagliflozin

Tablets, Oral, 0.3 mg, once on Day 1 only, 2 days

Intervention Type DRUG

dapagliflozin

Tablets, Oral, 1 mg, once on Day 1 only, 2 days

Intervention Type DRUG

dapagliflozin

Tablets, Oral, 2.5 mg, once on Day 1 only, 2 days

Intervention Type DRUG

Other Intervention Names

Discover alternative or legacy names that may be used to describe the listed interventions across different sources.

BMS-512148 BMS-512148 BMS-512148 BMS-512148 BMS-512148 BMS-512148

Eligibility Criteria

Check the participation requirements, including inclusion and exclusion rules, age limits, and whether healthy volunteers are accepted.

Inclusion Criteria

* Healthy men and women
* WOCBP who are using acceptable method of contraception
* Women who are not nursing

Exclusion Criteria

* History of GI disease
* Any GI surgery that could impact study drug absorption
* Glucosuria at screening or Day -2
* Abnormal liver function tests (ALT, AST or total bilirubin \> 10% above ULN)
* History of current or recurrent UTI
* History of Diabetes Mellitus
* History of chronic or recurrent vulvovaginal mycotic infections
* Estimated creatinine clearance (ClCr) \< 80 mL/min using Cockroft-Gault formula
* History of allergy to SGLT2 inhibitors or related compounds
Minimum Eligible Age

18 Years

Maximum Eligible Age

55 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

Yes

Sponsors

Meet the organizations funding or collaborating on the study and learn about their roles.

Bristol-Myers Squibb

INDUSTRY

Sponsor Role collaborator

AstraZeneca

INDUSTRY

Sponsor Role lead

Responsible Party

Identify the individual or organization who holds primary responsibility for the study information submitted to regulators.

Responsibility Role SPONSOR

Principal Investigators

Learn about the lead researchers overseeing the trial and their institutional affiliations.

Bristol-Myers Squibb

Role: STUDY_DIRECTOR

Bristol-Myers Squibb

Locations

Explore where the study is taking place and check the recruitment status at each participating site.

Ppd Development, Lp

Austin, Texas, United States

Site Status

Countries

Review the countries where the study has at least one active or historical site.

United States

Related Links

Access external resources that provide additional context or updates about the study.

Other Identifiers

Review additional registry numbers or institutional identifiers associated with this trial.

MB102-088

Identifier Type: -

Identifier Source: org_study_id

More Related Trials

Additional clinical trials that may be relevant based on similarity analysis.

A Phase 2b Diabetic Kidney Disease Study
NCT04170543 COMPLETED PHASE2
OPTIMISE-CKD Drug Utilization
NCT05932901 COMPLETED