A Pharmacokinetic/Pharmacodynamic Study of RO5185426 in Previously Treated Patients With Metastatic Melanoma

NCT ID: NCT01107418

Last Updated: 2015-08-26

Study Results

Results available

Outcome measurements, participant flow, baseline characteristics, and adverse events have been published for this study.

View full results

Basic Information

Get a concise snapshot of the trial, including recruitment status, study phase, enrollment targets, and key timeline milestones.

Recruitment Status

COMPLETED

Clinical Phase

PHASE1

Total Enrollment

52 participants

Study Classification

INTERVENTIONAL

Study Start Date

2010-05-31

Study Completion Date

2013-02-28

Brief Summary

Review the sponsor-provided synopsis that highlights what the study is about and why it is being conducted.

This open-label study will assess the pharmacokinetics, efficacy and safety of RO5185426 administered as 240mg tablets in previously treated patients with metastatic melanoma. Patients will be randomized to receive one of four dose-levels of RO5185426 \[RG7204; PLEXXIKON; PLX4032\] orally twice daily on days 1 to 15 (morning dose). Starting on day 22, treatment with RO5185426 may be resumed at a dose of 960 mg twice daily and continued until disease progression. Target sample size is \<100 patients.

Detailed Description

Dive into the extended narrative that explains the scientific background, objectives, and procedures in greater depth.

Conditions

See the medical conditions and disease areas that this research is targeting or investigating.

Malignant Melanoma

Study Design

Understand how the trial is structured, including allocation methods, masking strategies, primary purpose, and other design elements.

Allocation Method

NON_RANDOMIZED

Intervention Model

PARALLEL

Primary Study Purpose

TREATMENT

Blinding Strategy

NONE

Study Groups

Review each arm or cohort in the study, along with the interventions and objectives associated with them.

1

Group Type EXPERIMENTAL

RO5185426

Intervention Type DRUG

960 mg orally twice daily, from day 22 onward

RO5185426

Intervention Type DRUG

dosage a) orally twice daily, days 1-15 (morning dose)

2

Group Type EXPERIMENTAL

RO5185426

Intervention Type DRUG

dosage b) orally twice daily, days 1-15 (morning dose)

RO5185426

Intervention Type DRUG

960 mg orally twice daily, from day 22 onward

3

Group Type EXPERIMENTAL

RO5185426

Intervention Type DRUG

dosage c) orally twice daily, days 1-15 (morning dose)

RO5185426

Intervention Type DRUG

960 mg orally twice daily, from day 22 onward

4

Group Type EXPERIMENTAL

RO5185426

Intervention Type DRUG

dosage d) orally twice daily, days 1-15 (morning dose)

RO5185426

Intervention Type DRUG

960 mg orally twice daily, from day 22 onward

Interventions

Learn about the drugs, procedures, or behavioral strategies being tested and how they are applied within this trial.

RO5185426

dosage b) orally twice daily, days 1-15 (morning dose)

Intervention Type DRUG

RO5185426

dosage c) orally twice daily, days 1-15 (morning dose)

Intervention Type DRUG

RO5185426

dosage d) orally twice daily, days 1-15 (morning dose)

Intervention Type DRUG

RO5185426

960 mg orally twice daily, from day 22 onward

Intervention Type DRUG

RO5185426

dosage a) orally twice daily, days 1-15 (morning dose)

Intervention Type DRUG

Eligibility Criteria

Check the participation requirements, including inclusion and exclusion rules, age limits, and whether healthy volunteers are accepted.

Inclusion Criteria

* adult patients, \>/=18 years of age
* histologically confirmed metastatic melanoma, stage IIIc or IV (AJCC)
* failure of at least one prior standard of care regimen
* positive for BRAF V600E mutation (by Roche CoDx BRAF mutation assay)
* ECOG performance status 0 or 1
* adequate hematologic, renal and liver function

Exclusion Criteria

* active CNS lesions on CT/MRI within 28 days prior to enrollment
* history of spinal cord compression o carcinomatous meningitis
* anticipated or ongoing anti-cancer therapies other than those administered in this study
* previous treatment with BRAF inhibitor (sorafenib allowed) or MEK inhibitor
* severe cardiovascular disease within 6 months prior to study
* previous malignancy within the past 5 years except for basal or squamous cell carcinoma of the skin, melanoma in-situ and carcinoma in-situ of the cervix
Minimum Eligible Age

18 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

No

Sponsors

Meet the organizations funding or collaborating on the study and learn about their roles.

Hoffmann-La Roche

INDUSTRY

Sponsor Role lead

Responsible Party

Identify the individual or organization who holds primary responsibility for the study information submitted to regulators.

Responsibility Role SPONSOR

Principal Investigators

Learn about the lead researchers overseeing the trial and their institutional affiliations.

Clinical Trials

Role: STUDY_DIRECTOR

Hoffmann-La Roche

Locations

Explore where the study is taking place and check the recruitment status at each participating site.

La Jolla, California, United States

Site Status

San Francisco, California, United States

Site Status

Stanford, California, United States

Site Status

New Haven, Connecticut, United States

Site Status

Chicago, Illinois, United States

Site Status

Park Ridge, Illinois, United States

Site Status

Sioux City, Iowa, United States

Site Status

Omaha, Nebraska, United States

Site Status

Columbus, Ohio, United States

Site Status

East Providence, Rhode Island, United States

Site Status

Charlottesville, Virginia, United States

Site Status

Adelaide, South Australia, Australia

Site Status

Melbourne, Victoria, Australia

Site Status

Countries

Review the countries where the study has at least one active or historical site.

United States Australia

References

Explore related publications, articles, or registry entries linked to this study.

Frederick DT, Salas Fragomeni RA, Schalck A, Ferreiro-Neira I, Hoff T, Cooper ZA, Haq R, Panka DJ, Kwong LN, Davies MA, Cusack JC, Flaherty KT, Fisher DE, Mier JW, Wargo JA, Sullivan RJ. Clinical profiling of BCL-2 family members in the setting of BRAF inhibition offers a rationale for targeting de novo resistance using BH3 mimetics. PLoS One. 2014 Jul 1;9(7):e101286. doi: 10.1371/journal.pone.0101286. eCollection 2014.

Reference Type DERIVED
PMID: 24983357 (View on PubMed)

Lacouture ME, Duvic M, Hauschild A, Prieto VG, Robert C, Schadendorf D, Kim CC, McCormack CJ, Myskowski PL, Spleiss O, Trunzer K, Su F, Nelson B, Nolop KB, Grippo JF, Lee RJ, Klimek MJ, Troy JL, Joe AK. Analysis of dermatologic events in vemurafenib-treated patients with melanoma. Oncologist. 2013;18(3):314-22. doi: 10.1634/theoncologist.2012-0333. Epub 2013 Mar 1.

Reference Type DERIVED
PMID: 23457002 (View on PubMed)

Other Identifiers

Review additional registry numbers or institutional identifiers associated with this trial.

NP25163

Identifier Type: -

Identifier Source: org_study_id

More Related Trials

Additional clinical trials that may be relevant based on similarity analysis.