Study Of Safety And Efficacy Of Ertugliflozin (PF-04971729, MK-8835) In Participants With Type 2 Diabetes (MK-8835-016)

NCT ID: NCT01059825

Last Updated: 2018-09-13

Study Results

Results available

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Basic Information

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Recruitment Status

COMPLETED

Clinical Phase

PHASE2

Total Enrollment

375 participants

Study Classification

INTERVENTIONAL

Study Start Date

2010-02-24

Study Completion Date

2011-01-20

Brief Summary

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MK-8835-016 (B1521006) is designed to evaluate the safety and efficacy of an investigational drug, ertugliflozin (MK-8835, PF-04971729) in participants with Type 2 diabetes mellitus. Participants in the study will receive 1 of 6 treatments for 12 weeks including 1 treatment with an approved drug (sitagliptin) for the treatment of Type 2 diabetes mellitus.

Detailed Description

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Conditions

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Diabetes Mellitus, Type 2

Study Design

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Allocation Method

RANDOMIZED

Intervention Model

PARALLEL

Primary Study Purpose

TREATMENT

Blinding Strategy

DOUBLE

Participants Investigators

Study Groups

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Placebo

Placebo for ertugliflozin (1 mg or 5 mg and 25 mg) and placebo to sitagliptin, oral, once daily for 84 days

Group Type PLACEBO_COMPARATOR

Placebo to Ertugliflozin

Intervention Type DRUG

Tablet(s), 1 or 2, matching placebo to 1-mg, 5-mg and/or 25-mg tablets, once daily for 84 days

Placebo to Sitagliptin

Intervention Type DRUG

Tablet, matching placebo to 100 mg, once daily for 84 days

Metformin

Intervention Type DRUG

Participants continued pre-study stable doses of metformin during the run-in and treatment periods of the study (maximum dose up to 2500 mg/day or 3000 mg/day where the maximum metformin dose per the local country product labels was 3000 mg/day).

Ertugliflozin 1 mg

Ertugliflozin 1 mg, placebo for ertugliflozin (1 mg or 5 mg and 25 mg), and placebo to sitagliptin, oral, once daily for 84 days

Group Type EXPERIMENTAL

Placebo to Ertugliflozin

Intervention Type DRUG

Tablet(s), 1 or 2, matching placebo to 1-mg, 5-mg and/or 25-mg tablets, once daily for 84 days

Ertugliflozin 1 mg

Intervention Type DRUG

Tablet, 1 mg, once daily for 84 days

Placebo to Sitagliptin

Intervention Type DRUG

Tablet, matching placebo to 100 mg, once daily for 84 days

Metformin

Intervention Type DRUG

Participants continued pre-study stable doses of metformin during the run-in and treatment periods of the study (maximum dose up to 2500 mg/day or 3000 mg/day where the maximum metformin dose per the local country product labels was 3000 mg/day).

Ertugliflozin 5 mg

Ertugliflozin 5 mg, placebo for ertugliflozin (1 mg or 5 mg and 25 mg), and placebo to sitagliptin, oral, once daily for 84 days

Group Type EXPERIMENTAL

Placebo to Ertugliflozin

Intervention Type DRUG

Tablet(s), 1 or 2, matching placebo to 1-mg, 5-mg and/or 25-mg tablets, once daily for 84 days

Ertugliflozin 5 mg

Intervention Type DRUG

Tablet(s), 1 or 2, 5-mg tablets once daily for 84 days

Placebo to Sitagliptin

Intervention Type DRUG

Tablet, matching placebo to 100 mg, once daily for 84 days

Metformin

Intervention Type DRUG

Participants continued pre-study stable doses of metformin during the run-in and treatment periods of the study (maximum dose up to 2500 mg/day or 3000 mg/day where the maximum metformin dose per the local country product labels was 3000 mg/day).

Ertugliflozin 10 mg

Ertugliflozin 10 mg, placebo for ertugliflozin (25 mg), and placebo to sitagliptin, oral, once daily for 84 days

Group Type EXPERIMENTAL

Placebo to Ertugliflozin

Intervention Type DRUG

Tablet(s), 1 or 2, matching placebo to 1-mg, 5-mg and/or 25-mg tablets, once daily for 84 days

Ertugliflozin 5 mg

Intervention Type DRUG

Tablet(s), 1 or 2, 5-mg tablets once daily for 84 days

Placebo to Sitagliptin

Intervention Type DRUG

Tablet, matching placebo to 100 mg, once daily for 84 days

Metformin

Intervention Type DRUG

Participants continued pre-study stable doses of metformin during the run-in and treatment periods of the study (maximum dose up to 2500 mg/day or 3000 mg/day where the maximum metformin dose per the local country product labels was 3000 mg/day).

Ertugliflozin 25 mg

Ertugliflozin 25 mg, placebo for ertugliflozin (1 mg or 5 mg), and placebo to sitagliptin, oral, once daily for 84 days

Group Type EXPERIMENTAL

Placebo to Ertugliflozin

Intervention Type DRUG

Tablet(s), 1 or 2, matching placebo to 1-mg, 5-mg and/or 25-mg tablets, once daily for 84 days

Ertugliflozin 25 mg

Intervention Type DRUG

Tablet, 25 mg, once daily for 84 days

Placebo to Sitagliptin

Intervention Type DRUG

Tablet, matching placebo to 100 mg, once daily for 84 days

Metformin

Intervention Type DRUG

Participants continued pre-study stable doses of metformin during the run-in and treatment periods of the study (maximum dose up to 2500 mg/day or 3000 mg/day where the maximum metformin dose per the local country product labels was 3000 mg/day).

Sitagliptin 100 mg

Sitagliptin 100 mg, placebo for ertugliflozin (1 mg or 5 mg and 25 mg), oral, once daily for 84 days

Group Type ACTIVE_COMPARATOR

Placebo to Ertugliflozin

Intervention Type DRUG

Tablet(s), 1 or 2, matching placebo to 1-mg, 5-mg and/or 25-mg tablets, once daily for 84 days

Sitagliptin 100 mg

Intervention Type DRUG

Tablet, 100 mg, once daily for 84 days

Metformin

Intervention Type DRUG

Participants continued pre-study stable doses of metformin during the run-in and treatment periods of the study (maximum dose up to 2500 mg/day or 3000 mg/day where the maximum metformin dose per the local country product labels was 3000 mg/day).

Interventions

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Placebo to Ertugliflozin

Tablet(s), 1 or 2, matching placebo to 1-mg, 5-mg and/or 25-mg tablets, once daily for 84 days

Intervention Type DRUG

Ertugliflozin 1 mg

Tablet, 1 mg, once daily for 84 days

Intervention Type DRUG

Ertugliflozin 5 mg

Tablet(s), 1 or 2, 5-mg tablets once daily for 84 days

Intervention Type DRUG

Ertugliflozin 25 mg

Tablet, 25 mg, once daily for 84 days

Intervention Type DRUG

Sitagliptin 100 mg

Tablet, 100 mg, once daily for 84 days

Intervention Type DRUG

Placebo to Sitagliptin

Tablet, matching placebo to 100 mg, once daily for 84 days

Intervention Type DRUG

Metformin

Participants continued pre-study stable doses of metformin during the run-in and treatment periods of the study (maximum dose up to 2500 mg/day or 3000 mg/day where the maximum metformin dose per the local country product labels was 3000 mg/day).

Intervention Type DRUG

Other Intervention Names

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Januvia®, Tesavel®, Xelevia®, Ristaben® Fortamet®, Glucophage®, Glucophage® XR, Glumetza®, Riomet®, Metgluco®, Glycoran®

Eligibility Criteria

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Inclusion Criteria

* Participants with type 2 diabetes on stable doses of background medicines for management of the diabetes; aged 18-70 years; body mass index between 23-45 kg/m\^2

Exclusion Criteria

* Participants with type 1 diabetes, heart attack or stroke in last 6-months, uncontrolled blood pressure, significant kidney disease
Minimum Eligible Age

18 Years

Maximum Eligible Age

70 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

No

Sponsors

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Pfizer

INDUSTRY

Sponsor Role collaborator

Merck Sharp & Dohme LLC

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Principal Investigators

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Medical Director

Role: STUDY_DIRECTOR

Merck Sharp & Dohme LLC

References

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Amin NB, Wang X, Jain SM, Lee DS, Nucci G, Rusnak JM. Dose-ranging efficacy and safety study of ertugliflozin, a sodium-glucose co-transporter 2 inhibitor, in patients with type 2 diabetes on a background of metformin. Diabetes Obes Metab. 2015 Jun;17(6):591-598. doi: 10.1111/dom.12460. Epub 2015 Mar 31.

Reference Type RESULT
PMID: 25754396 (View on PubMed)

Fediuk DJ, Sahasrabudhe V, Dawra VK, Zhou S, Sweeney K. Population Pharmacokinetic Analyses of Ertugliflozin in Select Ethnic Populations. Clin Pharmacol Drug Dev. 2021 Nov;10(11):1297-1306. doi: 10.1002/cpdd.970. Epub 2021 Jul 2.

Reference Type DERIVED
PMID: 34213819 (View on PubMed)

Other Identifiers

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B1521006

Identifier Type: OTHER

Identifier Source: secondary_id

2009-017131-18

Identifier Type: EUDRACT_NUMBER

Identifier Source: secondary_id

8835-016

Identifier Type: -

Identifier Source: org_study_id

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