Efficacy and Safety of LCZ696A in Patients With Essential Hypertension

NCT ID: NCT00549770

Last Updated: 2015-08-25

Study Results

Results available

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Basic Information

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Recruitment Status

COMPLETED

Clinical Phase

PHASE2

Total Enrollment

1334 participants

Study Classification

INTERVENTIONAL

Study Start Date

2007-09-30

Study Completion Date

2008-07-31

Brief Summary

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This study was a dose-ranging efficiacy study in patients with essential hypertension to assess the blood pressure lowering effect, and safety of LCZ696 compared to valsartan and placebo. The study will also evaluate the efficacy and safety of AHU377 as compared to placebo.

Detailed Description

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Conditions

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Hypertension

Study Design

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Allocation Method

RANDOMIZED

Intervention Model

PARALLEL

Primary Study Purpose

TREATMENT

Blinding Strategy

DOUBLE

Participants Investigators

Study Groups

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LCZ696 100 mg

Participants received LCZ696 100 mg and matching placebo to LCZ696, Valsartan and AHU377 (5 tablets and 2 capsules) daily.

Group Type EXPERIMENTAL

LCZ696

Intervention Type DRUG

Placebo

Intervention Type DRUG

LCZ696 200 mg

Participants received LCZ696 200 mg and matching placebo to LCZ696, Valsartan and AHU377 (5 tablets and 2 capsules) daily.

Group Type EXPERIMENTAL

LCZ696

Intervention Type DRUG

Placebo

Intervention Type DRUG

LCZ696 400 mg

Participants received LCZ696 400 mg (200 mg LCZ696 for one week and then up-titration to 400 mg LCZ696 for 7 weeks) and matching placebo to LCZ696, Valsartan and AHU377 (5 tablets and 2 capsules) daily.

Group Type EXPERIMENTAL

LCZ696

Intervention Type DRUG

Placebo

Intervention Type DRUG

Valsartan 80 mg

Participants received Valsartan 80 mg and matching placebo to LCZ696, Valsartan and AHU377 (5 tablets and 2 capsules) daily.

Group Type ACTIVE_COMPARATOR

Valsartan

Intervention Type DRUG

Placebo

Intervention Type DRUG

Valsartan 160 mg

Participants received Valsartan 160 mg and matching placebo to LCZ696, Valsatan and AHU377 (5 tablets and 2 capsules) daily.

Group Type ACTIVE_COMPARATOR

Valsartan

Intervention Type DRUG

Placebo

Intervention Type DRUG

Valsartan 320 mg

Participants received Valsartan 320 mg (160 mg valsartan capsules for one week followed by 320 mg valsartan capsules for 7 weeks) and matching placebo to LCZ696, Valsartan and AHU377 (5 tablets and 2 capsules) daily.

Group Type ACTIVE_COMPARATOR

Valsartan

Intervention Type DRUG

Placebo

Intervention Type DRUG

AHU377 200 mg

Participants received AHU377 200 mg and matching placebo to LCZ696 and Valsartan (5 tablets and 2 capsules) daily.

Group Type EXPERIMENTAL

AHU377

Intervention Type DRUG

Placebo

Intervention Type DRUG

Placebo

Participants received matching placebo to LCZ696, Valsartan and AHU377 (5 tablets and 2 capsules) daily.

Group Type PLACEBO_COMPARATOR

Placebo

Intervention Type DRUG

Interventions

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LCZ696

Intervention Type DRUG

Valsartan

Intervention Type DRUG

AHU377

Intervention Type DRUG

Placebo

Intervention Type DRUG

Eligibility Criteria

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Inclusion Criteria

* Male or females from 18 up to and including 75 years
* Patients with mild-to-moderate uncomplicated essential hypertension, untreated or currently taking antihypertensive therapy (monotherapy or combination therapy of 2 drugs; therapy with a fixed dose combination of two active substances represents 2 drugs)
* Untreated patients must have had an office msDBP≥ 95 mmHg at the randomization visit (Visit 3) and the 2 preceding visits (Visits 1 and 2).
* Treated patients must have had an office msDBP≥ 90 mmHG after washout (Visit 2), and a msDBP\> 95 mmHg at baseline (Visit 3);

Exclusion Criteria

* Severe hypertension (msSBP ≥180 mmHg and/or msDBP ≥110 mmHg)
* History of angioedema, drug-related or otherwise, as reported by the patient
* Type 1 or Type 2 diabetes mellitus (according to the ADA criteria)
* History or evidence of a secondary form of hypertension, such as renal parenchymal hypertension, renovascular hypertension, coarctation of the aorta, primary hyperaldosteronism, Cushing's disease, drug-induced hypertension, unilateral or bilateral renal artery stenosis, pheochromocytoma, polycystic kidney disease, etc.
* History of angina pectoris, myocardial infarction, coronary bypass surgery, ischemic heart disease, surgical or percutaneous arterial intervention of any kind (coronary, carotid or peripheral intervention), stroke, TIA (transient ischemic attack), carotid artery stenosis, aortic aneurysm or peripheral arterial disease
Minimum Eligible Age

18 Years

Maximum Eligible Age

75 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

No

Sponsors

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Novartis Pharmaceuticals

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Principal Investigators

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Novartis Pharmaceuticals

Role: STUDY_DIRECTOR

Novartis Pharmaceuticals

Novartis Pharmaceuticals

Role: STUDY_CHAIR

Novartis Pharmaceuticals

Locations

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Novartis Investigative Site

Birmingham, Alabama, United States

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Muscle Shoals, Alabama, United States

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Chandler, Arizona, United States

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Buena Park, California, United States

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Fair Oaks, California, United States

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Long Beach, California, United States

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Los Angeles, California, United States

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Orangevale, California, United States

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Santa Ana, California, United States

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Stockton, California, United States

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Tustin, California, United States

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Jacksonville, Florida, United States

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Pembroke Pines, Florida, United States

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Pembroke Pines, Florida, United States

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Pensacola, Florida, United States

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Augusta, Georgia, United States

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Chicago, Illinois, United States

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Chicago, Illinois, United States

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Peoria, Illinois, United States

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Baton Rouge, Louisiana, United States

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Metairie, Louisiana, United States

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Chelsea, Michigan, United States

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Royal Oak, Michigan, United States

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Brooklyn Center, Minnesota, United States

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City of Saint Peters, Missouri, United States

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Toms River, New Jersey, United States

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Trenton, New Jersey, United States

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Cincinnati, Ohio, United States

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Cincinnati, Ohio, United States

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Oklahoma City, Oklahoma, United States

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Simpsonville, South Carolina, United States

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Dallas, Texas, United States

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Houston, Texas, United States

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Houston, Texas, United States

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Houston, Texas, United States

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Lake Jackson, Texas, United States

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Richmond, Virginia, United States

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Charleston, West Virginia, United States

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Caba, Buenos Aires, Argentina

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Caba, Buenos Aires, Argentina

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Caba, Buenos Aires, Argentina

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Corrientes, Corrientes Province, Argentina

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Rosario, Santa Fe Province, Argentina

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Cambridge, Ontario, Canada

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Mississauga, Ontario, Canada

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Toronto, Ontario, Canada

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Granby, Quebec, Canada

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Longueil, Quebec, Canada

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Montreal, Quebec, Canada

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Sherbrooke, Quebec, Canada

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Ste-Foy, Quebec, Canada

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Saskatoon, Saskatchewan, Canada

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Aalborg, , Denmark

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Aalborg SV, , Denmark

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Espergærde, , Denmark

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Greve, , Denmark

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Roslev, , Denmark

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Vaerloese, , Denmark

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Viborg, , Denmark

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Helsinki, , Finland

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Helsinki, , Finland

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Helsinki, , Finland

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Kerava, , Finland

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Oulu, , Finland

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Tampere, , Finland

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Bourges, , France

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La Chapelle-sur-Erdre, , France

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Saint-Avertin, , France

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Tours, , France

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Vihiers, , France

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Balve, , Germany

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Beckingen, , Germany

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Berlin, , Germany

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Berlin, , Germany

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Einbeck, , Germany

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Erfurt, , Germany

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Giengen an der Brenz, , Germany

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Hagen, , Germany

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Haigerloch, , Germany

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Hamburg, , Germany

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Kassel, , Germany

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Krefeld, , Germany

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Mahlberg, , Germany

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Messkirch, , Germany

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Reinfeld, , Germany

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Siegen, , Germany

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Wallerfing, , Germany

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Budapest, , Hungary

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Esztergom, , Hungary

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Miskolc, , Hungary

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Nyiregyháza, , Hungary

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Caserta, CE, Italy

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Cona, FE, Italy

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Florence, FI, Italy

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Pozzilli, IS, Italy

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Rozzano, MI, Italy

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Vimercate, MI, Italy

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Palermo, PA, Italy

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Padua, PD, Italy

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Pisa, PI, Italy

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Pisa, PI, Italy

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Casorate Primo, PV, Italy

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Pavia, PV, Italy

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Stradella, PV, Italy

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Mercato San Severino, SA, Italy

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Sassari, SS, Italy

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San Daniele del Friuli, UD, Italy

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Vibo Valentia, VV, Italy

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Daugavplis, , Latvia

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Kuldīga, , Latvia

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Ogre, , Latvia

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Alytus, , Lithuania

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Kaunas, , Lithuania

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Kaunas, , Lithuania

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Klaipėda, , Lithuania

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Losser, , Netherlands

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Oude Pekela, , Netherlands

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Poortvliet, , Netherlands

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Wamel, , Netherlands

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Ostrów Wielkopolski, , Poland

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Oława, , Poland

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Tarnów, , Poland

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Moscow, , Russia

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Moscow, , Russia

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S.-Petersburg, , Russia

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Saint Petersburg, , Russia

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Saint Petersburg, , Russia

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Banská Bystrica, Slovak Republic, Slovakia

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Bratislava, Slovak Republic, Slovakia

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Nitra, Slovak Republic, Slovakia

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Prešov, Slovak Republic, Slovakia

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Dunajská Streda, , Slovakia

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Žilina, , Slovakia

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Seville, Andalusia, Spain

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Palma de Mallorca, Balearic Islands, Spain

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Badalona, Catalonia, Spain

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Barcelona, Catalonia, Spain

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Barcelona, Catalonia, Spain

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Tàrrega, Catalonia, Spain

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Vic, Catalonia, Spain

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Begonte, Galicia, Spain

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Santiago de Compostela, Galicia, Spain

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Madrid, Madrid, Spain

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Alicante, Valencia, Spain

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Benidorm, Valencia, Spain

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Quart de Poblet, Valencia, Spain

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Valencia, Valencia, Spain

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Barcelona, , Spain

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Hospitalet de Llbregat, , Spain

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Petrel, , Spain

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Riudecols, , Spain

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Boden, Sweden, Sweden

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Skellefteå, Sweden, Sweden

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Arvidsjaur, , Sweden

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Karlstad, , Sweden

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Kil, , Sweden

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Kristianstad, , Sweden

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Lund, , Sweden

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Taipei, Taiwan, Taiwan

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Taipei, Taiwan, Taiwan

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Taichung, Taiwan ROC, Taiwan

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Tainan City, Taiwan ROC, Taiwan

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Changhua, , Taiwan

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Taichung County, , Taiwan

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Taipei, , Taiwan

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Countries

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United States Argentina Canada Denmark Finland France Germany Hungary Italy Latvia Lithuania Netherlands Poland Russia Slovakia Spain Sweden Taiwan

References

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Andersen MB, Simonsen U, Wehland M, Pietsch J, Grimm D. LCZ696 (Valsartan/Sacubitril)--A Possible New Treatment for Hypertension and Heart Failure. Basic Clin Pharmacol Toxicol. 2016 Jan;118(1):14-22. doi: 10.1111/bcpt.12453. Epub 2015 Sep 4.

Reference Type DERIVED
PMID: 26280447 (View on PubMed)

Ruilope LM, Dukat A, Bohm M, Lacourciere Y, Gong J, Lefkowitz MP. Blood-pressure reduction with LCZ696, a novel dual-acting inhibitor of the angiotensin II receptor and neprilysin: a randomised, double-blind, placebo-controlled, active comparator study. Lancet. 2010 Apr 10;375(9722):1255-66. doi: 10.1016/S0140-6736(09)61966-8. Epub 2010 Mar 16.

Reference Type DERIVED
PMID: 20236700 (View on PubMed)

Other Identifiers

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CLCZ696A2201

Identifier Type: -

Identifier Source: org_study_id

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