LY4268989 (MORF-057) Co-Administered With Mirikizumab in Adults With Moderately to Severely Active Ulcerative Colitis:

NCT ID: NCT07186101

Last Updated: 2025-11-12

Study Results

Results pending

The study team has not published outcome measurements, participant flow, or safety data for this trial yet. Check back later for updates.

Basic Information

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Recruitment Status

NOT_YET_RECRUITING

Clinical Phase

PHASE2

Total Enrollment

252 participants

Study Classification

INTERVENTIONAL

Study Start Date

2025-11-30

Study Completion Date

2029-03-31

Brief Summary

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The main purpose of the study is to evaluate the effectiveness and safety of LY4268989 when given with mirikizumab compared to mirikizumab alone in adult participants with moderately to severely active ulcerative colitis (UC).

Study participation will last approximately 118 weeks, including 104 weeks of treatment and may include up to 21 visits.

Detailed Description

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Conditions

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Ulcerative Colitis

Study Design

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Allocation Method

RANDOMIZED

Intervention Model

PARALLEL

Primary Study Purpose

TREATMENT

Blinding Strategy

DOUBLE

Participants Caregivers

Study Groups

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LY4268989 + Mirikizumab

LY4268989 administered orally (PO) + Mirikizumab administered intravenously (IV), then subcutaneously (SC). Responders will be re-randomized for Study Period 2.

Group Type EXPERIMENTAL

LY4268989

Intervention Type DRUG

Administered PO

Mirikizumab

Intervention Type DRUG

Administered IV then SC

Mirikizumab + LY4268989 Placebo

Mirikizumab administered IV, then SC + LY4268989 placebo administered PO. Responders and Non-responders will re-randomized for Study Period 2.

Group Type EXPERIMENTAL

Mirikizumab

Intervention Type DRUG

Administered IV then SC

LY4268989 Placebo

Intervention Type DRUG

Administered PO

Interventions

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LY4268989

Administered PO

Intervention Type DRUG

Mirikizumab

Administered IV then SC

Intervention Type DRUG

LY4268989 Placebo

Administered PO

Intervention Type DRUG

Other Intervention Names

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MORF-057 LY3074828

Eligibility Criteria

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Inclusion Criteria

* Have had an established diagnosis of ulcerative colitis (UC) of ≥3 months in before baseline, which includes endoscopic evidence of UC and a histopathology report that supports a diagnosis of UC
* Have moderately to severely active UC as defined by a Modified Mayo Score (mMS) of 5 to 9 with an Endoscopic Score (ES) ≥2 confirmed by central reader and rectal bleeding (RB) ≥1, with endoscopy performed within 21 days before baseline
* Participants with greater than 8 years of UC symptoms have documented evidence of having had a surveillance colonoscopy within 1 year, or according to local country or regional medical guidelines, to evaluate for polyps, dysplasia, or malignancy, prior to randomization
* Are up-to-date on colorectal cancer surveillance per local society guidelines
* Have an inadequate response to, loss of response to, or intolerance to at least 1 of the medications:
* Conventional-failed participants: Participants who have had an inadequate response to or a loss of response to or are intolerant to at least 1 of the following medications: corticosteroids or immunomodulators (Does not apply to US)

NOTE: After the interim analysis, participants with inadequate response, loss of response, or intolerance to conventional UC therapy without prior exposure to biologics may be enrolled if deemed appropriate (Applies to the US)

* Advanced therapy-failed participants: Participants who have an inadequate response to or a loss of response to, or are intolerant to advanced therapy for UC, defined as:

* a biologic or biosimilar medication such as anti-tumor necrosis factor (anti-TNF) antibodies or anti-interleukin antibodies (IL-12/23, or IL-23p19), except for

* mirikizumab.
* Janus kinase inhibitors (JAK) such as filgotinib, tofacitinib, or upadacitinib
* sphingosine 1-phosphate receptor 1 inhibitors (S1PR) such as etrasimod or ozanimod

Exclusion Criteria

* Have a current diagnosis of

* Crohn's disease
* Inflammatory Bowel Disease (IBD) unclassified (formerly known as indeterminate colitis), or
* primary sclerosing cholangitis
* Have had or will need bowel resection or intestinal or intra-abdominal surgery
* Have evidence of toxic megacolon, intra-abdominal abscess, or stricture or stenosis within small bowel or colon that cannot be traversed by a colonoscope or that are symptomatic
* Have any adenomatous polyp occurring in areas of the colon not involved by colitis, that has not been removed

Note: If such an adenomatous polyp has been completely removed and shows only low-grade dysplasia, this criterion would no longer apply

* Have a current or recent acute, active infection
Minimum Eligible Age

18 Years

Maximum Eligible Age

80 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

No

Sponsors

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Eli Lilly and Company

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Principal Investigators

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Call 1-877-CTLILLY (1-877-285-4559) or 1-317-615-4559 Mon - Fri 8 AM - 8 PM Eastern time (UTC/GMT - 5 hours, EST)

Role: STUDY_DIRECTOR

Eli Lilly and Company

Locations

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Mayo Clinic in Arizona - Scottsdale

Scottsdale, Arizona, United States

Site Status

Clinnova Research - Anaheim

Anaheim, California, United States

Site Status

Om Research LLC

Lancaster, California, United States

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Biopharma Informatic, LLC

Los Angeles, California, United States

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Peak Gastroenterology Associates

Colorado Springs, Colorado, United States

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NeoClinical Research

Hialeah, Florida, United States

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Encore Borland-Groover Clinical Research

Jacksonville, Florida, United States

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Clinical Research of Osceola

Kissimmee, Florida, United States

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Florida Research Institute

Lakewood Rch, Florida, United States

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Alliance Medical Research

Lighthouse PT, Florida, United States

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Atlantic Medical Research

Margate, Florida, United States

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Digestive and Liver Center of Florida

Orlando, Florida, United States

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Center for Gastrointestinal Health - Fairview Heights

Belleville, Illinois, United States

Site Status

Lakeshore Gastroenterology and Liver Disease Institute

Des Plaines, Illinois, United States

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GI Alliance - Glenview

Glenview, Illinois, United States

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Gi Alliance - Gurnee

Gurnee, Illinois, United States

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Gastroenterology Health Partners

New Albany, Indiana, United States

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Gastroenterology Health Partners

Louisville, Kentucky, United States

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Brigham and Women's Hospital

Boston, Massachusetts, United States

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Clinical Research Institute of Michigan, LLC

Clinton Township, Michigan, United States

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GI Associates - GIA and Endoscopy Center - Flowood

Flowood, Mississippi, United States

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Columbia University Irving Medical Center

New York, New York, United States

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Digestive Disease Medicine of Central New York

Utica, New York, United States

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Gastroenterology & Hepatology Specialists

Canton, Ohio, United States

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Dayton Gastroenterology, LLC

Dayton, Ohio, United States

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University Gastroenterology - Providence - West River Street

Providence, Rhode Island, United States

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Gastroenterology Associates, P.A. of Greenville

Greenville, South Carolina, United States

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Gastro One - Walnut Run Road

Cordova, Tennessee, United States

Site Status

Texas Digestive Disease Consultants - Cedar Park

Cedar Park, Texas, United States

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GI Alliance - Dallas - Gaston Avenue

Dallas, Texas, United States

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GI Alliance - Fort Worth

Fort Worth, Texas, United States

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GI Alliance - Garland

Garland, Texas, United States

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GI Alliance - Lubbock

Lubbock, Texas, United States

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Southern Star Research Institute

San Antonio, Texas, United States

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Tyler Research Institute

Tyler, Texas, United States

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GI Alliance-Webster

Webster, Texas, United States

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Care Access - Ogden

Ogden, Utah, United States

Site Status

Clinical Research Partners, LLC

Richmond, Virginia, United States

Site Status

GI Alliance - Richmond

Richmond, Virginia, United States

Site Status

Washington Gastroenterology - Bellevue

Bellevue, Washington, United States

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Uniklinikum Salzburg

Salzburg, , Austria

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Medizinische Universität Wien

Vienna, , Austria

Site Status

Chronos Pesquisa Clínica

Brasília, , Brazil

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CAEP - Synvia Labs

Campinas, , Brazil

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Fundação Universidade de Caxias do Sul (FUCS)

Caxias do Sul, , Brazil

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Centro Digestivo de Curitiba

Curitiba, , Brazil

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Galileo Medical Research

Juiz de Fora, , Brazil

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NewData Clinical Research - Maceió

Maceió, , Brazil

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Hospital Ernesto Dornelles

Porto Alegre, , Brazil

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Centro Internacional de Pesquisa Clínica (CIPES)

São José dos Campos, , Brazil

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CPQuali Pesquisa Clínica

São Paulo, , Brazil

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Solare Trials

São Paulo, , Brazil

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Hospital Santa Catarina - Paulista

São Paulo, , Brazil

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Clínica Hepatogastro JK

São Paulo, , Brazil

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Universidade Federal Do Piaui - Campos Universitario

Teresina, , Brazil

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Charlton Digestive Disease Centre

Hamilton, , Canada

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Victoria Hospital & Children's Hospital - London Health Sciences Centre

London, , Canada

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London Digestive Disease Institute

London, , Canada

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West GTA Research Inc.

Mississauga, , Canada

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C.I.C. Mauricie inc.

Trois-Rivières, , Canada

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Changzhou Second People's Hospital

Changzhou, , China

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Chongqing General Hospital

Chongqing, , China

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The First Affiliated Hospital Of Fujian Medical University

Fuzhou, , China

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Sir Run Run Shaw Hospital of Zhejiang University School of Medicine

Hangzhou, , China

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First Affiliated Hospital of Kunming Medical University

Kunming, , China

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Jiangsu Province Hospital

Nanjing, , China

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The Affiliated Hospital of Qingdao University

Qingdao, , China

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Shengjing Hospital of China Medical University

Shenyang, , China

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The Second Afilliated Hospital of Hebei Medical University

Shijiazhuang, , China

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Taian City Central Hospital

Taian, , China

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Wuhan Union Hospital

Wuhan, , China

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Wuxi People's Hospital

Wuxi, , China

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Aalborg Universitetshospital, Syd

Aalborg, , Denmark

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Aarhus Universitetshospital, Skejby

Aarhus, , Denmark

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Herlev and Gentofte Hospital

Copenhagen, , Denmark

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Odense Universitetshospital

Odense, , Denmark

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Charité Universitaetsmedizin Berlin - Campus Mitte

Berlin, , Germany

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Universitätsklinikum Regensburg

Regensburg, , Germany

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Universitaetsklinikum Ulm

Ulm, , Germany

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Békés Megyei Központi Kórház Dr. Réthy Pál Tagkórház

Békéscsaba, , Hungary

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Óbudai Egészségügyi Centrum

Budapest, , Hungary

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Semmelweis Egyetem

Budapest, , Hungary

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Pannónia Magánorvosi Centrum

Budapest, , Hungary

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Clinexpert Gyöngyös

Gyöngyös, , Hungary

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Komarom-Esztergom Varmegyei Szent Borbala Korhaz

Tatabánya, , Hungary

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Jávorszky Ödön Kórház

Vác, , Hungary

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Sardar Vallabhbhai Patel Institute of Medical Sciences and Research

Ahmedabad, , India

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Rajiv Gandhi Government General Hospital

Chennai, , India

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Ashwin Hospital

Coimbatore, , India

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Sushruta Multispeciality Hospital & Research Centre

Hubli, , India

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Mahavir Hospital & Research Centre - Hyderabad

Hyderabad, , India

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All India Institute of Medical Sciences

New Delhi, , India

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Medipoint Hospitals Pvt. Ltd.

Pune, , India

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Shree Giriraj Multispeciality Hospital

Rajkot, , India

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ASST Grande Ospedale Metropolitano Niguarda

Milan, , Italy

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Fondazione IRCCS Cà Granda Ospedale Maggiore Policlinico

Milan, , Italy

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Ospedale San Raffaele

Milan, , Italy

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Fondazione Policlinico Universitario Agostino Gemelli

Roma, , Italy

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Humanitas

Rozzano, , Italy

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Fukuoka University Hospital

Fukuoka, , Japan

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Gokeikai Ofuna Chuo Hospital

Kamakura, , Japan

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Tsujinaka Hospital - Kashiwanoha

Kashiwa, , Japan

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National Hospital Organization Osaka National Hospital

Osaka, , Japan

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Toho University Sakura Medical Center

Sakura, , Japan

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Sapporo Tokushukai Hospital

Sapporo, , Japan

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Scientia Investigacion Clinica S.C.

Chihuahua City, , Mexico

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Instituto de Investigaciones Aplicadas a la Neurociencia A.C.

Durango, , Mexico

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Boca Clinical Trials Mexico S.C.

Guadajalara, , Mexico

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Clinica de Investigacion en Reumatologia y Obesidad S. C.

Guadalajara, , Mexico

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Centro de Investigación y Gastroenterología - S.C.

Mexico City, , Mexico

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Centro de Investigación Clinica Chapultepec

Mexico City, , Mexico

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Instituto Nacional de Ciencias Medicas y Nutricion Salvador Zubiran

Mexico City, , Mexico

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Servicios de Oncología Médica Integral - Monterrey

San Pedro Garza García, , Mexico

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Scientia Investigacion Clinica S.C.

Tijuana, , Mexico

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Clinical Research Institute S.C.

Tlalnepantla, , Mexico

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Medimanage Research

Tlalpan, , Mexico

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FAICIC S. de R.L. de C.V.

Veracruz, , Mexico

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Radboudumc

Nijmegen, , Netherlands

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Elisabeth-TweeSteden Ziekenhuis

Tilburg, , Netherlands

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Gyncentrum sp. z o.o. NZOZ Holsamed - oddział Libero

Katowice, , Poland

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IRMED

Piotrkow Trybunalski, , Poland

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Pratia Poznań

Poznan, , Poland

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Uniwersyteckie Centrum Stomatologii i Medycyny Specjalistycznej

Poznan, , Poland

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Twoja Przychodnia SCM

Szczecin, , Poland

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Sonomed Sp. z o. o.

Szczecin, , Poland

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WSD MEDI

Warsaw, , Poland

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Medical Network Spółka z o.o. WIP Warsaw IBD Point Profesor Kierkuś

Warsaw, , Poland

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ETG Zamość

Zamość, , Poland

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Spitalul de Oncologie Monza

Bucharest, , Romania

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Delta Health Care

Bucharest, , Romania

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Spitalul Clinic Colentina

Bucharest, , Romania

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Constanta County Emergency Clinical Hospital Sf.Ap.Andrei

Constanța, , Romania

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Spital Judetean de Urgenta

Satu Mare, , Romania

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S.C Centrul de Gastroenterologie Dr. Goldis S.R.L

Timișoara, , Romania

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Centro Médico Teknon

Barcelona, , Spain

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Hospital Universitario de Fuenlabrada

Fuenlabrada, , Spain

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Hospital de Cabueñes

Gijón, , Spain

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Hospital Universitario La Paz

Madrid, , Spain

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Hospital Universitario Nuestra Señora de Candelaria

Santa Cruz de Tenerife, , Spain

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Adana City Hospital

Adana, , Turkey (Türkiye)

Site Status

Gazi University Health Research and Application Center Gazi Hospital

Ankara, , Turkey (Türkiye)

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Antalya Egitim ve Arastırma Hastanesi

Antalya, , Turkey (Türkiye)

Site Status

Eskisehir Osmangazi University

Eskişehir, , Turkey (Türkiye)

Site Status

Mustafa Kemal Universitesi

Hatay, , Turkey (Türkiye)

Site Status

Kocaeli University Medical Faculty Hospital

İzmit, , Turkey (Türkiye)

Site Status

İnönü Üniversitesi Turgut Özal Tıp Merkezi Eğitim ve Araştırma Hastanesi

Malatya, , Turkey (Türkiye)

Site Status

Mersin University

Mersin, , Turkey (Türkiye)

Site Status

Dicle Üniversitesi

Sur, , Turkey (Türkiye)

Site Status

Countries

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United States Austria Brazil Canada China Denmark Germany Hungary India Italy Japan Mexico Netherlands Poland Romania Spain Turkey (Türkiye)

Central Contacts

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Trial questions or participation questions: 1-877-CTLILLY (1-877-285-4559) or

Role: CONTACT

Phone: 1-317-615-4559

Email: [email protected]

Physicians interested in becoming principal investigators please contact

Role: CONTACT

Email: [email protected]

Facility Contacts

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Related Links

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https://trials.lilly.com/en-US/trial/655156

LY4268989 (MORF-057) Co-Administered With Mirikizumab in Adults With Moderately to Severely Active Ulcerative Colitis: (TOPAZ-UC)

Other Identifiers

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J6E-MC-KWAN

Identifier Type: OTHER

Identifier Source: secondary_id

MORF-057

Identifier Type: OTHER

Identifier Source: secondary_id

27704

Identifier Type: -

Identifier Source: org_study_id