A Study of DS5361b in Participants With Advanced Solid Tumors

NCT ID: NCT07182591

Last Updated: 2025-10-10

Study Results

Results pending

The study team has not published outcome measurements, participant flow, or safety data for this trial yet. Check back later for updates.

Basic Information

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Recruitment Status

RECRUITING

Clinical Phase

PHASE1

Total Enrollment

192 participants

Study Classification

INTERVENTIONAL

Study Start Date

2025-10-02

Study Completion Date

2030-12-03

Brief Summary

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This study aims to assess the safety, tolerability, and preliminary efficacy and to determine the MTD of DS5361b in monotherapy and combination with pembrolizumab in participants with advanced or metastatic solid tumors.

Detailed Description

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Conditions

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Advanced Solid Tumor

Keywords

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First-in-Human Advanced Solid Tumors

Study Design

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Allocation Method

NON_RANDOMIZED

Intervention Model

SEQUENTIAL

Primary Study Purpose

TREATMENT

Blinding Strategy

NONE

Study Groups

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Part 1: Monotherapy (Dose Escalation)

Participants will receive DS5361b at escalating doses.

Group Type EXPERIMENTAL

DS5361b

Intervention Type DRUG

Dose Escalation Part: DS5361b will be administered at escalating doses to determine the RDE.

Dose Expansion Part: DS5361b will be administered at RDE.

Part 2: Combination Therapy (Dose Escalation)

Participants will receive DS5361b at escalating doses in combination with Pembrolizumab.

Group Type EXPERIMENTAL

DS5361b

Intervention Type DRUG

Dose Escalation Part: DS5361b will be administered at escalating doses to determine the RDE.

Dose Expansion Part: DS5361b will be administered at RDE.

Pembrolizumab

Intervention Type DRUG

Dose Escalation Part: Pembrolizumab will be administered at a standard dose.

Dose Expansion Part: Pembrolizumab will be administered at a standard dose.

Part 3: Combination Therapy (Dose Expansion)

Participants will receive DS5361b in combination with Pembrolizumab at the recommended dose for expansion (RDE).

Group Type EXPERIMENTAL

DS5361b

Intervention Type DRUG

Dose Escalation Part: DS5361b will be administered at escalating doses to determine the RDE.

Dose Expansion Part: DS5361b will be administered at RDE.

Pembrolizumab

Intervention Type DRUG

Dose Escalation Part: Pembrolizumab will be administered at a standard dose.

Dose Expansion Part: Pembrolizumab will be administered at a standard dose.

Interventions

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DS5361b

Dose Escalation Part: DS5361b will be administered at escalating doses to determine the RDE.

Dose Expansion Part: DS5361b will be administered at RDE.

Intervention Type DRUG

Pembrolizumab

Dose Escalation Part: Pembrolizumab will be administered at a standard dose.

Dose Expansion Part: Pembrolizumab will be administered at a standard dose.

Intervention Type DRUG

Other Intervention Names

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Keytruda®

Eligibility Criteria

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Inclusion Criteria

1. Adults ≥18 years of age at the time the ICF is signed (Please follow local regulatory requirements if the legal age of consent for trial participation is \>18 years old).
2. Has histologically- or cytologically documented recurrent, metastatic, or unresectable solid tumors that are refractory to or intolerable with standard treatment or for which no standard treatment is available (For Part 1 and Part 2 only).
3. Participants need to have documented TMB or MSI status using a validated or approved genomic test as per applicable regulations prior to Cycle 1 Day 1. In Part 1 and Part 2, participants need to have documented TMB-H and/or MSI-H status. In Part 3, participants need to have documented TMB-H status.
4. Has measurable disease based on local CT/MRI imaging as assessment by the investigator using RECIST v1.1.
5. Eastern Cooperative Oncology Group (ECOG) Performance Status of 0-1.
6. Has adequate organ and bone marrow function as assessed by local laboratory within 14 days prior to initiation of trial intervention.
7. For HNSCC participants only: have documented results from local testing of HPV for oropharyngeal cancer. If HPV status has previously been tested using this procedure, no retesting is required.

Dose Expansion (Part 3) Only:
8. Has histologically or cytologically confirmed, Stage IV NSCLC without actionable gene alteration.

* No prior systemic therapy.
* Participants with PD-L1 TPS ≥1%.
9. Has histologically or cytologically confirmed recurrent or metastatic HNSCC that is considered incurable by local therapies.

* No prior systemic therapy administered in the recurrent or metastatic setting.
* Participants with PD-L1 CPS ≥1.

Exclusion Criteria

1. Has spinal cord compression or clinically active central nervous system metastases.
2. Has a history of leptomeningeal carcinomatosis.
3. Uncontrolled or significant cardiovascular disease.
4. Any of the following within the past 6 months prior to enrollment: cerebrovascular accident, transient ischemic attack, or other arterial thromboembolic event.
5. Has a history of (noninfectious) interstitial lung disease (ILD)/pneumonitis that required corticosteroids, has current ILD/pneumonitis, or where suspected ILD/pneumonitis cannot be ruled out.
6. Clinically severe pulmonary compromise (ie, requiring any supplemental oxygen).
7. Has any evidence of severe or uncontrolled systemic diseases.
8. Has active or uncontrolled HBV infection. Hepatitis B SCR testing is required.
9. Has active or uncontrolled HCV infection. Hepatitis C SCR testing is required.
10. For the dose escalation phase (Part 1 and Part 2), has HIV infection. For the dose expansion part (Part 3), has active or uncontrolled HIV infection.
11. Prior organ transplantation, including allogeneic stem cell transplantation.
12. Has an active, known, or suspected autoimmune disease.
13. Has a diagnosis of immunodeficiency or is receiving systemic steroid therapy or any other form of immunosuppressive therapy within 14 days prior to the trial intervention.
Minimum Eligible Age

18 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

No

Sponsors

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Daiichi Sankyo

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Locations

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Research Site

Irving, Texas, United States

Site Status RECRUITING

Research Site

San Antonio, Texas, United States

Site Status RECRUITING

Countries

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United States

Central Contacts

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Contact for Trial Information

Role: CONTACT

Phone: 908-992-6400

Email: [email protected]

Other Identifiers

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DS5361-061

Identifier Type: -

Identifier Source: org_study_id