A First-in-human, 3-part Study of MRT-8102 in Healthy Participants and Participants at Cardiovascular Risk With Elevated CRP

NCT ID: NCT07119125

Last Updated: 2025-10-10

Study Results

Results pending

The study team has not published outcome measurements, participant flow, or safety data for this trial yet. Check back later for updates.

Basic Information

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Recruitment Status

RECRUITING

Clinical Phase

PHASE1

Total Enrollment

100 participants

Study Classification

INTERVENTIONAL

Study Start Date

2025-06-27

Study Completion Date

2026-03-31

Brief Summary

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The principal aim of this study is to obtain safety and tolerability data when MRT-8102 is administered orally as single and multiple doses to healthy participants and participants at cardiovascular risk with elevated CRP. This information, together with the pharmacokinetic (PK) data, will help establish the dose and dosing regimen suitable for future studies.

The study drug, MRT-8102, is experimental. This is the first study in which MRT-8102 will be given to humans.

Part 1: Healthy participants will receive a single oral dose of MRT-8102 or placebo on Day 1

Part 2: Healthy participants will receive multiple oral doses of MRT-8102 or placebo for 7 consecutive days

Part 3: Participants at cardiovascular risk with elevated CRP will receive multiple oral doses of MRT-8102 or placebo for 28 consecutive days

Detailed Description

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The purpose of this study is to:

* Learn about the safety and tolerability of single and multiple ascending oral doses of MRT-8102 in healthy adult participants
* Learn about the safety and tolerability of 28-day daily dosing of MRT-8102 in participants at cardiovascular risk with elevated CRP

Conditions

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Healthy Volunteers Elevated CRP

Study Design

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Allocation Method

RANDOMIZED

Intervention Model

SEQUENTIAL

Primary Study Purpose

TREATMENT

Blinding Strategy

QUADRUPLE

Participants Caregivers Investigators Outcome Assessors

Study Groups

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Part 1: Single Ascending Dose (MRT-8102)

Single Dose of MRT-8102

Group Type EXPERIMENTAL

MRT-8102

Intervention Type DRUG

Oral capsules

Part 1: Single Ascending Dose (Placebo)

Single Dose of Placebo

Group Type PLACEBO_COMPARATOR

Placebo

Intervention Type DRUG

Oral capsules

Part 2: Multiple Ascending Dose (MRT-8102)

7-day Daily Dose of MRT-8102

Group Type EXPERIMENTAL

MRT-8102

Intervention Type DRUG

Oral capsules

Part 2: Multiple Ascending Dose (Placebo)

7-day Daily Dose of Placebo

Group Type PLACEBO_COMPARATOR

Placebo

Intervention Type DRUG

Oral capsules

Part 3: elevated CRP (MRT-8102)

28-day Daily Dose of MRT-8102

Group Type EXPERIMENTAL

MRT-8102

Intervention Type DRUG

Oral capsules

Part 3: elevated CRP (Placebo)

28-day Daily Dose of Placebo

Group Type PLACEBO_COMPARATOR

Placebo

Intervention Type DRUG

Oral capsules

Interventions

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MRT-8102

Oral capsules

Intervention Type DRUG

Placebo

Oral capsules

Intervention Type DRUG

Eligibility Criteria

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Inclusion Criteria

* Healthy, adult, male or females 18-65 years of age
* Non-smoker who has not used nicotine- and tobacco -containing products for at least 3 months prior to start of study
* Able to swallow oral medications
* Abstain from caffeine- and methylxanthine-containing beverages or food


* Elevated CRP value ≥3.0 mg/L at the time of screening
* Evidence of cardiovascular risk factors
* No signs or symptoms of acute disease
* No ECG finding of clinical significance

Exclusion Criteria

* History or presence of clinically significant medical or psychiatric condition or disease
* Underwent surgical intervention or an operation withing 6 weeks prior to start of study
* Has active TB, latent TB, a history of TB, or had close contact with a person with active TB within 8 weeks prior to the first dosing
* Pregnant, breastfeeding, or planning a pregnancy or fathering a child during the study or within 3 months after the last study drug administration.
* Positive urine drug or alcohol screen results
* Positive results for human immunodeficiency virus (HIV), hepatitis B or Hepatitis C virus or history of resolved hepatitis
* Participation in another clinical study within 30 days or within 5 half-live (if known) prior to start of study
* Currently receiving other immunomodulators
* History of immunodeficiency, chronic inflammatory and chronic inflammation
Minimum Eligible Age

18 Years

Maximum Eligible Age

65 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

Yes

Sponsors

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Monte Rosa Therapeutics, Inc

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Locations

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Clinical Pharmacology of Miami, LLC

Miami, Florida, United States

Site Status RECRUITING

ICON Clinical Research

Lenexa, Kansas, United States

Site Status RECRUITING

QPS

Springfield, Missouri, United States

Site Status RECRUITING

Endeavor Clinical Trials

San Antonio, Texas, United States

Site Status RECRUITING

Countries

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United States

Central Contacts

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Monte Rosa Therapeutics Inc. Sponsor

Role: CONTACT

617-949-2643

Facility Contacts

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Investigative Site 002

Role: primary

(305) 817-2900

Investigative Site 001

Role: primary

(913) 259-7100

Investigative Site 003

Role: primary

(417) 893-6188

Investigative Site 004

Role: primary

(210) 949-0807

Other Identifiers

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MRT-8102-001

Identifier Type: -

Identifier Source: org_study_id

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